DOI: 10.1055/s-00000131

Synfacts

Issue 09 · Volume 2011 · September 2011 DOI: 10.1055/s-002-22222

Synform

A76
Zanda, Matteo: SYNFORM ISSUE 2011/09

Synthesis of Natural Products and Potential Drugs

z925
All PDFs of this category
0925
Zu, L.; Boal, B. W.; Garg, N. K.: Synthesis of (±)-Aspidophylline A
0926
Yu, L.-F.; Hu, H.-N.; Nan, F.-J.: Synthesis of Lathyranoic Acid A
0927
Su, J.; Tang, H.; McKittrick, B. A.: Synthesis of a γ-Secretase Inhibitor
0928
Gallenkamp, D.; Fürstner, A.: Synthesis of Lactimidomycin
0929
Qin, H.; Xu, Z.; Cui, Y.; Jia, Y.: Synthesis of (±)-Decursivine and (±)-Serotobenin
0930
Mascal, M.; Modes, K. V.; Durmus, A.: Synthesis of (±)-Decursivine
0931
Gesinski, M. R.; Rychnovsky, S. D.: Synthesis of Cyanolide A Aglycon
0932
Cosner, C. C.; Helquist, P.: Synthesis of (±)-Trichostatin A
0933
Hodgetts et al., K. J.: Synthesis of a CRF-1 Receptor Antagonist
0934
Han-ya, Y.; Tokuyama, H.; Fukuyama, T.: Synthesis of (-)-Conophylline
0935
Knight, J. D.; Sauer, S. J.; Coltart, D. M.: Synthesis of (+)-Mefloquine Hydrochloride

Synthesis of Heterocycles

z937
All PDFs of this category
0937
Rogress, D. C.; Larock, R. C.: Arynes in the Synthesis of N-Arylisatins
0938
Li, P.; Zhao, J.; Wu, C.; Larock, R. C.; Shi, F.: Synthesis of NH-Free 3-Substituted Indazoles
0939
McAusland, D.; Seo, S.; Pintori, D. G.; Finlayson, J.; Greaney, M. F.: The Benzyne Fischer Indole Reaction
0940
Teller, H.; Fürstner, A.: Enyne Cycloisomerization Route to an Anti-depressant Drug Candidate, GSK1360707
0941
Xiao, B.; Gong, T.-J.; Liu, Z.-J.; Liu, J.-H.; Luo, D.-F.; Xu, J.; Liu, L.: Pd-Catalyzed Synthesis of Dibenzofurans by Phenol-Directed C-H Activation
0942
Han, B.; Wang, C.; Han, R.-F.; Yu, W.; Duan, X.-Y.; Fang, R.; Yang, X.-L.: (4-Hydroxy-TEMPO)-Catalyzed Synthesis of 2-Aryl Quinazolines
0943
Zhou, F.; Liu, J.; Ding, K.; Liu, J.; Cai, Q.: Copper-Catalyzed Synthesis of Pyrrolo[3,2-c]quinolin-4-nones
0944
Zheng, D.; Chen, Z.; Liu, J.; Wu, J.: Synthesis of 1-Aminoisoquinolines from 2-Alkynylbenzaldoximines
0945
Burkhard, J. A.; Tchitchanov, B. H.; Carreira, E. M.: Synthesis of Isoxazoles from the Reaction of Nitroalkanes with Oxetanes
0946
Wu, X.; Li, L.; Zhang, J.: Nickel-Catalyzed Diastereoselective Synthesis of Oxazolidines
0947
Neo, A. G.; Carrillo, R. M.; Marcos, C. F.: Conversion of Anilines into 2-Aminobenzo-thiazoles via Herz Compounds
0948
Kumar, M. R.; Park, A.; Park, N.; Lee, S.: Copper-Catalyzed Three-Component Synthesis of 2H-Indazoles
0949
Ryabukhin, S. V.; Naumchik, V. S.; Plaskon, A. S.; Grygorenko, O. O.; Tolmachev, A. A.: Synthesis of 3-Haloquinolines via the Friedländer Reaction
0950
Jepsen, T. H.; Larsen, M.; Jørgensen, M.; Nielsen, M. B.: An Efficient Protocol for the Synthesis of Dibenzodithiapentalene
0951
Verma, A. K.; Shukla, S. P.; Singh, J.; Rustagi, V.: Iodocyclization Route to Indolo- and Pyrroloquinolines

