DOI: 10.1055/s-00000131

Synfacts

Issue 10 · Volume 2011 · October 2011 DOI: 10.1055/s-002-22299

Synform

A89
Zanda, Matteo: SYNFORM ISSUE 2011/10

Synthesis of Natural Products and Potential Drugs

z1039
All PDFs of this category
1039
Day, J. J.; McFadden, R. M.; Virgil, S. C.; Kolding, H.; Alleva, J. L.; Stoltz, B. M.: Synthesis of (+)-Liphagal
1040
Slade, J.; Liu, H.; Prashad, M.; Prasad, K.: Synthesis of Aliskiren
1041
Liang, J. T.; Deng, X.; Mani, N. S.: Synthesis of a 5HT7/5HT2 Dual Antagonist
1042
Werness, J. B.; Tang, W.: Synthesis of (-)-Kumausallene
1043
Liu, G.; Romo, D.: Synthesis of (+)-Omphadiol
1044
Yoshikawa, N.; Xu, F.; Arredondo, J. D.; Itoh, T.: Synthesis of Glucokinase Activator MK-0941
1045
Zhang, X.; Mu, T.; Zhan, F.; Ma, L.; Liang, G.: Synthesis of (-)-Isatisine A
1046
Bish, G.; Hodgson et al., P. B.: Synthesis of Toll-like Receptor Agonist PF-4171455
1047
Wallace et al., D. J.: Synthesis of a PARP Inhibitor
1048
Donohoe, T. J.; Winship, P. C. M.; Tatton, M. R.; Szeto, P.: Synthesis of (-)-Neodysiherbaine A
1049
Cakmak, M.; Mayer, P.; Trauner, D.: Synthesis of the Loline Alkaloids
1050
Ghosh, A. K.; Cheng, X.: Synthesis of (-)-Zampanolide

Synthesis of Heterocycles

z1051
All PDFs of this category
1051
Pace, V.; Hoyos, P.; Sinisterra, J. V.; Alcántara, A. R.; Holzer, W.: Synthesis of 2-Aminoepoxides from Aminohalohydrins Using KF on Celite
1052
Ma, B.; Wang, Y.; Peng, J.; Zhu, Q.: Pd-Catalyzed Synthesis of Quinazolin-4(3H)-ones from N-Aryl Amidines
1053
Jiang, H.; Ji, X.; Li, Y.; Chen, Z.; Wang, A.: Pd-Catalyzed Synthesis of 1,4-Dihydro-pyridines via a Multicomponent Reaction
1054
Lopchuck, J. M.; Gribble, G. W.: A Convenient 1,3-Dipolar Cycloaddition Approach to Pyridylpyrroles
1055
Szatmári, I.; Fülöp, F.: Oxazinoisoquinoline Synthesis via the Unusual Reactivity of Aminomethylnaphthols
1056
Babinski, D. J.; Aguilar, H. R.; Still, R.; Frantz, D. E.: Pericyclic Approach to Synthesis of Substituted Pyrazoles
1057
Wetzel, A.; Gagosz, F.: Gold-Catalyzed Heteroannulation Route to Indolin-3-ones and Indoles
1058
Yu, X.; Lu, X.: 1-Benzoxepines from 2-Acylmethoxyaryl Boronic Acids and Allenoates
1059
Chen, L.; Fu, H.; Qiao, R.: Intramolecular Ullmann Cross-Coupling Route to Fused Pyridoquinazolinones
1060
Kumar, R.; Namboothiri, I. N. N.: Sulfonylpyrazoles via Base-Mediated Reaction of Diazosulfone with Nitroalkenes
1061
Li, W.; Li, X.; Wu, W.; Liang, X.; Ye, J.: One-Pot Enantioselective Michael-Aldol Approach to Imidazole Derivatives
1062
Jarvis, S. B. D.; Charette, A. B.: Synthesis of Enantiopure Piperidines via an Aziridinium Ring Expansion Reaction
1063
Nakanishi, M.; Katayev, M.; Besnard, C.; Kündig, E. P.: Palladium-Catalyzed C-H Activation Induced Enantioselective Route to Fused Indolines
1064
Nishino, M.; Hirano, K.; Satoh, T.; Miura, M.: Cu-Catalyzed Oxidative Synthesis of Tetrahydroquinolines from N-Methylanilines
1065
Nakai, K.; Kurahashi, T.; Matsubara, S.: Ni-Catalyzed Cycloaddition Approach to Coumarins by C-C σ-Bond Cleavage

