DOI: 10.1055/s-00000131

Synfacts

Issue 11 · Volume 2010 · November 2010 DOI: 10.1055/s-002-21416

Synform

A86
Zanda, Matteo: SYNFORM ISSUE 2010/10

Synthesis of Natural Products and Potential Drugs

z1211
All PDFs of this category
1211
Voight, E. A.; Yin, H.; Downing, S. V.; Calad, S. A.; Matsuhashi, H.; Giordano, I.; Hennessy, A. J.; Goodman, R. M.; Wood, J. L.: Synthesis of GSK966587
1212
Magnus, N. A.; Ley, C. P.; Pollock, P. M.; Wepsiec, J. P.: Synthesis of a Glycogen Synthase Kinase-3 Inhibitor
1213
Hickmann, V.; Alcarazo, M.; Fürstner, A.: Synthesis of the Ecklonialactones
1214
Espejo, V. R.; Rainier, J. D.: Synthesis of Kapakahine E
1215
Diethelm, S.; Schindler, C. S.; Carreira, E. M.: Synthesis of Microcin SF608
1216
Zhao, Y.-M.; Gu, P.; Tu, Y.-Q.; Zhang, H.-J.; Zhang, Q.-W.; Fan, C.-A.: Synthesis of Hexahydroapoerysopine
1217
Medeiros, M. R.; Wood, J. L.: Synthesis of (+)-Norsecurinine
1218
Zou, Y.; Deiters, A.: Synthesis of Cryptoacetalide
1219
Wu, J.; Panek, J. S.: Synthesis of (-)-Virginiamycin M2
1220
O’Neill et al., P. M.: Synthesis of RKA 182

Synthesis of Heterocycles

z1221
All PDFs of this category
1221
Spergel, S. H.; Okoro, D. R.; Pitts, W.: Palladium-Catalyzed α-Heteroarylation Route to 4-, 5-, 6- and 7-Azaindoles
1222
Yan, R.-L.; Luo, J.; Wang, C.-X.; Ma, C.-W.; Huang, G.-S.; Liang, Y.-M.: Copper-Catalyzed Synthesis of Poly-substituted Pyrroles from Enamino Ketones
1223
Wang, X.; Lu, Y.; Dai, H.-X.; Yu, J.-Q.: Palladium(II)-Catalyzed Heteroannulation Route to Dihydrobenzofurans
1224
Misra, N. C.; Ila, H.: 4-Bis(methylthio)methylene-2-phenyloxazol-5-one: Template for Oxazoles
1225
Kobatake, T.; Fujino, D.; Yoshida, S.; Yorimitsu, H.; Oshima, K.: Synthesis of Trifluoromethylbenzofurans by Extended Pummerer Reaction
1226
Pohjakallio, A.; Pihko, P. M.; Laitinen, U. M.: Synthesis of 2-Isoxazolines via Conjugate Additions
1227
Mai, D. N.; Wolfe, J. P.: Synthesis of Chiral Pyrrolidines by Palladium-Catalyzed Carboamination
1228
Zhang, J.; Senthilkumar, M.; Ghosh, S. C.; Hong, S. H.: Ruthenium-Catalyzed Synthesis of Cyclic Imides
1229
Lin, M.; Hao, L.; Ma, R.-d.; Zhan, Z.-p.: Indium-Mediated Multicomponent Synthesis of Pyrroles
1230
Liu, F.; Qian, D.; Li, L.; Zhao, X.; Zhang, J.: Gold(I)-Catalyzed Synthesis of Furo[3,4-d]-[1,2]oxazines
1231
Zhang, Q.; Fang, T.; Tong, X.: Triphenylphosphine-Catalyzed Synthesis of Dihydropyridines and Pyrans
1232
Jana, S.; Clements, M. D.; Sharp, B. K.; Zheng, N.: Synthesis of 2,3-Disubstituted Indoles by Iron(II)-Catalyzed Aromatic C-H Amination
1233
Crossley, J. A.; Browne, D. L.: Cycloaddition Route to 4-Iodoisoxazoles
1234
Chen, W.; Hu, M.; Wu, J.; Zou, H.; Yu, Y.: Synthesis of Pyrrolo[1,2-a]pyrazines from Vinyl Azides
1235
Kaïm, L. El; Grimaud, L.; Ronsseray, C.: One-Pot Modified Japp-Klingeman-Fischer Indole Synthesis

