DOI: 10.1055/s-00000131

Synfacts

Current Issue 05 · Volume 2010 · May 2010 DOI: 10.1055/s-002-20986

Synform

A39

Synthesis of Natural Products and Potential Drugs

0501
Seiple, I. B.; Su, S.; Young, I. S.; Lewis, C. A.; Yamaguchi, J.; Baran, P. S.: Synthesis of Palau’amine
0502
Stowe, G. N.; Silhár, P.; Hixon, M. S.; Silvaggi, N. R.; Allen, K. N.; Moe, S. T.; Jacobson, A. R.; Barbieri, J. T.; Janda, K. D.: Synthesis of a Botulinum Protease Inhibitor
0503
Liang, J.; Lalonde, J.; Borup, B.; Mitchell, V.; Mundorff, E.; Trinh, N.; Kochrekar, D. A.; Cherat, R. N.; Pai, G. G.: Synthesis of Montelukast
0504
0505
Nakamura, Y.; Burke, A. M.; Kotani, S.; Ziller, J. W.; Rychnovsky, S. D.: Synthesis of (-)-Lycoperine A
0506
Bouyssou, T.; Hoenke, C.; Rudolf, K.; Lustenberger, P.; Pestel, S.; Sieger, P.; Lotz, R.; Heine, C.; Büttner, F. H.; Schnapp, A.; Konetzki, I.: Synthesis of (R)-Olodaterol
0508
Lorenz, J. C.; al., C. A. Busacca et: Synthesis of a Cathepsin S Inhibitor
0509
Francais, A.; Leyva, A.; Etxebarria-Jardi, G.; Ley, S. V.: Synthesis of Iso- and Bongkrekic Acids
0510
Shimizu, Y.; Shi, S.-L.; Usuda, H.; Kanai, M.; Shibasaki, M.: Synthesis of ent-Hyperforin
0511
Nakajima, R.; Ogino, T.; Yokoshima, S.; Fukuyama, T.: Synthesis of (-)-Mersicarpine
0512
Björklund, C.; Oscarson, S.; Benkestock, K.; Borkakoti, N.; Jansson, K.; Lindberg, J.; Vrang, L.; Hallberg, A.; Rosenquist, Å.; Samuelsson, B.: Synthesis of a BACE-1 Inhibitor
0513
Magnus, N. A.; Campagna, S.; Confalone, P. N.; Savage, S.; Meloni, D. J.; Waltermire, R. E.; Wethman, R. G.; Yates, M.: Synthesis of BMS-561392

Synthesis of Heterocycles

0515
Vorobyeva, D. V.; Karimova, N. M.; Vasilyeva, T. P.; Osipov, S. N.; Shchetnikov, G. T.; Odinets, I. L.; Röschenthaler, G.-V.: Copper-Catalyzed Synthesis of Triazolyl-α-CF3-α-Aminophosphonates
0516
Oh, C. H.; Karmakar, S.; Park, H.; Ahn, Y.; Kim, J. W.: Silver-Catalyzed Heteroannulation Route to Indoles
0517
Pews-Davtyan, A.; Tillack, A.; Schmöle, A.-C.; Ortinau, S.; Frech, M. J.; Rolfs, A.; Beller, M.: Zinc Halide Mediated Synthesis of 3-Amidoindoles
0518
0519
Spiteri, C.; Sharma, P.; Zhang, F.; Macdonald, S. J. F.; Keeling, S.; Moses, J. E.: Synthesis of 1,2-Benzisoxazoles by 1,3-Dipolar Cycloaddition
0522
Reichelt, A.; Falsey, J. R.; Rzasa, R. M.; Thiel, O. R.; Achmatowicz, M. M.; Larsen, R. D.; Zhang, D.: Triazolopyridines via Selective Palladium-Catalyzed Monoarylation of Hydrazides
0524
0526
Gorugantula, S. P.; Carrero-Martínez, G. M.; Dantale, S. W.; Söderberg, B. C. G.: Palladium-Catalyzed Synthesis of Pyrrolo-Fused Compounds from Nitroarenes
0528

