DOI: 10.1055/s-00000131

Synfacts

Issue 10 · Volume 11 · October 2015 DOI: 10.1055/s-005-30172

Synform

A134
Zanda, Matteo: SYNFORM ISSUE 2015/10

Synthesis of Natural Products and Potential Drugs

z1011
All PDFs of this category
1011
Asymmetric Fluorination Approach to an SYK Inhibitor
1012
Total Synthesis of (–)-Hosieine A
1013
Total Synthesis of Pandamarine
1014
Synthesis of (+)-Zincophorin Methyl Ester
1015
Synthesis of (R)-Baclofen
1016
Total Synthesis of Fidaxomicin
1017
Synthesis of Axitinib
1018
Total Synthesis of Pallambins A and B
1019
Synthesis of AG-041 Analogues
1020
Synthesis of OZ439
1021
Synthesis of (R)-Lisophylline
1022
Synthesis and Stereochemical Reassignment of Propindilactone G
1023
Synthesis of Sonepiprazole by an Asymmetric Oxa-Michael Reaction
1024
Synthesis of Amathaspiramides
1025
Synthesis of a SYK Inhibitor
1026
Propargyl-Linked Antifolates Overcome Resistance in S. aureus

Synthesis of Heterocycles

z1027
All PDFs of this category
1027
Synthesis of Fused Imidazobenzodiazepinones by Ugi Reaction
1028
Oxabicycles from Gold-Catalyzed Prins-Type Cyclization of Enynols
1029
Nickel-Catalyzed Asymmetric Synthesis of Axially Chiral Isoquinolones
1030
Enantioselective Synthesis of Chiral Fluorinated Isoindolinones
1031
Synthesis of Oligocyclic Dienes by anti-Carbopalladation–Heck Reaction
1032
Copper-Catalyzed Synthesis of Phosphonylated Quinoline-2,4-diones
1033
Synthesis of Pyrazolo-triazolo[1,4]oxazepines by [2+3] Cycloaddition
1034
Palladium-Catalyzed Synthesis of Dibenzofurans from 2-Iododiaryl Ethers
1035
Synthesis of Pyrazoles from N-Propargyl Hydrazones Mediated by tert-BuOK
1036
Four-Component Reaction Approach to Uracil Analogues
1037
Lewis Acid Catalyzed Synthesis of Di/Trifluoromethyl-1,2,3,4-Tetrahydroquinazolines
1038
Gold-Catalyzed Synthesis of 2-Aminoindoles and β-Carbolines
1039
New Biocatalysts for the Efficient Synthesis of Enantiopure N-Heterocycles
1040
Synthesis of 2-Azabicyclo[3.2.0]hept-2-enes and Pyrroles from Aza-enynes
1041
Synthesis of Trisubstituted Isoxazoles from Morita–Baylis–Hillman Acetates

Synthesis of Materials and Unnatural Products

z1043
All PDFs of this category
1043
Hand Specific Rings
1044
Bridged Bithiophene Building Blocks
1045
Floppy Fullerene Sandwiches
1046
Flashing Hydrocarbons from Tetrazoles
1047
Carbazoles Made by a Simple Swap
1048
Azaborines Aligned: One, Two, Three, and More
1049
Tetraphenylhexaazaanthracenes: 16π Weakly Antiaromatic Species
1050
A New Member in the Family: Synthesis of a Pyrene Tetracarboxylic Diimide
1051
Carb(azole)-load Your Metallodendrimers: A New Regimen
1052
Novel Pyrene-Fused Chromophores
1053
Hole-y Charged Polymers, Ball Mill!
1054
Bridge the Gap with Light

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1055
All PDFs of this category
1055
Chiral γ-Lactams by Enantioselective Cyclopropane Functionalization
1056
Asymmetric Scandium-Catalyzed Bromocyclization of N-Tosylcarbamates
1057
Gold-Catalyzed Intramolecular Cyclopropanation of Sulfonium Ylides
1058
Asymmetric Pd(II)-Catalyzed Cyclization of Allenyl Aldehydes with Boronic Acids
1059
Diastereoselective Copper-Catalyzed Annulation of Hydrazones
1060
Palladium-Catalyzed Fluorination via sp3 C–H Functionalization
1061
Rhodium-Catalyzed Asymmetric Arylation of α-Aryl-α-diazoacetates
1062
Ruthenium-Catalyzed Asymmetric Lactonization through Tsuji–Trost Allylation
1063
Asymmetric Transfer Hydroformylation Using Paraformaldehyde
1064
Iridium-Catalyzed Hydroacylation of Strained Alkenes with Salicylaldehydes
1065
Silver-Catalyzed Asymmetric 1,3-Dipolar Cycloaddition
1066
Enantioselective Hydroformylation of Terminal Olefins
1067
Intermolecular Hydroarylations of Norbornenes
1068
Diastereoselective Trifluoromethylation via Photoredox Catalysis
1069
Scandium(III)-Catalyzed Asymmetric Opening of 2,3-Epoxy 3-Aryl Ketones
1070
Asymmetric Alkylation of Cyclic N-Acyl Hemiaminals with Aldehydes
1071
Iridium-Catalyzed Trichloromethylation of 2-Acylimidazoles and Pyridines
1072
Olefin-Directed Palladium-Catalyzed Stereoselective Arylation of Allenes
1073
Enantioselective Carbonyl (α-Cyclopropyl)-allylation via Transfer Hydrogenation
1074
Chiral Heterocycles Using a Rhodium/Zirconium–BINOL Catalyst
1075
Palladium-Catalyzed Asymmetric Intermolecular Heck Reaction of Dihydrofurans
1076
Rhodium-Catalyzed Desymmetrization of α-Quaternary Centers
1077
Asymmetric Arylation of Secondary Alkyl Electrophiles
1078
Enantioselective Ring Opening of Azabenzonorbornadienes
1079
Ruthenium-Catalyzed Asymmetric Allylic Alkylation
1080
Enantioselective One-Pot Copper- and Gold-Catalyzed Alkylation and Annulation

