DOI: 10.1055/s-00000131

Synfacts

Issue 05 · Volume 2010 · May 2010 DOI: 10.1055/s-002-20986

Synform

A39
Zanda, Matteo: SYNFORM ISSUE 2010/05

Synthesis of Natural Products and Potential Drugs

z501
All PDFs of this category
0501
Seiple, I. B.; Su, S.; Young, I. S.; Lewis, C. A.; Yamaguchi, J.; Baran, P. S.: Synthesis of Palau’amine
0502
Stowe, G. N.; Silhár, P.; Hixon, M. S.; Silvaggi, N. R.; Allen, K. N.; Moe, S. T.; Jacobson, A. R.; Barbieri, J. T.; Janda, K. D.: Synthesis of a Botulinum Protease Inhibitor
0503
Liang, J.; Lalonde, J.; Borup, B.; Mitchell, V.; Mundorff, E.; Trinh, N.; Kochrekar, D. A.; Cherat, R. N.; Pai, G. G.: Synthesis of Montelukast
0504
Menz, H.; Kirsch, S. F.: Synthesis of Polyrhacitides A and B
0505
Nakamura, Y.; Burke, A. M.; Kotani, S.; Ziller, J. W.; Rychnovsky, S. D.: Synthesis of (-)-Lycoperine A
0506
Bouyssou, T.; Hoenke, C.; Rudolf, K.; Lustenberger, P.; Pestel, S.; Sieger, P.; Lotz, R.; Heine, C.; Büttner, F. H.; Schnapp, A.; Konetzki, I.: Synthesis of (R)-Olodaterol
0507
Cheng, X.; Waters, S. P.: Synthesis of Nankakurines A and B via Luciduline
0508
Lorenz, J. C.; al., C. A. Busacca et: Synthesis of a Cathepsin S Inhibitor
0509
Francais, A.; Leyva, A.; Etxebarria-Jardi, G.; Ley, S. V.: Synthesis of Iso- and Bongkrekic Acids
0510
Shimizu, Y.; Shi, S.-L.; Usuda, H.; Kanai, M.; Shibasaki, M.: Synthesis of ent-Hyperforin
0511
Nakajima, R.; Ogino, T.; Yokoshima, S.; Fukuyama, T.: Synthesis of (-)-Mersicarpine
0512
Björklund, C.; Oscarson, S.; Benkestock, K.; Borkakoti, N.; Jansson, K.; Lindberg, J.; Vrang, L.; Hallberg, A.; Rosenquist, Å.; Samuelsson, B.: Synthesis of a BACE-1 Inhibitor
0513
Magnus, N. A.; Campagna, S.; Confalone, P. N.; Savage, S.; Meloni, D. J.; Waltermire, R. E.; Wethman, R. G.; Yates, M.: Synthesis of BMS-561392

Synthesis of Heterocycles

z515
All PDFs of this category
0515
Vorobyeva, D. V.; Karimova, N. M.; Vasilyeva, T. P.; Osipov, S. N.; Shchetnikov, G. T.; Odinets, I. L.; Röschenthaler, G.-V.: Copper-Catalyzed Synthesis of Triazolyl-α-CF3-α-Aminophosphonates
0516
Oh, C. H.; Karmakar, S.; Park, H.; Ahn, Y.; Kim, J. W.: Silver-Catalyzed Heteroannulation Route to Indoles
0517
Pews-Davtyan, A.; Tillack, A.; Schmöle, A.-C.; Ortinau, S.; Frech, M. J.; Rolfs, A.; Beller, M.: Zinc Halide Mediated Synthesis of 3-Amidoindoles
0518
Dheur, J.; Sauthier, M.; Castanet, Y.; Mortreux, A.: Rhodium-Catalyzed Carbonylative Addition-Cyclization Approach to Furans
0519
Spiteri, C.; Sharma, P.; Zhang, F.; Macdonald, S. J. F.; Keeling, S.; Moses, J. E.: Synthesis of 1,2-Benzisoxazoles by 1,3-Dipolar Cycloaddition
0520
Devarie-Baez, N. O.; Xian, M.: One-Pot Synthesis of Benzisothiazoles from ortho-Mercaptoacylphenones
0521
Saito, T.; Furukawa, N.; Otani, T.: Pyrrolo[2,3-b]quinolines via a Rhodium-Catalyzed Pauson-Khand-Type Reaction
0522
Reichelt, A.; Falsey, J. R.; Rzasa, R. M.; Thiel, O. R.; Achmatowicz, M. M.; Larsen, R. D.; Zhang, D.: Triazolopyridines via Selective Palladium-Catalyzed Monoarylation of Hydrazides
0523
Meng, T.-j.; Hu, Y.; Wang, S.: Palladium-Catalyzed Synthesis of Five-Membered Heterocycles from 1,6-Enynes
0524
Zhang, Z.; Zhang, Q.; Ni, Z.; Liu, Q.: Silver-Mediated Synthesis of Furo[3,2-b]-β/γ-Lactams
0525
Yang, Q.; Alper, H.: Ligand-Free Cyclocarbonylation of ortho-Iodophenols and Acetylenes to Chromones
0526
Gorugantula, S. P.; Carrero-Martínez, G. M.; Dantale, S. W.; Söderberg, B. C. G.: Palladium-Catalyzed Synthesis of Pyrrolo-Fused Compounds from Nitroarenes
0527
Li, J.; Li, S.; Li, C.; Liu, Y.; Jia, X.: Tandem Conjugate Addition-Cyclization Synthesis of 1,5-Benzodiazepines
0528
Ma, D.; Geng, Q.; Zhang, H.; Jiang, Y.: Copper/l-Proline-Catalyzed Synthesis of Phenothiazines