Synthesis of Materials and Unnatural Products

z1067
All PDFs of this category
1067
Ishii, A.; Yamaguchi, Y.; Nakata, N.: Highly Fluorescent Dyes, Never Mind the Heavy Atoms
1068
Takase, M.; Yoshida, N.; Nishinaga, T.; Iyoda, M.: Highly Charged Oxidized Tetrathiafulvalene Oligomers
1069
Ihara, E.; Hara, Y.; Itoh, T.; Inoue, K.: Multicomponent Polymerizations: It’s All about the Solvent
1070
Zhang, H.; Cao, D.; Liu, W.; Jiang, H.; Meier, H.: New Additions to the Triptycene Family
1071
Namba, K.; Osawa, A.; Ishizaka, S.; Kitamura, N.; Tanino, K.: Fluorescent Triazapentalenes
1072
Abbey, E. R.; Zakharov, L. N.; Liu, S.-Y.: Synthesis of a ‘Fused’ BN Indole
1073
Mochida, K.; Kawasumi, K.; Segawa, Y.; Itami, K.: Palladium Catalysis for Extended PAHs
1074
Rix, D.; Ballesteros-Garrido, R.; Zeghida, W.; Besnard, C.; Lacour, J.: One-Pot Synthesis of Unusual 15-Membered Polyether Macrocycles
1075
Chiu, C.-Y.; Kim, B.; Gorodetsky, A.; Sattler, W.; Wei, S.; Sattler, A.; Steigerwald, M.; Nuckolls, C.: Dibenzotetrathienocoronenes and Hexabenzocoronene in Three Steps
1076
Mastalerz, M.; Sieste, S.; Cenić, M.; Oppel, I. M.: Two’s Company, Six is a Crowded Triptycene
1077
Korovina, N. V.; Chang, M. L.; Nguyen, T. T.; Fernandez, R.; Walker, H. J.; Olmstead, M. M.; Gherman, B. F.; Spence, J. D.: Photodimerization of Arenediynes
1078
Purushothaman, B.; Bruzek, M.; Parkin, S. R.; Miller, A.-F.; Anthony, J. E.: Nine in a Row: Taming the Acenes
1079
Peng, P.; Strohecker, D.; Liao, Y.: Photochromism in Reverse

