DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 2009 · September 2009 DOI: 10.1055/s-002-20326

Synthesis of Natural Products and Potential Drugs

z939
All PDFs of this category
0939
Nicolaou, K. C.; Tang, Y.; Wang, J.: Synthesis of Sporolide B
0940
Nilewski, C.; Geisser, R. W.; Carreira, E. M.: Synthesis of a Polychlorinated Sulpholipid Cytotoxin
0941
Hamajima, A.; Isobe, M.: Synthesis of Ciguatoxin
0942
Tanaka, N.; Suzuki, T.; Matsumura, T.; Hosoya, Y.; Nakada, M.: Synthesis of (-)-FR182877
0943
Thalén, L. K.; Zhao, D.; Sortais, J.-B.; Paetzold, J.; Hoben, C.; Bäckvall, J. E.: Synthesis of Norsertraline
0944
Ishikawa, H.; Colby, D. A.; Seto, S.; Va, P.; Tam, A.; Kakei, H.; Rayl, T. J.; Hwang, I.; Boger, D. L.: Synthesis of Vinblastine
0945
Evans, D. A.; Welch, D. S.; Speed, A. W. H.; Moniz, G. A.; Reichelt, A.; Ho, S.: Synthesis of (+)-Peloruside A
0946
Chandra, A.; Pigza, J. A.; Han, J.-S.; Mutnick, D.; Johnston, J. N.: Synthesis of (+)-Serratezomine A
0947
Knott, K. E.; Auschill, S.; Jäger, A.; Knölker, H.-J.: Synthesis of Antiostatin B2
0948
Onoda, T.; Takikawa, Y.; Fujimoto, T.; Yasui, Y.; Suzuki, K.; Matsumoto, T.: Synthesis of (+)-11-Hydroxyerythratidine
0949
Kurokawa, T.; Isomura, M.; Tokuyama, H.; Fukuyama, T.: Synthesis of Lysergic Acid Methyl Ester
0950
Ruble, J. C.; Hurd, A. R.; Johnson, T. A.; Sherry, D. A.; Barbachyn, M. R.; Toogood, P. L.; Bundy, G. L.; Graber, D. R.; Kamilar, G. M.: Synthesis of (-)-PNU-286607
0951
Dockendorff, C.; Jin, S.; Olsen, M.; Lautens, M.; Coupal, M.; Hodzic, L.; Spear, N.; Payza, K.; Walpole, C.; Tomaszewski, M. J.: Synthesis of µ-Opioid Selective Ligands
0952
Georges, Y.; Ariza, X.; Garcia, J.: Synthesis of (-)-Spicigerolide
0953
Enomoto, M.; Kuwahara, S.: Synthesis of Bacilosarcin A

