DOI: 10.1055/s-00000131

Synfacts

Issue 07 · Volume 11 · July 2015 DOI: 10.1055/s-005-29358

Synform

A90
Zanda, Matteo: SYNFORM ISSUE 2015/07

Synthesis of Natural Products and Potential Drugs

z677
All PDFs of this category
0677
Synthesis of Glucagon Receptor Antagonist LY2409021
0678
Total Synthesis of Paspaline
0679
Synthesis of Diterpenoid Steenkrotin A
0680
Synthesis of Aliskiren
0681
Synthesis of DZ-2384
0682
Total Synthesis of Santalin Y
0683
Synthesis of rac-Efavirenz
0684
Formal Synthesis of Telaprevir
0685
Synthesis of 5,6-Dihydrocineromycin B
0686
Synthesis of Mycoleptodiscin A
0687
Synthesis of (+)-Muironolide A
0688
Total Synthesis of (–)-Galanthamine and (–)-Lycoramine
0689
Synthesis of a BACE1 Inhibitor

Synthesis of Heterocycles

z691
All PDFs of this category
0691
Rhodium(III)-Catalyzed Synthesis of 1,2-Benzothiazines
0692
Enantioselective Copper(I)-Catalyzed Construction of Spiroketals
0693
6-endo-dig versus 5-exo-dig. The Profound Effects of Acetonitrile
0694
Synthesis of Dihydropyridin-2-ones via an Ugi–Aldol Reaction
0695
Minisci-Type Synthesis of Tetrahydropyridopyridazines
0696
Single-Step Synthesis of Isoindolinones
0697
Synthesis of Fluorinated Diphenylpyrazole
0698
Four New Bonds in One Pot: Isoxazolines from Olefins and 2-Ethylquinolines
0699
Pyrido[2,3-c]coumarins via an Intramolecular Povarov Reaction
0700
Synthesis of 1,2-Borazaronaphthalenes
0701
Benzyne Route to Benzothiazoles
0702
Copper-Catalyzed Oxidative Annulation Approach to Oxadiazoles
0703
Enamide Umpolung for the Synthesis of Heterocycles
0704
Oxabicycles via Sequential Prins–Wagner–Ritter Processes
0705
Synthesis of Hexahydropyrano[3,4-c]chromenes via Prins Bicyclization

Synthesis of Materials and Unnatural Products

z707
All PDFs of this category
0707
Hexaaza Macrocycles Revisited
0708
Nestable Tetrakis(spiroborate) Nanocycles
0709
Circulene Flow
0710
A Mild Route to Quinoxalines Featuring Iodine
0711
Tiny Molecule, Big Fluorescence
0712
Synthesis of 2,5-Disubstituted Thiazoles
0713
Phospholify and Diversify
0714
Pitched Propeller PAHs
0715
Bowled Over! Nitrogen Takes Center Stage from Carbon in Azacorannulenes
0716
A Polymerization Displaying Great Tact
0717
Incorporating More Nitrogen Atoms in Hexacenes
0718
A Molecular Spring

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z719
All PDFs of this category
0719
Copper Hydride Catalyzed Synthesis of 2,3-Disubstituted Indolines
0720
Asymmetric Haloaminocyclization for the Synthesis of Cyclic Sulfamates
0721
Rhodium-Catalyzed Asymmetric Dearomatization of Naphthols with Alkynes
0722
Synthesis of Indanes and Indanones through Tandem Catalysis
0723
Iridium-Catalyzed Branched-Selective Hydroarylation of Vinyl Ethers
0724
Iridium-Catalyzed Asymmetric Hydrogenation of Ketones in Ethanol
0725
Gold-Catalyzed [2+2+2] of Allenamides, Alkenes and Aldehydes
0726
Catalytic Stereoselective Reaction of β-Lactams with Aldehydes
0727
Palladium-Catalyzed Enantioselective Reductive Heck Reactions
0728
Palladium- and Chiral Phosphoric Amide/Acid-Catalyzed C–H Arylation
0729
Enantioselective Allylic Alkylation of Ortho-Substituted Cinnamyl Bromides
0730
Enantioselective Synthesis of α-Trifluoromethylamines
0731
Iron-Catalyzed Z-Selective Olefin Synthesis
0732
Asymmetric Transfer Hydrogenation of Ketones by Macrocyclic Iron Complexes
0733
Addition of Allenes to Fluorinated Alcohols Catalyzed by Ruthenium
0734
Iridium-Catalyzed Intramolecular Asymmetric C–H Alkylations
0735
Zirconium-Catalyzed Asymmetric Hydroamination of Primary Aminoalkenes
0736
Enantioselective Scandium-Catalyzed 1,6-Addition of Oxindoles
0737
Synthesis of 3-Tetrasubstituted Oxindoles by Using a Chiral Calcium Catalyst
0738
Enantioselective Copper-Catalyzed Synthesis of Dispiropyrrolidines
0739
Copper-Catalyzed Synthesis of CF3-Substituted Oxazolines
0740
Asymmetric Mannich-Type Reaction of Ketimines and Aminoacetonitriles
0741
Formylation of Allylic Carbonates with Formaldehyde N,N-Dialkylhydrazones
0742
Asymmetric Transfer Hydrogenation by Means of Nickel Catalysis
0743
Diastereoselective Synthesis of cis-β-Fluorocyclopropane Carboxylates
0744
Catalytic Synthesis of Vinylcyclopropanes by Intramolecular Cyclopropanation
0745
Ring Enlargement of Alkynyl Donor–Acceptor Cyclopropanes
0746
Palladium-Catalyzed Dynamic Kinetic Asymmetric Spiroannulation

