DOI: 10.1055/s-00000131

Synfacts

Issue 11 · Volume 2006 · November 2006 DOI: 10.1055/s-002-5232

Synthesis of Natural Products and Potential Drugs

1083
Shen, X.; Wasmuth, A. S.; Zhao, J.; Zhu, C.; Nelson, S. G.: Synthesis of (-)-Pironetin
1084
Trost, B. M.; Dong, G.: Synthesis of (+)-Agelastatin A
1085
Chiba, S.; Kitamura, M.; Narasaka, K.: Synthesis of (-)-Sordarin
1086
Takahashi, K.; Matsumura, T.; Corbin, G. R. M.; Ishihara, J.; Hatakeyama, S.: Synthesis of (-)-Neodysiherbaine
1087
Tatsuta, K.; Suzuki, Y.; Furuyama, A.; Ikegami, H.: Synthesis of (-)-Tetrodecamycin
1088
Okano, K.; Tokuyama, H.; Fukuyama, T.: Synthesis of (+)-Yatakemycin
1089
Garg, N. K.; Hiebert, S.; Overman, L. E.: Synthesis of (-)-Sarain A
1090
Crimmins, M. T.; Zhang, Y.; Diaz, F. A.: Synthesis of (-)-Mucocin
1091
Fukumoto, H.; Takahashi, K.; Ishihara, J.; Hatakeyama, S.: Synthesis of (+)-β-Erythroidine
1092
Nicolaou, K. C.; Harrison, S. T.: Synthesis of Abyssomicin C
1093
Kim, J. G.; Walsh, P. J.: Synthesis of BMS 184394
1094
Brandau, S.; Landa, A.; Franzén, J.; Marigo, M.; Jørgensen, K. A.: Synthesis of (-)-Paroxetine
1095
Roy, A.; Gosselin, F.; O’Shea, P. D.; Chen, C.-y: Synthesis of a Cathepsin K Inhibitor
1096
Wang, Q.; Huang, Q.; Chen, B.; Lu, J.; Wang, H.; She, X.; Pan, X.: Synthesis of (+)-Machaeriol D
1097
Höck, S.; Borschberg, H.-J.: Synthesis of (-)-(19R)-Ibogamin-19-ol

Synthesis of Heterocycles

1099
Blaszykowski, C.; Aktoudianakis, E.; Bressy, C.; Alberico, D.; Lautens, M.: Synthesis of Annulated N-Containing Heterocycles via C-H Activation
1100
Morton, D.; Pearson, D.; Field, R. A.; Stockman, R. A.: Sulfur Ylide Mediated Asymmetric Synthesis of Aziridines from Sulfinylketimines
1101
Asao, N.; Iso, K.; S, Yudha: Three-Component Synthesis of 1,2-Dihydroisoquinolines
1102
Bhattacharya, A.; Cherukuri, S.; Plata, R. E.; Patel, N.; Tamez, V. Jr; Grosso, J. A.; Peddicord, M.; Palaniswamy, V. A.: One-Pot Synthesis of 3,4-Disubstituted Pyrrole-2-Esters
1103
Aparicio, D.; Attanasi, A.; Filippone, P.; Ignacio, R.; Lillini, S.; Mantellini, F.; Palacios, F.; de Santos, J. Mlos: Synthesis of Pyrazines from Diaza-butadienes and 1,2-Diamines
1104
Heller, S. T.; Natarajan, S. R.: A Classical but Short One-Pot Synthesis of Pyrazoles
1105
Komeyama, K.; Morimoto, T.; Takaki, K.: Synthesis of Pyrrolidines from Aminoolefins by Hydroamination
1106
McLaughlin, M.; Palucki, M.; Davies, I. W.: One-Pot Synthesis of Azaindoles and Indoles
1107
Muhuhi, J.; Spaller, M. R.: Synthesis of Tetrahydroquinolines via an Intramolecular Aza-Diels-Alder Reaction
1108
Kunetsky, R. A.; Dilman, A. D.; Struchkova, M. I.; Belyakov, P. A.; Tartakovsky, V. A.; Ioffe, S. L.: 1,3-Dipolar Cycloaddition Route to Isoxazoline N-Oxides
1109
Lu, B. Z.; Zhao, W.; Wei, H.-X.; Dufour, M.; Farina, V.; Senanayake, C. H.: One-Pot Synthesis of 2,3-Disubstituted Indoles
1110
Gwiazda, M.; Reissig, H.-U.: Synthesis of Highly Substituted Imidazoles from Lithiated Methoxyallene
1111
Kanazawa, C.; Kamijo, S.; Yamamoto, Y.: Cross-Cycloaddition of Two Different Isocyanides to Imidazoles
1112
Liu, J.; Shen, M.; Zhang, Y.; Li, G.; Khodabocus, A.; Rodriguez, S.; Qu, B.; Farina, V.; Senanayake, C. H.; Lu, B. Z.: Pd-Catalyzed Heteroannulation Route to Polycyclic Indoles
1113
Sanz, R.; Fernández, Y.; Castroviejo, M. P.; Pérez, A.; Fañanás, F. J.: Synthesis of Carbazoles, Dibenzofurans and -thiophenes via Benzynes