Synthesis of Materials and Unnatural Products

z953
All PDFs of this category
0953
Chen, X.; Lu, P.; Wang, Y.: One Step, Four Skeletons
0954
Iannazzo, L.; Vollhardt, K. P. C.; Malacria, M.; Aubert, C.; Gandon, V.: A Modular Approach to Oligoarenes: [2+2+2] Cycloadditions with a New Boramide
0955
Lee, J.-K.; Gwinner, M. C.; Berger, R.; Newby, C.; Zentel, R.; Friend, R. H.; Sirringhaus, H.; Ober, C. K.: N-Type Polymer from Suzuki Polycondensation
0956
Chen, Y.; Liu, Y.: A Mild Route to Substituted Fulvenes
0957
Chen, T.-A.; Liu, R.-S.: Large PAHs with Small HOMO-LUMO Gaps
0958
Juríček, M.; Stout, K.; Kouwer, P. H. J.; Rowan, A. E.: Click and Homocoupling for Extended π-Systems
0959
Mikami, K.; Daikuhara, H.; Kasama, J.; Yokoyama, A.; Yokozawa, T.: New Chain-Growth Living Polymerization Method
0960
Siamak, A. R.; Sakalauskas, M.; Arndtsen, B. A.: Modular Synthesis of Conjugated Imidazole-Based Oligomers
0961
Hsueh, S.-Y.; Ko, J.-L.; Lai, C.-C.; Liu, Y.-H.; Peng, S.-M.; Chiu, S.-H.: Rotaxanes under the Spotlight: A Metal-Free Synthesis
0962
Hirao, A.; Tanaka, S.; Goseki, R.; Ishizone, T.: Taming the Anion
0963
Luo, K.; Kim, S. J.; Cartwright, A. N.; Rzayev, J.: Polyacetylene by a Chain-Growth Approach
0964
Sugiyama, Y.; Kato, R.; Sakurada, T.; Okamoto, S.: [2+2+2] for Chain-Growth Polymerization

