Synfacts 2006(1): 0062-0062  
DOI: 10.1055/s-2005-921724
Metal-Mediated Synthesis
© Georg Thieme Verlag Stuttgart · New York

Cross-Coupling of Benzyl Phosphates with Arylboronic Acids

Contributor(s): Paul Knochel, Andrei Gavryushin
M. McLaughlin*
Merck Research Laboratories, Rahway, US
Weitere Informationen

Publikationsverlauf

Publikationsdatum:
16. Dezember 2005 (online)

Significance

An interesting approach for the formation of diarylmethanes from easily available arylboronic acids is described. The protocol is simple and excellent tolerance of functional groups can be expected. Also, a practical method for the synthesis of benzylic diethyl phosphates is described.