DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 2011 · August 2011 DOI: 10.1055/s-002-22161

Synform

A65
Zanda, Matteo: SYNFORM ISSUE 2011/08

Synthesis of Natural Products and Potential Drugs

z809
All PDFs of this category
0809
Tanino, K.; Takahashi, M.; Tomata, Y.; Tokura, H.; Uehara, T.; Narabu, T.; Miyashita, M.: Synthesis of Solanoeclepin A
0810
Reddy, P. G.; Chun, B.-K.; Zhang, H.-R.; Rachakonda, S.; Ross, B. S.; Sofia, M. J.: Synthesis of PSI-352938
0811
Abrecht, S.; Adam, J.-M.; Bromberger, U.; Diodone, R.; Fettes, A.; Fischer, R.; Goeckel, V.; Hildbrand, S.; Moine, G.; Weber, M.: Synthesis of Carmegliptin
0812
Bhat, V.; Allan, K. M.; Rawal, V. H.: Synthesis of N-Methylwelwitindolinone D Isonitrile
0813
Petronijevic, F. R.; Wipf, P.: Synthesis of (±)-Cycloclavine and (±)-5-epi-Cycloclavine
0814
Nelson, H. M.; Murakami, K.; Virgil, S. C.; Stoltz, B. M.: Syntheses of Basiliolide B and C8-Epimer and Transtaganolides C and D
0815
Inuki, S.; Iwata, A.; Oishi, S.; Fujii, N.; Ohno, H.: Synthesis of (+)-Lysergic Acid, (+)-Lysergol, and (+)-Isolysergol
0816
Anson, M. S.; Graham, J. P.; Roberts, A. J.: Synthesis of GSK1842799
0817
Werner, L.; Machara, A.; Adams, D. R.; Cox, D. P.; Hudlicky, T.: Synthesis of Buprenorphine
0818
Švenda, J.; Hill, N.; Myers, A. G.: Synthesis of DC-45-A2
0819
Dong, H.; Latka, R. T.; Driver, T. G.: Synthesis of Dimebolin
0820
Clausen, D. J.; Wan, S.; Floreancig, P. E.: Synthesis of Lactodehydrothyrsiferol
0821
Huang, Q.; Richardson, P. F.; Sach, N. W.; Zhu, J.; Liu, K. K.-C.; Smith, G. L.; Bowles, D. M.: Synthesis of P13K Inhibitors
0822
Strotman, N. A.; Baxter, C. A.; Brands, K. M. J.; Cleator, E.; Krska, S. W.; Reamer, R. A.; Wallace, D. J.; Wright, T. J.: Synthesis of Suvorexant

Synthesis of Heterocycles

z823
All PDFs of this category
0823
Churchill, G. H.; Raw, S. A.; Powell, L.: Effects of Addition Rate on the Synthesis of Pyridopyrimidinediones
0824
Zheng, Z.; Tang, L.; Fan, Y.; Qi, X.; Du, Y.; Zhang-Negrerie, D.: FeBr3-Mediated Heteroannulation Route to Yield N-Amino-3-Nitrile-Indoles
0825
Zhang, G.; Luo, Y.; Wang, Y.; Zhang, L.: Gold-Catalyzed Heteroannulation Route of N-Allyl Ureas to Tricyclic Indolines
0826
Wang, F.; Cai, S.; Wang, Z.; Xi, C.: Synthesis of 2-Mercaptobenzothiazoles via Metal-Free Heteroannulation
0827
Shi, L.; Liu, X.; Zhang, H.; Jiang, Y.; Ma, D.: Cu-Mediated Heteroannulation Route to 2-Thio-Substituted Benzothiazoles
0828
Francis, S.; Kiyoi, T.; Reid, M.; Davies, K.; Laats, S.; McArthur, D.; Feilden, H.; Easson, A. M.; Kiyoi, Y.; Wishart, G.; Ray, P.: Sythesis of Serotonin Antagonists Using an Intramolecular Diels-Alder Approach
0829
Neumann, J. J.; Rakshit, S.; Dröge, T.; Würtz, S.; Glorius, F.: Heteroannulation Route to Indoles from N-Aryl Enamines via C-H Activation
0830
Calvet, G.; Livecchi, M.; Schmidt, F.: Pd-Catalyzed Heteroannulation Route to Substituted 5-Azaindoles
0831
He, W.; Li, C.; Zhang, L.: Gold-Catalyzed [2+2+1] Synthesis of 2,5-Disubstituted Oxazoles
0832
Alsabeh, P. G.; Lundgren, R. J.; Longobardi, L. E.; Stradiotto, M.: Pd-Catalyzed Synthesis of Indoles via NH3 Cross-Coupling-Alkyne Cyclization
0833
Paradise, C. L.; Sarkar, P. R.; Razzak, M.; De Brabander, J. K.: AuCl3-Catalyzed Synthesis of 5-Bromomethyl Oxazoles from Amino Acids
0834
Surmont, R.; Verniest, G.; De Schrijver, M.; Thuring, J. W.; Holte, P. ten; Deroose, F.; De Kimpe, N.: Synthesis of 3-Amino-4-fluoropyrazoles Using Selectfluor
0835
Ascic, E.; Jensen, J. F.; Nielsen, T. E.: Ruthenium-Catalyzed Synthesis of Complex Indolizidinones
0836
Samanta, R.; Antonchick, A. P.: Palladium-Catalyzed C-H Activation Route to Dibenzothiophenes
0837
Ackermann, L.; Lygin, A. V.; Hofmann, N.: De Novo Ruthenium-Catalyzed Synthesis of 2-Pyridones