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1081
All PDFs of this category
1081
Turlington, M.; Pu, L.: Rh(I)-Catalyzed Pauson-Khand Cycloaddition
1082
Wu, Y.; Mao, F.; Meng, F.; Li, X.: Enantioselective Vanadium-Catalyzed Oxidation of 1,3-Dithianes
1083
Marinescu, S. C.; Levine, D. S.; Zhao, Y.; Schrock, R. R.; Hoveyda, A. H.: Purification of Alkene Stereoisomers through Z-Selective Ethenolysis
1084
Goto, T.; Takeda, K.; Shimada, N.; Nambu, H.; Anada, M.; Shiro, M.; Ando, K.; Hashimoto, S.: Asymmetric Dirhodium-Catalyzed Cyclopropenation of Terminal Alkynes
1085
Haddad, N.; Qu, B.; Rodriguez, S.; van der Veen, L.; Reeves, D. C.; Gonnella, N. C.; Lee, H.; Grinberg, N.; Ma, S. L.; Krishnamurthy, D.; Wunberg, T.; Senanayake, C. H.: Asymmetric Hydrogenation of Heterocyclic Ketone-Derived Hydrazones
1086
Gao, X.; Han, H.; Krische, M. J.: Iridium-Catalyzed Asymmetric Double Crotylation of 1,3-Diols
1087
Franckevičius, V.; Cuthbertson, J. D.; Pickworth, M.; Pugh, D. S.; Taylor, R. J. K.: Asymmetric Decarboxylative Allylation of Oxindoles
1088
Cao, H. T.; Roisnel, T.; Valleix, A.; Grée, R.: Nickel-Catalyzed Tandem Isomerization-Mannich Reaction
1089
McDonald, R. I.; White, P. B.; Weinstein, A. B.; Tam, C. P.; Stahl, S. S.: Enantioselective Pd(II)-Catalyzed Aerobic Oxidative Amidation of Alkenes
1090
Shibatomi, K.; Narayama, A.; Soga, Y.; Muto, T.; Iwasa, S.: Enantioselective gem-Chlorofluorination of Active Methylene Compounds
1091
Brooks, J. L.; Caruana, P. A.; Frontier, A. J.: Nazarov Cyclizations of Dienyl Diketones Initiated by Conjugate Addition
1092
Chen, F.; Ding, Z.; Qin, J.; Wang, T.; He, Y.; Fan, Q.-H.: Asymmetric Hydrogenation of Cyclic N-Alkyl Imines
1093
Ghosh, A. K.; Nicponski, D. R.: Cu(II)-Catalyzed Synthesis of Substituted Tetrahydropyrans
1094
Iqbal, M.; Mistry, N.; Clarke, P. A.: Catalytic Enantioselective Synthesis of Tetrahydro-4-ones
1095
Corberán, R.; Mszar, N. W.; Hoveyda, A. H.: Copper-Catalyzed Enantioselective Hydroboration
1096
Han, X.; Gan, M.; Qiu, H.; Ji, J.; Zhang, X.; Jiang, L.; Hu, W.: Rhodium-Catalyzed Trapping of Oxonium Ylides with Michael Acceptors
1097
Lv, C.; Cheng, Q.; Xu, D.; Wang, S.; Xia, C.; Sun, W.: Effects of Salen Ligands in Ti-Catalyzed Cyanosilylation of Aldehydes
1098
Gärtner, M.; Jäkel, M.; Achatz, M.; Sonnenschein, C.; Tverskoy, O.; Helmchen, G.: Enantioselective Allylic Substitutions with Hydroxamic Acid Derivatives
1099
Palmer, L. I.; de Alaniz, J. Read: Dysprosium(III) Triflate Catalyzed Aza-Piancatelli Rearrangement
1100
Fandrick, K. R.; Fandrick, D. R.; Reeves, J. T.; Gao, J.; Ma, S. L.; Li, W. J.; Lee, H.; Grinberg, N.; Lu, B.; Senanayake, C. H.: Cu-Catalyzed Asymmetric Propargylation of Ketones
1101
Lv, J.; Zhang, L.; Zhou, Y.; Nie, Z.; Cheng, J.-P.; Luo, S.: Binary Acid System for Asymmetric Regioselective 1,2- and 1,4- Addition
1102
Chuprakov, S.; Malik, J. A.; Zibinsky, M.; Fokin, V. V.: Catalytic Asymmetric C-H Insertions of Rhodium(II) Azavinyl Carbenes
1103
Soni, R.; Collinson, J.-M.; Clarkson, G. C.; Wills, M.: Asymmetric Transfer Hydrogenation of α,α-Disubstituted Ketones
1104
Xue, Z.-Y.; Li, Q.-H.; Tao, H.-Y.; Wang, C.-J.: Conjugate Addition Approach Towards Unnatural Amino Acid Derivatives
1105
Gao, Q.; Lu, S.-M.; Liu, Y.; Li, C.: Chiral Diamine-Polyoxometalate (POM) Acid Catalyzed Aldol Reaction
1106
Deng, Z. H.; Feng, J. H.; Cao, W. D.; Liu, X. H.; Lin, L. L.; Feng, X. M.: N,N′-Dioxide-Ni Complex Catalyzed Asymmetric Michael Addition
1107
Xie, J.-H.; Liu, X.-Y.; Xie, J.-B.; Wang, L.-X.; Zhou, Q.-L.: Iridium-Catalyzed Asymmetric Hydrogenation of Ketones
1108
Trost, B. M.; Thaisrivongs, D. A.; Hartwig, J.: Asymmetric Allylic Alkylation of Diverse Nitrogen-Containing Heterocycles
1109
Cui, Z.; Yu, H.-J.; Yang, R.-F.; Gao, W.-Y.; Feng, C.-G.; Lin, G.-Q.: Asymmetric Arylation of Aliphatic Aldimines

