DOI: 10.1055/s-00000131

Synfacts

Issue 11 · Volume 2009 · November 2009 DOI: 10.1055/s-002-20475

Synform

A68
Zanda, Matteo: SYNFORM ISSUE 2009/08

Synthesis of Natural Products and Potential Drugs

z1181
All PDFs of this category
1181
Yoo, K.; Kim, H.; Yun, J.: Synthesis of (R)-Tolterodine
1182
Williams, D. R.; Walsh, M. J.; Miller, N. A.: Synthesis of 4-Hydroxydictyolactone
1183
Newhouse, T.; Lewis, C. A.; Baran, P. S.: Synthesis of Kapakahines B and F
1184
Takamura, H.; Kikuchi, S.; Nakamura, Y.; Yamagami, Y.; Kishi, T.; Kadota, I.; Yamamoto, Y.: Synthesis of Brevenal
1185
Sullivan, B.; Carrera, I.; Drouin, M.; Hudlicky, T.: Synthesis of Oseltamivir
1186
Snyder, S. A.; Tang, Z.-Y.; Gupta, R.: Synthesis of (-)-Napyradiomycin A1
1187
Pereira, C. L.; Chen, Y.-H.; McDonald, F. E.: Synthesis of Fumonisin B1
1188
Maligres, P. E.; Humphrey, G. R.; Marcoux, J.-F.; Hillier, M. C.; Zhao, D.; Krska, S.; Grabowski, E. J. J.: Synthesis of a Selective PPARγ Modulator
1189
Li, Y.; Kobayashi, T.; Katsumura, S.: Synthesis of (-)-Corynantheidol
1190
Savage, S. A.; Waltermire, R. E.; Campagna, S.; Bordawekar, S.; Toma, J. D. R.: Synthesis of an Oral TACE Inhibitor
1191
Pérez, M.; Pérez, D. I.; Martínez, A.; Castro, A.; Gómez, G.; Fall, Y.: Synthesis of Palinurin
1192
Lee, B.; Kwon, J.; Yu, C.-M.: Synthesis of (-)-Adaline
1193
Shenvi, R. A.; Corey, E. J.: Synthesis of (-)-7-Methylomuralide
1194
Nicolaou, K. C.; Wu, T. R.; Kang, Q.; Chen, D. Y.-K.: Synthesis of ()-Hopeanol

Synthesis of Heterocycles

z1195
All PDFs of this category
1195
Wang, Y.-F.; Chiba, S.: Mn(III)-Mediated Synthesis of Pyridines
1196
Facoetti, D.; Abbiati, G.; d’Avolio, L.; Ackermann, L.; Rossi, E.: TiCl4-Catalyzed Synthesis of Pyrimido[1,6-a]indol-1-ones
1197
Donets, P. A.; van Hecke, K.; van Meervelt, L.; van der Eycken, E. V.: Synthesis of Indoloazocine by Hg(OTf)2-Catalyzed Intramolecular Carbocyclization
1198
Bryan, C. S.; Braunger, J. A.; Lautens, M.: Pd-Catalyzed Synthesis of Benzothiophenes from gem-Dihalovinyl Thiophenols
1199
Duguet, N.; Salwin, A. M. Z.; Smith, A. D.: Asymmetric Synthesis of 3-Alkyl-3-aryl-oxindoles
1200
Savitha, G.; Felix, K.; Perumal, P. T.: Pd-Catalyzed Synthesis of 3-Bromo-2H-Chromenes
1201
Azizi, N.; Khajeh-Amiri, A.; Ghafuri, H.; Bolourtchian, M.; Saidi, M. Reza: FeCl3-Catalyzed Synthesis of N-Substituted Pyrroles in Water
1202
Friedman, R. Keller; Rovis, T.: Rh-Catalyzed Cycloadditions of Unsymmetrical Alkynes with Isocyanates
1203
Allen, C. P.; Benkovics, T.; Turek, A. K.; Yoon, T. P.: Synthesis of Tetrahydroisoquinolines and Tetrahydropyridines from Oxaziridines
1204
Lu, W.; Song, W.; Hong, D.; Lu, P.; Wang, Y.: Cu-Catalyzed Multicomponent Synthesis of 1,2,3,4-Tetrahydropyrimidines
1205
Tang, S.; He, J.; Sun, Y.; He, L.; She, X.: Regioselective One-Pot Straightforward Synthesis of Isoxazoles
1206
Chandra, A.; Singh, B.; Khanna, R. S.; Singh, R. M.: Pd-Catalyzed One-Pot Coupling-Annulation Synthesis of Pyrano[4,3-b]quinolines
1207
Zhao, X.; Zhang, E.; Tu, Y.-Q.; Zhang, Y.-Q.; Yuan, D.-Y.; Cao, K.; Fan, C.-A.; Zhang, F.-M.: Au(I)-Catalyzed Synthesis of Cycloalkene-Fused Pyrroles
1208
Burton, D. J.; Hansen, S. W.: Synthesis of Fluorinated α-Pyrans
1209
Yang, D.; Liu, H.; Yang, H.; Fu, H.; Hu, L.; Jiang, Y.; Zhao, Y.: Efficient Cu-Catalyzed Synthesis of 1,2,4-Benzothiadiazine-1,1-dioxides