Synthesis of Materials and Unnatural Products

z1237
All PDFs of this category
1237
Criado, A.; Peña, D.; Cobas, A.; Guitián, E.: Cascade Cycloadditions for the Synthesis of Perylenes
1238
Konishi, A.; Hirao, Y.; Nakano, M.; Shimizu, A.; Botek, E.; Champagne, B.; Shiomi, D.; Sato, K.; Takui, T.; Matsumoto, K.; Kurata, H.; Kubo, T.: A Singlet Biradical Polycyclic Aromatic Hydrocarbon
1239
Li, S.; Zheng, B.; Chen, J.; Dong, S.; Ma, Z.; Huang, F.; Gibson, H. W.: Mechanically Interlocked Polymers
1240
Zhang, L.; Ang, G. Y.; Chiba, S.: Phenanthridine Derivatives Made Easy
1241
Lepeltier, M.; Lukoyanova, O.; Jacobson, A.; Jeeva, S.; Perepichka, D. F.: Interplay of Heteroatoms
1242
Wu, Y.-L.; Bureš, F.; Jarowski, P. D.; Schweizer, W. B.; Boudon, C.; Gisselbrecht, [nl]J.-P.; Diederich, F.: A Proof of Concept for Proaromaticity
1243
Bura, T.; Retailleau, P.; Ziessel, R.: Panchromatic Fluorescent Materials
1244
Fort, E. H.; Scott, L. T.: Acetylene Equivalent for Bay Region Diels-Alder Cycloaddition
1245
Zhang, X.; Li, J.; Qu, H.; Chi, C.; Wu, J.: Conjugate Additions When You Least Expect Them
1246
Hierold, J.; Gray-Weale, A.; Lupton, D. W.: Swollen-up Molecules by Fragmentation
1247
Jin, Y.; Voss, B. A.; Noble, R. D.; Zhang, W.: Gas Profiling Rampant: CO2 Detained
1248
Liu, W.; Huang, W.; Pink, M.; Lee, D.: Metal-Containing Conducting Polymers
1249
Cambrea, L. R.; Davis, M. C.; Groshens, T. J.; Guenthner, A. J.; Lamison, K. R.; Mabry, J. M.: Novel Adhesive via Cyclotrimerization
1250
Peart, P. A.; Tovar, J. D.: Inclusion of Cyclopropenium in a Conductive Polymer
1251
Qiu, Z.; Wang, S. R.; Xie, Z.: Rings on Carboranes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1253
All PDFs of this category
1253
Chen, I.-H.; Kanai, M.; Shibasaki, M.: Enantioselective Copper-Catalyzed Boration
1254
Guijarro, D.; Pablo, Ó.; Yus, M.: Ruthenium-Catalyzed Asymmetric Transfer Hydrogenation to Chiral Primary Amines
1255
Zhang, P.; Brozek, L. A.; Morken, J. P.: Pd-Catalyzed Asymmetric Cross-Coupling of Allyl Carbonates and Allyl Boronates
1256
Shintani, R.; Soh, Y.-T.; Hayashi, T.: Asymmetric Synthesis of 1-(Diarylmethyl)-pyrazolidin-3-ones
1257
Tsuji, H.; Ueda, Y.; Ilies, L.; Nakamura, E.: Synthesis of Tetrasubstituted Alkenes through a Stannyllithiation
1258
Shintani, R.; Takatsu, K.; Hayashi, T.: Asymmetric Addition to Isatins
1259
Roggen, M.; Carreira, E. M.: Stereospecific Substitution of Allylic Alcohols
1260
Kirchberg, S.; Fröhlich, R.; Studer, A.: Palladium-Catalyzed Oxidative Carbofunctionalization of Indenes
1261
Cai, Y.; Liu, X.; Hui, Y.; Jiang, J.; Wang, W.; Chen, W.; Lin, L.; Feng, X.: Catalytic Asymmetric Bromoamination of Chalcones
1262
Arai, N.; Akashi, M.; Sugizaki, S.; Ooka, H.; Inoue, T.; Ohkuma, T.: Ruthenium-Catalyzed Asymmetric Hydrogenation of Bicyclic Ketones
1263
Takenaka, K.; Mohanta, S. C.; Patil, M. L.; Rao, C. V. L.; Takizawa, S.; Suzuki, T.; Sasai, H.: Asymmetric Wacker-Type Cyclization Catalyzed by Pd-SPRIX
1264
Sakai, Y.; Mitote, J.; Matsumoto, K.; Katsuki, T.: Vanadium-Catalyzed Asymmetric Synthesis of Cyanohydrins
1265
Hashimoto, T.; Naganawa, Y.; Maruoka, K.: Desymmetrizing Asymmetric Ring Expansion of Cyclohexanones
1266
Wang, G.; Zhao, J.; Zhou, Y.; Wang, B.; Qu, J.: Asymmetric Vinylogous Aldol Reaction Cata-lyzed by a Combined Acid Titanium Complex
1267
Ito, M.; Kobayashi, C.; Himizu, A.; Ikariya, T.: Ruthenium-Catalyzed Hydrogenative Desymmetrization of Bicyclic Amides
1268
Hatano, M.; Horibe, T.; Ishihara, K.: Mg(II)-BINOLate Salt Catalyzed Asymmetric Mannich-Type Reaction
1269
Zhong, C.; Kunii, S.; Kosaka, Y.; Sawamura, M.; Ito, H.: Novel Asymmetric Synthesis of Substituted Cyclopropylboronates
1270
Geherty, M. E.; Dura, R. D.; Nelson, S. G.: Ruthenium-Catalyzed Asymmetric Claisen Rearrangement
1271
Nishimura, T.; Sawano, T.; Tokuji, S.; Hayashi, T.: Asymmetric Alkynylation of Nitroalkenes
1272
O’Brien, J. M.; Lee, K.-s.; Hoveyda, A. H.: NHC Copper Catalyzed Enantioselective Conjugate Addition
1273
Han, S. B.; Gao, X.; Krische, M. J.: anti-Diastereo- and Enantioselective Carbonyl (Trimethylsilyl)allylation
1274
Kang, S.; Han, J.; Lee, E. S.; Choi, E. B.; Lee, H.-K.: Enantioselective Synthesis of Cyclic Sulfamidates
1275
Wang, Z.-Q.; Feng, C.-G.; Zhang, S.-S.; Xu, M.-H.; Lin, G.-Q.: Asymmetric Conjugate Addition of Arylboronic Acids to Nitroolefins
1276
Zhou, C.-Y.; Zhu, S.-F.; Wang, L.-X.; Zhou, Q.-L.: Enantioselective Reductive Coupling of Alkynes and Imines
1277
Lundin, P. M.; Fu, G. C.: Asymmetric Suzuki Cross-Coupling of Secondary Alkyl Electrophiles
1278
Chen, Z.; Li, J.; Jiang, H.; Zhu, S.; Li, Y.; Qi, C.: Regio- and Stereoselective Difunctionalization of Alkynes
1279
Guo, L.-N.; Gao, H.; Mayer, P.; Knochel, P.: Preparation and Diastereoselective Additions of Organoaluminum Reagents
1280
Nolin, K. A.; Ahn, R. W.; Kobayashi, Y.; Kennedy-Smith, J. J.; Toste, F. D.: Enantioselective Reduction Catalyzed by (CN-Box)ReV-Oxo Complexes
1281
Guzman-Martinez, A.; Hoveyda, A. H.: Enantioselective Synthesis of Allylboronates by NHC Copper Catalyzed Substitution
1282
Li, D.; Tanaka, T.; Ohmiya, H.; Sawamura, M.: α-Aryl Allylsilanes from Palladium-Catalyzed Allyl-Aryl Coupling