Synthesis of Materials and Unnatural Products

z529
All PDFs of this category
0529
Chen, G.; Mahmud, I.; Dawe, L. N.; Zhao, Y.: Conformation Switching
0530
Matsumoto, K.; Inokuchi, D.; Hirao, Y.; Kurata, H.; Sato, K.; Takui, T.; Kubo, T.: Stable Triplet TMM Diradical
0531
Ishida, M.; Naruta, Y.; Tani, F.: Phenanthroline-Porphyrin Hybrid as a Fluorescence Sensor for Magnesium(II)
0532
Arroyave, F. A.; Reynolds, J. R.: Decarboxylative Cross-Coupling
0533
Xue, Z.; Mayer, M. F.: Self-Entangling in a [1]Rotaxane
0534
Amb, C. M.; Beaujuge, P. M.; Reynolds, J. R.: Switchable Electrochromic Polymers
0535
Ueda, A.; Nishida, S.; Fukui, K.; Ise, T.; Shiomi, D.; Sato, K.; Takui, T.; Nakasuji, K.; Morita, Y.: Radical Corannulene
0536
Gidron, O.; Diskin-Posner, Y.; Bendikov, M.: Furan Oligomers
0537
Yoshida, H.; Okada, K.; Kawashima, S.; Tanino, K.; Ohshita, J.: 1,2-Diborylation of Arynes
0538
Cangelosi, V. M.; Zakharov, L. N.; Johnson, D. W.: Self-Assembled Cryptands with Sulfur-Phosphorus Bonds
0539
Shinamura, S.; Miyazaki, E.; Takimiya, K.: New Heteroarene Cores for Organic Semiconductors
0540
Rivera-Fuentes, P.; Alonso-Gómez, J. L.; Petrovic, A. G.; Santoro, F.; Harada, N.; Berova, N.; Diederich, F.: Alleno-Acetylenic Oligomers
0541
Figueira-Duarte, T. M.; Rosso, P. G. Del; Trattnig, R.; Sax, S.; List, E. J. W.; Müllen, K.: High Molecular Weight Polypyrene
0542
Wang, F.; Zhang, J.; Ding, X.; Dong, S.; Liu, M.; Zheng, B.; Li, S.; Wu, L.; Yu, Y.; Gibson, H. W.; Huang, F.: Reversible Conversion between Linear and Cross-Linked Supramolecular Polymers
0543
Bouffard, J.; Watanabe, M.; Takaba, H.; Itami, K.: Active Material and Photoresist in One Novel Polymer

