DOI: 10.1055/s-00000131

Synfacts

Issue 02 · Volume 2011 · February 2011 DOI: 10.1055/s-002-21628

Synform

A11
Zanda, Matteo: SYNFORM ISSUE 2011/02

Synthesis of Natural Products and Potential Drugs

z119
All PDFs of this category
0119
Xu et al., F.: Synthesis of Telcagepant
0120
Gauvreau, D.; Hughes, G. J.; Lau, S. Y. W.; McKay, D. J.; O’Shea, P. D.; Sidler, R. R.; Yu, B.; Davies, I. W.: Synthesis of MK-8141
0121
Han, S. B.; Hassan, A.; Ku, I. S.; Krische, M. J.: Total Synthesis of (+)-Roxaticin
0122
Slavov, N.; Cvengroš, J.; Neudörfl, J.-M.; Schmalz, H.-G.: Synthesis of Pestalone and Pestalalactone
0123
Kim, J.; Movassaghi, M.: Synthesis of (+)-Chaetocin A
0124
Zacharia, J. T.; Tanaka, T.; Hayashi, M.: Synthesis of (+)- and (-)-Fluvastatin
0125
Ramharter, J.; Weinstabl, H.; Mulzer, J.: Synthesis of (+)-Lycoflexine
0126
Micoine, K.; Fürstner, A.: Synthesis of Lactimidomycin
0127
O’Keefe, B. M.; Mans, D. M.; Kaelin, Jr, D. E.; Martin, S. F.: Total Synthesis of Isokidamycin
0128
Deng et al., X.: Synthesis of a CCK1 Receptor Antagonist
0129
Lemonnier, G.; Charette, A.: Synthesis of (-)-209I and (-)-223J
0130
Soulé, J.-F.; Mathieu, A.; Norsikian, S.; Beau, J.-M.: Synthesis of Zanamivir Congeners

Synthesis of Heterocycles

z131
All PDFs of this category
0131
Li, Y.; Wheeler, K. A.; Dembinski, R.: Au/Ag-Catalyzed Synthesis of 3-Fluorofurans
0132
Kurochkin, N. N.; Fesenko, A. A.; Cheshkov, D. A.; Davudi, M. M.; Shutalev, A. D.: Acid-Catalyzed Rearrangement of Ureido-dihydrofurans to N-Pyrrole Ureas
0133
Lin, S.; Zhao, G.-L.; Deiana, L.; Sun, J.; Zhang, Q.; Leijonmarck, H.; Córdova, A.: Enantioselective Synthesis of Dihydrofurans Using Dynamic Kinetic Resolution
0134
Wang, C.; Li, S.; Liu, H.; Jiang, Y.; Fu, H.: Copper-Catalyzed Ullmann-Type Coupling Route to Quinazolines
0135
Jiang, H.; Huang, H.; Cao, H.; Qi, C.: Synthesis of Oxazoles via TBHP/I2-Mediated Reaction of Alkenes with Benzylic Amines
0136
Ermolat’ev, D. S.; Bariwal, J. B.; Steenackers, H. P. L.; De Keersmaecker, S. C. J.; Van der Eycken, E. V.: Silver-Catalyzed Synthesis of 2-Amino-imidazole Alkaloids
0137
De Sarkar, S.; Studer, A.: NHC-Catalyzed Michael Addition for the Synthesis of Dihydropyranones
0138
Ozawa, T.; Horie, H.; Kurahashi, T.; Matsubara, S.: A Nickel-Catalyzed [2+2+1]-Cycloaddition Approach to Lactams
0139
Cioffi, C. L.; Lansing, J. J.; Yüksel, H.: Synthesis of 2-Aminobenzoxazoles from 2-Aminophenols
0140
Cikotiene, I.; Sazinas, R.; Mazeikaite, R.; Labanauskas, L.: Synthesis of Fused Thiophene-Isoxazoles from 2-Alkynyl-3-Nitro-Thiophenes
0141
Zeng, F.; Alper, H.: Synthesis of 1,4-Benzothiazepin-5-ones from N-Tosyl Aziridines and 2-Iodothiophenols
0142
Campbell, J. B.; Dedinas, R. F.; Trumbower-Walsh, S.: Synthesis of Isoindolones from Imines and ortho-Iodobenzoyl Acid Chlorides
0143
Sanz, R.; Guilarte, V.; Hernando, E.; Sanjuán, A. M.: Directed ortho-Metalation-Halocyclization Route to Benzothiophenes
0144
Huang, J.; Macdonald, S. J. F.; Harrity, J. P. A.: Palladium-Catalyzed Heterannulation Synthesis of 3-Borylated Indoles
0145
Li, C.; Zhang, Q.; Tong, X.: Tertiary Amine Catalyzed Annulation Route to Tetrasubstituted Pyrans

