DOI: 10.1055/s-00000083

Synlett

Issue 20 · Volume 28 · December 2017 DOI: 10.1055/s-007-35789

editorial

I
Editorial

account

2685
Quiclet-Sire, Béatrice; Zard, Samir Z.: Convergent Routes to Pyrroles Exploiting the Unusual Radical Chemistry of Xanthates – An Overview
https://www.thieme-connect.de/media/synlett/201720/i_r0364_ga_10-1055_s-0036-1590809.gif
2697
Davies, Stephen G.; Fletcher, Ai M.; Roberts, Paul M.; Thomson, James E.: Asymmetric Synthesis of Pyrrolizidines, Indolizidines and Quinolizidines via a Double Reductive Cyclisation Protocol
https://www.thieme-connect.de/media/synlett/201720/i_r0464_ga_10-1055_s-0036-1590975.gif
2707
Shaaban, Saad; Maulide, Nuno: Metal-Free Redox Transformations for C–C and C–N Bond Construction
https://www.thieme-connect.de/media/synlett/201720/i_r0098_ga_10-1055_s-0036-1588776.gif
2714
Liu, Wenbo; Li, Chao-Jun: Recent Synthetic Applications of Catalyst-Free Photochemistry
https://www.thieme-connect.de/media/synlett/201720/i_r0490_ga_10-1055_s-0036-1590900.gif

