DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 12 · August 2016 DOI: 10.1055/s-006-32122

Synform

A111
Zanda, Matteo: SYNFORM ISSUE 2016/08

Synthesis of Natural Products and Potential Drugs

z767
All PDFs of this category
0767
Total Synthesis of (−)-6-epi-Ophiobolin N
0768
Synthesis of Darunavir
0769
Synthesis of PDE4 Inhibitors
0770
Large Scale Synthesis of Eupalinilide E
0771
Synthesis of (+)-Dictyoxetane
0772
Synthesis of an Inhibitor of Influenza Virus Replication
0773
Syntheses of Decinnamoyltaxinine E and Taxabaccatin III
0774
Synthesis of (R)-JM 1232 by Asymmetric Alkynylation
0775
Synthesis of a Glucocorticoid Receptor Modulator
0776
Synthesis of a tRNA–Guanine Transglycosylase Inhibitor
0777
Total Syntheses of Erythrina Alkaloids
0778
Synthesis of LpxC Inhibitor LP-058
0779
Synthesis of Strongylophorine-2
0780
Synthesis of Indolactam V
0781
Synthesis of (+)-Minfiensine

Synthesis of Heterocycles

z783
All PDFs of this category
0783
Minisci-Type Reaction of Nonactivated Ethers with Heterocycles
0784
Fluorinated Triazoles by Using a Heterobifunctional Fluoroalkylation Reagent
0785
1,3-Dipolar Cycloaddition of Azomethine Imines with Enecarbamates
0786
Synthesis of Chiral Piperazinones from Aziridine Aldehyde Dimers
0787
[3+2] Cycloaddition Route to Imidazopyrrolo-Fused Isoxazoles
0788
Synthesis of Enantiomerically Enriched Isoquinoline Derivatives
0789
Synthesis of Pyrroles by Rhodium-Catalyzed Hydroacylation of Alkynylamines
0790
Synthesis of 3-Bromoquinoline-2(1H)-thiones
0791
Functionalized Arynes from Aryl Iodonium Salts
0792
Four-Component Palladium-Catalyzed Synthesis of Pyrroles
0793
Palladium-Catalyzed Synthesis of (Spiro)polyheterocycles by Domino Post-Ugi Route
0794
Halogenated Piperidines and Tetrahydropyrans by the Prins Reaction
0795
Palladium-Catalyzed Synthesis of Phenanthridinones by Dual C–H Activation
0796
Heteroannulation Route to Fluorinated Purine Derivatives

Synthesis of Materials and Unnatural Products

z797
All PDFs of this category
0797
Synthesis of Symmetrical and Unsymmetrical 1,4-Dithiins
0798
Two Dots in One ‘DIAn’
0799
Bottoms Up! Ball Mill Synthesis of Water-Soluble ZnO from Molecular Precursors
0800
A Novel TBI Building Unit for Semiconducting Polymers
0801
Synthesis of Twisted PAH via [4+4] Dimerization
0802
Switch-Hitter but Primarily a Dienophile
0803
Cyclic Polyacetylenes by Tungsten Catalysis
0804
One-Pot Synthesis of Tetraphene and Construction of Expanded Conjugated Aromatics
0805
Calcium-Sensitive Photocage: An In Situ Ca2+ Sensor
0806
Let Me Reiterate…Sequence Control in Living Radical Polymerizations
0807
Making the Most of γ-Butyrolactones: Catalytic, Chemoselective, Clickable
0808
Feeling Lucky? Making d20 Dice Stand On a Vertex

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z809
All PDFs of this category
0809
Asymmetric Michael Addition Reaction via Rhodium Catalyst Fragmentation
0810
Rhodium-Catalyzed Asymmetric Cycloisomerization of (E)-1,6-Enynes
0811
Quaternary Stereocenters by Asymmetric Allylic Alkylation
0812
Pd-Catalyzed Diastereoselective Synthesis of Borylated Chromans
0813
Enantioselective Rhodium-Catalyzed Silylation of C−H Bonds
0814
Enantio- and Regioselective Copper-Catalyzed Hydroboration of Internal Alkenes
0815
Enantioselective and Diastereoselective Scandium-Catalyzed [3+3] Annulation
0816
Asymmetric Nickel-Catalyzed Diels–Alder Reaction
0817
Iridium-Catalyzed Asymmetric C–H Functionalization with Ethyl Diazoacetate
0818
Cobalt-Catalyzed Regioselective Alkenylation of 8-Methylquinoline with Alkynes
0819
Synthesis of Chiral Spiro-nitroprolinates by Silver(I) Catalysis
0820
Desymmetrization of Cyclohexadienones by Conjugate Hydrosilylation
0821
Asymmetric Iridium-Catalyzed Hydrogenation of Pyridinium Salts
0822
Desymmetrization of Cyclopentenes by Rh-Catalyzed Hydroformylation Reaction
0823
Synthesis of Indolines from 1,2,3-Triazoles by a Rhodium-Catalyst
0824
Titanium-Catalyzed Asymmetric Epoxidation of N-Alkenyl Sulfonamides
0825
Site- and Stereoselective Functionalization of Nonactivated Alkanes
0826
Asymmetric [3+2] Cycloaddition by Synergistic Catalysis
0827
Asymmetric Photoinduced Copper-Catalyzed C–N Coupling of Alkyl Chlorides
0828
Enantioselective Rhodium-Catalyzed C−H Insertion of Carbenes
0829
Asymmetric Hydrogenation of 1,8-Naphthyridines by Ruthenium(II) Catalysis
0830
Copper-Catalyzed [3+2] Cycloaddition of Enones with a Trifluoromethyl Group
0831
Highly Asymmetric Synthesis of α-Aryl Ketones
0832
Palladium-Catalyzed Asymmetric Synthesis of Functionalized 2,3-Dihydrofurans
0833
Axially Chiral Boron Catalyst for Asymmetric Piers Hydrosilylation
0834
Palladium-Catalyzed Asymmetric Hydrogenation of Fluorinated Hydrazones
0835
Copper-Catalyzed Mannich Type Reaction of Alkylamides
0836
Copper(II)-Catalyzed (E)-Selective Hydrosilylation of Allenes
0837
Rhodium-Catalyzed Stepwise Asymmetric Arylation of Cyclic Sulfamidates