Metal-Mediated Synthesis

z747
All PDFs of this category
0747
Rhodium-Catalyzed Asymmetric Cyclopropylation
0748
Gallium-Promoted Halocyclization
0749
Cobalt-Catalyzed Hydroboration of Alkynes
0750
Synthesis of Fluoren-9-ones via Carbonylative C–C Bond Formation
0751
Asymmetric Addition of Arylboronic Acids to Nitrostyrenes
0752
1,4-Hydroboration of Pyridines
0753
Synthesis of Vinyl Boronates
0754
Iron(II)-Mediated C–N Bond Formation Towards 2-Aminothiazoles
0755
Asymetric Nickel-Catalyzed Synthesis of Azetidines and Aziridines
0756
Carbolithiation of Heterosubstituted Alkynes
0757
Copper-Mediated Radical Trifluoromethylation
0758
Trifluoromethylation of Substituted Arenes and Heteroarenes
0759
Copper-Mediated Cyclization Approach to 3H- and 1H-Indoles
0760
Desymmetrization of 1,1-Diborylalkanes via Suzuki–Miyaura Cross-Coupling
0761
Grignard Addition to Aldimino Esters

Organo- and Biocatalysis

z763
All PDFs of this category
0763
Enantioselective Intramolecular Aza-Diels–Alder Reactions
0764
A Mild Neutral Silicon Lewis Acid for Hydro- and Cyanosilylations
0765
Radical Alkylation of Aldehydes via Asymmetric Photo-Organocatalysis
0766
Organocatalytic CO2 Trapping Using Alkynyl Indoles
0767
NHC-Catalyzed Benzannulation via 1,6-Addition to Conjugated Dienals
0768
Quaternary Stereocenters via NHC-Catalyzed Sulfa-Michael Addition
0769
Desymmetrizing Michael Reactions via Enol Catalysis
0770
Facile Net Cycloaddition Approach to Optically Active 1,5-Benzothiazepines

Polymer-Supported Synthesis

z771
All PDFs of this category
0771
Silica-Supported Iridium Complex Catalyst for Asymmetric Allylic Amination
0772
C–P Bond Formation Catalyzed by a Magnetic Nanoparticle-Supported Palladium Catalyst
0773
A Cellulose-Supported DNA-Based Ligand for Asymmetric Catalysis
0774
Cross-Coupling of Iodides with Nucleophiles by Using Copper Clusters
0775
Aerial Oxidation of Alcohols on a Silica–γ-Iron(III) Oxide Supported Palladium Complex
0776
Dendrimer-Encapsulated Palladium Nanoparticles for Flow Cross-Couplings
0777
Aerobic Oxidation of Alcohols with Gold–Platinum/Polystyrene Nanoparticles
0778
Deoxygenation of Carbonyls by Poly(methylhydrosiloxane) on Palladium/Carbon
0779
Gold Nanoparticle Promoted Cycloisomerization of Alkynoic Acids
0780
Huisgen Cycloaddition on a Polymer-Supported Copper Catalyst
0781
Well-Defined Adenosine Diphosphate Ribose Oligomers
0782
Double Carbonylation of Aryl Iodides with Amines on Palladium Nanoparticles
0783
Dehydrogenation of Alcohols to Carboxylic Acids on Palladium/Carbon
0784
Ruthenium-Catalyzed Oxidative Decarboxylation of Amino Acids
0785
C–O and C–X Bond-Forming Reactions with Pd(II)/MWCNT