Synthesis of Materials and Unnatural Products

z147
All PDFs of this category
0147
Haberhauer, G.: Controlling Supramolecular Chirality
0148
Li, C.-Z.; Matsuo, Y.; Niinomi, T.; Sato, Y.; Nakamura, E.: Perfluorobenzene Captures Fullerene
0149
Baumes, J. M.; Gassensmith, J. J.; Giblin, J.; Lee, J.-J.; White, A. G.; Culligan, W. J.; Leevy, W. M.; Kuno, M.; Smith, B. D.: Supramolecular Glow-Sticks
0150
Kou, Y.; Tao, H.; Cao, D.; Fu, Z.; Schollmeyer, D.; Meier, H.: Pillar[5]arenes
0151
Kaloudi-Chantzea, A.; Karakostas, N.; Raptopoulou, C. P.; Psycharis, V.; Saridakis, E.; Griebel, J.; Hermann, R.; Pistolis, G.: Unquenched Fluorescent Metal Nanocages
0152
Fan, H.; Zhang, T.; Lv, S.; Jin, Q.: Polyelectrolytes: Fluorescence Turn-On Sensors in Aqueous Media
0153
Thirion, D.; Poriel, C.; Rault-Berthelot, J.; Barrière, F.; Jeannin, O.: (2,1-a)-Indenofluorene with Clapping Fluorenes
0154
Cant, A. A.; Roberts, L.; Greaney, M. F.: Cheap Precursor for Arynes
0155
Galán, H.; de Mendoza, J.; Prados, P.: Microwaveable Calixarenes
0156
Ding, L.; Ying, H.-Z.; Zhou, Y.; Lei, T.; Pei, J.: Polycyclic Imide Derivatives: Getting in Tune with Your Inner LUMO
0157
Dommerholt, J.; Schmidt, S.; Temming, R.; Hendriks, L. J. A.; Rutjes, F. P. J. T.; van Hest, J. C. M.; Lefeber, D. J.; Friedl, P.; van Delft, F. L.: Bicyclononynes: New Ring-Strained Alkynes for Bioorthogonal Labeling
0158
Du, C.; Ye, S.; Liu, Y.; Guo, Y.; Wu, T.; Liu, H.; Zheng, J.; Cheng, C.; Zhu, M.; Yu, G.: Facile Synthesis of Benzobisthioxanthene
0159
Zhang, X.; Jiang, X.; Zhang, K.; Mao, L.; Luo, J.; Chi, C.; Chan, H. S. O.; Wu, J.: Novel Synthesis of Tetrabenzocoronenes
0160
Shi, P.; Amb, C. M.; Knott, E. P.; Thompson, E. J.; Liu, D. Y.; Mei, J.; Dyer, A. L.; Reynolds, J. R.: Black to Transmissive Electrochromic Polymers
0161
Kuninobu, Y.; Seiki, T.; Kanamaru, S.; Nishina, Y.; Takai, K.: Synthesis of Functionalized Pentacenes from Isobenzofurans