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z965
All PDFs of this category
0965
Hashimoto, T.; Naganawa, Y.; Maruoka, K.: Aluminum-Catalyzed Cyclohexanone Ring Expansion with α-Diazoacetates
0966
Tosatti, P.; Campbell, A. J.; House, D.; Nelson, A.; Marsden, S. P.: Catalytic Asymmetric Synthesis of Unnatural Amino Acids
0967
Ohshima, T.; Kawabata, T.; Takeuchi, Y.; Kakinuma, T.; Iwasaki, T.; Yonezawa, T.; Murakami, H.; Nishiyama, H.; Mashiama, K.: Asymmetric Rhodium-Catalyzed Synthesis of Tertiary Propargyl Alcohols
0968
Matsumura, K.; Arai, N.; Hori, K.; Saito, T.; Sayo, N.; Ohkuma, T.: Enantioselective Ketone Hydrogenation Using a Novel Ruthenium Catalyst
0969
Wang, M.; Wang, Z.; Shi, Y.-H.; Shi, X.-X.; Fossey, J. S.; Deng, W.-P.: Functionalized Pyrrolidines via Enantioselective 1,3-Dipolar Cycloaddition
0970
Arai, T.; Awata, A.; Wasai, M.; Yokoyama, N.; Masu, H.: Copper(I)-Catalyzed Asymmetric Conjugate Addition-Protonation of Nitroalkenes
0971
Wang, J.; Crane, E. A.; Scheidt, K. A.: Brønsted Acid Catalyzed Synthesis of Spirooxindole Pyrans
0972
Barba, A.; Barroso, S.; Blay, G.; Cardona, L.; Melegari, M.; Pedro, J. R.: New Ligand for Inverse-Electron-Demand Hetero-Diels-Alder Reaction
0973
Mejuch, T.; Botoshansky, M.; Marek, I.: Diastereoselective Alkoxyallylation of Aldehydes
0974
Lowe, M. A.; Ostovar, M.; Ferrini, S.; Chen, C. C.; Lawrence, P. G.; Fontana, F.; Calabrese, A. A.; Aggarwal, V. K.: Palladium-Catalyzed Synthesis of Substituted Pyrrolidines
0975
Ji, J.; Zhang, X.; Zhu, Y.; Qian, Y.; Zhou, J.; Yang, L.; Hu, W.: Diastereoselective Rhodium-Catalyzed Switchable Three-Component Couplings
0976
Xu, X.; Hu, W.-H.; Doyle, M. P.: Cu/Box-Catalyzed Mukaiyama-Michael Additions towards Chiral Diazoacetoacetates
0977
Crouch, I. T.; Dreier, T.; Frantz, D. E.: Palladium-Catalyzed Elimination-Isomerization of Enol Triflates into 1,3-Dienes
0978
Nishimura, T.; Maeda, Y.; Hayashi, T.: Chiral Tridentate Ligand for Rhodium-Catalyzed Cycloisomerization
0979
Endo, K.; Grubbs, R. H.: Z-Selective Ruthenium-Catalyzed Olefin Cross Metathesis
0980
Peed, J.; Domínguez, I. Periñán; Davies, I. R.; Cheeseman, M.; Taylor, J. E.; Kociok-Köhn, G.; Bull, S. D.: Synthesis of δ-Lactones via Aldol, Cyclo-propanation, and Ring-Opening Cascade
0981
Moure, A. L.; Arrayás, R. Gómez; Carretero, J. C.: Asymmetric Conjugate Boration of α,β-Unsaturated Sulfones
0982
Wang, Z.; Yang, Z.; Chen, D.; Liu, X.; Lin, L.; Feng, X.: Catalytic Asymmetric Conjugate Addition of Pyrazolin-5-ones
0983
Feng, X.; Wang, Y.; Wei, B.; Yang, J.; Du, H.: Rhodium-Catalyzed Asymmetric Conjugate Addition with N-Sulfinyl Ligands
0984
Tanaka, K.; Kukita, K.; Ichibakase, T.; Kotani, S.; Nakajima, M.: Lithium Binaphtholate-Catalyzed Asymmetric Alkynylation of Ketones
0985
Jin, S.-S.; Wang, H.; Xu, M.-H.: New Sulfonamide-Olefin Ligand for Rh-Catalyzed 1,4-Addition
0986
Fukumoto, Y.; Hagihara, M.; Kinashi, F.; Chatani, N.: Controlling E/Z Selectivity in the Formation of Alkenyl Imines
0987
Trost, B. M.; Miller, J. R.; Hoffman, Jr., C. M.: Asymmetric Mo-Catalyzed Allylic Alkylation of Cyano Esters
0988
Vicario, J.; Aparicio, D.; Palacios, F.: Synthesis of Tetrahydropyridines by an Aza-Diels-Alder Reaction
0989
Hussain, M. M.; Toribio, J. H.; Carroll, P. J.; Walsh, P. J.: Synthesis of 2-Keto-anti-1,3-Diols by Chemoselective Tandem Oxidation
0990
Kang, Y. K.; Kwon, B. K.; Mang, J. Y.; Kim, D. Y.: Pd-Catalyzed Indole Alkylation with γ,δ-Unsaturated β-Keto Phosphonates
0991
Takenaka, K.; Akita, M.; Tanigaki, Y.; Takizawa, S.; Sasai, H.: Asymmetric Cyclization of 4-Alkenoic Acids via Oxidative Allylic C-H Esterification
0992
Li, H.; He, A.; Falck, J. R.; Liebeskind, L. S.: Copper-Catalyzed Coupling of Peptidic Thiol Esters and α-Alkoxyalkylstannanes
0993
Hamashima, Y.; Nagi, T.; Shimizu, R.; Tsuchimoto, T.; Sodeoka, M.: Nickel-Catalyzed Enantioselective α-Chlorination
0994
Zhang, X.-C.; Wu, F.-F.; Li, S.; Zhou, J.-N.; Wu, J.; Li, N.; Fang, W.; Lam, K. H.; Chan, A. S. C.: Copper-Catalyzed Asymmetric Hydrosilylation