Synthesis of Heterocycles

z955
All PDFs of this category
0955
Liang, J.; Chen, J.; Du, F.; Zeng, X.; Li, L.; Zhang, H.: Synthesis of Spiro β-Lactams and Oxoindoles by Oxidative Dearomatization
0956
Ñunez, A.; Abarca, B.; Cuadro, A. M.; Alvarez-Builla, J.; Vaquero, J. J.: Ring-Closing Metathesis Approach to Quinolizinium Salts
0957
Han, Z.-G.; Tu, S.-J.; Jiang, B.; Yan, S.; Zhang, X.-H.; Wu, S.-S.; Hao, W.-J.; Cao, X.-D.; Shi, F.; Zhang, G.; Ma, N.: Chemoselective Synthesis of Naphthyridines and Pyrano[3,2-c]pyridines
0958
Budén, M. E.; Vaillard, V. A.; Martin, S. E.; Rossi, R. A.: Photostimulated Intramolecular SRN1 Reaction of Diarylamines to Carbazoles
0959
Ueda, S.; Nagasawa, H.: Copper-Catalyzed C-H Activation for the Synthesis of Benzoxazoles
0960
Suzuki, Y.; Ohta, Y.; Oishi, S.; Fujii, N.; Ohno, H.: Synthesis of Pyrroloindoles and Dipyrrolo-pyridines by a Hydroamination Route
0961
Heydari, A.; Khaksar, S.; Tajbakhsh, M.; Bijanzadeh, H. R.: General Synthesis of Hantzsch Esters in 2,2,2-Trifluoroethanol
0962
Spitz, C.; Lohier, J.-F.; Reboul, V.; Metzner, P.: Synthesis of 1,3-Benzothiazines by Catalytic Generation of Cesium Acetylide
0963
Joyce, L. L.; Batey, R. A.: Synthesis of 2-Aminobenzothiazoles via Oxidative C-H Functionalization
0964
Schuler, M.; Monney, A.; Gouverneur, V.: Synthesis of 4,4-Difluorodihydrofuran-3(2H)-ones
0965
Li, L.; Li, Z.; Wang, Q.: Organocatalytic Synthesis of Benzo[b]thiepines
0966
Gising, J.; Örtqvist, P.; Sandström, A.; Larhed, M.: An Improved Synthesis of Dichloro-pyrazinones
0967
Wender, P. A.; Strand, D.: Silver-Catalyzed Synthesis of 2,3-Dihydro-pyrroles
0968
Han, B.; He, Z.-Q.; Li, J.-L.; Li, R.; Jiang, K.; Liu, T.-Y.; Chen, Y.-C.: Piperidines from Organocatalytic Inverse-Demand Aza-Diels-Alder Reaction
0969
Fukamachi, S.; Konishi, H.; Kobayashi, K.: One-Pot Synthesis of 2-Sulfanylindoles

Synthesis of Materials and Unnatural Products

z971
All PDFs of this category
0971
Buehrdel, G.; Beckert, R.; Herzigova, P.; Petrlikova, E.; Schuch, D.; Birckner, E.; Goerls, H.: Synthesis of Push-Pull Pyrroles and their Oxidative Anellation Reaction
0972
Liu, W.; Pink, M.; Lee, D.: Conjugated Borasiloxane Cages
0973
Ortiz, A. L.; Rivera, D. M.; Athans, A. J.; Echegoyen, L.: Functional Fullerenes for Electronics
0974
Juspin, T.; Terme, T.; Vanelle, P.: Rapid Access to Diphenyl- and Acenaphthoquinoline Derivatives
0975
Liang, Y.; Feng, D.; Wu, Y.; Tsai, S.-T.; Li, G.; Ray, C.; Yu, L.: Fluorine-Containing Semiconducting Polymers
0976
Zhong, W.; Lin, F.; Chen, R.; Su, W.: Benzonaphthyridines from Morita-Baylis-Hillman Adduct Acetates
0977
Jiang, Z.; Yao, H.; Zhang, Z.; Yang, C.; Liu, Z.; Tao, Y.; Qin, J.; Ma, D.: Synthesis of ortho-Linked Oligo-9,9′-spirobifluorenes
0978
Petersen, M. Å.; Broman, S. L.; Kadziola, A.; Kilså, K.; Nielsen, M. B.: Azulene Photochromes
0979
Allen, M. J.; Wangkanont, K.; Raines, R. T.; Kiessling, L. L.: Graft Copolymers from a Double ROMP
0980
Bricks, J.; Ryabitskii, A.; Kachkovskii, A.: Azulenated Cyanine Dyes
0981
Hudson, Z. M.; Zhao, S.-B.; Wang, R.-Y.; Wang, S.: A Breakdown in Communication
0982
Wijsboom, Y. H.; Patra, A.; Zade, S. S.; Sheynin, Y.; Li, M.; Shimon, L. J. W.; Bendikov, M.: Planar Polyselenophenes
0983
Mullen, K. M.; Mercurio, J.; Serpell, C. J.; Beer, P. D.: Giving a Use to Triazoles
0984
Wharton, S. I.; Henry, J. B.; McNab, H.; Mount, A. R.: Selective Dimerization of Indolocarbazoles
0985
Kim, Y.; Zhao, H.; Gabbaï, F. P.: A Highly Selective Cyanide Sensor

