DOI: 10.1055/s-00000131

Synfacts

Issue 02 · Volume 14 · February 2018 DOI: 10.1055/s-008-37541

Synform

A16
Zanda, Matteo: SYNFORM ISSUE 2018/02

Synthesis of Natural Products and Potential Drugs

z0111
All PDFs of this category
0111
Synthesis of (–)-Himalensine A
0112
Modular Synthesis of (+)-Pleuromutilin
0113
Synthesis of an Inhibitor of Histone Lysine Demethylases KDM2/7
0114
Synthesis of BMS-986020 by a Tandem Borylation–Suzuki Procedure
0115
Modular Synthesis of Cyclotryptamine Alkaloids
0116
Synthesis of (+)-CP-99,994
0117
Total Synthesis of Bryostatin 1
0118
Synthesis of (+)-Sarcophytin
0119
Synthesis of Periconianone A
0120
Synthesis of a Dual Leucine Zipper Kinase Inhibitor
0121
Asymmetric Syntheses of Xanthanolides
0122
Synthesis of Ubrogepant

Synthesis of Heterocycles

z0123
All PDFs of this category
0123
[8+2] Cycloannulation: Synthesis of Dihydrocyclohepta[b]pyrrol-2(1H)-ones
0124
Copper-Catalyzed Aerobic Indole Synthesis through Nitrogen Radical Cyclization
0125
Oxidative Cross-Coupling of Nonactivated Substrates to Yield 1-Benzazepines
0126
Cobalt-Catalyzed Synthesis of 5-Aminooxazoles
0127
Palladium-Catalyzed Enantioselective Synthesis of Fused Benzofurans
0128
Synthesis of β-(Hetero)Aryl Ketones through sp3 C–H Activation
0129
Photochemical Synthesis of Chloromethylated Pyrrolidines
0130
Synthesis of Heteroaryl Amino Acids
0131
Copper-Catalyzed Synthesis of 1-(2-Hydroxyaryl)-1H-indazoles
0132
N-Heterocyclic Carbene Catalyzed Synthesis of Substituted Pyridines
0133
Synthesis of Functionalized Spiro-Oxetanes for Combinatorial Chemistry
0134
Manganese-Catalyzed Minisci Alkylation of Heteroarenes
0135
Copper-Catalyzed Synthesis of Dihydropyrroles and Pyrroles

Synthesis of Materials and Unnatural Products

z0137
All PDFs of this category
0137
Butterfly-Shaped Semiconductor Molecules
0138
Triazoliptycenes: Solution-Like Fluorescence in the Solid State
0139
Rhodium(III)-Catalyzed C–H Activation Towards Polyarylated Naphthols
0140
Easy as Di(mer)
0141
Visible-Light-Promoted C–S Cross-Coupling
0142
Over the Rim of Cycloaddition
0143
Helical Radicals with NIR Circular Dichroism
0144
Expanded N-Heterocycles through C(sp3)–H Amination
0145
Iodonium Trifluoroborates: New Bifunctional Reagents
0146
A Library of PPYPs with Unique Fluorescence Properties
0147
Molecular Crabs Can Catalyze Transfer Hydrogenation of Quinolines
0148
A New Addition to the APEX Family

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z0149
All PDFs of this category
0149
Coupling of Boronic Acids, 1,3-Enynes and Cyclic Imines
0150
Protocol for the Synthesis of Allylic Aryl Ethers
0151
Cooperative Catalysis for Asymmetric Decarboxylative Cyanation
0152
Asymmetric Alkylation of Quinoline N-Oxides with Vinylarenes
0153
Silver-Catalyzed Enantioselective Allylation of Aldehydes
0154
Gold-Catalyzed Synthesis of Cyclohepta[b]indoles
0155
Ruthenium-Catalyzed Cycloaddition
0156
Ion Pair Directed Hydrogenation of α,α-Disubstituted Terminal Olefins
0157
Visible-Light-Activated Asymmetric β-C–H Functionalization of Ketones
0158
Iron(II)-Catalyzed Michael Addition
0159
Cobalt-Catalyzed Asymmetric Allylation
0160
Scandium-Catalyzed Asymmetric Dearomatization of β-Naphthols
0161
Asymmetric Reduction of Allyl Bromides by Copper Catalysis
0162
Copper-Catalyzed Enantioselective Borylation of Alkenes
0163
Enantioselective Synthesis of Lactones by Ternary Catalysis
0164
Nickel-Catalyzed N-Alkylation of Acylhydrazines and Arylamines
0165
Copper-Catalyzed Stereospecific Synthesis of α-Silylated Nitriles and Esters
0166
Palladium-Catalyzed [3+2] Cycloaddition
0167
Nickel-Catalyzed C(sp3) Cross-Coupling
0168
Disubstituted Pyrrolidines through C–H Bond Amination
0169
α-Hydroxyallenes through β-Oxygen Elimination of α-Epoxy Vinyl Boronates
0170
Nickel/Zinc Co-Catalyzed Asymmetric [2+2] Cycloaddition
0171
Rhodium-Catalyzed Enantioselective Hydroarylation of 1,3-Dienes by Indoles
0172
Gold-Catalyzed Intramolecular Cyclization of N-Allenamides
0173
Enantioselective N–H Functionalization of Quinazolinones
0174
Zinc-Catalyzed Asymmetric Synthesis of β,β-Diaryl α-Hydroxy Ketones
0175
Enantioselective α-Arylative Desymmetrization of 1,3-Diketones
0176
Enantioselective Synthesis of Hydropyrimidines by Allylic C–H Amination
0177
Enantioselective Cu-Catalyzed Reductive Hydroxymethylation of Styrenes and 1,3-Dienes
0178
Aqueous Copper-Catalyzed Henry Reaction

