DOI: 10.1055/s-00000084

Synthesis

Issue 06 · Volume 57 · March 2025 DOI: 10.1055/s-015-61218

table of contents

V
Linked PDF of Table of Contents

review

1081
Kim, Eunbi; Baik, Eunji; Shin, Jihye; Hwang, Junha; Dongbang, Sun: Aziridines as Versatile C(sp3) Precursors in Transition-Metal-Catalyzed Cross-Coupling Strategies
https://www.thieme-connect.de/media/synthesis/202506/i_r0325_ga_10-1055_a-2427-9162.gif

short review

1102
Gerlach, Tabea; Turner, Nicholas J.: Biocatalytic Dearomatisation Reactions
https://www.thieme-connect.de/media/synthesis/202506/i_r0274_ga_10-1055_a-2385-4073.gif
1117
Abd El Sater, Mariam; Popek, Lucas; Blanchard, Nicolas; Bizet, Vincent: Recent Advances in the Chemistry and Application of SF5-Compounds
https://www.thieme-connect.de/media/synthesis/202506/i_r0305_ga_10-1055_a-2383-6620.gif

Special Topic Dedicated to Prof. Erick Carreira

1138
Miguélez, Rubén; Arto, Omar; Rodríguez-Arias, Carlos; Barrio, Pablo: Gold(I)-Catalyzed Intramolecular C(sp3)–H Bond Functionalization
https://www.thieme-connect.de/media/synthesis/202506/i_r0320_ga_10-1055_a-2389-7434.gif

Bioisosteres

1153
Nagasawa, Shota; Iwabuchi, Yoshiharu: Recent Progress in Accessing Multi-functionalized Caged Hydrocarbons: En Route to Highly Functionalized Saturated (Bio)isosteres of Benzene Rings
https://www.thieme-connect.de/media/synthesis/202506/i_r0248_ga_10-1055_a-2360-8218.gif
1171
Fang, Zhuohan; Xu, Qian; Lu, Xuehe; Wan, Nianfeng; Yang, Wu-Lin: The Application of Bicyclo[1.1.1]pentane as a Bioisostere of the Phenyl Ring in Pharmaceutical Chemistry
https://www.thieme-connect.de/media/synthesis/202506/i_r0266_ga_10-1055_s-0043-1775395.jpg

feature

1180
Qian, Huijun; Liu, Wenhao; Su, Junqi; Shi, Zhengjun; Hu, Meng-Yang; Lv, Leiyang; Li, Zhiping: Pd/IHept-Catalyzed Regioselective Annulation of 2-Fluoroallyl Carbonates with Enaminones: Synthesis of Fully Substituted Pyrroles
https://www.thieme-connect.de/media/synthesis/202506/i_b0335_ga_10-1055_a-2436-0471.gif
Supporting Information

paper

1189
Gao, Jun-Nan; Tan, Wen-Xin; Yang, Shuang; Wang, Ning-Yi; Han, Jiebin; Wang, Da-Hua; Zhang, Yu-Chen; Shi, Feng: Lewis Acid Catalyzed Regioselective Substitution of 2-Indolylmethanols with Pyrroles
https://www.thieme-connect.de/media/synthesis/202506/i_f0437_ga_10-1055_a-2503-3181.gif
Supporting Information CIF File
1199
Manna, Priyadarshi; Chatterjee, Arunima; Kundu, Mrinalkanti; Rao, G. Prabhakar; Mukherjee, Rusmita; Podder, Swarnali; Datta, Bandita; Adhikari, Susanta: 3-Amino-1-methyl-1H-pyridin-2-one as Inbuilt Directing Group for Additive-Free Late-Stage ortho-Amination under Copper Catalysis towards Biologically Relevant Molecules
https://www.thieme-connect.de/media/synthesis/202506/i_m0441_ga_10-1055_s-0040-1720160.gif
1213
Ďurina, Lukáš; Kerti, Lukáš; Litecká, Miroslava; Moncol, Ján; Žídeková, Ivana; Fischer, Róbert: Zinc-Mediated Diastereoselective Acyloxyallylation of Isoxazolidine-4,5-diols
https://www.thieme-connect.de/media/synthesis/202506/i_t0401_ga_10-1055_a-2503-2981.gif
Supporting Information CIF File
1223
Niu, Yu-Dan; Lv, Pei; Hu, Hao-Lan; Shi, Jianghuan; Chen, Peng; Jiang, Yi-Jun: Scandium(III)-Catalyzed N-Alkylation of Carbazoles with Alcohols
https://www.thieme-connect.de/media/synthesis/202506/i_g0415_ga_10-1055_a-2502-7704.gif
Supporting Information

Bioisosteres

1230
Huang, Long-Ling; Li, Jia-Yi; Sun, Qigang; Zhao, Gui-Yang; Wang, Honggen; Li, Qingjiang: Hypervalent Iodine Mediated Ring-Opening 1,3-Difluorination of Benzylidenecyclopropanes
https://www.thieme-connect.de/media/synthesis/202506/i_m0261_ga_10-1055_a-2373-0304.gif
Supporting Information