Metal-Mediated Synthesis

z1111
All PDFs of this category
1111
Yu, D.-G.; Shi, Z.-J.: Direct Suzuki-Miyaura Coupling of Phenol Derivatives via Mutual Activation
1112
Kawai, H.; Furukawa, T.; Nomura, Y.; Tokunaga, E.; Shibata, N.: Cu-Mediated Trifluoromethylation of Benzyl Bromides
1113
Zhang, Y.; Gao, J.; Li, W.; Lee, H.; Lu, B. Z.; Senanayake, C. H.: Pd-Catalyzed One-Pot Process to Yield 8-Arylquinolines
1114
Zhang, X.; Liu, H.; Hu, X.; Tang, G.; Zhu, J.; Zhao, Y.: Ni-Catalyzed Cross-Coupling of Aryl Halides with Diphenylphosphine Oxide
1115
Schnapperelle, I.; Breitenlechner, S.; Bach, T.: Regioselective Oxidative Couplings of 3-Substituted Thiophenes
1116
Schneider, C.; Broda, E.; Snieckus, V.: One-Pot ortho-Borylation and Subsequent Cross-Coupling-Reaction
1117
Molander, G. A.; Shin, I.: Suzuki Coupling of an Aminomethyl Equivalent with (Hetero)Aryl Halides
1118
Ramachandran, P. V.; Tafelska-Kaczmarek, A.; Sakavuyi, K.: Preparation and Reaction of Chiral Difluoroallylboronates
1119
Teverovskiy, G.; Surry, D. S.; Buchwald, S. L.: Pd-Catalyzed Synthesis of (Het)Ar-SCF3 Compounds
1120
Maekawa, T.; Sekizawa, H.; Itami, K.: Ni-Catalyzed Alcohol-Carbonyl Interconversions
1121
Sueda, T.; Oshima, A.; Teno, N.: Cu-Catalyzed Coupling Reaction to Yield Ynimides
1122
Liu, C.; Deng, Y.; Wang, J.; Yang, Y.; Tang, S.; Lei, A.: Pd-Catalyzed Construction of 2,3-Diaryl 1,4-Diketones
1123
DeLuca, R. J.; Sigman, M. S.: Pd-Catalyzed Anti-Markovnikov Hydroalkylation of Allylic Amines
1124
Prakash, G. K. S.; Paknia, F.; Mathew, T.; Mlostoń, G.; Joshek, J. P.; Olah, G. A.: Synthesis of Polyfluoro-2,2-diarylethanes

