DOI: 10.1055/s-00000083

Synlett

Issue 01 · Volume 27 · January 2016 DOI: 10.1055/s-005-30663

editorial

I
Editorial

synform

A1
Zanda, Matteo: SYNFORM ISSUE 2016/01

letter

1
Lewis, Frank W.; Harwood, Laurence M.; Hudson, Michael J.; Núñez, Ana; Galán, Hitos; Espartero, Amparo G.: Synthesis and Evaluation of a Novel Hydrophilic 6,6′-Bis(1,2,4-triazin-3-yl)-2,2′-bipyridine Ligand for Separating Actinide(III) from Lanthanide(III)
https://www.thieme-connect.de/media/synlett/201601/i_b0731_ga_10-1055_s-0035-1560541.gif
Supporting Information
6
Armstrong, Roly J.; D’Ascenzio, Melissa; Smith, Martin D.: Cation-Directed Enantioselective N-Functionalization of Pyrroles
https://www.thieme-connect.de/media/synlett/201601/i_d0738_ga_10-1055_s-0035-1560813.gif
Supporting Information
11
Bisterfeld, Carolin; Küberl, Irene; Dick, Markus; Pietruszka, Jörg: A Fluorogenic Screening for Enantio- and Diastereoselectivity of 2-Deoxy-d-ribose-5-phosphate Aldolases
https://www.thieme-connect.de/media/synlett/201601/i_d0693_ga_10-1055_s-0035-1560723.jpg
Supporting Information
17
Al-Ani, Widad; Shankland, Kenneth; Cobb, Alexander J. A.: Asymmetric Organocatalytic Synthesis of Cyclopentane γ-Nitroketones
https://www.thieme-connect.de/media/synlett/201601/i_d0726_ga_10-1055_s-0035-1560504.gif
21
Robertson, Gerard P.; Farley, Alistair J. M.; Dixon, Darren J.: Bifunctional Iminophosphorane Catalyzed Enantioselective Ketimine Phospha-Mannich Reaction
https://www.thieme-connect.de/media/synlett/201601/i_d0800_ga_10-1055_s-0035-1560530.gif
Supporting Information
25
Verhoog, Stefan; Pfeifer, Lukas; Khotavivattana, Tanatorn; Calderwood, Samuel; Collier, Thomas Lee; Wheelhouse, Katherine; Tredwell, Matthew; Gouverneur, Véronique: Silver-Mediated 18F-Labeling of Aryl-CF3 and Aryl-CHF2 with 18F-Fluoride
https://www.thieme-connect.de/media/synlett/201601/i_d0820_ga_10-1055_s-0035-1560592.gif
Supporting Information
29
Kim, Yo-Han; Han, Jusung; Jung, Byeong Yeon; Baek, Heeyoel; Yamada, Yoichi M. A.; Uozumi, Yasuhiro; Lee, Yoon-Sik: Production of Valuable Esters from Oleic Acid with a Porous Polymeric Acid Catalyst without Water Removal
https://www.thieme-connect.de/media/synlett/201601/i_d0448_ga_10-1055_s-0035-1560584.gif
Supporting Information
33
Rota, Filippo; Benhamou, Laure; Sheppard, Tom D.: Asymmetric Synthesis of Secondary Alcohols and 1,2-Disubstituted Epoxides via Organocatalytic Sulfenylation
https://www.thieme-connect.de/media/synlett/201601/i_d0635_ga_10-1055_s-0035-1560769.gif
Supporting Information
37
Blunt, Christopher E.; Nawrat, Christopher C.; LeBozec, Lucille; Liutkus, Mantas; Liu, Yang; Lewis, William; Moody, Christopher J.: Oxidative Routes to the Heterocyclic Cores of Benzothiazole Natural Products
https://www.thieme-connect.de/media/synlett/201601/i_d0651_ga_10-1055_s-0035-1560722.gif
Supporting Information
41
Anderson, James C.; Rundell, Christopher D.: Stereoselective Synthesis of Densely Substituted Tetrahydroquinolines by a Conjugate Addition Nitro-Mannich Reaction with Carbon Nucleophiles
https://www.thieme-connect.de/media/synlett/201601/i_d0752_ga_10-1055_s-0035-1560815.gif
Supporting Information
45
Broadley, Kenneth J.; Buffat, Maxime G. P.; Davies, Robin H.; Thomas, Eric J.: A Stereoselective Synthesis of a 3,4,5-Substituted Piperidine of Interest as a Selective Muscarinic (M1) Receptor Agonist
https://www.thieme-connect.de/media/synlett/201601/i_d0758_ga_10-1055_s-0035-1560753.gif
Supporting Information
51
Buckley, Benjamin R.; Figueres, Maria M. P.; Khan, Amna N.; Heaney, Harry: A New Simplified Protocol for Copper(I) Alkyne–Azide Cycloaddition Reactions Using Low Substoichiometric Amounts of Copper(II) Precatalysts in Methanol
https://www.thieme-connect.de/media/synlett/201601/i_d0767_ga_10-1055_s-0035-1560526.gif
Supporting Information
57
