DOI: 10.1055/s-00000131

Synfacts

Issue 05 · Volume 2011 · May 2011 DOI: 10.1055/s-002-21867

Synform

A37
Zanda, Matteo: SYNFORM ISSUE 2011/05

Synthesis of Natural Products and Potential Drugs

z461
All PDFs of this category
0461
Molinaro et al., C.: Synthesis of Renin Inhibitor MK-1597
0462
Zhou, Q.; Snider, B. B.: Synthesis of (±)-Phantasmidine
0463
Martin, D. B. C.; Vanderwal, C. D.: Synthesis of Strychnine
0464
Keck, G. E.; Poudel, Y. B.; Cummins, T. J.; Rudra, A.; Covel, J. A.: Synthesis of Bryostatin 1
0465
Knowles, R. R.; Carpenter, J.; Blakey, S. B.; Kayano, A.; Mangion, I. K.; Sinz, C. J.; MacMillan, D. W. C.: Synthesis of Diazonamide A
0466
Jousseaume, T.; Wurz, N. E.; Glorius, F.: Synthesis of Kynurenine 3-Hydroxylase Inhibitor FCE28833
0467
Green, J. C.; Pettus, T. R. R.: Syntheses of α-Cedrene, α-Pipitzol, and sec-Cedrenol
0468
di Fabio et al., R.: Synthesis of Casopitant
0469
Yang, L.; Wang, X.; Pan, Z.; Zhou, M.; Chen, W.; Yang, X.: Synthesis of (±)-Oxocrinine and Formal Synthesis of (±)-Crinine
0470
Hu, D. X.; Clift, M. D.; Lazarski, K. E.; Thompson, R. J.: Synthesis of Streptorubin B
0471
Ramgren, S. D.; Silberstein, A. L.; Yang, Y.; Garg, N. K.: Synthesis of Linezolid
0472
Yamamoto, T.; Suzuki, Y.; Ito, E.; Tokunaga, E.; Shibata, N.: Synthesis of (R)- and (S)-3′-Fluorothalidomide
0473
Shao, C.; Yu, H.-J.; Wu, N.-Y.; Tian, P.; Wang, R.; Feng, C.-G.; Lin, G.-Q.: Synthesis of (R)-Baclofen and (R)-Rolipram

Synthesis of Heterocycles

z475
All PDFs of this category
0475
Salman, G. A.; Hussain, M.; Iaroshenko, V.; Villinger, A.; Langer, P.: Thienopyrroles and Benzothienoquinolines via Palladium-Catalyzed Domino Reactions
0476
Vedachalam, S.; Wong, Q.-L.; Maji, B.; Zeng, J.; Ma, J.; Liu, X.-W.: Synthesis of Chromones via an Intramolecular Hydroacylation
0477
Castanedo, G. M.; Seng, P. S.; Blaquiere, N.; Trapp, S.; Staben, S. T.: Metal-Free Synthesis of 1,3,5-Trisubstituted 1,2,4-Triazoles
0478
Chunavala, K. C.; Joshi, G.; Suresh, E.; Adimurthy, S.: Catalyst- and Solvent-Free Synthesis of Substituted Imidazo[1,2-a]pyridines
0479
Guru, M. M.; Ali, M. A.; Punniyamurthy, T.: Cu(II)-Catalyzed Synthesis of Benzoxazoles from Bisaryloxime Ethers
0480
Wang, Z.-J.; Yang, F.; Lv, X.; Bao, W.: One-Pot Synthesis of Fused Unsymmetrical 2,2′-Biindolyls
0481
Pews-Davtyan, A.; Beller, M.: Zinc-Catalyzed Hydroamination Route to Di- and Trisubstituted Imidazoles
0482
Frolova, L. V.; Evdokimov, N. M.; Hayden, K.; Malik, I.; Rogelj, S.; Kornienko, A.; Magedov, I. V.: Synthesis of Polysubstituted 2-Aminopyrroles via a Multicomponent Reaction
0483
Gurunathan, S.; Perumal, P. T.: Synthesis of Dihydroquinolines via Pd/Cu-Catalyzed Heteroannulation
0484
Chen, Z.; Huang, G.; Jiang, H.; Huang, H.; Pan, X.: Palladium-Catalyzed Sonogashira Coupling and Iodocyclization Route to 3-Iodofurans
0485
Xiong, Z.; Qiu, X.-L.; Huang, Y.; Qing, F.-L.: TBS-Directed 1,3-Dipolar Cycloaddition to 5-Trifluoromethyl-1,2,3-triazoles
0486
Kunzer, A. R.; Wendt, M. D.: Synthesis of 2-Halo-3-carboxyindoles
0487
Gross, U.; Gross, P. J.; Shi, M.; Bräse, S.: NHC-Catalyzed Synthesis of Coumarins
0488
Adib, M.; Ansari, S.; Bijanzadeh, H. R.: Synthesis of N-Amino-Succinimides by a Multicomponent Reaction
0489
Saito, T.; Ogawa, S.; Takei, N.; Kutsumura, N.; Otani, T.: Palladium-Catalyzed Heteroannulation Route to 4-Alkylidene-4H-3,1-benzoxazines