Synthesis of Materials and Unnatural Products

z1211
All PDFs of this category
1211
Isobe, H.; Hitosugi, S.; Matsuno, T.; Iwamoto, T.; Ichikawa, J.: Synthesis of Chrysenes through an Unexpected Skeletal Rearrangement
1212
Robinson, S. G.; Sauro, V. A.; Mitchell, R. H.: Switchable Molecular Wires
1213
Clever, G. H.; Tashiro, S.; Shionoya, M.: A Molecular Cage with Electrostatic Anchors
1214
Hayashi, S.; Inagi, S.; Fuchigami, T.: Electro-Fluorination of Polymers
1215
Robbins, S. J.; Thibault, M. E.; Masuda, J. D.; Ward, D. R.; Boeré, R. T.; Dibble, P. W.: Isobenzofurans and Cyclophanes
1216
Nakazono, S.; Imazaki, Y.; Yoo, H.; Yang, J.; Sasamori, T.; Tokitoh, N.; Cédric, T.; Kageyama, [nl]H.; Kim, D.; Shinokubo, H.; Osuka, A.: Regioselective Functionalization of Perylene through C-H Bond Activation
1217
Morinaka, K.; Ubukata, T.; Yokoyama, Y.: Synthesis and Cyclization of Photochromic Bisarylindenones
1218
Binauld, S.; Hawker, C. J.; Fleury, E.; Drockenmuller, E.: High-Yielding Click Route to Macrocycles
1219
Ni, Y.; Nakajima, K.; Kanno, K.-i.; Takahashi, T.: Thiophene-Fused Acenes
1220
Matsuo, Y.; Maruyama, M.; Gayathri, S. S.; Uchida, T.; Guldi, D. M.; Kishida, H.; Nakamura, A.; Nakamura, E.: Symmetric Fullerene Dumbbells
1221
Sehnal, P.; Stará, I. G.; Šaman, D.; Tichý, M.; Míšek, J.; Cvačka, J.; Rulíšek, L.; Chocholšouova, J.; Vacek, J.; Goryl, G.; Szymonski, M.; Císařová, I.; Star, I.: Long Helicenes by Alkyne Cycloisomerization
1222
Newman, S. G.; Aureggi, V.; Bryan, C. S.; Lautens, M.: 2-Bromo Benzofurans and Benzothiophenes via Cu-Catalyzed Cross-Coupling
1223
Zhang, F.; Götz, G.; Winkler, H. D. F.; Schalley, C. A.; Bäuerle, P.: A Platinum Template Strategy to Cyclo[n]thio-phenes
1224
Takaba, H.; Omachi, H.; Yamamoto, Y.; Bouffard, J.; Itami, K.: Hooping it up
1225
Arai, S.; Sato, T.; Nishida, A.: Catalytic Dicyanation