Metal-Mediated Synthesis

z839
All PDFs of this category
0839
Enantioselective Addition of Organoboron Reagents to Fluoroketones
0840
Oxidative Trifluoromethylation of Alkynes with Fluoroform-Derived CuCF3
0841
Magnesium-Catalyzed Hydroboration of Carbodiimides
0842
Palladium-Catalyzed Carboperfluoroalkylation
0843
Iron-Catalyzed Cross-Coupling of Tosylates
0844
2,3-Dihydroisoxazole Synthesis from Alkynes and Nitrones
0845
Palladium-Catalyzed Cross-Coupling of Allylboronic Acids with α-Diazoketones
0846
Cobalt-Catalyzed Arylative Cyclization of Acetylenic Esters and Ketones
0847
Coupling of Organocuprates with Propargyl Electrophiles
0848
Nickel-Catalyzed Cyclization of Alkyne-Nitriles
0849
Photoredox/Nickel Dual Catalytic Cross-Coupling
0850
Nickel-Catalyzed Cross-Coupling of Anisoles with Alkylmagnesium Reagents
0851
Carboxylation of Alkenes and Heteroaromatics
0852
Multicomponent Cascade Synthesis
0853
Chemoselective Primary Amination of Boronic Acids

Organo- and Biocatalysis

z855
All PDFs of this category
0855
N-Hydroxyphthalimide-Catalyzed Electrochemical Allylic Oxidation
0856
A New Substituent for BINOL-Phosphate Catalysis
0857
Proline-Catalyzed Enantioselective Synthesis of 2,3-Disubstituted Piperidines
0858
Triflic Acid Catalyzed Enyne Cyclization
0859
Iminium Catalysis in a Supramolecular Host
0860
An Organocatalytic Approach to Enantiopure 2H- and 3H-Pyrroles
0861
Organocatalytic Construction of Spiroindane Derivatives
0862
Visible-Light-Promoted Synthesis of Benzo[b]phosphole Oxides
0863
One-Pot Biocatalytic Cascade to Substituted Piperidines and Pyrrolidines

Polymer-Supported Synthesis

z865
All PDFs of this category
0865
Arylation of Pyrroles and Imidazoles with Bromobenzenes Using Pd@PPy
0866
Peptide-Catalyzed Epoxidation with Inverted Juliá–Colonna Stereoselectivity
0867
Organocatalyzed Asymmetric Michael Addition of Ketones and Nitrostyrenes
0868
Chemoselective Reduction of Aldehydes with Pd-Nanoparticles
0869
Homocoupling of Alkynes on Polystyrene-Supported Copper Catalyst
0870
Gold/Titania-Catalyzed Semireduction of Alkynes by Formic Acid
0871
Solid-Phase Syntheses of Polysubstituted 2-Sulfanylbenzimidazoles
0872
A Functionalized Covalent Organic Framework for Formylation of Amines
0873
Three-Component Synthesis of Propargylamines with Supported Au Nanoparticles
0874
Reduction of Nitroarenes on Microsphere-Supported Silver Nanoparticles
0875
An Activated Metal–Organic Framework Catalyst with a Lewis Acid
0876
Gold-Catalyzed Oxidation of Anilines to Nitrosobenzenes by Hydrogen Peroxide
0877
Hydrogenation of Enals and Enones on Supported Palladium Nanoparticles
0878
Copper-Catalyzed Coupling of Arylboronic Acids with Sulfonyl Azides
0879
Pd-Catalyzed Carbonylative Coupling of Triarylbismuthines with Aryl Iodides
0880
Copper-Catalyzed Oxidative Coupling of Amines with Disulfides or Thiols
0881
Ferrite Nanoparticle/Montmorillonite-Catalyzed Baeyer–Villiger Oxidation
0882
Hydrosilylation of Terminal Alkynes with a Copper/Carbene-Functionalized Polymer