Metal-Mediated Synthesis

z995
All PDFs of this category
0995
Gao, M.; Thorpe, S. B.; Kleeberg, C.; Slebodnick, C.; Marder, T. B.; Santos, W. L.: Catalytic Regioselective Boration of α,β-Unsaturated Compounds
0996
Nielsen, D. K.; Doyle, A. G.: Ni-Catalyzed Opening of Styrenyl Epoxides with Boronic Acids
0997
Shintani, R.; Takeda, M.; Soh, Y.-T.; Ito, T.; Hayashi, T.: Rh-Catalyzed Asymmetric Addition of Trifluoroborates to Sulfonylketimines
0998
Ohtaka, A.; Teratani, T.; Fujii, R.; Ikeshita, K.; Kawashima, T.; Tatsumi, K.; Shimomura, O.; Nomura, R.: Polystyrene-Stabilized PdO Nanoparticles-Catalyzed Cross-Coupling
0999
Popov, I.; Lindeman, S.; Daugulis, O.: Cu-Catalyzed 1H-Perfluoroalkane Arylation by Aryl Iodide
1000
Endo, K.; Ohkubo, T.; Shibata, T.: Access to Benzyl Boronates via Suzuki Coupling of Diborylmethane
1001
Rudolph, A.; Bos, P. H.; Meetsma, A.; Minnaard, A. J.; Feringa, B. L.: Sequential Asymmetric Conjugate Addition and Oxidative Dearomatization
1002
Ortial, S.; Montchamp, J.-L.: Hydroalumination and Carbocupration of Alkynylphosphine-Borane Complexes
1003
Ishida, N.; Ikemoto, W.; Narumi, M.; Murakami, M.: Pd-Catalyzed Synthesis of Pyridine-N-Oxide-Borane Complexes
1004
Hirose, T.; Sugawara, K.; Kodama, K.: Enantioselective Addition of Diethylzinc to Aldehydes
1005
Meza-Aviña, M. E.; Pater, M. K.; Lee, C. B.; Dietz, T. J.; Croatt, M. P.: Synthesis of 1,5-Substituted Sulfonyl Triazoles
1006
Rodríguez-Solla, H.; Concellón, C.; Blanco, E. G.; Sarmiento, J. I.; Díaz, P.; Soengas, R. G.: Cr-Mediated Stereoselective Synthesis of α,β-Unsaturated Esters and Amides
1007
Patti, R. Kumar; Waynant, K. V.; Herndon, J. W.: Two-Component Coupling to Form Benzocycloheptanones
1008
Chen, Q.; Ilies, L.; Yoshikai, N.; Nakamura, E.: C-H Coupling of Grignard Reagents to Benzamides and Phenylpyridines
1009
Lauer, A. M.; Mahmud, F.; Wu, J.: Copper(I)-Catalyzed α-Selective Allylic Alkylation