Organo- and Biocatalysis

z1125
All PDFs of this category
1125
Jones, S. B.; Simmons, B.; Mastracchio, A.; MacMillan, D. W. C.: Collective, Organocatalytic Syntheses of Natural Products: Strychnos Alkaloids
1126
Zhao, D.; Yang, D.; Wang, Y.; Wang, Y.; Wang, L.; Mao, L.; Wang, R.: Asymmetric Mannich Reaction of a HWE Reagent to Afford MBH-Type Products
1127
Xiao, X.; Xie, Y.; Su, C.; Liu, M.; Shi, Y.: Synthesis of α-Amino Acid Derivatives by Biomimetic Transamination
1128
Lozano, O.; Blessley, G.; Campo, T. Martinez del; Thompson, A. L.; Giuffredi, G. T.; Bettati, M.; Walker, M.; Borman, R.; Gouverneur, V.: Organocatalytic Enantioselective Fluorocyclizations
1129
Antonchick, A. P.; Samanta, R.; Kulikov, K.; Lategahn, J.: Metal-Free Intra- and Intermolecular Oxidative C-N Bond Formation
1130
Wu, Y.; Singh, R. P.; Deng, L.: Asymmetric Olefin Isomerization of Butenolides
1131
Beck, E. M.; Hyde, A. M.; Jacobsen, E. N.: Enantioselective Protonation of Enol Silanes by Protonated Chiral Sulfinamides
1132
Chen, L.-Y.; He, H.; Chan, W.-H.; Lee, A. W. M.: Brønsted Acid Catalysis: Friedel-Crafts Alkylation with Chiral Disulfonimides
1133
Henseler, A.; Kato, M.; Mori, K.; Akiyama, T.: Chiral Phosphoric Acid Catalyzed Transfer Hydrogenation of Ketimines
1134
Jia, Z.-J.; Zhou, Q.; Zhou, Q.-Q.; Chen, P.-Q.; Chen, Y.-C.: exo-Selective Diels-Alder Reaction of 2,4-Dienals and Nitroalkenes

Polymer-Supported Synthesis

z1135
All PDFs of this category
1135
Chen, J. M.; Zeng, X. M.; Middleton, K.; Yusubov, M. S.; Zhdankin, V. V.: Polystyrene-Supported Iodosylbenzene as an Oxidizing Reagent
1136
Miura, T.; Imai, K.; Kasuga, H.; Ina, M.; Tada, N.; Imai, N.; Itoh, A.: Asymmetric Aldol Reactions in Brine with Fluorous Organocatalysts
1137
Lykakis, I. N.; Psyllaki, A.; Stratakis, M.: Cycloaddition of Tetramethyldisiloxane to Alkynes with [Au]/TiO2
1138
Yang, J.; Li, P.; Wang, L.: Synthesis of 2-Aminobenzothiazoles with a Polymeric Phen-Cu(I) Complex
1139
Banerjee, S.; Khatri, H.; Balasanthiran, V.; Koodali, R. T.; Sereda, G.: Cross-Coupling Using Mesoporous Pd-MCM-48
1140
Rahman, M.; Bagdi, A. K.; Majee, A.; Hajra, A.: Synthesis of Propargylamines with In2O3 Nanoparticles
1141
Zhang, W.; Zeng, Q.; Zhang, X.; Tian, Y.; Yue, Y.; Guo, Y.; Wang, Z.: Arylation of Heterocycles with a CuO Nanospindle
1142
Hermannsdörfer, J.; Kempe, R.: Pd Nanoparticles in the Metal-Organic Framework MIL-101
1143
Song, F.; Wang, C.; Lin, W.: Asymmetric Epoxidation with a Chiral Metal-Organic Framework
1144
Dhahagani, K.; Rajesh, J.; Kannan, R.; Rajagopal, G.: Asymmetric Henry Reaction with MCM-41-Supported Cu-Salen Complex
1145
Hong, H.; Hu, L.; Li, M.; Zheng, J.; Sun, X.; Lu, X.; Cao, X.; Lu, J.; Gu, H.: Oxidation of Olefins and Alcohols with Pt@Fe2O3 Nanowires
1146
Murugan, K.; Srimurugan, S.; Chen, C.: Hosomi-Sakurai Reaction with Silicomolybdic Acid
1147
Liu, Z.; Chen, W.; Giulianotti, M. A.; Houghten, R. A.: Solid-Phase Synthesis of Tetrahydrobenzo-diazepine Derivatives
1148
Hankari, S. El; Kadib, A. El; Finiels, A.; Bouhaouss, A.; Moreau, J. J. E.; Crudden, C. M.; Brunel, D.; Hesemann, P.: An Organosilica-Supported Pd Catalyst