Synthesis of Materials and Unnatural Products

z491
All PDFs of this category
0491
Evans, N. H.; Serpell, C. J.; Beer, P. D.: Chlorides in Handcuffs
0492
Qu, H.; Cui, W.; Li, J.; Shao, J.; Chi, C.: Pentacene: Going Above and Beyond
0493
Iwaniuk, D. P.; Wolf, C.: A Well-Oiled Stereodynamic Probe
0494
Rostami, A.; Wei, C. J.; Guérin, G.; Taylor, M. S.: Poly(squaramide) for Dihydrogenphosphate Detection
0495
Wessig, P.; Matthes, A.: (1,5)Naphthalenophanes via Photo-dehydro-Diels-Alder Cycloaddition
0496
Gessner, V. H.; Tilley, T. D.: Macrocycles from Reductive Zirconocene Coupling: On the Edge of Steric Overload
0497
Nambo, M.; Segawa, Y.; Itami, K.: A Versatile Route to Functionalized Fullerenes
0498
Prakash, G. K. S.; Ni, C.; Wang, F.; Hu, J.; Olah, G. A.: New Difluoro(sulfonato)methylation Method
0499
Kan, L.; Xu, Z.; Gao, C.: Efficient Access to Densely Functionalized Graphene Oxide Materials
0500
Mohebbi, A. R.; Wudl, F.: Emeraldicene Derivatives
0501
Motokuni, K.; Okada, T.; Takeuchi, D.; Osakada, K.: Everything is Falling into Place!
0502
Li, X.; Zhang, X.; Li, W.; Wang, Y.; Liu, T.; Zhang, B.; Yang, W.: Efficient TPA Cross-Conjugated Polymers
0503
Tsuneishi, A.; Okamoto, K.; Ikeda, Y.; Murai, M.; Miki, K.; Ohe, K.: One-Pot Chromophore Synthesis