letter

2755
Thullen, Scott M.; Rubush, David M.; Rovis, Tomislav: A Photochemical Two-Step Formal [5+2] Cycloaddition: A Condensation–Ring-Expansion Approach to Substituted Azepanes
https://www.thieme-connect.de/media/synlett/201720/i_b0169_ga_10-1055_s-0036-1589049.gif
Supporting Information
2759
Vásquez-Céspedes, Suhelen; Holtkamp, Michael; Karst, Uwe; Glorius, Frank: Reusable and Magnetic Palladium and Copper Oxide Catalysts in Direct ortho and meta Arylation of Anilide Derivatives
https://www.thieme-connect.de/media/synlett/201720/i_r0147_ga_10-1055_s-0036-1589007.gif
Supporting Information
2765
Aeyad, Tahani; Williams, Jason D.; Meijer, Anthony J. H. M.; Coldham, Iain: Lithiation–Substitution of N-Boc-2-phenylazepane
https://www.thieme-connect.de/media/synlett/201720/i_r0412_ga_10-1055_s-0036-1590857.gif
Supporting Information
2769
Piras, Monica; Andriu, Alexandra; Testa, Andrea; Wienecke, Paul; Fleming, Ian N.; Zanda, Matteo: Design and Synthesis of an RGD Peptidomimetic-Paclitaxel Conjugate Targeting αvβ3 Integrin for Tumour-Directed Drug Delivery
https://www.thieme-connect.de/media/synlett/201720/i_r0479_ga_10-1055_s-0036-1590898.gif
Supporting Information
2777
Chen, Jun; Lu, Lingxiao; Wulff, Jeremy E.: Radical Stabilization Algorithm as a Predictive Tool for Novel and Reported Noncanonical Thiele’s Acid Analogues
https://www.thieme-connect.de/media/synlett/201720/i_r0579_ga_10-1055_s-0036-1588583.gif
Supporting Information
2783
Schleper, A. Lennart; Voll, Constantin-Christian A.; Engelhart, Jens U.; Swager, Timothy M.: Iptycene-Containing Azaacenes with Tunable Luminescence
https://www.thieme-connect.de/media/synlett/201720/i_r0234_ga_10-1055_s-0036-1589503.jpg
Supporting Information
2790
Bagdžiūnas, Gintautas; Stončius, Sigitas; Butkus, Eugenijus: Synthesis of Star-Shaped Aromatic Derivatives with Chirality Predetermined by Bicyclo[3.3.1]nonane Framework
https://www.thieme-connect.de/media/synlett/201720/i_r0374_ga_10-1055_s-0036-1590833.gif
Supporting Information
2795
Afsar, Ashfaq; Cowell, Joseph; Distler, Petr; Harwood, Laurence M.; John, Jan; Westwood, James: Synthesis of Novel BTPhen-Functionalized Silica-Coated Magnetic Nanoparticles for Separating Trivalent Actinides and Lanthanides
https://www.thieme-connect.de/media/synlett/201720/i_r0433_ga_10-1055_s-0036-1590865.gif
Supporting Information
2800
Chernichenko, Nataliya M.; Shevchuk, Vadim N.; Averin, Alexei D.; Maloshitskaya, Olga A.; Beletskaya, Irina P.: Synthesis of Dansyl-Substituted Cryptands Containing Triaza­cycloalkane Moieties and their Evaluation as Fluorescent Chemosensors
https://www.thieme-connect.de/media/synlett/201720/i_r0525_ga_10-1055_s-0036-1590883.gif
Supporting Information
2807
Chui, Tin-Ki; Chow, Hak-Fun: New Triazole-Containing Branched Bis(dipeptidomimetic) – Switching from Self-Dimerization to Anion-Binding Properties
https://www.thieme-connect.de/media/synlett/201720/i_r0531_ga_10-1055_s-0036-1590884.gif
Supporting Information
2812
Ichioka, Fumiki; Itai, Yuhei; Nishii, Yuji; Miura, Masahiro: Palladium-Catalyzed Direct C2-Arylation of Benzo[b]thiophenes with Electron-Rich Aryl Halides: Facile Access to Thienoacene Derivatives
https://www.thieme-connect.de/media/synlett/201720/i_r0128_ga_10-1055_s-0036-1588994.gif
Supporting Information
2817
Ketels, Marthe; Ziegler, Dorothée S.; Knochel, Paul: Selective Zincation of 1,2-Dicyanobenzene and Related Benzonitriles in Continuous Flow Using In Situ Trapping Metalations
https://www.thieme-connect.de/media/synlett/201720/i_r0246_ga_10-1055_s-0036-1588837.gif
Supporting Information
2823
Hamel, Jean-Denys; Beaudoin, Meggan; Cloutier, Mélissa; Paquin, Jean-François: Hydrogen-Bond-Promoted Friedel–Crafts Reaction of Secondary Propargylic Fluorides: Preparation of 1-Alkyl-1-aryl-2-alkynes
https://www.thieme-connect.de/media/synlett/201720/i_r0278_ga_10-1055_s-0036-1589057.gif
Supporting Information
2829
Gao, Ang; Liu, Xiu-Yan; Ding, Chang-Hua; Hou, Xue-Long: Diastereoselective Palladium-Catalyzed Conjugate Addition of Arylboronic Acids to α-Substituted Cyclic Enones
https://www.thieme-connect.de/media/synlett/201720/i_r0385_ga_10-1055_s-0036-1590742.gif
Supporting Information
2833