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z163
All PDFs of this category
0163
Pradal, A.; Nasr, A.; Toullec, P. Y.; Michelet, V.: Stereoselective Iodocarbocyclization
0164
Coulter, M. M.; Kou, K. G. M.; Galligan, B.; Dong, V. M.: Intermolecular Hydroacylation of Homoallylic Sulfides
0165
Zhu, S.-F.; Song, X.-G.; Li, Y.; Cai, Y.; Zhou, Q.-L.: Enantioselective Synthesis of 2-Carboxy Cyclic Ethers
0166
Dias, L. C.; de Lucca, Jr, E. C.; Ferreira, M. A. B.; Garcia, D. C.; Tormena, C. F.: The Effect of β-Substituents in Aldol Reactions of Boron Enolates
0167
Park, J. K.; Lackey, H. H.; Rexford, M. D.; Kovnir, K.; Shatruk, M.; McQuade, D. T.: Design of a New Six-Membered NHC Ligand for Copper-Catalyzed β-Borylation
0168
Akai, S.; Hanada, R.; Fujiwara, N.; Kita, Y.; Egi, M.: Enantioenriched Allyl Esters via Lipase-Vanadium Combo Catalysis
0169
Boersma, A. J.; Coquière, D.; Geerdink, D.; Rosati, F.; Feringa, B. L.; Roelfes, G.: Enantioselective syn Hydration of Enones in Water Using a DNA-Based Catalyst
0170
Konrad, T. M.; Fuentes, J. A.; Slawin, A. M. Z.; Clarke, M. L.: Alkene Alkoxycarbonylation Using Novel Chiral Dipalladium Catalysts
0171
Yan, H.; Jang, H. B.; Lee, J.-W.; Kim, H. K.; Lee, S. W.; Yang, J. W.; Song, C. E.: Chiral Fluoride Generator and Its Application in Kinetic Resolution
0172
Murai, M.; Uenishi, J.; Uemura, M.: Enantioselective Synthesis of Planar Chiral Arene Chromium Complexes
0173
Nave, S.; Sonawane, R. P.; Elford, T. G.; Aggarwal, V. K.: Asymmetric Synthesis of Tertiary Stereogenic Centers
0174
Shono, T.; Harada, T.: Titanium-Catalyzed Reaction of Alkenylboron Reagents with Aldehydes
0175
Shen, A.; Liu, M.; Jia, Z.-S.; Xu, M.-H.; Lin, G.-Q.: Selective aza-Barbier Allylations of N-tert-Butanesulfinylimines
0176
Reznichenko, A. L.; Nguyen, H. P.; Hultzsch, K. C.: Rare Earth Metal Catalyzed Asymmetric Intermolecular Hydroamination
0177
Denmark, S. E.; Wilson, T. W.: Lewis Base Catalyzed Asymmetric Aldol Addition of Oxyketene Imines to Aldehydes
0178
Benkovics, T.; Guzei, I. A.; Yoon, T. P.: Copper-Catalyzed Synthesis of 3-Aminoindoles and Pyrroloindolines
0179
Barluenga, J.; Suero, M. G.; De la Campa, R.; Flórez, J.: Synthesis of Chiral Cyclohexenones Using a Multicomponent Reaction
0180
Miura, T.; Morimoto, M.; Murakami, M.: Nickel-Catalyzed [2+2+2] Cycloaddition of Isocyanates and Allenes
0181
Wang, L.; Li, P.; Menche, D.: Domino Synthesis of Complex Tetrahydropyrans
0182
Feng, X.; Yun, J.: Synthesis of Chiral Tertiary Organoboronic Esters by Conjugate Addition
0183
Boyd, W. C.; Crimmin, M. R.; Rosebrugh, L. E.; Schomaker, J. M.; Bergman, R. G.; Toste, F. D.: Enantioselective Synthesis of C2 and C1 Dienes
0184
Shen, K.; Liu, X.; Wang, W.; Wang, G.; Cao, W.; Li, W.; Hu, X.; Lin, L.; Feng, X.: Neodymium-Catalyzed Asymmetric Synthesis of 1,3-Bis(hydroxymethyl)-2-oxindoles
0185
Miao, L.; Haque, I.; Manzoni, M. R.; Tham, W. S.; Chemler, S. R.: Enantioselective Copper-Catalyzed Intramolecular Carboamination of Alkenes
0186
Gao, F.; Lee, Y.; Mandai, K.; Hoveyda, A. H.: Copper-Catalyzed Asymmetric Allylic Substitution with Arylaluminum Reagents
0187
Fackler, P.; Berthold, C.; Voss, F.; Bach, T.: Hydrogen Bond Assisted Asymmetric Metal Catalysis
0188
Chen, M.-W.; Duan, Y.; Chen, Q.-A.; Wang, D.-S.; Yu, C.-B.; Zhou, Y.-G.: Asymmetric Hydrogenation of Fluorinated Imines
0189
Long, Y.; Yang, D.; Zhang, Z.; Wu, Y.; Zeng, H.; Chen, Y.: Iridium-Catalyzed Enantioselective Ring Opening of Azanorbornene Derivatives
0190
Ito, H.; Kunii, S.; Sawamura, M.: Enantioconvergent Synthesis of Allyl Boronates
0191
Seashore-Ludlow, B.; Villo, P.; Häcker, C.; Somfai, P.: Dynamic Kinetic Resolution under Ruthenium-Catalyzed Transfer Hydrogenation
0192
Phan, D. H. T.; Kou, K. G. M.; Dong, V. M.: Enantioselective Desymmetrization of Cyclopropenes