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z505
All PDFs of this category
0505
Zhang, Z.; Zheng, W.; Antilla, J. C.: Calcium-Catalyzed Asymmetric Benzoyloxylation of 3-Aryloxindoles
0506
Gärtner, M.; Mader, S.; Seehafer, K.; Helmchen, G.: Iridium-Catalyzed Allylic Hydroxylation
0507
Trost, B. M.; Luan, X.: Pd/V Contemporaneous Dual Catalysis
0508
Guijarro, D.; Pablo, Ó.; Yus, M.: Ruthenium-Catalyzed Asymmetric Transfer Hydrogenation of Sulfinylimines
0509
Manna, K.; Xu, S.; Sadow, A. D.: Enantioselective Intramolecular Hydroamination of Alkenes
0510
Zheng, W.; Zhang, Z.; Kaplan, M. Z.; Antilla, J. C.: Calcium-Catalyzed Asymmetric Chlorination and Michael Additions
0511
Mori, F.; Fukawa, N.; Noguchi, K.; Tanaka, K.: Rhodium-Catalyzed Asymmetric Synthesis of Axially Chiral Diphosphine Ligands
0512
Langlois, J.-B.; Alexakis, A.: Copper-Catalyzed Asymmetric Allylic Alkylation
0513
Morandi, B.; Mariampillai, B.; Carreira, E. M.: Enantioselective Synthesis of Trifluoromethyl-Substituted Cyclopropanes
0514
Barroso, S.; Blay, G.; Muñoz, M. C.; Pedro, J. R.: Enantioselective Nitrone Cycloadditions with 2-Alkenoyl Pyridine N-Oxides
0515
Vieira, E. M.; Snapper, M. L.; Hoveyda, A. H.: Copper-Catalyzed Synthesis of Homoallylic Amines Using C1-Symmetric NHCs
0516
Slattery, C. N.; Maguire, A. R.: Copper-Catalyzed C-H Insertion in α-Sulfonyl Cyclopentanone Synthesis
0517
Li, Q.; Yu, Z.-X.: Enantioselective Rhodium-Catalyzed Allylic C-H Activation
0518
Peng, H.; Liu, G.: Palladium-Catalyzed Fluorination of Enynes
0519
Quintard, A.; Alexakis, A.; Mazet, C.: One-Pot Iridium and Enamine Catalysis
0520
Jadhav, A. M.; Bhunia, S.; Liao, H.-Y.; Liu, R.-S.: Gold-Catalyzed Stereoselective Synthesis of Azacyclic Compounds
0521
Han, Y.; Zhu, L.; Gao, Y.; Lee, C.-S.: Cascade Diels-Alder/Carbocyclization Approach to Hydrindanes
0522
Zhang, H.; Zhou, C.-B.; Chen, Q.-Y.; Xiao, J.-C.; Hong, R.: Synthesis and Suzuki Coupling of Monofluorovinyl Tosylates
0523
Sun, T.; Hou, G.; Ma, M.; Zhang, X.: Asymmetric Rhodium-Catalyzed Hydrogenation of α-Dehydroamino Ketones
0524
Sasaki, Y.; Horita, Y.; Zhong, C.; Sawamura, M.; Ito, H.: Selective Hydroboration of 1,3-Enynes Containing Internal Alkynes
0525
Cui, X.; Xu, X.; Lu, H.; Zhu, S.; Wojtas, L.; Zhang, X. P.: Enantioselective Cyclopropenation of Alkynes
0526
Aponick, A.; Biannic, B.: Gold-Catalyzed Synthesis of Chiral Tetrahydropyrans
0527
Bao, H.; Qi, X.; Tambar, U. K.: Palladium-Catalyzed Asymmetric [2,3] Rearrangements of Amine N-Oxides
0528
Cao, W.; Liu, X.; Wang, W.; Lin, L.; Feng, X.: Lewis Acid Catalyzed Asymmetric Synthesis of Tetrahydroquinolines
0529
Thaler, T.; Guo, L.-N.; Mayer, P.; Knochel, P.: Diastereoselective Palladium-Catalyzed C(sp³)-C(sp) Cross-Couplings
0530
Irrgang, T.; Friedrich, D.; Kempe, R.: Iridium-Catalyzed Asymmetric Hydrogenation of Aryl Ketones
0531
Balázsik, K.; Szőri, K.; Szőllősi, G.; Bartók, M.: New Insights in Heterogeneous Catalytic Asymmetric Hydrogenation
0532
Ibrahem, I.; Santoro, S.; Himo, F.; Córdova, A.: Asymmetric Conjugate Silyl Addition by Combined Copper/Chiral Amine Catalysis
0533
Mazuela, J.; Tolstoy, P.; Pàmies, O.; Andersson, P. G.; Diéguez, M.: Heck Reaction Catalyzed by Chiral Phosphite-Oxazole/Imidazole Ligands
0534
MacLellan, P.; Clayden, J.: Asymmetric Synthesis of Tertiary Thiols

