DOI: 10.1055/s-00000131

Synfacts

Issue 12 · Volume 2011 · December 2011 DOI: 10.1055/s-002-22456

Synform

A109
Zanda, Matteo: SYNFORM ISSUE 2011/12

Synthesis of Natural Products and Potential Drugs

z1265
All PDFs of this category
1265
Tsuna, K.; Noguchi, N.; Nakada, M.: Synthesis of (+)-Ophiobolin A
1266
Scott, J. P.; Alam, M.; Bremeyer, N.; Goodyear, A.; Lam, T.; Wilson, R. D.; Zhou, G.: Synthesis of MK-3281
1267
Berliner, M. A.; Dubant, S. P. A.; Makowski, T.; Ng, K.; Sitter, B.; Wager, C.; Zhang, Y.: Synthesis of PF-03463275
1268
Furst, L.; Narayanam, J. M. R.; Stephenson, C. R. J.: Synthesis of (+)-Gliocladin C
1269
Dirat et al., O.: Synthesis of Fesoterodine
1270
Konkol, L. C.; Guo, F.; Sarjeant, A. A.; Thomson, R. J.: Synthesis of the Bismurrayaquinone A
1271
Cha, J. Y.; Yeoman, J. T. S.; Reisman, S. E.: Synthesis of (-)-Maoecrystal Z
1272
Snell, R. H.; Woodward, R. L.; Willis, M. C.: Synthesis of (-)-Hodgkinsine B
1273
Wang, X.-J.; Frutos et al., R. P.: Synthesis of BIRT2584
1274
de Koning et al., P. D.: Synthesis of Crizotinib (PF-02341066)
1275
de Koning, P. D.; Murtagh, L.; Lawson, J. P.; Vonder Embse, R. A.; Kunda, S. A.; Kong, W.: Synthesis of PF-04191834
1276
Girardin, M.; Dolman, S. J.; Lauzon, S.; Ouellet, S. G.; Hughes, G.; Fernandez, P.; Zhou, G.; O’Shea, P. D.: Synthesis of MK-8245
1277
Campeau, L.-C.; Dolman, S. J.; Gauvreau, D.; Corley, E.; Liu, J.; Guidry, E. N.; Ouellet, S. G.; Steinhuebel, D.; Weisel, M.; O’Shea, P. D.: Synthesis of a Renin Inhibitor
1278
Cuthbertson, J. D.; Godfrey, A. A.; Taylor, R. J. K.: Synthesis of (+)-Grandisine D
1279
Butcher, K. J.; Denton, S. M.; Field, S. E.; Gillmore, A. T.; Harbottle, G. W.; Howard, R. M.; Laity, D. A.; Ngono, C. J.; Pibworth, B. A.: Synthesis of a TRPV1 Antagonist
1280
Goto, M.; Konishi, T.; Kawaguchi, S.; Yamada, M.; Nagata, T.; Yamano, M.: Synthesis of TAK-475
1281
Huters, A. D.; Quasdorf, K. W.; Styduhar, E. D.; Garg, N. K.: Synthesis of (-)-N-Methylwelwitindolinone C Isothiocyanate