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z545
All PDFs of this category
0545
He, A.; Falck, J. R.: Stereospecific Suzuki Cross-Coupling
0546
Smith, S. M.; Takacs, J. M.: Asymmetric Hydroboration of Trisubstituted Alkenes
0547
Baeza, A.; Pfaltz, A.: Asymmetric Hydrogenation of N-Protected Indoles Catalyzed by Iridium Complexes
0548
Poisson, T.; Tsubogo, T.; Yamashita, Y.; Kobayashi, S.: Calcium-PyBox Catalyzed Asymmetric Mannich Reaction of Imines
0549
Weickgenannt, A.; Mewald, M.; Muesmann, T. W. T.; Oestreich, M.: Kinetic Resolution of Alcohols Through Si-O Coupling
0550
Yeom, H.-S.; Lee, Y.; Jeong, J.; So, E.; Hwang, S.; Lee, J.-E.; Lee, S. S.; Shin, S.: Gold-Catalyzed Cascade Reaction of Tethered Nitrone-Propargyl Alcohols
0551
Fandrick, D. R.; Johnson, C. S.; Fandrick, K. R.; Reeves, J. T.; Tan, Z.; Lee, H.; Song, J. J.; Yee, N. K.; Senanayake, C. H.: Diastereoselective Zinc-Catalyzed Propargylation of Chiral Imines
0552
Woo, C. M.; Lu, L.; Gholap, S. L.; Smith, D. R.; Herzon, S. B.: Expedient Total Synthesis of Kinamycin F
0553
Hargrave, J. D.; Allen, J. C.; Kociok-Köhn, G.; Bish, G.; Frost, C. G.: Asymmetric Dieckmann-Type Annulation
0554
Hou, G.; Tan, R.; Sun, Y.; Zhang, X.; Gosselin, F.: Iridium-Catalyzed Asymmetric Hydrogenation of Benzophenone N-H Imines
0555
Nishimura, T.; Kawamoto, T.; Nagaosa, M.; Kumamoto, H.; Hayashi, T.: Rhodium-Catalyzed Asymmetric Cycloisomerization of 1,6-Enynes
0556
Brichacek, M.; Batory, L. A.; Njardarson, J. T.: Copper-Catalyzed Stereoselective Ring Expansion of Vinyl Oxiranes
0557
Xu, Q.-L.; Dai, L.-X; You, S.-L.: Synthesis of Vinyl Sulfones by Isomerization of Allyl Sulfinates
0558
Cérat, P.; Gritsch, P. J.; Goudreau, S. R.; Charette, A. B.: Synthesis of Enantioenriched Allenes from 1,1-Cyclopropanediesters
0559
Bedke, D. K.; Shibuya, G. M.; Pereira, A. R.; Gerwick, W. H.; Vanderwal, C. D.: Enantioselective Synthesis of Malhamensilipin A
0560
Zhi, S.-J.; Sun, H.; Zhang, G.; Li, G.; Pan, Y.: Reverse Regioselectivity in Amino-halogenation of Electron-Deficient Olefins
0561
Chakrabarti, A.; Konishi, H.; Yamaguchi, M.; Schneider, U.; Kobayashi, S.: Indium(I)-Catalyzed Allylation and Crotylation of Imines
0562
Wender, P. A.; Stemmler, R. T.; Sirois, L. E.: Rhodium-Catalyzed [5+2] Cycloaddition-Nazarov Cyclization Strategy
0563
Mukherjee, S.; Corey, E. J.: Asymmetric Oxazaborolidine-Catalyzed Diels-Alder Reaction of Maleimides
0564
Giacomina, F.; Riat, D.; Alexakis, A.: Chiral Cycloalkenes by an Asymmetric Allylic Alkylation-RCM Procedure
0565
Cheng, H.; Stark, C. B. W.: Ruthenium-Catalyzed Oxidative Cylization of 5,6-Dihydroxy Alkenes
0566
Limanto, J.; Krska, S. W.; Dorner, B. T.; Vazquez, E.; Yoshikawa, N.; Tan, L.: Ru-Catalyzed Dynamic Kinetic Resolution of β-Keto Amides via Transfer Hydrogenation
0567
Grünanger, C. U.; Breit, B.: Rh-Catalyzed Regio- and Diastereoselective Hydroformylation of Bishomoallylic Alcohols
0568
Guan, X.-Y; Yang, L.-P.; Hu, W.: Multicomponent Asymmetric Synthesis of γ-Hydroxy Ketones
0569
Brekan, J. A.; Reynolds, T. E.; Scheidt, K. A.: Enantioselective Synthesis of Substituted Indanones
0570
Grimster, N.; Zhang, L.; Fokin, V. V.: Rhodium-Catalyzed Asymmetric Cyclopropanation via Azavinyl Carbenoids
0571
Han, S. B.; Han, H.; Krische, M. J.: Iridium-Catalyzed Asymmetric Alkoxy-allylation of Aldehydes
0572
Heitbaum, M.; Fröhlich, R.; Glorius, F.: Diastereoselective Hydrogenation of Substituted Quinolines
0573
Hadfield, M. S.; Lee, A.-L.: Synthesis of Tertiary Allylic Ethers by Gold(I) Catalysis

