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Synfacts 2020; 16(11): 1269
DOI: 10.1055/s-0040-1706324
Synthesis of Natural Products and Potential Drugs

Synthesis of LSZ102

Contributor(s):
Philip Kocienski
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Key words

LSZ102 - selective estrogen receptor degrader - benzothiophene ring formation - Krubsack–Higa reaction - C–H activation - arene hydroxylation - palladium catalysis


Publication History

Article published online:
20 October 2020

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