Synthesis of Heterocycles

z1283
All PDFs of this category
1283
Karthikeyan, J.; Cheng, C.-H.: Pd-Catalyzed Synthesis of Phenanthridinones by Double C-H Activation
1284
Shintani, R.; Moriya, K.; Hayashi, T.: Palladium-Catalyzed Enantioselective Synthesis of Silacyles
1285
Denmark, S. E.; Kornfilt, D. J. P.; Vogler, T.: Ethers via Catalytic Asymmetric Thiofunctionalization of Alkenyl Alcohols
1286
Estrada, A. A.; Lyssikatos, J. P.; St-Jean, F.; Bergeron, P.: Synthesis of Pyrimidines via N-Vinyl Tertiary Enamides
1287
Anas, S.; Cordi, A.; Kagan, H. B.: Pd-Catalyzed Enantioselective Synthesis of 2-Methyl Indolines
1288
Wang, Y.; Luo, Y.-C.; Hu, X.-Q.; Xu, P.-F.: Metal-Free Synthesis of 2-Trifluoromethyl Furans
1289
Chai, G.; Qiu, Y.; Fu, C.; Ma, S.: Synthesis of Chromones from 2,3-Allenoic Acids and Benzynes
1290
Patil, S. S.; Patil, S. V.; Bobade, V. D.: Iron-Catalyzed Synthesis of Aminoindolizines and Quinolines
1291
Reddy, C. R.; Reddy, M. D.; Srikanth, B.; Prasad, K. R.: Metal-Free Synthesis of Pyrroles From Morita-Baylis-Hillman Acetates
1292
Li, Y.; Hong, D.; Zhu, Y.; Lu, P.; Wang, Y.: Copper-Catalyzed One-Pot Synthesis of 5-Sulfonamidopyrazoles
1293
Yamagishi, M.; Nishigai, K.; Hata, T.; Urabe, H.: Two-Step Heck-Mediated Synthesis of Pyrroles from Sulfonamides and Bromoacetylenes
1294
Nandi, G. C.; Samai, S.; Singh, M. S.: Cycloaddition Approach to Substituted Thiophenes
1295
Sun, L.-L.; Deng, C.-L.; Tang, R.-Y.; Zhang, X.-G.: Heteroannulation Route to Benzothiophenes from 2-Bromo Alkynylbenzenes
1296
Panteleev, J.; Zhang, L.; Lautens, M.: A Multicatalytic Domino Heteroannulation Approach to Dihydroquinolines
1297
Kuninobu, Y.; Yoshida, T.; Takai, K.: Pd-Catalyzed C-H Activation Route to Dibenzophosphole Oxides