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1227
All PDFs of this category
1227
Yanagisawa, A.; Terajima, Y.; Sugita, K.; Yoshida, K.: Dibutyltin Dimethoxide and Ag(I)-BINAP-Catalyzed Aldol Reactions of Ketones
1228
Wang, D.-Y.; Hu, X.-P.; Hou, C.-J.; Deng, J.; Yu, S.-N.; Duan, Z.-C.; Huang, J.-D.; Zheng, Z.: Enantioselective Rh-Catalyzed Hydrogena-tion of 3-Aryl-2-phosphonomethylpropenoates
1229
Geng, H.; Zhang, W.; Chen, J.; Hou, G.; Zhou, L.; Zou, Y.; Wu, W.; Zhang, X.: Rhodium-Catalyzed Hydrogenation of β-Keto Enamides
1230
Mothe, S. R.; Chan, P. W. H.: Brønsted Acid Catalyzed Formation of Enynes
1231
Pouy, M. J.; Stanley, L. M.; Hartwig, J. F.: Enantioselective Monoallylation of Ammonia
1232
Moro, A. Venturini; Cardoso, F. Sega Pareira; Correia, C. Roque Duarte: Stereoselective Heck Reaction of Allylic Esters with Arenediazonium Salts
1233
Park, Y.; Kang, S.; Lee, Y. J.; Kim, T.-S.; Jeong, B.-S.; Park, H.-g.; Jew, S.-s.: Asymmetric Phase-Transfer Catalytic Alkylation of Imidazoline-4-carboxylates
1234
Noh, D.; Chea, H.; Ju, J.; Yun, J.: Copper-Catalyzed Asymmetric Hydroboration of Styrenes
1235
Uchida, T.; Katsuki, T.: Cu(I)-Catalyzed Asymmetric Conjugate Alkylation with New NHC Ligands
1236
Li, F.-Q.; Zhong, S.; Lu, G.; Chan, A. S. C.: Alkynylation of Acylsilanes via Zinc-Salen Catalysis
1237
Lu, Y.; Johnstone, T. C.; Arndtsen, B. A.: Coupling of Imines and Alkynes through Amino Acid and Metal Catalysis
1238
Wilkinson, S. C.; Lozano, O.; Schuler, M.; Pacheco, M. C.; Salmon, R.; Gouverneur, V.: Stereospecific Synthesis of Fluorinated Tetrahydrofurans
1239
Wang, C.; Li, C.; Wu, X.; Pettman, A.; Xiao, J.: pH-Regulated Asymmetric Transfer Hydrogenation of Quinolines in Water
1240
Tan, Q.; Hayashi, M.: Copper-Catalyzed Allylic Oxidation of 4,5-Epoxycyclohex-1-ene
1241
Aikawa, K.; Kojima, M.; Mikami, K.: Chiral Anion-Controlled Axial Chirality of Gold(biphep) Complexes
1242
Chen, I-H.; Yin, L.; Itano, W.; Kanai, M.; Shibasaki, M.: Copper-Catalyzed Asymmetric Conjugate Boration of Cyclic Enones
1243
Biradar, D. B.; Zhou, S.; Gau, H.-M.: Titanium-Catalyzed Thienylation to Ketones
1244
Alladoum, J.; Vrancken, E.; Mangeney, P.; Roland, S.; Kadouri-Puchot, C.: Syntheses of Enantiopure Bicyclic Oxazolidines Using Pd(II) Catalysts
1245
Wu, M.; Wang, B.; Wang, S.; Xia, C.; Sun, W.: Novel Chiral Mn(II) Complexes for Asymmetric Epoxidation of Olefins
1246
da Silva, W. A.; Rodrigues Jr., M. T.; Shankaraiah, N.; Ferreira, R. B.; Andrade, C. K. Z.; Pilli, R. A.; Santos, L. S.: Supramolecular Pd Catalyst for the Reduction of Dihydro-β-Carbolines
1247
Hashimoto, T.; Miyamoto, H.; Naganawa, Y.; Maruoka, K.: Auxiliary-Based Diastereoselective Roskamp Reaction
1248
Yamaguchi, A.; Matsunaga, S.; Shibasaki, M.: Direct Aldol Reaction via Dynamic Kinetic Asymmetric Transformation
1249
Nishihara, Y.; Saito, D.; Tanemura, K.; Noyori, S.; Takagi, K.: Zirconocene-Mediated Stereoselective Synthesis of Multisubstituted Vinylsilanes
1250
Mangion, I.; Strotman, N.; Drahl, M.; Imbriglio, J.; Guidry, E.: Dynamic Kinetic Asymmetric Allylation of Hydrazines and Hydroxylamines
1251
Taniguchi, H.; Ohmura, T.; Suginome, M.: Synthesis of γ,δ-Unsaturated Ketones from Methylenecyclopropanes
1252
Miura, T.; Shimada, M.; de Mendoza, P.; Deutsch, C.; Krause, N.; Murakami, M.: Rhodium-Catalyzed Formation of syn-α-Allenols
1253
Ghorai, M. K.; Shukla, D.; Das, K.: A Modular Approach to the Synthesis of Morpholines
1254
Trost, B. M.; Thaisrivongs, D. A.: Benzylic Allylation of 2-Substituted Pyridines