Synthesis of Materials and Unnatural Products

z839
All PDFs of this category
0839
Teraoka, T.; Hiroto, S.; Shinokubo, H.: Iridium-Catalyzed Direct Tetraborylation of Perylene Bisimides
0840
Fischer, G. M.; Daltrozzo, E.; Zumbusch, A.: Selective NIR-Absorbing Dyes
0841
Muschelknautz, C.; Frank, W.; Müller, T. J. J.: Merocyanines Made Easy
0842
Silvestri, F.; Jordan, M.; Howes, K.; Kivala, M.; Rivera-Fuentes, P.; Boudon, C.; Gisselbrecht, J.-P.; Schweizer, W. B.; Seiler, P.; Chiu, M.; Diederich, F.: Multiple CA-CR Reactions
0843
Varotto, A.; Treat, N. D.; Jo, J.; Shuttle, C. G.; Batara, N. A.; Brunetti, F. G.; Seo, J. H.; Chabinyc, M. L.; Hawker, C. J.; Heeger, A. J.; Wudl, F.: Tuning the Electronic Properties of Fullerene
0844
Zhao, Z.; Ma, X.; Zhang, A.; Song, N.: Numbers of Substitutions to Order: 2, 4, 5, 6, or Polymer
0845
Al-Afyouni, M. H.; Huang, T. A.; Hung-Low, F.; Bradley, C. A.: A Radically Different Approach to the Synthesis of Bifluorenes
0846
Zhang, J.; Sarrafpour, S.; Pawle, R. H.; III, S. W. Thomas: Conjugated Polymers for ¹O2 Sensing
0847
Maeda, K.; Mochizuki, H.; Osato, K.; Yashima, E.: It’s all about the Twist!
0848
Zhang, Y.; Matsuo, Y.; Li, C.-Z.; Tanaka, H.; Nakamura, E.: Methanofullerenes for Improved OPVs
0849
Karlsson, K. M.; Jiang, X.; Eriksson, S. K.; Gabrielsson, E.; Rensmo, H.; Hagfeldt, A.; Sun, L.: Phenoxazine Dyes
0850
Hirose, K.; Yachi, Y.; Tobe, Y.: Chirality Sensor Based on Non-Linear Transmittance Change
0851
Jiao, C.; Zhu, L.; Wu, J.: Porphyrin Stability and Absorption Red Shift via BODIPY Extension