Synthesis of Materials and Unnatural Products

z1299
All PDFs of this category
1299
Gu, Z.; Boursalian, G. B.; Gandon, V.; Padilla, R.; Shen, H.; Timofeeva, T. V.; Tongwa, P.; Vollhardt, K. P. C.; Yakovenko, A. A.: Nickel-Catalyzed Synthesis of Strained Phenacenes
1300
Wu, T.-C.; Chen, J.-J.; Wu, Y.-T.: One Step to Polyenes
1301
Vaid, T. P.: An All-Organic Porphyrin and its Properties
1302
Nagata, Y.; Suginome, M.: Polymerization of Diisocyanobenzenes Bearing Alkoxy Side Chains
1303
Shao, N.; Pang, G.-X.; Yan, C.-X.; Shi, G.-F.; Cheng, Y.: A One-Pot Approach to ‘Shutting the Lights Off’ in the Presence of Mercury Ion
1304
Kubo, T.; Katada, Y.; Shimizu, A.; Hirao, Y.; Sato, K.; Takui, T.; Uruichi, M.; Yakushi, K.; Haddon, R. C.: Delocalized Radicals
1305
Bautista, R.; Bernal, P.; Herrera, R.; Santoyo, B. M.; Lazcano-Seres, J. M.; Delgado, F.; Tamariz, J.: Synthesis of a New exo-Heterocyclic Diene
1306
Zhao, W.; Carreira, E. M.: High-Yielding One-Pot Synthesis of Oxazine Photochromes
1307
Evans, N. H.; Beer, P. D.: Anion-Templated Yin Yang: Janus [2]Rotaxanes
1308
Pammer, F.; Lalancette, R. A.; Jäkle, F.: Putting a B in Polymer
1309
Sisto, T. J.; Golder, M. R.; Hirst, E. S.; Jasti, R.: The Smaller the Redder
1310
Gordo, J.; Avó, J.; Parola, A. J.; Lima, J. C.; Pereira, A.; Branco, P. S.: A One-Pot Route to 3-Vinyl Coumarins
1311
Amaya, T.; Hifumi, M.; Okada, M.; Shimizu, Y.; Moriuchi, T.; Segawa, K.; Ando, Y.; Hirao, T.: Route to Functionalized Sumanenes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1313
All PDFs of this category
1313
Jiang, G.; List, B.: Asymmetric α-Allylation of Aldehydes with Simple Allylic Alcohols
1314
Bigot, A.; Williamson, A. E.; Gaunt, M. J.: Copper-Catalyzed Asymmetric α-Arylation of N-Acyloxazolidinones
1315
Harvey, J. S.; Simonovich, S. P.; Jamison, C. R.; MacMillan, D. W. C.: Cu-Catalyzed Asymmetric α-Arylation of Carbonyls
1316
Katcher, M. H.; Sha, A.; Doyle, A. G.: Palladium-Catalyzed Enantioselective Fluorination of Allylic Halides
1317
Karlow, J. A.; Doyle, A. G.: Enantioselective Fluorination of Epoxides via Cooperative Catalysis
1318
Feng, X.; Wei, B.; Yang, J.; Du, H.: Enantioselective Rhodium-Catalyzed Conjugate Addition
1319
Kawato, Y.; Iwata, M.; Yazaki, R.; Kumagai, N.; Shibasaki, M.: A Simplified Catalytic System for Direct Asymmetric Aldol Reaction of Thioamides
1320
Kanno, O.; Kuriyama, W.; Wang, Z. J.; Toste, F. D.: Hydroamination of Dienes by Gold(I)/Menthol Cooperative Catalysis
1321
Yamashita, Y.; Imaizumi, T.; Guo, X.-X.; Kobayashi, S.: Silver-Catalyzed Enantioselective [3+2] Cycloadditions
1322
Yamamoto, T.; Akai, Y.; Nagata, Y.; Suginome, M.: Helical Macromolecular Ligand for Asymmetric Suzuki Coupling
1323
Zheng, B.-H.; Ding, C.-H.; Hou, X.-L.: Pd-Catalyzed Asymmetric Allylic Amination
1324
Huang, Z.; Liu, Z.; Zhou, J.: Palladium-Catalyzed Enantioselective α-Arylation
1325
Trost, B. M.; Burns, A. C.; Tautz, T.: Readily Accessible Diene Ligands for Enantioselective Conjugate Additions
1326
Ichinose, M.; Suematsu, H.; Yasutomi, Y.; Nishioka, Y.; Uchida, T.; Katsuki, T.: Enantioselective Intramolecular Benzylic C-H Bond Amination
1327
Matsumoto, K.; Feng, C.; Handa, S.; Oguma, T.; Katsuki, T.: Asymmetric Epoxidation Catalyzed by Titanium(salalen) Complex
1328
Capozzi, M. A. M.; Centrone, C.; Fracchiolla, G.; Naso, F.; Cardellicchio, C.: Titanium-Catalyzed Enantioselective Oxidation of Aryl Sulfides
1329
Karmakar, A.; Maji, T.; Wittmann, S.; Reiser, O.: Diastereo- and Enantioselective Direct Aldol Reactions Mediated by CoCl2/l-Proline
1330
Kobayashi, S.; Arai, K.; Yamakawa, T.; Chen, Y.-J.; Salter, M. M.; Yamashita, Y.: Niobium-Catalyzed Asymmetric Aldol-Type Reactions
1331
Xue, F.; Li, X.; Wan, B.: Rh-Catalyzed Enantioselective Addition of Arylboronic Acids to Enones
1332
Guo, S.; Xie, Y.; Hu, X.; Huang, H.: Cu-Catalyzed Asymmetric Tandem Dual Michael Reaction of Dialkylzinc to Enones
1333
Teng, H.-L.; Luo, F.-L.; Tao, H.-Y.; Wang, C.-J.: Cu(I)/BINAP-Catalyzed Synthesis of Pyro-glutamates
1334
Ji, Y. Q.; Qi, G.; Judeh, Z. M. A.: Copper-Catalyzed Asymmetric Henry Reaction
1335
Lebel, H.; Spitz, C.; Leogane, O.; Trudel, C.; Parmentier, M.: Stereoselective Rhodium-Catalyzed Amination of Alkenes
1336
Akashi, M.; Arai, N.; Inoue, T.; Ohkuma, T.: Catalyst-Controlled Diastereo- and Enantioselective Hydrogenation
1337
Chow, T. W.-S.; Liu, Y.; Che, C.-M.: Manganese-Catalyzed Enantioselective cis-Dihydroxylation
1338
Wang, L.; Meng, W.; Zhu, C.-L.; Zheng, Y.; Nie, J.; Ma, J.-A.: Copper-Catalyzed Tandem 1,4-Addition-Fluorination Sequence
1339
Chien, C.-W.; Shi, C.; Lin, C.-F; Ojima, I.: Pd-Catalyzed Intramolecular Asymmetric Allylic Amination
1340
Pan, S.; Endo, K.; Shibata, T.: Ir(I)-Catalyzed C-H Bond Activation of 2-(Alkylamino)pyridines with Alkenes
1341
Hu, B.; Meng, M.; Fossey, J. S.; Mo, W.; Hu, X.; Deng, W.-P.: Synthesis of Optically Pure Bulky Carbinols via Kinetic Resolution
1342
Lian, Y.; Hardcastle, K. I.; Davies, H. M. L.: Stereocontrol of the Combined C-H Functionalization/Cope Rearrangement