Seiple, Ian B.; Hog, Daniel T.; Myers, Andrew G.: Practical Protocols for the Preparation of Highly Enantioenriched Silyl Ethers of (R)-3-Hydroxypentan-2-one, Building Blocks for the Synthesis of Macrolide Antibiotics
https://www.thieme-connect.de/media/synlett/201601/i_d0780_ga_10-1055_s-0035-1560972.gif
Supporting Information
61
Muhammad, Rehmani N.; Draffan, Alistair G.; Banwell, Martin G.; Willis, Anthony C.: A Second-Generation Chemoenzymatic Total Synthesis of Platencin
https://www.thieme-connect.de/media/synlett/201601/i_d0783_ga_10-1055_s-0035-1560814.gif
Supporting Information
67
Honraedt, Aurélien; Gallagher, Timothy: Concise Entries to 4-Halo-2-pyridones and 3-Bromo-4-halo-2-pyridones
https://www.thieme-connect.de/media/synlett/201601/i_d0455_ga_10-1055_s-0035-1560469.gif
Supporting Information
70
Osler, Jonathan D.; Unsworth, William P.; Taylor, Richard J. K.: Synthetic Studies towards the Africanane Sesquiterpenes via the Cope Rearrangement of gem-Dimethyl-Substituted Divinyl Cyclopropanes
https://www.thieme-connect.de/media/synlett/201601/i_d0456_ga_10-1055_s-0035-1560176.gif
Supporting Information
75
Sonneck, Marcel; Kuhrt, David; Kónya, Krisztina; Patonay, Tamás; Villinger, Alexander; Langer, Peter: Regioselective Suzuki–Miyaura Cross-Coupling Reactions of the Bis(triflate) of 1,4-Dihydroxy-9H-fluoren-9-one
https://www.thieme-connect.de/media/synlett/201601/i_d0468_ga_10-1055_s-0035-1560211.gif
80
Bulman Page, Philip C.; Buckley, Benjamin R.; Elliott, Claire; Chan, Yohan; Dreyfus, Nicolas; Marken, Frank: Chemoselective Oxidation of Sulfides to Sulfoxides with Urea–Hydrogen Peroxide Complex Catalysed by Diselenide
https://www.thieme-connect.de/media/synlett/201601/i_d0481_ga_10-1055_s-0034-1378827.gif
Supporting Information
83
Monteiro, Julia L.; Pieber, Bartholomäus; Corrêa, Arlene G.; Kappe, C. Oliver: Continuous Synthesis of Hydantoins: Intensifying the Bucherer–Bergs Reaction
https://www.thieme-connect.de/media/synlett/201601/i_d0549_ga_10-1055_s-0035-1560317.gif
Supporting Information
88
McPherson, Christopher G.; Livingstone, Keith; Jamieson, Craig; Simpson, Iain: Palladium-Catalyzed Synthesis of Aryl Amides through Silanoate-Mediated Hydrolysis of Nitriles
https://www.thieme-connect.de/media/synlett/201601/i_d0636_ga_10-1055_s-0035-1560724.gif
Supporting Information
93
Bates, Roderick W.; Vilaivan, Tirayut; Apparao, Suryavanshi Padmakar; Ho, Tu Thanh: Synthesis of a Tetrahydrofuranyl β-Amino Acid for Peptide Nucleic Acid Construction
https://www.thieme-connect.de/media/synlett/201601/i_d0655_ga_10-1055_s-0035-1560649.gif
Supporting Information
96
Tietze, Lutz F.; Jackenkroll, Stefan; Ganapathy, Dhandapani; Reiner, Johannes R.: Formal Synthesis of (–)-Siccanin Using an Enantioselective Domino Wacker/Carbonylation/Methoxylation Reaction
https://www.thieme-connect.de/media/synlett/201601/i_d0705_ga_10-1055_s-0035-1560752.gif
Supporting Information
101
Flegeau, Emmanuel Ferrer; Harrison, Jack M.; Willis, Michael C.: One-Pot Sulfonamide Synthesis Exploiting the Palladium-Catalyzed Sulfination of Aryl Iodides
https://www.thieme-connect.de/media/synlett/201601/i_d0714_ga_10-1055_s-0035-1560578.gif
Supporting Information
106
Morgan, Kate F.; Doran, Robert; Croft, Rosemary A.; Hollingsworth, Ian A.; Bull, James A.: 2-Sulfinyl Oxetanes: Synthesis, Stability and Reactivity
https://www.thieme-connect.de/media/synlett/201601/i_d0749_ga_10-1055_s-0035-1560588.gif
Supporting Information
111
Cross, Paul W. C.; Herbert, John M.; Kerr, William J.; McNeill, Alan H.; Paterson, Laura C.: Isotopic Labelling of Functionalised Arenes Catalysed by Iridium(I) Species of the [(cod)Ir(NHC)(py)]PF6 Complex Class
https://www.thieme-connect.de/media/synlett/201601/i_d0757_ga_10-1055_s-0035-1560518.gif
116