Metal-Mediated Synthesis

z575
All PDFs of this category
0575
Çalimsiz, S.; Sayah, M.; Mallik, D.; Organ, M. G.: Pd-PEPPSI-IPent as Catalyst for the Synthesis of Highly Congested Biaryls
0576
Mo, F.; Jiang, Y.; Qiu, D.; Zhang, Y.; Wang, J.: Direct Conversion of Aryl Amines to Pinacol Boronates
0577
Das, S.; Addis, D.; Zhou, S.; Junge, K.; Beller, M.: Zinc(II)-Catalyzed Chemoselective Reduction of Amides to Amines
0578
Fujihara, T.; Katafuchi, Y.; Iwai, T.; Terao, J.; Tsuji, Y.: Palladium-Catalyzed Intermolecular Addition of Formamides to Alkynes
0579
Vallée, F.; Mousseau, J. J.; Charette, A. B.: Iron(II)-Catalyzed Radical Arylation of Arenes with Aryl and Heteroaryl Iodides
0580
Lundgren, R. J.; Sappong-Kumankumah, A.; Stradiotto, M.: A General Catalyst System for Amination of Aryl Chlorides
0581
Xi, P.; Yang, F.; Qin, S.; Zhao, D.; Lan, J.; Gao, G.; Hu, C.; You, J.: Oxidative C-H/C-H Cross-Coupling of Heteroarenes
0582
Nagaki, A.; Kim, H.; Usutani, H.; Matsuo, C.; Yoshida, J.-i.: Bromine-Lithium Exchange on Cyano-Substituted Arenes Using Microreactors
0583
Kondoh, A.; Jamison, T. F.: Rhodium-Catalyzed Dehydrogenative Borylation of Cyclic Alkenes
0584
Shade, R. E.; Hyde, A. M.; Olsen, J.-C.; Merlic, C. A.: Allyl Vinyl Ethers by Copper-Promoted Coupling of Vinyl Boronates to Alcohols
0585
Voituriez, A.; Zimmer, L. E.; Charette, A. B.: A New Phosphate Zinc Carbenoid
0586
Saidi, O.; Blacker, A. J.; Farah, M. M.; Marsden, S. P.; Williams, J. M. J.: Iridium-Catalyzed Amine Alkylation with Alcohols in Water
0587
Ishiyama, T.; Isou, H.; Kikuchi, T.; Miyaura, N.: Iridium-Catalyzed ortho-Borylation of Benzoate Esters with Bis(pinacolato)diboron
0588
Xu, H.-J.; Zheng, F.-Y.; Liang, Y.-F.; Cai, Z.-Y.; Feng, Y.-S.; Che, D.-Q.: Simple Copper Chloride Catalyzed Arylation of Amines and Pyrrole in Water
0589
Kang, F.-A.; Lanter, J. C.; Cai, C.; Sui, Z.; Murray, W. V.: Dehydrative Pd/Cu-Catalyzed Coupling of Heterocycles with Terminal Alkynes