Synthesis of Materials and Unnatural Products

1115
Takahashi, M.; Masui, K.; Sekiguchi, H.; Kobayashi, N.; Mori, A.; Funahashi, M.; Tamaoki, N.: Activating C-H Bonds Over C-Br Bonds to Make Oligothiophenes
1116
Liu, Y.; Jessop, P. G.; Cunningham, M.; Eckert, C. A.; Liotta, C. L.: Switchable Surfactants
1117
Gupta, I.; Fröhlich, R.; Ravikanth, M.: Preparation of Thiaphlorins and Related Dyads
1118
Kumbaraci, V.; Talinli, N.; Yagci, Y.: Synthesis of Oligoesters by Photochemical Reaction
1119
Chen, C.; Xi, C.; Ai, Z.; Hong, X.: Synthesizing Higher para-Quinones Using Zirconacyclopentadienes
1120
Li, Y.; Lokitz, B. S.; McCormick, C. L.: Vesicles Formed Thermally and Cross-Linked Ionically
1121
Knapton, D.; Burnworth, M.; Rowan, S. J.; Weder, C.: Organophosphate Sensors by Fluorescent Ligands
1122
Siegel, J. S.; Baldridge, K. K.; Linden, A.; Dorta, R.: Curved Carbon Fragment of C60 as a Ligand
1123
Riddle, J. A.; Lathrop, S. P.; Bollinger, J. C.; Lee, D.: Synthesis of Stackable Pseudo-Triphenylenes
1124
Adachi, K.; Takasugi, H.; Tezuka, Y.: Macrocyclization via Ring-Emitting Covalent Fixation
1125
Mori, H.; Masuda, S.; Endo, T.: Chain Growth of Polymers with Fluorescent Main-Chain Units
1126
Ueno, T.; Urano, Y.; Kojima, H.; Nagano, T.: Fluorescence-Based Detection of Nitrating Agents in vivo