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z987
All PDFs of this category
0987
He, H.; Liu, W.-B.; Dai, L.-X.; You, S.-L.: Ir-Catalyzed Cross-Coupling of Styrene Derivatives with Allylic Carbonates
0988
Burks, H. E.; Kliman, L. T.; Morken, J. P.: Platinum-Catalyzed Asymmetric 1,4-Dihydroxylation of 1,3-Dienes
0989
Hatano, M.; Hattori, Y.; Furuya, Y.; Ishihara, K.: Lanthanum(III)-Binaphthyldisulfonate Complex Catalyzed Strecker Reaction
0990
Duplessis, M.; Waltz, M.-E.; Bencheqroun, M.; Cardinal-David, B.; Guindon, Y.: Synthesis of Quaternary Stereocenters through a Radical Cyclization
0991
Kureshy, R. I.; Prathap, K. J.; Agrawal, S.; Kumar, M.; Khan, N. H.; Abdi, S. H. R.; Bajaj, H. C.: Co-Salen Complexes Catalyzed Kinetic Resolution of Terminal Epoxides
0992
Tang, X.; Woodward, S.; Krause, N.: Synthesis of α-Hydroxyallenes by SN2′ of Propargylic Dioxolanones
0993
Lee, K.-s.; Hoveyda, A. H.: Copper-NHC Catalysts for Asymmetric Conjugate Addition
0994
Korenaga, T.; Osaki, K.; Maenishi, R.; Sakai, T.: Rhodium-Catalyzed 1,4-Addition of Arylboronic Acids
0995
Ogura, T.; Yoshida, K.; Yanagisawa, A.; Imamoto, T.: Chiral Dinuclear Palladium Complexes in Ring-Opening Reactions
0996
Wang, J.; Shao, Z.; Yu, K. D. W. Y.; Chan, A. S. C.: Asymmetric Addition of Terminal Alkynes to Imines Catalyzed by Copper(I)
0997
Lu, Y.; Kim, I. S.; Hassan, A.; Valle, D. J. Del; Krische, M. J.: Iridium-Catalyzed Stereoselective Two-Directional Elongation of 1,3-Polyols
0998
Liu, L.; Floreancig, P. E.: Oxidative Addition of Nucleophiles to Vinyl Oxazolidinones
0999
Lysenko, I. L.; Lee, H. G.; Cha, J. K.: Titanium-Mediated Cross-Coupling of Aldimines and Allylic Alcohols
1000
Mantilli, L.; Gérard, D.; Torche, S.; Besnard, C.; Mazet, C.: Asymmetric Isomerization of Primary Allylic Alcohols
1001
Lim, H. J.; Smith, C. R.; RajanBabu, T. V.: Metal-Mediated Isomerization of Terminal Olefins
1002
Schmidtmann, E. S.; Oestreich, M.: Generation and Applications of α-Chiral Allylic Stannanes
1003
Lu, W.-J.; Hou, X.-L.: Iridium-Catalyzed Hydrogenation of
α,β-Unsaturated Amides
1004
Hassan, A.; Lu, Y.; Krische, M. J.: Transfer Hydrogenation in Iterative Elongation of Alcohols
1005
Duan, S.; Jana, R.; Tunge, J. A.: Diastereoselective Hydroarylation for the Synthesis of Dihydrocoumarins
1006
Ye, Y.; Zheng, C.; Fan, R.: Divergent Cyclization towards Cyclopropanes and Oxetanes
1007
Mihara, H.; Xu, Y.; Shepherd, N. E.; Matsunaga, S.; Shibasaki, M.: Catalytic Asymmetric α-Addition of Isocyanoacetamides to Aldehydes
1008
Turlington, M.; DeBerardinis, A. M.; Pu, L.: H8BINOL-Catalyzed Enantioselective Alkyl Propiolate Addition to Aliphatic Aldehydes
1009
Shaikh, T. M.; Karabal, P. U.; Suryavanshi, G.; Sudalai, A.: Titanium Superoxide Catalyzed Aminobromination of Olefins
1010
Kleinbeck, F.; Toste, F. D.: Cyclobutanones via Ring Expansion of Allenylcyclopropanols
1011
Würtz, S.; Lohre, C.; Fröhlich, R.; Bergander, K.; Glorius, F.: A Sterically Demanding NHC Ligand
1012
Nishimoto, Y.; Moritoh, R.; Yasuda, M.; Baba, A.: Ketene Silyl Acetal Addition to Alkynes Gives Alkenylindiums
1013
ConcellÓn, J. M.; RodrÍguez-Solla, H.; Simal, C.: Nucleophilic Addition of Samarium Enolates to Imines
1014
Huang, K.; Ortiz-Marciales, M.; Correa, W.; Pomales, E.; López, X. Y.: Chiral β-Hydroxy Ethers from Spiroborate Ester Mediated Reductions