Metal-Mediated Synthesis

z193
All PDFs of this category
0193
Ueda, K.; Yanagisawa, S.; Yamaguchi, J.; Itami, K.: β-Selective Arylation of Thiophenes
0194
Song, Z.; Lei, Z.; Gao, L.; Wu, X.; Li, L.: 3,3-Bissilyl Carbonyl and Enol Derivatives via Brook Rearrangement
0195
Sandrock, D. L.; Jean-Gérard, L.; Chen, C.-y.; Dreher, S. D.; Molander, G. A.: Stereospecific Cross-Coupling of Secondary Alkyl Trifluoroborates
0196
Lindh, J.; Sjöberg, P. J. R.; Larhed, M.: Palladium(II)-Catalyzed Decarboxylative Addition of Benzoic Acids to Nitriles
0197
Zhou, L.; Ye, F.; Zhang, Y.; Wang, J.: Coupling of N-Tosylhydrazone, Terminal Alkyne, and Aryl Halide
0198
Hiroshima, S.; Matsumura, D.; Kochi, T.; Kakiuchi, F.: Control of Product Selectivity in Ruthenium-Catalyzed C-H Arylation
0199
Fors, B. P.; Buchwald, S. L.: A Multiligand-Based Palladium Catalyst for C-N Cross-Coupling Reactions
0200
Shen, Z.-L.; Goh, K. K. K.; Cheong, H.-L.; Wong, C. H. A.; Lai, Y.-C.; Yang, Y.-S.; Loh, T.-P.: Coupling of Indium Homoenolates with Acid Chlorides
0201
Wang, C.; Rakshit, S.; Glorius, F.: Palladium-Catalyzed Decarboxylative Cross-Coupling of 2-Phenylbenzoic Acids
0202
Yeung, P. Y.; So, C. M.; Lau, C. P.; Kwong, F. Y.: Palladium-Catalyzed Cyanation of Aryl Mesylates
0203
Qin, C.; Jiao, N.: Iron-Catalyzed Oxidative C-H Transformation of Allylarenes or Alkenes to Alkenyl Nitriles
0204
Lundgren, R. J.; Stradiotto, M.: Palladium-Catalyzed Cross-Coupling with Hydrazine
0205
Simmons, E. M.; Hartwig, J. F.: Iridium-Catalyzed ortho-Silylation of Arenes by Hydroxyl-Directed C-H Activation
0206
Tsui, G. C.; Lautens, M.: Rhodium-Catalyzed 1,4-Addition of Arylboronic Acids to Allyl Sulfones
0207
Zhang, L.; Cheng, J.; Ohishi, T.; Hou, Z.: Copper-Catalyzed Direct Carboxylation of C-H Bonds Using Carbon Dioxide