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

1127
Murakami, M.; Sakita, K.; Igawa, K.; Tomooka, K.: 1,2,3-Triols: Partial Oxidation of γ-Silyl Allylic Alcohols with Ozone
1128
Falciola, C. A.; Tissot-Croset, K.; Alexakis, A.: Cu-Catalyzed Asymmetric SN2′ Reaction onβ-Disubstituted Allylic Chlorides
1129
Hatano, M.; Miyamoto, T.; Ishihara, K.: Enantioselective Dialkylzinc Addition to Aldehydes
1130
Martín-Matute, B.; Edin, M.; Bäckvall, J.-E.: Ruthenium-Catalyzed Enzymatic Dynamic Kinetic Resolution of Diols
1131
Khan, N.-u H.; Agrawal, S.; Kureshy, R. I.; Abdi, S. H. R.; Mayani, V. J.; Jasra, R. V.: Recyclable Ti(IV)/V(V) Catalysts for ChiralO-Acetylcyanohydrin Formation
1132
Liu, J.; Wang, Y.; Li, G.: Cu(I)-Catalyzed anti-Selective Aminochlorination of Enones
1133
Weihofen, R.; Tverskoy, O.; Helmchen, G.: Enantioselective Allylic Aminations
1134
Tanaka, T.; Yasuda, Y.; Hayashi, M.: A Chiral Tridentate Schiff Base Catalyst for Alkylzinc Addition to Aldehydes
1135
Saruhashi, K.; Kobayashi, S.: Air-Stable Zr(IV) Catalysts for Asymmetric Mannich Reactions
1136
Kaiser, S.; Smidt, S. P.; Pfaltz, A.: Iridium-Catalyzed Hydrogenation of Olefins and Furan Derivatives
1137
Rhee, J. U.; Krische, M. J.: Reductive Cyclization of Acetylenic Aldehydes via Hydrogenation
1138
Manickam, G.; Siddappa, U.; Li, Y.: One-Pot Synthesis of Z-Iodoallylic Iodides from Propargyl Alcohols
1139
Evans, D. A.; Aye, Y.: Sc(III)-Catalyzed Vinylsilane Addition toN-Phenylglyoxamide
1140
Hernandez, E.; Burgos, C. H.; Alicea, E.; Soderquist, J. A.: Asymmetric Synthesis of Propargyl andα-Allenyl Alcohols from Ketones
1141
Huang, B.; Yao, X.; Li, C.-J.: 3-Component Couplings of α-Oxyaldehydes, Alkynes, and Amines in Water
1142
Walter, C.; Auer, G.; Oestreich, M.: Rh-Catalyzed Enantioselective 1,4-Addition of Silyl Boronic Esters
1143
Capriati, V.; Florio, S.; Luisi, R.; Salomone, A.; Cuocci, C.: Stereoselective Synthesis of Epoxyhydroxylamines and 1,2-Oxazetidines
1144
Blay, G.; Fernández, I.; Marco-Aleixandre, A.; Pedro, J. R.: Mandelamide-Zn-Catalyzed Enantioselective Alkyne Addition to Aldehydes
1145
Goossen, L. J.; Deng, G.; Levy, L. M.: Synthesis of Biaryls via Decarboxylative Coupling
1146
Wang, S.; Seto, C. T.: Enantioselective Addition of Vinylzinc Reagents to a Cyclic Nitrone
1147
Kobayashi, S.; Ogawa, C.: Using Rare-Earth Metals for Water-Tolerable Lewis Acid Catalysis
1148
Tanaka, K.; Hagiwara, Y.; Hirano, M.: Rh(I)-Catalyzed Stereoselective Carbocyclization of Alkynals and Alkenes
1149
Nájera, C.; Retamosa, M. G.; Sansano, J. M.: Diastereoselective 1,3-Dipolar Cylcoaddition Catalyzed by Silver Acetate
1150
Harada, T.; Kanda, K.: Unsymmetric BINOL-Titanium Complex for Enantioselective Alkylation
1151
Clark, T. B.; Woerpel, K. A.: Stereoselective Synthesis of 1,2,4-Triols from Silylenol Ethers
1152
Weiss, M. E.; Fischer, D. F.; Xin, Z.-q; Jautze, S.; Schweizer, W. B.; Peters, R.: Ferrocenyl Imidazoline Palladacycle Catalyzed aza-Claisen Rearrangement
1153
Lam, H. W.; Joensuu, P. M.; Murray, G. J.; Fordyce, E. A. F.; Prieto, O.; Luebbers, T.: Co-Catalyzed Reductive Aldol Cyclizations Using Diethylzinc as Reductant
1154
Plietker, B.: Fe-Catalyzed Allylic Amination

Metal-Mediated Synthesis

1155
Waser, J.; Gaspar, B.; Nambu, H.; Carreira, E. M.: Co-Catalyzed Hydrohydrazination and Hydroazidation of Olefins
1156
Schaffner, A.-P.; Darmency, V.; Renaud, P.: Radical Functionalization of B-Alkylcatecholboranes
1157
Korivi, R. P.; Cheng, C.-H.: Synthesis of Quinolines from Acylalkynes and 2-Iodoanilines
1158
Langille, N. F.; Jamison, T. F.: trans-Hydroalumination-Alkylation of Propargylic Alcohols
1159
Laitar, D. S.; Tsui, E. Y.; Sadighi, J. P.: Cu-Catalyzed Catalytic Diboration of Aldehydes
1160
Kofink, C. C.; Knochel, P.: Diarylmethanes from Benzylic Phosphates and Arylmagnesium Halides
1161
Friestad, G. K.; Marié, J.-C.; Suh, Y. S.; Qin, J.: Mn-Mediated Radical Diastereoselective Alkylation of N-Acylhydrazones
1162
Kabalka, G. W.; Yao, M.-L.; Borella, S.: C-Allylation of Propargyl and Benzhydryl Alcohols with Allylsilanes
1163
Anderson, K. W.; Ikawa, T.; Tundel, R. E.; Buchwald, S. L.: Pd-Catalyzed Synthesis of Phenols and Aromatic Ethers from Aryl Halides
1164
Su, W.; Raders, S.; Verkade, J. G.; Liao, X.; Hartwig, J. F.: Pd-Catalyzed α-Arylation of Trimethylsilyl Enol Ethers
1165
Cammidge, A. N.; Goddard, V. H. M.; Gopee, H.; Harrison, N. L.; Hughes, D. L.; Schubert, C. J.; Sutton, B. M.; Watts, G. L.; Whitehead, A. J.: Aryl Trihydroxyborates as Convenient Species for Cross-Coupling Reactions
1166
Hatano, M.; Suzuki, S.; Ishihara, K.: ZnCl2-Catalyzed Addition of Grignard Reagents to Ketones and Aldimines
1167
Huang, Z.; Negishi, E.-i: Cp2ZrCl2-DIBAL-H As a Convenient in situ Equivalent to Cp2ZrHCl