Metal-Mediated Synthesis

z1015
All PDFs of this category
1015
Han, C.; Buchwald, S. L.: Coupling of Secondary Alkylzinc Halides with Aryl Bromides and Chlorides
1016
Cheng, K.; Huang, L.; Zhang, Y.: CuBr-Mediated Oxyalkylation of Styrenes by Cyclic Ethers
1017
Wang, X.; Mei, T.-S.; Yu, J.-Q.: Pd(OTf)2˙2H2O-Catalyzed ortho-Fluorination of Benzyl Triflamides
1018
Gao, Y.; Wang, G.; Chen, L.; Xu, P.; Zhao, Y.; Zhou, Y.; Han, L.-B.: Cu-Catalyzed Aerobic Oxidative Coupling of Alkynes to H-Phosphonates
1019
Kleeberg, C.; Dang, L.; Lin, Z.; Marder, T. B.: Copper(I)-Catalyzed Room-Temperature Borylation of Aryl Halides
1020
Ihara, H.; Suginome, M.: 2-Pyrazol-5-ylaniline as ortho-Directing Agent for Arylboronic Acids in C-H Silylation
1021
Nowrouzi, F.; Thadani, A. N.; Batey, R. A.: Allylation and Crotylation of Carbonyls Using Organotrifluoroborates
1022
Maegawa, T.; Akashi, A.; Yaguchi, K.; Iwasaki, Y.; Shigetsura, M.; Monguchi, Y.; Sajiki, H.: Practical Arene Hydrogenation by Heterogeneous Catalysts
1023
Lam, K.; Markó, I. E.: Chemoselective Chemical and Electrochemical Deprotections of Toluates
1024
Furuya, T.; Ritter, T.: AgOTf-Mediated Fluorination of Boronic Acids
1025
Schmink, J. R.; Leadbeater, N. E.: Synthesis of Diarylmethanes via Pd-Catalyzed α-Arylation of Benzylketones
1026
Watson, A. J. A.; Maxwell, A. C.; Williams, J. M. J.: Ruthenium-Catalyzed Oxidation of Primary Alcohols into Amides
1027
Kobayashi, O.; Uraguchi, D.; Yamakawa, T.: Direct C-H Arylation of Benzene, Naphthalene, and Pyridine
1028
Cui, L.; Peng, Y.; Zhang, L.: Gold-Catalyzed Synthesis of Piperidin-4-ones
1029
Ueno, S.; Shimizu, R.; Kuwano, R.: Ni-Catalyzed C-N Bond Formation at the β-Position of Saturated Ketones

