DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 2011 · September 2011 DOI: 10.1055/s-002-22222

Synform

A76
SYNFORM ISSUE 2011/09

Synthesis of Natural Products and Potential Drugs

z925
All PDFs of this category
0925
Synthesis of (±)-Aspidophylline A
0926
Synthesis of Lathyranoic Acid A
0927
Synthesis of a γ-Secretase Inhibitor
0928
Synthesis of Lactimidomycin
0929
Synthesis of (±)-Decursivine and (±)-Serotobenin
0930
Synthesis of (±)-Decursivine
0931
Synthesis of Cyanolide A Aglycon
0932
Synthesis of (±)-Trichostatin A
0933
Synthesis of a CRF-1 Receptor Antagonist
0934
Synthesis of (-)-Conophylline
0935
Synthesis of (+)-Mefloquine Hydrochloride

Synthesis of Heterocycles

z937
All PDFs of this category
0937
Arynes in the Synthesis of N-Arylisatins
0938
Synthesis of NH-Free 3-Substituted Indazoles
0939
The Benzyne Fischer Indole Reaction
0940
Enyne Cycloisomerization Route to an Anti-depressant Drug Candidate, GSK1360707
0941
Pd-Catalyzed Synthesis of Dibenzofurans by Phenol-Directed C-H Activation
0942
(4-Hydroxy-TEMPO)-Catalyzed Synthesis of 2-Aryl Quinazolines
0943
Copper-Catalyzed Synthesis of Pyrrolo[3,2-c]quinolin-4-nones
0944
Synthesis of 1-Aminoisoquinolines from 2-Alkynylbenzaldoximines
0945
Synthesis of Isoxazoles from the Reaction of Nitroalkanes with Oxetanes
0946
Nickel-Catalyzed Diastereoselective Synthesis of Oxazolidines
0947
Conversion of Anilines into 2-Aminobenzo-thiazoles via Herz Compounds
0948
Copper-Catalyzed Three-Component Synthesis of 2H-Indazoles
0949
Synthesis of 3-Haloquinolines via the Friedländer Reaction
0950
An Efficient Protocol for the Synthesis of Dibenzodithiapentalene
0951
Iodocyclization Route to Indolo- and Pyrroloquinolines

Synthesis of Materials and Unnatural Products

z953
All PDFs of this category
0953
One Step, Four Skeletons
0954
A Modular Approach to Oligoarenes: [2+2+2] Cycloadditions with a New Boramide
0955
N-Type Polymer from Suzuki Polycondensation
0956
A Mild Route to Substituted Fulvenes
0957
Large PAHs with Small HOMO-LUMO Gaps
0958
Click and Homocoupling for Extended π-Systems
0959
New Chain-Growth Living Polymerization Method
0960
Modular Synthesis of Conjugated Imidazole-Based Oligomers
0961
Rotaxanes under the Spotlight: A Metal-Free Synthesis
0962
Taming the Anion
0963
Polyacetylene by a Chain-Growth Approach
0964
[2+2+2] for Chain-Growth Polymerization

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z965
All PDFs of this category
0965
Aluminum-Catalyzed Cyclohexanone Ring Expansion with α-Diazoacetates
0966
Catalytic Asymmetric Synthesis of Unnatural Amino Acids
0967
Asymmetric Rhodium-Catalyzed Synthesis of Tertiary Propargyl Alcohols
0968
Enantioselective Ketone Hydrogenation Using a Novel Ruthenium Catalyst
0969
Functionalized Pyrrolidines via Enantioselective 1,3-Dipolar Cycloaddition
0970
Copper(I)-Catalyzed Asymmetric Conjugate Addition-Protonation of Nitroalkenes
0971
Brønsted Acid Catalyzed Synthesis of Spirooxindole Pyrans
0972
New Ligand for Inverse-Electron-Demand Hetero-Diels-Alder Reaction
0973
Diastereoselective Alkoxyallylation of Aldehydes
0974
Palladium-Catalyzed Synthesis of Substituted Pyrrolidines
0975
Diastereoselective Rhodium-Catalyzed Switchable Three-Component Couplings
0976
Cu/Box-Catalyzed Mukaiyama-Michael Additions towards Chiral Diazoacetoacetates
0977
Palladium-Catalyzed Elimination-Isomerization of Enol Triflates into 1,3-Dienes
0978
Chiral Tridentate Ligand for Rhodium-Catalyzed Cycloisomerization
0979
Z-Selective Ruthenium-Catalyzed Olefin Cross Metathesis
0980
Synthesis of δ-Lactones via Aldol, Cyclo-propanation, and Ring-Opening Cascade
0981
Asymmetric Conjugate Boration of α,β-Unsaturated Sulfones
0982
Catalytic Asymmetric Conjugate Addition of Pyrazolin-5-ones
0983
Rhodium-Catalyzed Asymmetric Conjugate Addition with N-Sulfinyl Ligands
0984
Lithium Binaphtholate-Catalyzed Asymmetric Alkynylation of Ketones
0985
New Sulfonamide-Olefin Ligand for Rh-Catalyzed 1,4-Addition
0986
Controlling E/Z Selectivity in the Formation of Alkenyl Imines
0987
Asymmetric Mo-Catalyzed Allylic Alkylation of Cyano Esters
0988
Synthesis of Tetrahydropyridines by an Aza-Diels-Alder Reaction
0989
Synthesis of 2-Keto-anti-1,3-Diols by Chemoselective Tandem Oxidation
0990
Pd-Catalyzed Indole Alkylation with γ,δ-Unsaturated β-Keto Phosphonates
0991
Asymmetric Cyclization of 4-Alkenoic Acids via Oxidative Allylic C-H Esterification
0992
Copper-Catalyzed Coupling of Peptidic Thiol Esters and α-Alkoxyalkylstannanes
0993
Nickel-Catalyzed Enantioselective α-Chlorination
0994
Copper-Catalyzed Asymmetric Hydrosilylation