Metal-Mediated Synthesis

z0179
All PDFs of this category
0179
Organolithium Chemistry in an Environmentally Friendly Medium
0180
Nickel-Catalyzed 1,2-Diarylation of Unactivated Olefins
0181
Hydrogenolysis and Conjugate Addition of 2-(Hydroxymethyl)pyridines
0182
Enantiospecific Coupling of Phenols with Boronic Esters
0183
Phenanthrene Synthesis via Annulation of Grignard Reagents and Alkynes
0184
Iron-Catalyzed Remote Arylation
0185
Asymmetric Synthesis of α-Tertiary Amines
0186
Hydroarylation of Styrenes and 1,3-Dienes
0187
Late-Stage C–H Functionalization of Arenes
0188
Photoredox/Nickel Dual-Catalysis: Synthesis of Secondary Benzylic Alcohols
0189
Novel Intermolecular Pummerer Coupling Protocol
0190
Palladium-Catalyzed Diastereoselective 1,4-Addition
0191
Transition-Metal-Free Cross-Coupling of (Hetero)aryl Thiols
0192
Stereocomplementary Cross-Coupling of Diols with Boronic Acids
0193
Nucleophilic Arylation of N,O-Ketene Acetals

Organo- and Biocatalysis

z0195
All PDFs of this category
0195
Organocatalytic C(sp3)–H Amination through Nitrenoid Transfer
0196
Asymmetric Silylium Catalysis Enabled by Hydrogen-Bond Donors
0197
Iminium Catalysis inside a Self-Assembled Supramolecular Capsule
0198
Visible-Light-Mediated Metal-Free Hydrosilylation of Alkenes
0199
Cinchona Squaramide Catalyzed Asymmetric Domino Reaction
0200
Biocatalytic Highly Enantioselective Oxidative Dearomatization of Phenols
0201
BINOL-Catalyzed Reductive Petasis Borono-Mannich Reaction of Enals
0202
Anthraquinones as Photoredox Organocatalysts
0203
A Catalytic Enantioselective Prototopic Shift/Furan Diels–Alder Cascade
0204
Atroposelective Synthesis of Axially Chiral Biaryl Amino Alcohols

Polymer-Supported Synthesis

z0205
All PDFs of this category
0205
Visible-Light-Mediated [4+2] Annulation of N-Cyclobutylanilines on Self-Doped Titania
0206
Photocatalytic Click Reactions on a Two-Dimensional Cu(II) Coordination Polymer
0207
Synthesis of (±)-Pregabalin in a Sequential Flow System
0208
Copper/Nickel-Catalyzed Reduction of Nitroarenes by Borazane
0209
Resorcinarene Salt Catalyzed Epoxide–Carbon Dioxide Coupling Reactions
0210
Stabilized Pd Nanoparticle Catalyzed Conjugate Addition of Aryl Halides to Enones
0211
A Sulfated Polyborate Catalyst for the Synthesis of 1,5-Benzodiazepines
0212
Heterogenized CuI Catalyst for Ullmann-Type C–N Coupling
0213
Heterogeneous Iron Catalyst for Aerobic Oxi-dation of Alcohols and Benzylic Compounds
0214
Pd/Zeolite-Catalyzed Annulation of o-Haloaromatic Amines with Terminal Alkynes
0215
Selective Hydrogenation of Enals and Enones on Ionic Liquid–Rhodium Nanoparticles
0216
Platinum Nanoparticle Catalyzed Selective Flow Hydrogenation of Aldehydes
0217
Batch and Continuous-Flow Huisgen Reactions on Dendrimer-Supported CuSO4
0218
NiGa Layered Double-Hydroxide Catalyst for Tandem Condensation Reactions
0219
Gold-Catalyzed Conversion of Alkynes into Amides
0220
Copper-Catalyzed Glaser–Hey Homocoupling of Terminal Alkynes