Benoit, Emeline; Dansereau, Julien; Gagnon, Alexandre: Palladium-Catalyzed Carbonylative Cross-Coupling Reaction between Aryl(Heteroaryl) Iodides and Tricyclopropylbismuth: Expedient Access to Aryl Cyclopropylketones
https://www.thieme-connect.de/media/synlett/201720/i_r0394_ga_10-1055_s-0036-1590832.gif
Supporting Information
2839
Xu, Lanting; Tan, Lushi; Ma, Dawei: Rhodium-Catalyzed Regioselective C7-Functionalization of Indole Derivatives with Acrylates by Using an N-Imino Directing Group
https://www.thieme-connect.de/media/synlett/201720/i_r0441_ga_10-1055_s-0036-1588530.gif
Supporting Information
2845
Corbett, Michael T.; Caille, Seb: A Bench-Stable Vilsmeier Reagent for in situ Alcohol Activation: Synthetic Application in the Synthesis of 2-Amino-2-Thiazolines
https://www.thieme-connect.de/media/synlett/201720/i_r0476_ga_10-1055_s-0036-1589086.gif
Supporting Information
2851
Isbrandt, Eric S.; Vandavasi, Jaya Kishore; Zhang, Wanying; Jamshidi, Mohammad P.; Newman, Stephen G.: Catalytic Deuteration of Aldehydes with D2O
https://www.thieme-connect.de/media/synlett/201720/i_r0495_ga_10-1055_s-0036-1588540.gif
Supporting Information
2855
Labes, Ricardo; González-Calderón, Davir; Battilocchio, Claudio; Mateos, Carlos; Cumming, Graham R.; de Frutos, Oscar; Rincón, Juan A.; Ley, Steven V.: Rapid Continuous Ruthenium-Catalysed Transfer Hydrogenation of Aromatic Nitriles to Primary Amines
https://www.thieme-connect.de/media/synlett/201720/i_r0508_ga_10-1055_s-0036-1589096.gif
Supporting Information
2859
Irwin, Lauren C.; Kerr, Michael A.: One-Pot Michael Addition/Radical Cyclization Reaction of N-Acryloyl Indoles
https://www.thieme-connect.de/media/synlett/201720/i_r0529_ga_10-1055_s-0036-1589105.gif
Supporting Information
2865
Ramadhar, Timothy R.; Kawakami, Jun-ichi; Batey, Robert A.: Sequential O-Arylation/Lanthanide(III)-Catalyzed [3,3]-Sigmatropic Rearrangement of Bromo-Substituted Allylic Alcohols
https://www.thieme-connect.de/media/synlett/201720/i_r0540_ga_10-1055_s-0036-1590890.gif
Supporting Information
2871
Eljo, Jasmin; Carle, Myriam S.; Murphy, Graham K.: Hypervalent Iodine-Based Activation of Triphenylphosphine for the Functionalization of Alcohols
https://www.thieme-connect.de/media/synlett/201720/i_r0272_ga_10-1055_s-0036-1589069.gif
Supporting Information
2876
Zhi, Ying; Zhao, Kun; von Essen, Carolina; Rissanen, Kari; Enders, Dieter: Thiourea-Catalyzed Domino Michael–Mannich [3+2] Cycloadditions: A Strategy for the Asymmetric Synthesis of 3,3′-Pyrrolidinyl-dispirooxindoles
https://www.thieme-connect.de/media/synlett/201720/i_r0387_ga_10-1055_s-0036-1589070.gif
Supporting Information
2881
Papatzimas, James W.; Gorobets, Evgueni; Brownsey, Duncan K.; Maity, Ranjan; Bahlis, Nizar J.; Derksen, Darren J.: A General Strategy for the Preparation of Thalidomide-Conjugate Linkers
https://www.thieme-connect.de/media/synlett/201720/i_r0401_ga_10-1055_s-0036-1588539.gif
Supporting Information
2886
Fahandej-Sadi, Anis; Lundgren, Rylan J.: Copper-Mediated Synthesis of Monofluoro Aryl Acetates via Decarboxylative Cross-Coupling
https://www.thieme-connect.de/media/synlett/201720/i_r0405_ga_10-1055_s-0036-1588516.gif
Supporting Information
2891
Barraza, Scott J.; Denmark, Scott E.: Unexpected Rearrangement of 2-Bromoaniline under Biphasic Alkylation Conditions
https://www.thieme-connect.de/media/synlett/201720/i_r0502_ga_10-1055_s-0036-1590882.gif
Supporting Information
2896
Lapinskaite, Ringaile; Ghavre, Mukund; Rintelmann, Chelsea L.; Bedard, Korey; Dela Paz, Helen E.; Hudlicky, Tomas: Chemoenzymatic Formal Total Synthesis of Pancratistatin from Narciclasine-Type Compounds via Myers Transposition: Model Study for a Short Conversion of Narciclasine to Pancratistatin
https://www.thieme-connect.de/media/synlett/201720/i_r0439_ga_10-1055_s-0036-1588515.gif
Supporting Information
2901
Emberson, Kassandra; Tran, Ngan; Metallinos, Costa: Diastereoselective Lithiation of N-Benzyl Pyrroloimidazolones Derived from l-Proline Hydantoin
https://www.thieme-connect.de/media/synlett/201720/i_r0443_ga_10-1055_s-0036-1591206.gif
Supporting Information
2906
Ma, Zhi-Xiong; Fang, Li-Chao; Haugen, Bryan J.; Bruckbauer, Daniel; Feltenberger, John B.; Hsung, Richard P.: Facile Synthesis of 3-Amido-Dienynes via a Tandem α-Propargylation–Isomerization of Chiral Allenamides and their Applications in Diels–Alder Cycloadditions