Organo- and Biocatalysis

z209
All PDFs of this category
0209
Padmanaban, M.; Biju, A. T.; Glorius, F.: NHC-Catalyzed C-H Alkylation of Aldehydes
0210
Shirakawa, S.; Liu, K.; Ito, H.; Maruoka, K.: Asymmetric α-Alkylation of Cyanocarbolines by Phase-Transfer Catalysis
0211
Gómez-Bengoa, E.; Landa, A.; Lizarraga, A.; Mielgo, A.; Oiarbide, M.; Palomo, C.: α-Allylation of Aldehydes via a Conjugate Addition-Elimination Pathway
0212
Tsutsumi, Y.; Yamakawa, K.; Yoshida, M.; Ema, T.; Sakai, T.: Betaine-Catalyzed Synthesis of Cyclic Carbonates
0213
Thai, K.; Wang, L.; Dudding, T.; Bilodeau, F.; Gravel, M.: NHC-Catalyzed Intramolecular Redox Lactamization
0214
Li, X.; Luo, S.; Cheng, J.-P.: An Efficient Entry to Chiral Pyrroloindolines
0215
Uyeda, C.; Rötheli, A. R.; Jacobsen, E. N.: Chiral Guanidinium-Catalyzed Enantioselective Claisen Rearrangement
0216
Moteki, S. A.; Xu, S.; Arimitsu, S.; Maruoka, K.: A New Chiral Primary Amine Catalyst: Application in Conjugate Additions
0217
Albrecht, Ł.; Ransborg, L. K.; Gschwend, B.; Jørgensen, K. A.: 2-Hydroxyalkyl, 2-Aminoalkyl Furanes, and 2,3-Dihydrofuranes
0218
Mancheño, O. García; Tangen, P.; Rohlmann, R.; Fröhlich, R.; Alemán, J.: Michael Addition of β-Ketosulfones to Nitroalkenes
0219
Xu, F.; Huang, D.; Han, C.; Shen, W.; Lin, X.; Wang, Y.: SPINOL-Derived Phosphoric Acids for Addition of Indoles to Imines
0220
Čorić, I.; Müller, S.; List, B.: A Highly Efficient Approach to Chiral Homoaldols
0221
Takizawa, S.; Inoue, N.; Hirata, S.; Sasai, H.: An Asymmetric Domino Aza-Morita-Baylis-Hillman/Aza-Michael Reaction

Polymer-Supported Synthesis

z223
All PDFs of this category
0223
Liu, X.; Wang, P.; Zhang, L.; Yang, J.; Li, C.; Yang, Q.: Asymmetric Addition of Diethyl Zinc to Benzaldehydes with Ti(Oi-Pr)4 and NS(a)
0224
Rueping, M.; Bootwicha, T.; Sugiono, E.: Flow Hydroalkylation of Styrenes under Microwave Irradiation
0225
Leung, P. S.-W.; Teng, Y.; Toy, P. H.: Wittig Reactions Using a Bifunctional Polymeric Reagent
0226
Wang, B. G.; Ma, B. C.; Wang, Q.; Wang, W.: A Supported Organic Catalyst for Asymmetric Michael Addition
0227
Sawamura, T.; Kuribayashi, S.; Inagi, S.; Fuchigami, T.: Fluorination with Polystyrene-Supported Iodobenzenes in Ionic Liquid
0228
Sueoka, S.; Mitsudome, T.; Mizugaki, T.; Jitsukawa, K.; Kaneda, K.: Dehydration of Amides with Hydrotalcite-Supported Vanadium Catalyst
0229
Hu, L.; Shi, L.; Hong, H.; Li, M.; Bao, Q.; Tang, J.; Ge, J.; Lu, J.; Cao, X.; Gu, H.: Aerobic Epoxidation of Stilbene with Copper on FePt Nanowires
0230
Oda, Y.; Hirano, K.; Yoshii, K.; Kuwabata, S.; Torimoto, T.; Miura, M.: Aqueous Suzuki-Miyaura Coupling with Palladium Nanoparticles/BMI-TFSI
0231
Tucker-Schwartz, A. K.; Garrell, R. L.: TEMPO-Coated Fe3O4 Nanoparticles for Selective Oxidation of Alcohols
0232
Preedasuriyachai, P.; Kitahara, H.; Chavasiri, W.; Sakurai, H.: N-Formylation of Amines with Methanol or Formalin Using Gold Nanoclusters
0233
Stolze, S. C.; Meltzer, M.; Ehrmann, M.; Kaiser, M.: Solid-Phase Total Synthesis of Symplocamide A
0234
Dhakshinamoorthy, A.; Alvaro, M.; Garcia, H.: Acetalization with Methanol Using Metal-Organic Frameworks
0235
Maechling, S.; Good, J.; Lindell, S. D.: Solid-Phase Synthesis of an Amino Imidazotriazine Library

Addenda and Errata

0236
Alkenylative Cross-Coupling between Alkyl Sulfides and Grignard Reagents