Synthesis of Materials and Unnatural Products

0529
Chen, G.; Mahmud, I.; Dawe, L. N.; Zhao, Y.: Conformation Switching
0530
Matsumoto, K.; Inokuchi, D.; Hirao, Y.; Kurata, H.; Sato, K.; Takui, T.; Kubo, T.: Stable Triplet TMM Diradical
0532
Arroyave, F. A.; Reynolds, J. R.: Decarboxylative Cross-Coupling
0533
0534
Amb, C. M.; Beaujuge, P. M.; Reynolds, J. R.: Switchable Electrochromic Polymers
0535
Ueda, A.; Nishida, S.; Fukui, K.; Ise, T.; Shiomi, D.; Sato, K.; Takui, T.; Nakasuji, K.; Morita, Y.: Radical Corannulene
0536
Gidron, O.; Diskin-Posner, Y.; Bendikov, M.: Furan Oligomers
0537
Yoshida, H.; Okada, K.; Kawashima, S.; Tanino, K.; Ohshita, J.: 1,2-Diborylation of Arynes
0538
Cangelosi, V. M.; Zakharov, L. N.; Johnson, D. W.: Self-Assembled Cryptands with Sulfur-Phosphorus Bonds
0539
Shinamura, S.; Miyazaki, E.; Takimiya, K.: New Heteroarene Cores for Organic Semiconductors
0540
Rivera-Fuentes, P.; Alonso-Gómez, J. L.; Petrovic, A. G.; Santoro, F.; Harada, N.; Berova, N.; Diederich, F.: Alleno-Acetylenic Oligomers
0541
Figueira-Duarte, T. M.; Rosso, P. G. Del; Trattnig, R.; Sax, S.; List, E. J. W.; Müllen, K.: High Molecular Weight Polypyrene
0542
Wang, F.; Zhang, J.; Ding, X.; Dong, S.; Liu, M.; Zheng, B.; Li, S.; Wu, L.; Yu, Y.; Gibson, H. W.; Huang, F.: Reversible Conversion between Linear and Cross-Linked Supramolecular Polymers
0543
Bouffard, J.; Watanabe, M.; Takaba, H.; Itami, K.: Active Material and Photoresist in One Novel Polymer

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0548
Poisson, T.; Tsubogo, T.; Yamashita, Y.; Kobayashi, S.: Calcium-PyBox Catalyzed Asymmetric Mannich Reaction of Imines
0549
Weickgenannt, A.; Mewald, M.; Muesmann, T. W. T.; Oestreich, M.: Kinetic Resolution of Alcohols Through Si-O Coupling
0550
Yeom, H.-S.; Lee, Y.; Jeong, J.; So, E.; Hwang, S.; Lee, J.-E.; Lee, S. S.; Shin, S.: Gold-Catalyzed Cascade Reaction of Tethered Nitrone-Propargyl Alcohols
0551
Fandrick, D. R.; Johnson, C. S.; Fandrick, K. R.; Reeves, J. T.; Tan, Z.; Lee, H.; Song, J. J.; Yee, N. K.; Senanayake, C. H.: Diastereoselective Zinc-Catalyzed Propargylation of Chiral Imines
0552
Woo, C. M.; Lu, L.; Gholap, S. L.; Smith, D. R.; Herzon, S. B.: Expedient Total Synthesis of Kinamycin F
0553
Hargrave, J. D.; Allen, J. C.; Kociok-Köhn, G.; Bish, G.; Frost, C. G.: Asymmetric Dieckmann-Type Annulation
0554
Hou, G.; Tan, R.; Sun, Y.; Zhang, X.; Gosselin, F.: Iridium-Catalyzed Asymmetric Hydrogenation of Benzophenone N-H Imines
0555
Nishimura, T.; Kawamoto, T.; Nagaosa, M.; Kumamoto, H.; Hayashi, T.: Rhodium-Catalyzed Asymmetric Cycloisomerization of 1,6-Enynes
0556
0558
Cérat, P.; Gritsch, P. J.; Goudreau, S. R.; Charette, A. B.: Synthesis of Enantioenriched Allenes from 1,1-Cyclopropanediesters
0559
Bedke, D. K.; Shibuya, G. M.; Pereira, A. R.; Gerwick, W. H.; Vanderwal, C. D.: Enantioselective Synthesis of Malhamensilipin A
0561
Chakrabarti, A.; Konishi, H.; Yamaguchi, M.; Schneider, U.; Kobayashi, S.: Indium(I)-Catalyzed Allylation and Crotylation of Imines
0562
0566
Limanto, J.; Krska, S. W.; Dorner, B. T.; Vazquez, E.; Yoshikawa, N.; Tan, L.: Ru-Catalyzed Dynamic Kinetic Resolution of β-Keto Amides via Transfer Hydrogenation
0569
Brekan, J. A.; Reynolds, T. E.; Scheidt, K. A.: Enantioselective Synthesis of Substituted Indanones
0572