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z853
All PDFs of this category
0853
Zhou, S.; Fleischer, S.; Junge, K.; Beller, M.: Cooperative Transition-Metal and Chiral Brønsted Acid Catalysis
0854
Wu, Q.-F.; Liu, W.-B.; Zhuo, C.-X.; Rong, Z.-Q.; Ye, K.-Y.; You, S.-L.: Iridium-Catalyzed Enantioselective Allylic Dearomatization of Phenols
0855
Pérez, M.; Fañanás-Mastral, M.; Bos, P. H.; Rudolph, A.; Harutyunyan, S. R.; Feringa, B. L.: Copper-Catalyzed Asymmetric Allylic Alkylation with Organolithium Reagents
0856
Kuwano, R.; Kameyama, N.; Ikeda, R.: Asymmetric Hydrogenation of Heterocyclic Compounds
0857
White, J. D.; Shaw, S.: New Scaffold for Asymmetric Catalysis via Salen-Metal Complexes
0858
Thaler, T.; Guo, L.-N.; Steib, A. K.; Raducan, M.; Karaghiosoff, K.; Mayer, P.; Knochel, P.: Sulfoxide-Alkene Hybrid Ligands in Rhodium-Catalyzed 1,4-Addition
0859
Zhu, S.-F.; Qiao, X.-C.; Zhang, Y.-Z.; Wang, L.-X.; Zhou, Q.-L.: Palladium-Catalyzed Umpolung Allylation of Aldehydes
0860
Yoshida, A.; Hattori, G.; Miyake, Y.; Nishibayashi, Y.: Enantioselective Propargylic Amination of Nonaromatic Propargylic Esters
0861
Lu, G.; Yoshino, T.; Morimoto, H.; Matsunaga, S.; Shibasaki, M.: Stereodivergent Asymmetric Reactions of α-Isothiocyanato Ester with Ketimines
0862
Larson, S. E.; Li, G. L.; Rowland, G. B.; Junge, D.; Huang, R. C.; Woodcock, H. L.; Antilla, J. C.: Asymmetric Aza-Darzens Reaction Catalyzed by Mg Phosphate Salt
0863
Rauniyar, V.; Wang, Z. J.; Burks, H. E.; Toste, F. D.: Synthesis of Chiral Furans by a Copper-Catalyzed Domino Process
0864
Roggen, M.; Carreira, E. M.: Enantioselective Allylic Etherification
0865
Nishikawa, Y.; Yamamoto, H.: Asymmetric Epoxidations of Disubstituted Enones with Iron
0866
Kurono, N.; Nii, N.; Sakaguchi, Y.; Uemura, M.; Ohkuma, T.: Asymmetric Hydrocyanation of α,β-Unsaturated Ketones
0867
Huang, G.; Yang, J.; Zhang, X.: Asymmetric Alkynylation of α-Trifluoromethyl Ketoimine Esters
0868
Yu, C.-B.; Gao, K.; Wang, D.-S.; Shi, L.; Zhou, Y.-G.: Palladium-Catalyzed Asymmetric Hydrogenation of Enesulfonamides
0869
Takatsu, K.; Shintani, R.; Hayashi, T.: Copper-Catalyzed 1,4-Addition of Organo-boronates to Alkylidene Cyanoacetates
0870
Cao, Z.; Liu, Y.; Liu, Z.; Feng, X.; Zhuang, M.; Du, H.: Pd-Catalyzed Asymmetric Allylic Alkylation of Indoles and Pyrroles
0871
Trost, B. M.; Bringley, D. A.; Silverman, S. M.: Synthesis of Chiral Tetrahydrofurans by a Palladium-Catalyzed Cycloaddition
0872
Bentley, S. A.; Davies, S. G.; Lee, J. A.; Roberts, P. M.; Thomson, J. E.: Diastereoselective 1,4-Addition of Asymmeric Lithium Amides
0873
Li, J.; Chen, G.; Wang, Z.; Zhang, R.; Zhang, X.; Ding, K.: New Ligand for Zinc-Catalyzed Hydroxylation of β-Keto Esters and 1,3-Diesters
0874
Bolte, B.; Gagosz, F.: Gold- and Acid-Catalyzed Synthesis of Tetrahydropyrans and Tetrahydrofurans
0875
Kim, H.; Ho, S.; Leighton, J.: Highly Selective Scandium-Catalyzed Aldehyde Crotylation
0876
Kanbayashi, N.; Onitsuka, K.: Ruthenium-Catalyzed Regio- and Enantio-selective Allylic Substitution with Water
0877
Kang, Y. K.; Suh, K. H.; Kim, D. Y.: Friedel-Crafts Alkylation of Indoles Catalyzed by a Chiral Palladium Complex
0878
Yao, M.; Lu, C.-D.: Asymmetric Domino Synthesis of N-Sulfonylamidines
0879
Gulías, M.; Collado, A.; Trillo, B.; López, F.; Oñate, E.; Esteruelas, M. A.; Mascareñas, J. L.: Diastereoselective Ruthenium-Catalyzed [2+2] Cycloadditions of Allenenes
0880
Yamashita, Y.; Imaizumi, T.; Kobayashi, S.: Silver-Catalyzed Asymmetric [3+2] Cycloaddition of Amino Esters to Olefins
0881
Bonollo, S.; Lanari, D.; Pizzo, F.; Vaccaro, L.: Scandium-Catalyzed Asymmetric Sulfa-Michael Addition in Water
0882
Lang, F.; Chen, G.; Li, L.; Xing, J.; Han, F.; Cun, L.; Liao, J.: Asymmetric Addition of Arylboronic Acids to 2-Nitrostyrenes