Organo- and Biocatalysis

z1011
All PDFs of this category
1011
Enders, D.; Yang, X.; Wang, C.; Raabe, G.; Runsik, J.: Controlling the Reaction Mechanism to Construct Dihydrocoumarins
1012
Hatcher, J. M.; Kohler, M. C.; Coltart, D. M.: Asymmetric Synthesis of α-Sulfenyl Ketones Using Thiols
1013
Sun, X.; Worthy, A. D.; Tan, K. L.: Desymmetrization of meso-Diols via Covalent Substrate Binding Catalysis
1014
DiRocco, D. A.; Rovis, T.: Asymmetric Intermolecular Stetter Reaction of Enals with Nitroalkenes
1015
Liu, Y.-L.; Shi, T.-D.; Zhou, F.; Zhao, X.-L.; Wang, X.; Zhou, J.: Asymmetric Strecker Reaction of Di- and Trifluoromethyl Ketoimines
1016
Lu, J.; Toy, P. H.: New Developments in Putting Waste to Work
1017
Kwiatkowski, P.; Dudziński, K.; Łyżwa, D.: High Pressure in Organocatalysis
1018
Gualandi, A.; Emer, E.; Capdevila, M. G.; Cozzi, P. G.: Enantioselective α-Alkylation of Aldehydes Using 1,3-Benzodithiolylium Tetrafluoroborate
1019
Furukawa, T.; Nishimine, T.; Tokunaga, E.; Hasegawa, K.; Shiro, M.; Shibata, N.: Organocatalytic Trifluoromethylations
1020
Zhong, F.; Han, X.; Wang, Y.; Lu, Y.: [3+2] Annulation of MBH Adducts Promoted by Bifunctional Phosphines
1021
Zhu, Z.-Q.; Zheng, X.-L.; Jiang, N.-F.; Wan, X.; Xiao, J.-C.: Chiral NHC-Catalyzed Annulations of Ynals and Enals

Polymer-Supported Synthesis

z1023
All PDFs of this category
1023
Di, L.; Hua, Z.: Oxidation of Alcohols with PSB-TEMPO/NOx
1024
Wu, L.; Ling, J.; Wu, Z.-Q.: The Suzuki Coupling with Phosphine Dendrimer-Stabilized Nano Nickel
1025
Karimi, B.; Akhavan, P. F.: Suzuki-Miyaura Coupling in Water Using an NHC-Pd Polymer
1026
Arakawa, Y.; Wiesner, M.; Wennemers, H.: Asymmetric Addition of Aldehydes to Nitroalkenes with an Immobilized Peptide
1027
Akagawa, K.; Kudo, K.: Asymmetric α-Oxyamination with a Peptide Catalyst and Laccase
1028
Nandi, M.; Mondal, J.; Sarkar, K.; Yamauchi, Y.; Bhaumik, A.: A Silica-Supported Organocatalyst for the Preparation of Xanthenes
1029
Arundhathi, R.; Damodara, D.; Likhar, P. R.; Kantam, M. L.; Saravanan, P.; Magdaleno, T.; Kwon, S. H.: A Magnetically Separable Catalyst for O-Arylation
1030
Sreedhar, B.; Kumar, A. S.; Yada, D.: Hiyama Coupling in Water with Fe3O4-Supported Pd Nanoparticles
1031
Figlus, M.; Wellaway, N.; Cooper, W. J.; Sollis, S. L.; Hartley, R. C.: The Mitsunobu Reaction with MPEG-Supported Ph3P and DEAD
1032
Sreedhar, B.; Kumar, A. S.; Yada, D.: Synthesis of 5-Substituted 1H-Tetrazoles with CuFe2O4 Nanoparticles
1033
Yang, Y.; Rioux, R. M.: Hydrothiolation of Acetylenes Using an SBA-15-Supported Rh Complex
1034
Xu, W.; Wang, H.; Liu, X.; Ren, J.; Wang, Y.; Lu, G.: Direct Conversion of Furfural to 1,5-Pentanediol Using Pt/Co2AlO4
1035
Pandarus, V.; Ciriminna, R.; Béland, F.; Pagliaro, M.: Pt Nanoparticle Catalyzed Chemoselective Reduction of Nitroarenes
1036
He, J.; Yamaguchi, K.; Mizuno, N.: Synthesis of Nitriles from Primary Azides with Ru(OH)x/Al2O3

Addenda and Errata

1037
Synthesis of (-)-Viriditoxin