Metal-Mediated Synthesis

z535
All PDFs of this category
0535
Tsuchimoto, T.; Kanbara, M.: Indium-Catalyzed Reductive Alkylation of Indoles
0536
Lumbroso, A.; Koschker, P.; Vautravers, N. R.; Breit, B.: Rhodium-Catalyzed Coupling of Terminal Alkynes with Carboxylic Acids
0537
Kirchberg, S.; Tani, S.; Ueda, K.; Yamaguchi, J.; Studer, A.; Itami, K.: Palladium-Catalyzed Coupling of Thiophenes and Thiazoles with Arylboronic Acids
0538
Han, W.; Mayer, P.; Ofial, A. R.: Palladium-Catalyzed Cross-Coupling of Benzazoles with Azoles
0539
Kitahara, M.; Umeda, N.; Hirano, K.; Satoh, T.; Miura, M.: Palladium-Free, Copper-Mediated Intermolecular Direct Biaryl Coupling
0540
Krämer, K.; Leong, P.; Lautens, M.: Enantioselective Palladium-Catalyzed Carbozincation of Cyclopropenes
0541
Fleming, P.; O’Shea, D. F.: Benzylic Metalation with a Mixed Metal Li/K-TMP Amide
0542
Grosso, A. Del; Singleton, P. J.; Muryn, C. A.; Ingleson, M. J.: Direct Arene Borylation with Borenium Cations to Yield Pinacol Boronates
0543
Lee, K. S.; Ready, J. M.: Titanium-Mediated Oxidative Arylation of Homoallylic Alcohols
0544
Zhou, L.; Shi, Y.; Xiao, Q.; Liu, Y.; Ye, F.; Zhang, Y.; Wang, J.: CuBr-Catalyzed Synthesis of Benzofurans and Indoles
0545
Satterfield, A. D.; Kubota, A.; Sanford, M. S.: Palladium-Catalyzed 1,1-Arylacetoxylation of Terminal Olefins
0546
Zhang, C.-P.; Wang, Z.-L.; Chen, Q.-Y.; Zhang, C.-T.; Gu, Y.-C.; Xiao, J.-C.: Copper-Mediated Trifluoromethylation of Heteroaromatic Iodides
0547
DeBerardinis, A. M.; Turlington, M.; Pu, L.: Activation of Vinyl Iodides for the Highly Enantioselective Addition to Aldehydes
0548
Chen, H.; Jiang, H.; Cai, C.; Dong, J.; Fu, W.: Palladium-Catalyzed Oxygenation of Allyl Arenes and Allyl Alkenes
0549
de Carné-Carnavalet, B.; Archambeau, A.; Meyer, C.; Cossy, J.; Folléas, B.; Brayer, J.-L.; Demoute, J.-P.: Copper-Free Sonogashira Coupling of Cyclopropyl Iodides with Terminal Alkynes