Metal-Mediated Synthesis

z883
All PDFs of this category
0883
Stanton, G. R.; Koz, G.; Walsh, P. J.: Highly Diastereoselective Additions to α-Silyloxy Ketones
0884
Lamas, M.-C.; Studer, A.: Radical Alkylphosphanylation of Olefins
0885
Lu, Z.; Wilsily, A.; Fu, G. C.: Amine-Directed Alkyl-Alkyl Suzuki Reactions
0886
Velcicky, J.; Soicke, A.; Steiner, R.; Schmalz, H.-G.: Palladium-Catalyzed Cyanomethylation of Aryl Halides
0887
Berhal, F.; Esseiva, O.; Martin, C.-H.; Tone, H.; Genêt, J.-P.; Ayad, T.; Ratovelomanana-Vidal, V.: Room-Temperature Rh-Catalyzed Asymmetric Conjugate Addition
0888
Hodgson, D. M.; Talbot, E. P. A.; Clark, B. P.: Synthesis of β-(Hydroxymethylaryl/alkyl)-α-methylene-γ-butyrolactones
0889
Havlik, S. E.; Simmons, J. M.; Winton, V. J.; Johnson, J. B.: Ni-Mediated Decarbonylative Cross-Coupling of Diorganozinc Reagents
0890
Sun, A. D.; Love, J. A.: Nickel-Catalyzed Cross-Coupling of Polyfluoroarenes with Arylboronic Acids
0891
Manabe, K.; Ohba, M.; Matsushima, Y.: Pd-Catalyzed Chemoselective Cross-Couplings for Oligoarene Synthesis
0892
Chan, D. G.; Winternheimer, D. J.; Merlic, C. A.: Silyl Enol Ethers via Copper(II)-Catalyzed C-O Bond Formation
0893
Xie, L.-G.; Wang, S.-X.: Ni-Catalyzed Cross-Coupling of Aryltrimethylammonium Iodides
0894
Gottumukkala, A. L.; Teichert, J. F.; Heijnen, D.; Eisink, N.; van Dijk, S.; Ferrer, C.; van den Hoogenband, A.; Minnaard, A. J.: Novel Base-Free Oxidative Heck Reaction
0895
Ihara, H.; Koyanagi, M.; Suginome, M.: Anthranilamide as Protecting and Directing Group for Arylboronic Acids
0896
Ilies, L.; Asako, S.; Nakamura, E.: Iron-Catalyzed Stereospecific C-H Bond Activation
0897
Joshi-Pangu, A.; Wang, C.-Y.; Biscoe, M. R.: Ni-Catalyzed Cross-Couplings of Tertiary Alkyl Grignards and Aryl Bromides