Metal-Mediated Synthesis

z1343
All PDFs of this category
1343
Zultanski, S. L.; Fu, G. C.: Catalytic Enantioselective γ-Alkylation of Carbonyl Compounds
1344
Morandi, B.; Carreira, E. M.: Synthesis of Trifluoroethyl-Substituted Ketones
1345
Lim, D. S. W.; Anderson, E. A.: Takai-Analogous One-Step Preparation of (E)-Vinylsilanes
1346
Genna, D. T.; Posner, G. H.: Direct Conversion of Carboxylic Acids into Ketones
1347
Urabe, D.; Yamaguchi, H.; Inoue, M.: Bridgehead Radicals for Coupling of Oxygenated Carbocycles
1348
Wang, Z.-Q.; Zhang, W.-W.; Gong, L.-B.; Tang, R.-Y.; Yang, X.-H.; Liu, Y.; Li, J.-H.: Copper-Catalyzed Intramolecular Oxidative Cyclization
1349
Sternativo, S.; Calandriello, A.; Constantino, F.; Testaferri, L.; Tiecco, M.; Marini, F.: An Organocatalyzed Michael Addition-Cyclization Sequence to Spirolactones
1350
Ramharter, J.; Mulzer, J.: One-Pot Synthesis of 2,4-Dienols from Cycloalkenones
1351
Pan, J.; Wang, X.; Zhang, Y.; Buchwald, S. L.: Improved Conversion of Aryl and Vinyl Triflates into Bromides and Chlorides
1352
Zhang, G.; Ren, X.; Chen, J.; Hu, M.; Cheng, J.: Cu-Mediated Cyanation of Aryl Halides
1353
Das, P. P.; Lysenko, I. L.; Cha, J. K.: Ti-Mediated Tandem Ethylation and Functionalization of Allylic Alcohols
1354
III, A. B. Smith; Tong, R.; Kim, W.-S.; Maio, W. A.: New Insights into Anion Relay Chemistry
1355
Zhao, Y.; Huang, W.; Zheng, J.; Hu, J.: Difluoromethylation of Carbonyls and Imines with TMSCF2H
1356
Saadi, J.; Akakura, M.; Yamamoto, H.: Mukaiyama Cross-Aldol Reaction to Yield anti-β-Siloxy-α-haloaldehydes
1357
Ohashi, M.; Taniguchi, T.; Ogoshi, S.: Nickel-Catalyzed Formation of Cyclo-pentenones via Cycloaddition