Metal-Mediated Synthesis

z995
All PDFs of this category
0995
Catalytic Regioselective Boration of α,β-Unsaturated Compounds
0996
Ni-Catalyzed Opening of Styrenyl Epoxides with Boronic Acids
0997
Rh-Catalyzed Asymmetric Addition of Trifluoroborates to Sulfonylketimines
0998
Polystyrene-Stabilized PdO Nanoparticles-Catalyzed Cross-Coupling
0999
Cu-Catalyzed 1H-Perfluoroalkane Arylation by Aryl Iodide
1000
Access to Benzyl Boronates via Suzuki Coupling of Diborylmethane
1001
Sequential Asymmetric Conjugate Addition and Oxidative Dearomatization
1002
Hydroalumination and Carbocupration of Alkynylphosphine-Borane Complexes
1003
Pd-Catalyzed Synthesis of Pyridine-N-Oxide-Borane Complexes
1004
Enantioselective Addition of Diethylzinc to Aldehydes
1005
Synthesis of 1,5-Substituted Sulfonyl Triazoles
1006
Cr-Mediated Stereoselective Synthesis of α,β-Unsaturated Esters and Amides
1007
Two-Component Coupling to Form Benzocycloheptanones
1008
C-H Coupling of Grignard Reagents to Benzamides and Phenylpyridines
1009
Copper(I)-Catalyzed α-Selective Allylic Alkylation

Organo- and Biocatalysis

z1011
All PDFs of this category
1011
Controlling the Reaction Mechanism to Construct Dihydrocoumarins
1012
Asymmetric Synthesis of α-Sulfenyl Ketones Using Thiols
1013
Desymmetrization of meso-Diols via Covalent Substrate Binding Catalysis
1014
Asymmetric Intermolecular Stetter Reaction of Enals with Nitroalkenes
1015
Asymmetric Strecker Reaction of Di- and Trifluoromethyl Ketoimines
1016
New Developments in Putting Waste to Work
1017
High Pressure in Organocatalysis
1018
Enantioselective α-Alkylation of Aldehydes Using 1,3-Benzodithiolylium Tetrafluoroborate
1019
Organocatalytic Trifluoromethylations
1020
[3+2] Annulation of MBH Adducts Promoted by Bifunctional Phosphines
1021
Chiral NHC-Catalyzed Annulations of Ynals and Enals

Polymer-Supported Synthesis

z1023
All PDFs of this category
1023
Oxidation of Alcohols with PSB-TEMPO/NOx
1024
The Suzuki Coupling with Phosphine Dendrimer-Stabilized Nano Nickel
1025
Suzuki-Miyaura Coupling in Water Using an NHC-Pd Polymer
1026
Asymmetric Addition of Aldehydes to Nitroalkenes with an Immobilized Peptide
1027
Asymmetric α-Oxyamination with a Peptide Catalyst and Laccase
1028
A Silica-Supported Organocatalyst for the Preparation of Xanthenes
1029
A Magnetically Separable Catalyst for O-Arylation
1030
Hiyama Coupling in Water with Fe3O4-Supported Pd Nanoparticles
1031
The Mitsunobu Reaction with MPEG-Supported Ph3P and DEAD
1032
Synthesis of 5-Substituted 1H-Tetrazoles with CuFe2O4 Nanoparticles
1033
Hydrothiolation of Acetylenes Using an SBA-15-Supported Rh Complex
1034
Direct Conversion of Furfural to 1,5-Pentanediol Using Pt/Co2AlO4
1035
Pt Nanoparticle Catalyzed Chemoselective Reduction of Nitroarenes
1036
Synthesis of Nitriles from Primary Azides with Ru(OH)x/Al2O3

Addenda and Errata

1037
Synthesis of (-)-Viriditoxin