Metal-Mediated Synthesis

z1081
All PDFs of this category
1081
Transnitrilation of Grignard Reagents and Aryllithiums
1082
Palladium-Catalyzed Tandem Cross-Coupling towards 9H-Fluorenes
1083
Iron-Catalyzed Cross-Coupling of Alkenyl Acetates
1084
Nickel-Catalyzed Alkyl–Alkyl Cross-Coupling
1085
Allylic Alkylation of α-Amino Ketones
1086
Catalytic Asymmetric Vinylation of Imines
1087
Hydroxyl-Directed Cross-Coupling
1088
Copper-Catalyzed Cross-Coupling of Allylboronic Acid Pinacol Ester with Haloalkanes
1089
Cross-Coupling of Unactivated Trialkyl(aryl)boranes with Aryl Halides
1090
Cobalt-Catalyzed Cross-Coupling of Piperidines with Grignard Reagents
1091
Lithiation–Borylation–Protodeboronation Methodology
1092
Rhodium-Catalyzed Vinylation
1093
Mild Gold(I)-Catalyzed Protodeboronation
1094
Nickel-Catalyzed Fluoromethylation of Arylboronic Acids
1095
Ruthenium-Catalyzed C–O/C–N Alkenylation of Aromatic Ketones

Organo- and Biocatalysis

z1097
All PDFs of this category
1097
Catalytic Asymmetric Umpolung of Imines
1098
Glycosylation by Using Electron-Deficient Pyridinium Salts
1099
NHC-Catalyzed Dimerization and Cross-Coupling of Enals to Cyclopentanones
1100
Hydrogen Activation and Hydrogenation with Fluorophosphonium Cations
1101
para Vinylation of Unprotected Phenols by a Biocatalytic Cascade
1102
Asymmetric Organocatalytic Conjugate Addition of Trifluoroborates
1103
Phosphine-Catalyzed Doubly Stereoconvergent γ-Additions to Allenoates
1104
Sulfenate-Catalyzed Alkyne Synthesis

Polymer-Supported Synthesis

z1105
All PDFs of this category
1105
Asymmetric Carbonyl Reduction with a Supported Ketoreductase
1106
A Magnetic Nickel Ferrate–Glutamate–Copper Catalyst for 1,2,3-Triazole Synthesis
1107
One-Pot Reduction–Isomerization of α,β-Unsaturated Ketones
1108
Deoxygenative Coupling of Nitroarenes on Ceria-Supported Gold Catalysts
1109
α-Acyloxylation of (Thio)Ethers Catalyzed by a Copper–Iron Mixed Oxide
1110
Zinc Oxide-Supported Palladium: Cross-Coupling at ppb Catalyst Loadings
1111
Nano Copper Ferrite-Catalyzed C–H Arylation of Benzothiazoles with Aryl Iodides
1112
Nucleophilic Hydroxylation of Alkyl Halides by Using an Oligoglycol-Bridged Ionic Liquid
1113
A Rasta Resin Supported Base Catalyst for the Morita–Baylis–Hillman Reaction of Allenones
1114
Reductive N-Alkylation with Supported Rhodium Nanoparticles
1115
Dehydrogenation of Cyclohexanones with Palladium/Carbon Under Hydrogen
1116
Dehydrogenative Synthesis of Benzazoles with Platinum Catalysts
1117
Supported Molybdenum-Catalyzed Oxidation of Sulfides to Sulfoxides
1118
Pyrazoloisoquinolines and Pyrazolopyridines by Carbonaceous Sulfonic Acid Catalysis
1119
Metal–Organic Framework-Supported Palladium Nano-Catalyst for Suzuki–Miyaura Coupling