Organo- and Biocatalysis

z899
All PDFs of this category
0899
Sakakura, A.; Sakuma, M.; Ishihara, K.: Chiral Lewis Base Assisted Brønsted Acids
0900
Deiana, L.; Dziedzic, P.; Zhao, G.-L.; Vesely, J.; Ibrahem, I.; Rios, R.; Sun, J.; Córdova, A.: Catalytic Asymmetric Aziridination of α,β-Unsaturated Aldehydes
0901
Nicolaou, K. C.; Simmons, N. L.; Ying, Y.; Heretsch, P. M.; Chen, J. S.: Catalytic Asymmetric Dichlorination of Allylic Alcohols
0902
Bugaut, X.; Liu, F.; Glorius, F.: Intermolecular Hydroacylation of Cyclopropenes
0903
Leon, R.; Jawalekar, A.; Redert, T.; Gaunt, M. J.: Assembly of Complex Molecules via Dearomatization-Catalytic Desymmetrization
0904
Duque, M. del Mar Sanchez; Baslé, O.; Isambert, N.; Gaudel-Siri, A.; Génisson, Y.; Plaquevent, J.-C.; Rodriguez, J.; Constantieux, T.: Asymmetric Michael Addition of α-Substituted β-Keto Amides
0905
Huang, first article: L.; Wulff, W. D.; Hashimoto, second article: T.; Nakatsu, H.; Yamamoto, K.; Maruoka, K.: Catalytic Asymmetric Synthesis of Trisub-stituted Aziridines
0906
Moccia, M.; Fini, F.; Scagnetti, M.; Adamo, M. F. A.: Catalytic Asymmetric Conjugate Addition of NaHSO3 to Chalcones
0907
Pham, P. V.; Ashton, K.; MacMillan, D. W. C.: Intramolecular Asymmetric α-Allylation of Aldehydes via SOMO Umpolung
0908
Liu, L.; Zhang, S.; Xue, F.; Lou, G.; Zhang, H.; Ma, S.; Duan, W.; Wang, W.: Catalytic Asymmetric Henry Reaction of Isatins
0909
Xie, Y.; Zhao, Y.; Qian, B.; Yang, L.; Xia, C.; Huang, H.: Chiral Brønsted Acid Catalyzed N-Functional-ization of Indoles

Polymer-Supported Synthesis

z911
All PDFs of this category
0911
Riva, E.; Rencurosi, A.; Gagliardi, S.; Passarella, D.; Martinelli, M.: Flow Synthesis of Alkaloids
0912
Shi, J. Y.; Wang, C. A.; Li, Z. J.; Wang, Q.; Zhang, Y.; Wang, W.: A Mesoporous Organosilica-Supported Organocatalyst
0913
Chen, Z.; Guan, Z.; Li, M.; Yang, Q.; Li, C.: A Platinum Nanocatalyst Confined within Carbon Nanotubes
0914
Karimi, B.; Badreh, E.: Aerobic Oxidation of Alcohols Using IL@SBA-15-TEMPO
0915
Karimi, B.; Farhangi, E.: Aerobic Oxidation of Alcohols with Fe3O4/SiO2-Supported TEMPO in Water
0916
Fujita, K.; Umeki, S.; Yamazaki, M.; Ainoya, T.; Tsuchimoto, T.; Yasuda, H.: Magnetic Nanoparticle Supported Osmium for Olefin Dihydroxylation
0917
Dhakshinamoorthy, A.; Alvaro, M.; Garcia, H.: NHPI/Fe(BTC)-Catalyzed Aerobic Oxidation of Alkanes
0918
He, W.; Zhang, F.; Li, H.: C-C Bond-Forming Reactions in Water with Pd-PPh2-MSN
0919
Qu, X.; Sun, P.; Li, T.; Mao, J.: Mizoroki-Heck Reaction of Hypervalent Iodine with Pd Nanocatalyst
0920
Kumar, V. K. R.; Gopidas, K. R.: Chemoselective Hydrogenation with Pd Nanoparticle Cored Dendrimer
0921
Tanaka, S.; Kaneko, T.; Asao, N.; Yamamoto, Y.; Chen, M.; Zhang, W.; Inoue, A.: Suzuki-Miyaura Coupling with Nanoporous Metallic Glass Pd
0922
Thummanagoti, S.; Yellol, G. S.; Sun, C.-M.: Ionic Liquid Supported Synthesis of Benzimidazolones
0923
Jeong, K. S.; Go, Y. B.; Shin, S. M.; Lee, S. J.; Kim, J.; Yaghi, O. M.; Jeong, N.: Chiral MOF for Carbonyl-Ene and Hetero-Diels-Alder Reactions
0924
Peng, Q.; Zhang, Y.; Shi, F.; Deng, Y.: Reductive N-Alkylation of Nitroarenes with Alcohols Catalyzed by Au/Fe2O3