(untitled) - Rudolph, J; Aliagas, I; Crawford, J J; Mathieu, S; Lee, W; Chao, Q; Dong, P; Rouge, L; Wang, W; Heise, C; Murray, L J; La, H; Liu, Y; Manning, G; Diederich, F; Hoeflich, K P (ACS Med. Chem. Lett., 2015)