Metal-Mediated Synthesis

0575
0576
Mo, F.; Jiang, Y.; Qiu, D.; Zhang, Y.; Wang, J.: Direct Conversion of Aryl Amines to Pinacol Boronates
0577
Das, S.; Addis, D.; Zhou, S.; Junge, K.; Beller, M.: Zinc(II)-Catalyzed Chemoselective Reduction of Amides to Amines
0578
Fujihara, T.; Katafuchi, Y.; Iwai, T.; Terao, J.; Tsuji, Y.: Palladium-Catalyzed Intermolecular Addition of Formamides to Alkynes
0580
Lundgren, R. J.; Sappong-Kumankumah, A.; Stradiotto, M.: A General Catalyst System for Amination of Aryl Chlorides
0581
Xi, P.; Yang, F.; Qin, S.; Zhao, D.; Lan, J.; Gao, G.; Hu, C.; You, J.: Oxidative C-H/C-H Cross-Coupling of Heteroarenes
0582
Nagaki, A.; Kim, H.; Usutani, H.; Matsuo, C.; Yoshida, J.-i.: Bromine-Lithium Exchange on Cyano-Substituted Arenes Using Microreactors
0584
0585
Voituriez, A.; Zimmer, L. E.; Charette, A. B.: A New Phosphate Zinc Carbenoid
0586
Saidi, O.; Blacker, A. J.; Farah, M. M.; Marsden, S. P.; Williams, J. M. J.: Iridium-Catalyzed Amine Alkylation with Alcohols in Water
0588
Xu, H.-J.; Zheng, F.-Y.; Liang, Y.-F.; Cai, Z.-Y.; Feng, Y.-S.; Che, D.-Q.: Simple Copper Chloride Catalyzed Arylation of Amines and Pyrrole in Water
0589
Kang, F.-A.; Lanter, J. C.; Cai, C.; Sui, Z.; Murray, W. V.: Dehydrative Pd/Cu-Catalyzed Coupling of Heterocycles with Terminal Alkynes

Organo- and Biocatalysis

0593
Lehwald, P.; Richter, M.; Röhr, C.; Liu, H.-W.; Müller, M.: Enzyme-Catalyzed Carboligations by Thiamine Diphosphate Dependent YerE
0596
Köhler, V.; Bailey, K. R.; Znabet, A.; Raftery, J.; Helliwell, M.; Turner, N. J.: Desymmetrization of meso-Pyrrolidines via Biocatalytic C-H Oxidation
0597
Whitehead, D. C.; Yousefi, R.; Jaganathan, A.; Borhan, B.: Organocatalytic Enantioselective Chlorolactonization
0598
Wang, X.-F.; Chen, J.-R.; Cao, Y.-J.; Cheng, H.-G.; Xiao, W.-J.: A Hydrogen Bonding Catalyzed Asymmetric Cascade to Tetrahydrocarbazoles
0599
Itsuno, S.; Paul, D. K.; Salam, M. A.; Haraguchi, N.: An Ionic Network as Catalyst for Asymmetric Benzylation
0600
Chen, Y.-J.; Seki, K.; Yamashita, Y.; Kobayashi, S.: Synthesis of Amines Using Aminoalkane Surrogates
0601
Xu, H.; Zuend, S. J.; Woll, M. G.; Tao, Y.; Jacobsen, E. N.: Asymmetric Povarov Reactions Cobalt-Catalyzed by Chiral Ureas/Achiral Acids
0603
0604
Fowler, B. S.; Mikochik, P. J.; Miller, S. J.: Kinetic Resolution of Thioformamides

Polymer-Supported Synthesis

0605
Itsuno, S.; Paul, D. K.; Ishimoto, M.; Haraguchi, N.: A Chiral Ionene for Asymmetric Benzylation
0606
Lee, T.; Lee, D.; Lee, I. Y.; Gong, Y.-D.: Solid-Phase Synthesis of Thiazolo[4,5-b]-pyridines
0607
Wittmann, S.; Schätz, A.; Grass, R. N.; Stark, W. J.; Reiser, O.: Graphene-Coated Cobalt Nanoparticles-Supported Palladium Catalyst
0610
0611
Shylesh, S.; Wagener, A.; Seifert, A.; Ernst, S.; Thiel, W. R.: One-Pot Reaction with Bifunctional Mesoporous Organosilicas
0612
Fang, W.; Zhang, Q.; Chen, J.; Deng, W.; Wang, Y.: Oxidant-Free Dehydrogenation of Alcohols with Au/HT
0613
Iwanami, K.; Seo, H.; Choi, J.-C.; Sakakura, T.; Yasuda, H.: Three-Component Strecker-Type Reaction with Al-MCM-41

Addenda and Errata