Metal-Mediated Synthesis

z1255
All PDFs of this category
1255
Yu, D.-G.; Yu, M.; Guan, B.-T.; Li, B.-J.; Zheng, Y.; Wu, Z.-H.; Shi, Z.-J.: Suzuki-Miyaura Coupling through C-CN Bond Cleavage
1256
Barluenga, J.; Tomás-Gamasa, M.; Aznar, F.; Valdés, C.: Direct Metal-Catalyst-Free Reductive Cou-pling of Boronic Acids and Tosylhydrazones
1257
Tobisu, M.; Ano, Y.; Chatani, N.: Pd-Catalyzed Direct Alkynylation of C-H Bonds in Benzenes
1258
Wei, Y.; Kan, J.; Wang, M.; Su, W.; Hong, M.: Direct Arylation of Polyfluoroarenes with Arylboronic Acids
1259
Söderberg, B. C. G.; Gorugantula, S. P.; Howerton, C. R.; Petersen, J. L.; Dantale, S. W.: Pd-Catalyzed Synthesis of Isatins from (2-Haloethynyl)nitrobenzenes
1260
Awuah, E.; Capretta, A.: Microwave-Assisted Pd-Catalyzed Flavone Synthesis from Arenes
1261
Han, W.; Ofial, A. R.: Fe-Catalyzed Oxidative Cyanation of Tertiary Amines
1262
Rice, G. T.; White, M. C.: Allylic C-H Amination for the Synthesis of syn-1,3-Amino Alcohols
1263
Shapiro, N. D.; Shi, Y.; Toste, F. D.: Au-Catalyzed [3+3] Annulation of Azomethine Imines with Propargyl Esters
1264
Ye, L.; Zhang, L.: Au/Mo-Catalyzed Synthesis of α-Halo-α,β-unsaturated Carbonyls
1265
Yu, W.-Y.; Sit, W. N.; Zhou, Z.; Chan, A. S. C.: Pd-Catalyzed Decarboxylative Arylation of C-H Bonds
1266
Candito, D. A.; Lautens, M.: Direct Synthesis of Phenanthridines via Domino Arylation/N-Arylation
1267
Hilt, G.; Danz, M.; Treutwein, J.: Co-Catalyzed 1,4-Hydrovinylation
1268
Hatakeyama, T.; Hashimoto, S.; Ishizuka, K.; Nakamura, M.: Biaryl Cross Coupling Catalyzed by Fe/Co/Ni-Fluorides and NHC Ligands
1269
Li, S.; Qu, H.; Zhou, L.; Kanno, K.; Guo, Q.; Shen, B.; Takahashi, T.: Zr-Mediated Synthesis of 1,2,4,5-Tetra-substituted Benzenes from Alkynes