Organo- and Biocatalysis

z1359
All PDFs of this category
1359
Sohtome, Y.; Yamaguchi, T.; Shin, B.; Nagasawa, K.: Friedel-Crafts Alkylation, Internal Redox Reaction, and Umpolung Cascade
1360
Xiao, Y.-C.; Wang, C.; Yao, Y.; Sun, J.; Chen, Y.-C.: Asymmetric Reduction of Unprotected Indoles
1361
Hein, J. E.; Tse, E.; Blackmond, D. G.: Enantiopure RNA Precursors from Nearly Racemic Starting Materials
1362
Xiang, S.-K.; Zhang, B.; Zhang, L.-H.; Cui, Y.; Jiao, N.: Morpholine-Catalyzed C3 Alkenylation of Indoles with Enals
1363
Martin, A.; Casto, K.; Morris, W.; Morgan, J. B.: Phosphine-Catalyzed Heine Reaction
1364
Zhang, Z.; Jain, P.; Antilla, J. C.: Asymmetric Reduction of Ketones
1365
De, C. Kanta; Mittal, N.; Seidel, D.: Dual-Catalytic Asymmetric Reactions
1366
Herlé, B.; Wanner, M. J.; van Maarseveen, J. H.; Hiemstra, H.: Organocatalytic Pictet-Spengler Reaction in Natural Product Synthesis
1367
Belkheira, M.; Abed, D. El; Pons, J.-M.; Bressy, C.: Organo-Click Synthesis of 1,2,3-Triazoles from Unactivated Ketones
1368
Ren, L.; Lei, T.; Gong, L.-Z.: Phosphoric Acid Catalyzed Enantioselective Friedländer Condensations
1369
Liu, J.-D.; Chen, Y.-C.; Zhang, G.-B.; Li, Z.-Q.; Chen, P.; Du, J.-Y.; Tu, Y.-Q.; Fan, C.-A.: Synthesis of Piperidines through Intramolecular Aza-Michael Addition
1370
Asano, K.; Matsubara, S.: Catalytic Cycloetherification Using Bifunctional Thiourea Catalysts

Polymer-Supported Synthesis

z1371
All PDFs of this category
1371
Jagadeesh, R. V.; Wienhöfer, G.; Westerhaus, F. A.; Surkus, A.-E.; Pohl, M.-M.; Junge, H.; Junge, K.; Beller, M.: Reduction of Nitroarenes with N2H4˙H2O Using Fe-Phen/C
1372
Wang, Y.; Zhu, D.; Tang, L.; Wang, S.; Wang, Z.: Oxidative Amidation of Alcohols with Amines Catalyzed by Au/DNA
1373
Kong, G.-Q.; Xu, X.; Zou, C.; Wu, C.-D.: Suzuki-Miyaura Reaction with NHC-Cu-Pd MOF Catalysts
1374
Yanase, T.; Mori, S.; Monguchi, Y.; Sajiki, H.: Pd/C-Catalyzed Hiyama Cross-Coupling
1375
Alza, E.; Sayalero, S.; Kasaplar, P.; Almai, D.; Pericàs, M. A.: Solid-Supported Prolinol Ether Catalysts
1376
Karimi, B.; Esfahani, F. K.: Ullmann Reaction of Aryl Iodides with Au@PMO
1377
Zhi, J.; Song, D.; Li, Z.; Lei, X.; Hu, A.: Suzuki-Miyaura Coupling in Water with Pd@SBA-15©
1378
Zeng, X.-M.; Chen, J.-M.; Middleton, K.; Zhdankin, V. V.: Oxidation with SiO2-Supported Iodoarene-RuCl3 Bifunctional Catalysts
1379
Lagiakos, H. R.; Walker, A.; Aguilar, M.-I.; Perlmutter, P.: Microwave-Assisted Thionation of Amides Using a Solid-Supported P2S5
1380
Sarkar, S. M.; Uozumi, Y.; Yamada, Y. M. A.: A Poly(Imidazole-Palladium) Catalyst for Allylic Arylation/Alkenylation
1381
Swapna, K.; Murthy, S. N.; Jyothi, M. T.; Nageswar, Y. V. D.: CuO on Alumina for C-O Coupling of Halides with Alcohols
1382
Verdié, P.; Ronga, L.; Cristau, M.; Amblard, M.; Cantel, S.; Enjalbal, C.; Puget, K.; Martinez, J.; Subra, G.: Disulfide Bond Formation with Polymer-Supported Reagent
1383
Zhang, X.; Li, P.; Ji, Y.; Zhang, L.; Wang, L.: Suzuki Coupling of Alkynyl Bromides with Boronic Acids by Pd-SiO2@Fe3O4
1384
Hirai, Y.; Uozumi, Y.: C-N and C-S Bond-Forming Cross-Coupling in Water with PS-PEG-Pd

Addenda and Errata

1385
Trienamines in Organocatalysis
1385
exo-Selective Diels-Alder Reaction of 2,4-Dienals and Nitroalkenes