DOI: 10.1055/s-00000084

Synthesis

Issue 23 · Volume 44 · December 2012 DOI: 10.1055/s-002-24066

synform

A122
Zanda, Matteo: SYNFORM ISSUE 2012/12

review

3551
Trstenjak, Uroš; Ilaš, Janez; Kikelj, Danijel: Advances in the Synthesis of Morpholin-3-ones and Morpholin-2-ones
https://www.thieme-connect.de/media/synthesis/201223/e0609_ga.gif

feature article

3579
Ghosh, Arun K.; Kass, Jorden; Nicponski, Daniel R.; Keyes, Chad: Diastereoselective Synthesis of Substituted Tetrahydropyrans by Copper(II)–Bisphosphine-Catalyzed Olefin Migration and Prins Cyclization
https://www.thieme-connect.de/media/synthesis/201223/z0569_ga.gif

practical synthetic procedures

3590
Blay, Gonzalo; Fernández, Isabel; Pedro, José R.; Vila, Carlos: Enantioselective Synthesis of Substituted Indoles Through Zirconium(IV)-Catalyzed Friedel–Crafts Alkylation
https://www.thieme-connect.de/media/synthesis/201223/z0488_ga.gif

short paper

3595
Edelbach, Brian L.; Pharoah, Blaze M.; Bellows, Sarina M.; Thayer, Peter R.; Fennie, Charles N.; Cowley, Ryan E.; Holland, Patrick L.: An Expedient Synthesis of 2,4,6-Tris(trifluoromethyl)aniline
https://www.thieme-connect.de/media/synthesis/201223/m0747_ga.gif

paper

3598
Ni, Feng; Li, Jianqi: A New Route to Roflumilast via Copper-Catalyzed Hydroxylation
https://www.thieme-connect.de/media/synthesis/201223/h0689_ga.gif
Supporting Information
3603
Koguchi, Shinichi; Izawa, Kazuki: A New Method for the Synthesis of 1,5-Disubstituted 1,2,3-Triazoles via Triazolium Salt Intermediates
https://www.thieme-connect.de/media/synthesis/201223/f0633_ga.gif
3609
Bae, Hoon; Jeon, Hongjun; Baek, Dong Jae; Lee, Dongjoo; Kim, Sanghee: Stereochemically Reliable Syntheses of Pachastrissamine and Its 2-epi-Congener via Oxazolidinone Precursors from an Established Starting Material N-tert-Butoxycarbonyl-Protected Phytosphingosine
https://www.thieme-connect.de/media/synthesis/201223/f0644_ga.gif
Supporting Information
3613
Ahn, Sang-Hyun; Kim, Young Keun; Hyun, Jina; Lee, Kee-Jung: A Synthetic Pathway to the 1,4-Dihydro-2H-3-benzoxocine System from Morita–Baylis–Hillman Cinnamyl Alcohols with 2,5-Dimethoxy-2,5-dihydrofuran via the Heck Reaction
https://www.thieme-connect.de/media/synthesis/201223/f0656_ga.gif
3623
Kimura, Tsutomu; Kobayashi, Gen; Ishigaki, Masashi; Inumaru, Mio; Sakurada, Jo; Satoh, Tsuyoshi: Coupling Reaction of Magnesium Alkylidene Carbenoids with α-Sulfonyl­allyllithiums: An Efficient Route to Multi-Substituted Vinylallenes
https://www.thieme-connect.de/media/synthesis/201223/f0694_ga.gif
Supporting Information
3633
Jiang, Hui; Na, Risong; Zhang, Lei; Liu, Honglei; Li, Zhen; Wang, Bo; Guo, Hongchao: Samarium Diiodide Mediated Highly Diastereoselective Conjugate Reduction of the α,β-Unsaturated Ester Moiety in Heterocyclic Compounds
https://www.thieme-connect.de/media/synthesis/201223/h0661_ga.gif
Supporting Information
3639
McDonald, Frank E.; Pereira, Claney L.: Stereo- and Regioselective Synthesis of 2-Amino-3,5-diols via Stereospecific Crotyl Transfer and Regioselective Aminohydroxylation
https://www.thieme-connect.de/media/synthesis/201223/m0648_ga.gif
3649
Mahdavi, Mohammad; Asadi, Mehdi; Saeedi, Mina; Ebrahimi, Mostafa; Rasouli, Mohammad A.; Ranjbar, Parviz R.; Foroumadi, Alireza; Shafiee, Abbas: One-Pot, Four-Component Synthesis of Novel Imidazo[2,1-b]thiazol-5-amine Derivatives
https://www.thieme-connect.de/media/synthesis/201223/n0418_ga.gif
3655
Kálai, Tamás; Bognár, Balázs; Zsolnai, Dániel; Berente, Zoltán; Hideg, Kálmán: Synthesis of Nitroxide-Annulated Carbocycles and Heterocycles
https://www.thieme-connect.de/media/synthesis/201223/n0671_ga.gif
Supporting Information
3661
Gratzer, Katharina; Waser, Mario: Investigations Concerning the Syntheses of TADDOL-Derived Secondary Amines and Their Use To Access Novel Chiral Organocatalysts
https://www.thieme-connect.de/media/synthesis/201223/t0707_ga.jpg
Supporting Inform.ation
3671
Ahmad, Anees; Silva, Luiz F.: Synthesis of Chromanes and 4H-Chromenes: Exploring the Oxidation of 2H-Chromenes and Dihydro-1-benzoxepines by Hypervalent Iodine(III)
https://www.thieme-connect.de/media/synthesis/201223/m0654_ga.gif
Supporting Information
3678
Goud, D. Raghavender; Pathak, Uma: A Mild and Efficient Synthesis of 2-Oxazolines via Transamidation–Cyclodehydrosulfurisation­ of Thioamides with 2-Aminoethanol
https://www.thieme-connect.de/media/synthesis/201223/z0598_ga.gif
Supporting Information
3683
Skonieczny, Kamil; Charalambidis, Georgios; Tasior, Mariusz; Krzeszewski, Maciej; Kalkan-Burat, Ayfer; Coutsolelos, Athanassios G.; Gryko, Daniel T.: General and Efficient Protocol for Formylation of Aromatic and Heterocyclic Phenols
https://www.thieme-connect.de/media/synthesis/201223/z0640_ga.gif
Supporting Information
3688
Scarpi, Dina; Avataneo, Ottavia; Prandi, Cristina; Venturello, Paolo; Occhiato, Ernesto G.: Synthesis of Both Enantiomers of the Streptomyces Alkaloid 4-epi-SS20846A
https://www.thieme-connect.de/media/synthesis/201223/z0642_ga.gif
Supporting Information
3693
Cheng, Xue-Ming; Chen, Min; Huang, Zhi-Tang; Zheng, Qi-Yu: Stereocontrolled Photodimerization of (E)-3-Benzylidene-4-chromanones in the Crystalline State: The Effect of a Halogen Group on the Chromanone Moiety
https://www.thieme-connect.de/media/synthesis/201223/h0683_ga.gif
Supporting Information