Organo- and Biocatalysis

z1271
All PDFs of this category
1271
Gong, B.; Meng, Q.; Su, T.; Lian, M.; Wang, Q.; Gao, Z.: Lappaconitine Catalysis
1272
B. Jones, S.; Simmons, B.; MacMillan, D. W. C.: Nine-Step Total Synthesis of (+)-Minfiensine
1273
Scroggins, S. T.; Chi, Y.; Fréchet, J. M. J.: Cascade Reactions Directed by Polarity
1274
O’Brien, C. J.; Tellez, J. L.; Nixon, Z. S.; Kang, L. J.; Carter, A. L.; Kunkel, S. R.; Przeworski, K. C.; Chass, G. A.: Catalytic Wittig Reaction via in situ Phosphine Oxide Recycling
1275
Cheng, Y.-Q.; Bian, Z.; He, Y.-B.; Han, F.-S.; Kang, C.-Q.; Ning, Z.-L.; Gao, L.-X.: An Effective Combination of Prolinamides and BINOLs
1276
Marqués-López, E.; Herrera, R. P.; Marks, T.; Jacobs, W. C.; Könning, D.; de Figueiredo, R. M.; Christmann, M.: Dienamine Activation in Enantioselective Intramolecular Rauhut-Currier Reactions
1277
Momiyama, N.; Tabuse, H.; Terada, M.: anti-Diastereoselective and Enantioselective Hetero-Diels-Alder Reaction
1278
Galzerano, P.; Pesciaioli, F.; Mazzanti, A.; Bartoli, G.; Melchiorre, P.: Aminocatalysis Cascades of α-Branched α,β-Unsaturated Aldehydes
1279
Chen, X.-H.; Wei, Q.; Luo, S.-W.; Xiao, H.; Gong, L.-Z.: Organocatalytic Synthesis of Spiro[pyrrolidin-3,3′-oxindoles]
1280
Lathrop, S. P.; Rovis, T.: Secondary Amine/N-Heterocyclic Carbene Catalyzed Cascade Sequence
1281
Fu, X.; Loh, W.-T.; Zhang, Y.; Chen, T.; Ma, T.; Liu, H.; Wang, J.; Tan, C.-H.: Guanidinium Salt Catalyzed Imine Hydrophosphonylation
1282
Zhu, C.; Akiyama, T.: A New Organic Hydrogenation Reagent
1283
Wu, L.-Y.; Bencivenni, G.; Mancinelli, M.; Mazzanti, A.; Bartoli, G.; Melchiorre, P.: Aminocatalysis Cascades of Enones
1284
Jones, C. R.; Panto, G. D.; Morrison, A. J.; Smith, M. D.: Hydrogen-Bond-Assisted Hydrogen-Bonding Catalysis
1285
Alza, E.; Rodríguez-Escrich, C.; Sayalero, S.; Bastero, A.; Pericàs, M. A.: Continuous-Flow Mannich Reactions Using a Solid-Supported Hydroxyproline

Polymer-Supported Synthesis

z1287
All PDFs of this category
1287
Oishi, T.; Yamaguchi, K.; Mizuno, N.: Synthesis of Nitriles from Primary Alcohols and NH3 with Ru(OH)x/Al2O3
1288
Mitsudome, T.; Noujima, A.; Mizugaki, T.; Jitsukawa, K.; Kaneda, K.: Aerobic Oxidation of Alcohols with Au/HT
1289
Hagiwara, H.; Sekifuji, M.; Tsubokawa, N.; Hoshi, T.; Suzuki, T.: Henry Reaction with Nano-NAP
1290
Chakraborti, A. K.; Singh, B.; Chankeshwara, S. V.; Patel, A. R.: HClO4-SiO2 Catalyst for Esterification of Carboxylic Acids with Alcohols
1291
Shylesh, S.; Schweizer, J.; Demeshko, S.; Schünemann, V.; Ernst, S.; Thiel, W. R.: Epoxidation of Olefins with Nanoparticle-Supported Mo Complexes
1292
Niknam, K.; Saberi, D.: SBNPSA-Catalyzed Formylation and Acetylation of Alcohols and Amines
1293
Lang, L.; Li, B.; Liu, W.; Li, X.; Xu, Z.: The Aerobic Oxidation of Benzylic Alcohols with F-MSS Catalyst
1294
Wei, J.-F.; Jiao, J.; Feng, J.-J.; Lv, J.; Zhang, X.-R.; Shi, X.-Y.; Chen, Z.-G.: Aqueous Suzuki Reactions with PdEDTA in SiO2-Ionic Liquid
1295
Jung, N.; Bräse, S.: SPOS of Natural Products via Ullmann Condensation
1296
Cheng, C.; Sun, J.; Xing, L.; Xu, J.; Wang, X.; Hu, Y.: Pd/C-Catalyzed N-Debenzylation of Benzylamines
1297
Snelders, D. J. M.; van Koten, G.; Gebbink, R. J. M. Klein: Hexacationic Dendriphos-Pd Complexes for Suzuki-Miyaura Reaction
1298
Akagawa, K.; Yamashita, T.; Sakamoto, S.; Kudo, K.: Asymmetric Alkylation Using Resin-Supported Peptide Catalysts
1299
Kristensen, T. E.; Vestli, K.; Fredriksen, K. A.; Hansen, F. K.; Hansen, T.: Aldol Reaction with Polymer-Supported Proline Derivatives
1300
Sedelmeier, J.; Ley, S. V.; Lange, H.; Baxendale, I. R.: Microwave-Assisted Sonogashira-Type Reaction Using Pd-EnCat

Addenda and Errata

1301
Cyclization/[3+2]-Cycloaddition Reaction of N′-(2-Alkynylbenzylidene) Hydrazides