Williamson, Alice E.; Ngouansavanh, Tifelle; Pace, Robert D. M.; Allen, Anna E.; Cuthbertson, James D.; Gaunt, Matthew J.: Rapid Generation of Complex Molecular Architectures by a Catalytic Enantioselective Dearomatization Strategy
https://www.thieme-connect.de/media/synlett/201601/i_d0759_ga_10-1055_s-0035-1560514.gif
Supporting Information
121
Gregory, Mark; Catimel, Bruno; Yin, Meng-Xin; Condron, Melanie; Burgess, Antony W.; Holmes, Andrew B.: Synthesis of a Tethered myo-Inositol (1,3,4,5,6)Pentakisphosphate (IP5) Derivative as a Probe for Biological Studies
https://www.thieme-connect.de/media/synlett/201601/i_d0764_ga_10-1055_s-0035-1560381.gif
Supporting Information
126
Bulman Page, Philip C.; Farah, Mohamed M.; Buckley, Benjamin R.; Chan, Yohan; Blacker, A. John: Preparation of C2-Symmetric Biaryl Bisiminium Salts and Their Use as Organocatalysts for Asymmetric Epoxidation
https://www.thieme-connect.de/media/synlett/201601/i_d0770_ga_10-1055_s-0035-1560540.gif
Supporting Information
131
Cranwell, Philippa B.; Russell, Andrew T.; Smith, Christopher D.: Methyl Hydrazinocarboxylate as a Practical Alternative to Hydrazine in the Wolff–Kishner Reaction
https://www.thieme-connect.de/media/synlett/201601/i_d0771_ga_10-1055_s-0035-1560805.gif
Supporting Information
136
Clemente-Tejeda, David; Zard, Samir Z.: O-Ethyl-S-(1,2,2,2-Tetrafluoroethyl)-Dithiocarbonate: A Convenient Reagent for the Generation and Capture of 1,2,2,2-Tetra­fluoroethyl Radicals
https://www.thieme-connect.de/media/synlett/201601/i_d0773_ga_10-1055_s-0035-1560539.gif
Supporting Information
141
Nixon, Gemma L.; Billington, Helen; Kalindjian, S. Barret; Steiner, Alexander; O’Neil, Ian A.: Tripodal Tris-N-oxides: Synthesis and Hydrogen Bonding Capabilities
https://www.thieme-connect.de/media/synlett/201601/i_d0782_ga_10-1055_s-0035-1560533.gif
Supporting Information
146
Watson, Emma L.; Ball, Anthony; Raw, Steven A.; Marsden, Stephen P.: Synthetic Studies on Psychotrimine: Palladium-Catalysed Arylation of 2-(N-Indolyl) Amides
https://www.thieme-connect.de/media/synlett/201601/i_d0786_ga_10-1055_s-0035-1560519.gif
151
Armstrong, Alan; Pullin, Robert D. C.; Scutt, James N.: Tertiary Amine Promoted Aziridination: Preparation of NH-Aziridines from Aliphatic α,β-Unsaturated Ketones
https://www.thieme-connect.de/media/synlett/201601/i_d0787_ga_10-1055_s-0035-1560583.gif
Supporting Information
156
Kaib, Philip S. J.; List, Benjamin: Highly Acidic BINOL-Derived Phosphoramidimidates and their Application in the Brønsted Acid Catalyzed Synthesis of α-Tocopherol
https://www.thieme-connect.de/media/synlett/201601/i_d0862_ga_10-1055_s-0035-1560971.gif
Supporting Information
159
Baumann, Marcus; Baxendale, Ian R.: Continuous-Flow Synthesis of 2H-Azirines and Their Diastereoselective Transformation to Aziridines
https://www.thieme-connect.de/media/synlett/201601/i_d0920_ga_10-1055_s-0035-1560391.gif
Supporting Information
164
O’Brien, Matthew; Cooper, Dennis: Continuous Flow Liquid–Liquid Separation Using a Computer-Vision Control System: The Bromination of Enaminones with N-Bromosuccinimide
https://www.thieme-connect.de/media/synlett/201601/i_d0789_ga_10-1055_s-0035-1560975.gif
Supporting Information
169
Beadle, Jonathan D.; Powell, Nicola H.; Raubo, Piotr; Clarkson, Guy J.; Shipman, Michael: Synthesis of Oxetane- and Azetidine-Containing Spirocycles Related to the 2,5-Diketopiperazine Framework
https://www.thieme-connect.de/media/synlett/201601/i_d0812_ga_10-1055_s-0035-1560593.gif
Supporting Information

errata

e1
Al-Ani, Widad; Shankland, Kenneth; Cobb, Alexander J. A.: Asymmetric Organocatalytic Synthesis of Cyclopentane γ-Nitroketones
e2
Williamson, Alice E.; Ngouansavanh, Tifelle; Pace, Robert D. M.; Allen, Anna E.; Cuthbertson, James D.; Gaunt, Matthew J.: Rapid Generation of Complex Molecular Architectures by a Catalytic Enantioselective Dearomatization Strategy