Organo- and Biocatalysis

z551
All PDFs of this category
0551
Zhong, F.; Wang, Y.; Han, X.; Huang, K.-W.; Lu, Y.: A Novel Bifunctional Phosphine Catalyst for Aza-Morita-Baylis-Hillman Reactions
0552
Nielsen, M.; Jacobsen, C. B.; Jørgensen, K. A.: Asymmetric C-P Bond Formation Using Phosphine Electrophiles
0553
Wang, J.; Feringa, B. L.: Control of Reaction Enantioselectivity with a Molecular Motor Switch
0554
Hashimoto, T.; Omote, M.; Maruoka, K.: Umpolung 1,3-Dipolar Cycloaddition of C,N-Cyclic Azomethine Imines
0555
Shapiro, N. D.; Rauniyar, V.; Hamilton, G. L.; Wu, J.; Toste, F. D.: Dithiophosphoric Acid Catalyzed Hydro-amination of Dienes
0556
Ma, T.; Fu, X.; Kee, C. W.; Zong, L.; Pan, Y.; Huang, K.-W.; Tan, C.-H.: Pentanidium-Type Chiral Phase-Transfer Catalysts
0557
Huang, H.; Jin, Z.; Zhu, K.; Liang, X.; Ye, J.: Vinylogous Michael Addition of α,β-Unsaturated γ-Butyrolactams to Enones
0558
Ryan, S. J.; Candish, L.; Lupton, D. W.: All-Carbon [4+2] Cycloaddition Catalyzed by an NHC
0559
Palacio, C.; Connon, S. J.: A Powerful Cinchona Alkaloid Derivative for the Henry Reaction
0560
Zhang, S.-L.; Xie, H.-X.; Zhu, J.; Li, H.; Zhang, X.-S.; Li, J.; Wang, W.: Enantioselective β-Functionalization of Aldehydes via Oxidative Enamine Catalysis
0561
Xiao, J.; Lu, Y.-P.; Liu, Y.-L.; Wong, P.-S.; Loh, T.-P.: Michael Addition of Aldehydes to Vinyl Sulfones
0562
Wu, B.; Liu, G.-G.; Li, M.-Q.; Zhang, Y.; Zhang, S.-Y.; Qiu, J.-R.; Xu, X.-P.; Ji, S.-J.; Wang, X.-W.: An Intermolecular Organocatalytic Entry to 4-Nitrocyclohexanones

Polymer-Supported Synthesis

z563
All PDFs of this category
0563
Yan, N.; Yuan, Y.; Dyson, P. J.: Rhodium Nanoparticle Catalysts Stabilized with Modified Polyvinylpyrrolidones
0564
Shi, L. X.; Wu, C. D.: A Copper Metal-Organic Framework Catalyst for Henry Reaction
0565
Egi, M.; Azechi, K.; Akai, S.: Polymer-Supported Gold(I) Catalysts for Intramolecular Cyclization
0566
Li, M.; Hu, L.; Cao, X.; Hong, H.; Lu, J.; Gu, H.: Hydrogenation of Nitro Groups and Reductive Amidation with Platinum Nanowires
0567
Olmos, A.; Sommer, J.; Pale, P.: [4+2] Cyclocondensation of Aryl Imines with Alkenes Using Sc(III) Zeolites
0568
Mikami, Y.; Noujima, A.; Mitsudome, T.; Mizugaki, T.; Jitsukawa, K.; Kaneda, K.: Deoxygenation of Amides, Sulfoxides, and Pyridine N-Oxides with AuHAP
0569
Polyzos, A.; O’Brien, M.; Petersen, T. P.; Baxendale, I. R.; Ley, S. V.: A Tube-in-Tube Gas-Liquid Flow Synthesis of Carboxylic Acids Using CO2
0570
Sakthivel, S.; Punniyamurthy, T.: Asymmetric Cyanosilylation with a Polymeric Chiral Titanium Complex
0571
Zeng, T.; Yang, L.; Hudson, R.; Song, G.; Moores, A. R.; Li, C.-J.: Enantioselective Imine Alkynylation with Fe3O4-Supported Copper Pybox
0572
Fukaya, N.; Onozawa, S.; Ueda, M.; Miyaji, T.; Takagi, Y.; Sakakura, T.; Yasuda, H.: Silica-Supported Chiral Rhodium Complex for Asymmetric Hydrogenation
0573
Grirrane, A.; Corma, A.; Garcia, H.: Borylation of Alkynes with MgO-Supported CuO or Pt Nanoparticles
0574
Khorsandi, Z.; Khosropour, A. R.; Mirkhani, V.; Baltork, I. M.; Moghadam, M.; Tangestaninejad, S.: Synthesis of 3-Hydroxyphthalans via Oxa-Pictet-Spengler Reaction
0575
Reddy, B. V. S.; Krishna, A. S.; Ganesh, A. V.; Kumar, G. G. K. S. N.: Synthesis of α-Aminophosphonates with Nano Fe3O4

Addenda and Errata

0576
Chromium-Catalyzed Enantioselective Alkynylation of Aldehydes