Organo- and Biocatalysis

z1031
All PDFs of this category
1031
Goswami, P.; Baruah, A.; Das, B.: A Highly Enantioselective α-Bromination?
1032
Reyes, E.; Talavera, G.; Vicario, J. L.; Badía, D.; Carrillo, L.: One-Step Synthesis of Furofuranes
1033
Cui, H.-L.; Feng, X.; Peng, J.; Lei, J.; Jiang, K.; Chen, Y.-C.: N-Allylic Alkylation of Indoles
1034
Zhu, D.; Lu, M.; Dai, L.; Zhong, G.: One-Pot Synthesis of Bicyclic Isoxazolidines with Five Stereogenic Centers
1035
Zeng, X.; Xu, Z.; Lu, M.; Zhong, G.: Enantioselective Aziridination Using Chiral Phosphoric Acids
1036
Sala, G. Della; Lattanzi, A.: Enantioselective Ring Opening of meso-Aziridines with TMS-Protected Thiophenol
1037
Nielsen, M.; Jacobsen, C. B.; Paixão, M. W.; Holub, N.; Jørgensen, K. A.: Formal Alkynylation and Alkenylation of α,β-Unsaturated Aldehydes
1038
Wu, J.; Ni, B.; Headley, A.: Highly Enantioselective Michael Addition to Nitroolefins in Water
1039
Gioia, C.; Fini, F.; Mazzanti, A.; Bernardi, L.; Ricci, A.: Formal [3+2] Cycloaddition with in situ Generated N-Carbamoyl Nitrones
1040
Pu, X.; Qi, X.; Ready, J. M.: Lewis Base Catalysts Containing Axial Chirality of Allenes
1041
Zheng, C.; Li, Y.; Yang, Y.; Wang, H.; Cui, H.; Zhang, J.; Zhao, G.: Asymmetric Epoxidation of Electron-Deficient α,β-Enones
1042
Chiang, P.-C.; Kim, Y.; Bode, J. W.: NHC-Catalyzed Redox Amidation of α-Hydroxyenones
1043
Liu, Y.-k.; Ma, C.; Jiang, K.; Liu, T.-Y.; Chen, Y.-C.: Highly Selective Formal [3+3] Cyclohexenone Annulation
1044
Garrabou, X.; Castillo, J. A.; Guérard-Hélaine, C.; Parella, T.; Joglar, J.; Lemaire, M.; Clapés, P.: Enzymatic Control over Self- and Cross-Aldol Reactions

Polymer-Supported Synthesis

z1045
All PDF of this category
1045
Lee, K. S.; Woo, M. H.; Kim, H. S.; Lee, E. Y.; Lee, I. S.: Optical Resolution with Immobilized Enzymes on Nanoparticles
1046
Motokura, K.; Tada, M.; Iwasawa, Y.: Tandem Condensation Reactions with H-mont-NH2
1047
Niknam, K.; Saberi, D.; Sefat, M. N.: Benzylidene Diacetate Formation with Silica-Bonded S-Sulfonic Acid
1048
Peuchmaur, M.; Lisowski, V.; Gandreuil, C.; Maillard, L. T.; Martinez, J.; Hernandez, J.-F.: Solid-Phase Synthesis of Isocoumarins via Halocyclization
1049
Wang, N.; Matsumoto, T.; Ueno, M.; Miyamura, H.; Kobayashi, S.: A Gold-Immobilized Capillary Column Reactor for Oxidation of Alcohols
1050
Gill, C. S.; Venkatasubbaiah, K.; Jones, C. W.: Asymmetric Cyclopropanation with Immobilized Ru(II)-Salen-Py2
1051
Karimi, B.; Akhavan, P. F.: Suzuki-Miyaura Coupling with NHC-Palladium Polymer
1052
Lee, E. Y.; Kim, Y.; Lee, J. S.; Park, J.: One-Pot Oxidation-Wittig Reaction with Ruthenium Catalyst
1053
Kadib, A. El; Chimenton, R.; Sachse, A.; Fajula, F.; Galarneau, A.; Coq, B.: MonoSil Microreactor for Knoevenagel Reaction and Transesterification
1054
Kantam, M. L.; Yadav, J.; Laha, S.; Srinivas, P.; Sreedhar, B.; Figueras, F.: Asymmetric Hydrosilylation of Ketones by Copper Ferrite Nanoparticles
1055
Tan, M.; Zhang, Y.; Ying, J. Y.: Cyanosilylation and Hydrosilylation with Poly-NHC Particles
1056
Zhang, P.-P.; Zhang, X.-X.; Sun, H.-X.; Liu, R.-H.; Wang, B.; Lin, Y.-H.: Suzuki-Miyaura Cross-Coupling of Aryl Bromides with Pd-CNT
1057
Nguyen, Q. P. B.; Kim, J. N.; Kim, T. H.: Solid-Supported 2-Imidazolidinone Chiral Auxiliary for Alkylation

Addenda and Errata

1058
Synthesis of BYK 405879