Organo- and Biocatalysis

1169
Gröger, H.; Chamouleau, F.; Orologas, N.; Rollmann, C.; Drauz, K.; Hummel, W.; Weckbecker, A.; May, O.: Biocatalytic Asymmetric Reduction of Ketones Using Designer Cells
1170
Lalonde, M. P.; Chen, Y.; Jacobsen, E. N.: Conjugate Addition of α,α-Disubstituted Aldehydes to Nitroalkenes
1171
Lee, S.; MacMillan, D. W. C.: Organocatalytic Epoxidation Using Hypervalent Iodine Reagents
1172
McGilvra, J. D.; Unni, A. K.; Modi, K.; Rawal, V. H.: Asymmetric Mukaiyama Aldol Reaction Catalyzed by Hydrogen Bonding
1173
Ooi, T.; Miki, T.; Fukumoto, K.; Maruoka, K.: Phase-Transfer-Catalyzed Asymmetric Alkylation of α-Acyl-γ-butyrolactones
1174
Zhao, Y.; Rodrigo, J.; Hoveyda, A. H.; Snapper, M. L.: Desymmetrization of meso-Diols via Enantioselective Silylation
1175
Staben, S. T.; Linghu, X.; Toste, F. D.: Organocatalytic Asymmetric Kornblum-DeLaMare Rearrangement
1176
Berkessel, A.; Sebastian-Ibarz, M. L.; Müller, T. N.: Dynamic Kinetic Resolution of Secondary Alcohols
1177
Tuttle, J. B.; Ouellet, S. G.; MacMillan, D. W. C.: Asymmetric Organocatalytic Transfer Hydrogenation of Cyclic Enones

Polymer-Supported Synthesis

1179
Glegoa, K.; Framery, E.; Pietrusiewicz, K. M.; Sinou, D.: PS-PEG-Supported Aryldicyclohexylphosphine Ligand for Pd-Catalyzed Suzuki Coupling
1180
Yamaguchi, K.; Imago, T.; Ogasawara, Y.; Kasai, J.; Kotani, M.; Mizuno, N.: An Immobilized Organocatalyst for Cyanosilylation
1181
Forrat, V. J.; Ramón, D. J.; Yus, M.: Polymer-Support Synthesis of Chiral Tertiary Alcohols
1182
Bandini, M.; Benaglia, M.; Quinto, T.; Tommasi, S.; Umani-Ronchi, A.: PEG-Supported Chiral Diamine Ligand for Pd-Catalyzed Allylic Alkylation
1183
Jimenez, O.; Müller, T. E.; Sievers, C.; Spirkl, A.; Lercher, J. A.: Hydroamination Catalyzed by a Pd Catalyst Immobilized in a Thin Film
1184
Lee, S. S.; Hadinoto, S.; Ying, J. Y.: Asymmetric Cyclopropanation Catalyzed by MCF-Supported Bisoxazoline-Cu(I)
1185
Wu, L.; Li, B.-L.; Huang, Y.-Y.; Zhou, H.-F.; He, Y.-M.; Fan, Q.-H.: Phosphine Dendrimer-Stabilized Pd Nanoparticles for Suzuki-Miyaura Coupling
1186
Nakamura, Y.; Maki, T.; Wang, X.; Ishihara, K.; Yamamoto, H.: A Polymer-Supported Fe-Zr Catalyst for Dehydrative Esterfication
1187
Wu, H.; Shen, Y.; Fan, L.-y; Wan, Y.; Shi, D.-q: Solid Silica Sulfuric Acid (SSA)-Catalyzed Acetylation of Aldehydes and Sugars
1188
Gheorghe, A.; Matsuno, A.; Reiser, O.: Immobilization of TEMPO onto Polystyrene Resin
1189
Struss, J. A.; Barnhart, W. D.; Velasco, M. R.; Bronley-DeLancey, A.: Polymeric DABCO-Bromine Complex for Oxidation of Alcohols
1190
Liang, Y.; Wang, Z.; Ding, K.: Self-Supported Noyori-Type Catalysts Using Achiral Bridged-BIPHEPs
1191
Lee, S.-C.; Choi, S. Y.; Chung, Y. K.; Park, S. B.: Solid-Phase Synthesis of Tetrahydroβ-carboline Alkaloid