Organo- and Biocatalysis

z591
All PDFs of this category
0591
Vora, H. U.; Rovis, T.: Asymmetric Synthesis of α-Halo Carboxylic Acids from α,α-Dihalo Aldehydes
0592
Rana, N. K.; Selvakumar, S.; Singh, V. K.: Sulfa-Michael Addition Catalyzed by a Quinine-Derived Urea Catalyst
0593
Lehwald, P.; Richter, M.; Röhr, C.; Liu, H.-W.; Müller, M.: Enzyme-Catalyzed Carboligations by Thiamine Diphosphate Dependent YerE
0594
Hrdina, R.; Müller, C. E.; Schreiner, P. R.: Enantioselective Steglich Esterification for the Resolution of 1,2-Diols
0595
Abermil, N.; Masson, G.; Zhu, J.: Aza-Morita-Baylis-Hillman Reaction Using Aliphatic Imine Precursors
0596
Köhler, V.; Bailey, K. R.; Znabet, A.; Raftery, J.; Helliwell, M.; Turner, N. J.: Desymmetrization of meso-Pyrrolidines via Biocatalytic C-H Oxidation
0597
Whitehead, D. C.; Yousefi, R.; Jaganathan, A.; Borhan, B.: Organocatalytic Enantioselective Chlorolactonization
0598
Wang, X.-F.; Chen, J.-R.; Cao, Y.-J.; Cheng, H.-G.; Xiao, W.-J.: A Hydrogen Bonding Catalyzed Asymmetric Cascade to Tetrahydrocarbazoles
0599
Itsuno, S.; Paul, D. K.; Salam, M. A.; Haraguchi, N.: An Ionic Network as Catalyst for Asymmetric Benzylation
0600
Chen, Y.-J.; Seki, K.; Yamashita, Y.; Kobayashi, S.: Synthesis of Amines Using Aminoalkane Surrogates
0601
Xu, H.; Zuend, S. J.; Woll, M. G.; Tao, Y.; Jacobsen, E. N.: Asymmetric Povarov Reactions Cobalt-Catalyzed by Chiral Ureas/Achiral Acids
0602
Uyanik, M.; Yasui, T.; Ishihara, K.: Kita’s Oxidative Spirolactonization Catalyzed by a Hypervalent Iodine(III) Species
0603
Shao, P.-L.; Chen, X.-Y.; Sun, L.-H.; Ye, S.: NHC-Catalyzed Cycloaddition of Ketenes and 9,10-Phenanthrenequinone
0604
Fowler, B. S.; Mikochik, P. J.; Miller, S. J.: Kinetic Resolution of Thioformamides

Polymer-Supported Synthesis

z605
All PDFs of this category
0605
Itsuno, S.; Paul, D. K.; Ishimoto, M.; Haraguchi, N.: A Chiral Ionene for Asymmetric Benzylation
0606
Lee, T.; Lee, D.; Lee, I. Y.; Gong, Y.-D.: Solid-Phase Synthesis of Thiazolo[4,5-b]-pyridines
0607
Wittmann, S.; Schätz, A.; Grass, R. N.; Stark, W. J.; Reiser, O.: Graphene-Coated Cobalt Nanoparticles-Supported Palladium Catalyst
0608
Hirai, Y.; Uozumi, Y.: Buchwald-Hartwig Reaction with Amphiphilic Resin-Supported Palladium
0609
Rong, Z.; Du, W.; Wang, Y.; Lu, L.: Controlled Hydrogenation of ArNO2 Using Carbon-Supported Platinum Colloid
0610
Shiraishi, Y.; Sugano, Y.; Tanaka, S.; Hirai, T.: Photocatalytic Synthesis of Benzimidazoles on Pt@TiO2 Nanoparticles
0611
Shylesh, S.; Wagener, A.; Seifert, A.; Ernst, S.; Thiel, W. R.: One-Pot Reaction with Bifunctional Mesoporous Organosilicas
0612
Fang, W.; Zhang, Q.; Chen, J.; Deng, W.; Wang, Y.: Oxidant-Free Dehydrogenation of Alcohols with Au/HT
0613
Iwanami, K.; Seo, H.; Choi, J.-C.; Sakakura, T.; Yasuda, H.: Three-Component Strecker-Type Reaction with Al-MCM-41
0614
Jin, M.-J.; Lee, D.-H.: Pd-SiO2@Fe3O4: A Catalyst for Cross-Coupling of Aryl Chlorides
0615
Shylesh, S.; Wang, L.; Thiel, W. R.: Suzuki-Miyaura Coupling with Palladium(II) Phosphine Complexes on MNPs
0616
Haraguchi, N.; Takemura, Y.; Itsuno, S.: Polymer-Supported Chiral Organocatalysts for Diels-Alder Reaction
0617
Liu, Y.; Zhang, R.; He, C.; Dang, D.; Duan, C.: Palladium Cross-Linked Crystal-Catalyzed Knoevenagel Reaction-Cyclization

Addenda and Errata

0618
Asymmetric Addition of Deactivated Grignard Reagents to Aldehydes
0618
Poly-Chirality