https://www.thieme-connect.de/media/synlett/201720/i_r0444_ga_10-1055_s-0036-1590899.gif
Supporting Information
2913
Yamamoto, Yasutomo; Yamaguchi, Tatsuya; Kaneshige, Atsunori; Hashimoto, Aiko; Kaibe, Sachiho; Miyawaki, Akari; Yamada, Ken-ichi; Tomioka, Kiyoshi: Consecutive Aminolithiation–Carbolithiation of a Linear Aminoalkene Bearing Terminal Vinyl Sulfide Moiety to Give Hydro­indolizine
https://www.thieme-connect.de/media/synlett/201720/i_r0445_ga_10-1055_s-0036-1588522.gif
Supporting Information
2918
Jia, Zhi-Jun; Merten, Christian; Knauer, Lena; Murarka, Sandip; Strohmann, Carsten; Waldmann, Herbert: Biology-Oriented Synthesis of Decahydro-4,8-epoxyazulene Scaffolds
https://www.thieme-connect.de/media/synlett/201720/i_r0463_ga_10-1055_s-0036-1588558.gif
Supporting Information
2923
Onge, Brent St.; Green, James R.: Nicholas Reactions of Alkynyl- and Alkenyltrifluoroborates
https://www.thieme-connect.de/media/synlett/201720/i_r0465_ga_10-1055_s-0036-1588528.gif
Supporting Information
2928
Cooze, Christopher; Manchoju, Amarender; Pansare, Sunil V.: Synthesis of (–)-Muricatacin and (–)-(R,R)-L-Factor Involving an Organocatalytic Direct Vinylogous Aldol Reaction
https://www.thieme-connect.de/media/synlett/201720/i_r0466_ga_10-1055_s-0036-1590858.gif
Supporting Information
2933
Wang, Tao; Oswood, Christian J.; Hoye, Thomas R.: Trapping of Hexadehydro-Diels–Alder Benzynes with Exocyclic, Conjugated Enals as a Route to Fused Spirocyclic Benzopyran Motifs
https://www.thieme-connect.de/media/synlett/201720/i_r0467_ga_10-1055_s-0036-1589091.gif
Supporting Information
2936
Nambo, Masakazu; Yim, Jacky C.-H.; Fowler, Kevin G.; Crudden, Cathleen M.: Synthesis of Tetraarylmethanes by the Triflic Acid-Promoted Formal Cross-Dehydrogenative Coupling of Triarylmethanes with Arenes
https://www.thieme-connect.de/media/synlett/201720/i_r0475_ga_10-1055_s-0036-1588563.gif
Supporting Information
2941
Morimoto, Koji; Koseki, Doichi; Dohi, Toshifumi; Kita, Yasuyuki: Oxidative Biaryl Coupling of N-Aryl Anilines by Using a Hypervalent Iodine(III) Reagent
https://www.thieme-connect.de/media/synlett/201720/i_r0483_ga_10-1055_s-0036-1590875.gif
2946
Mohr, Lisa-Marie; Bach, Thorsten: Intermolecular [2+2] Photocycloaddition of β-Nitrostyrenes to Olefins upon Irradiation with Visible Light
https://www.thieme-connect.de/media/synlett/201720/i_r0492_ga_10-1055_s-0036-1588524.gif
Supporting Information Primary Data
2951
Hurtak, Jessica A.; McDonald, Frank E.: Regioselectivity of Mercury-Promoted Oxacyclizations of Alkynyl Diols
https://www.thieme-connect.de/media/synlett/201720/i_r0506_ga_10-1055_s-0036-1588562.gif
Supporting Information
2956
Gao, Ke; Yamamoto, Keita; Nogi, Keisuke; Yorimitsu, Hideki: Palladium-Catalyzed Arylation of Benzylic C–H Bonds of Azaarylmethanes with Aryl Sulfides
https://www.thieme-connect.de/media/synlett/201720/i_r0514_ga_10-1055_s-0036-1589098.gif
Supporting Information
2961
Narayanappa, Arkesh; Hurem, David; McNulty, James: Regioselective Ylide Formation on Acetal-Functionalized Trialkyl Phosphonium Salts: Extending the Scope of Carbonyl Homologation
https://www.thieme-connect.de/media/synlett/201720/i_r0528_ga_10-1055_s-0036-1588551.gif
Supporting Information
2966
Hirai, Yoshinori; Uozumi, Yasuhiro: Preparation of Aryl(dicyclohexyl)phosphines by C–P Bond-Forming Cross-Coupling in Water Catalyzed by an Amphiphilic-Resin-Supported Palladium Complex
https://www.thieme-connect.de/media/synlett/201720/i_r0609_ga_10-1055_s-0036-1590926.gif
Supporting Information
2971
Zhao, Changjia; Sibi, Mukund P.: Enantioselective and Diastereoselective Conjugate Radical Additions to α-Arylidene Ketones and Lactones
https://www.thieme-connect.de/media/synlett/201720/i_r0625_ga_10-1055_s-0036-1590930.gif
Supporting Information
2976
Aldmairi, Abdul Hadi; Knight, David W.; Wirth, Thomas: Acid-Catalyzed Tandem Process for the One-Pot Synthesis of Oxazolidines
https://www.thieme-connect.de/media/synlett/201720/i_r0719_ga_10-1055_s-0036-1591513.gif
Supporting Information

errata

e8
Piras, Monica; Andriu, Alexandra; Testa, Andrea; Wienecke, Paul; Fleming, Ian N.; Zanda, Matteo: Design and Synthesis of an RGD Peptidomimetic-Paclitaxel Conjugate Targeting αvβ3 Integrin for Tumour-Directed Drug Delivery