Metal-Mediated Synthesis

z1283
All PDFs of this category
1283
Huang, D. S.; Hartwig, J. F.: Pd-Catalyzed γ-Arylation of α,β-Unsaturated Esters from Silyl Ketene Acetals
1284
Maimone, T. J.; Buchwald, S. L.: O-Arylhydroxylamines and Benzofurans via O-Arylation of Ethyl Acetohydroximate
1285
Tang, W.; Capacci, A. G.; Wei, X.; Li, W.; White, A.; Patel, N. D.; Savoie, J.; Gao, J. J.; Rodriguez, S.; Qu, B.; Haddad, N.; Lu, B. Z.; Krishnamurthy, D.; Yee, N. K.; Senanayake, C. H.: A Novel General Phosphine Ligand for Suzuki-Miyaura Cross-Coupling
1286
Liao, L.; Sigman, M. S.: Palladium-Catalyzed Oxidative Hydro-arylation of 1,3-Dienes with Boronic Esters
1287
Kawamura, S.; Ishizuka, K.; Takaya, H.; Nakamura, M.: A New Iron-Catalyzed Aluminum Variant of the Negishi Coupling
1288
Wang, B.; Wang, S.; Li, P.; Wang, L.: Iron-Catalyzed Addition of Acid Chlorides to Alkynes
1289
McNeill, E.; Bois, J. Du: Ruthenium-Catalyzed Csp³-H Oxidation of Tertiary Alkanes
1290
Hatakeyama, T.; Hashimoto, T.; Kondo, Y.; Fujiwara, Y.; Seike, H.; Takaya, H.; Tamada, Y.; Ono, T.; Nakamura, M.: Iron-Catalyzed Suzuki-Miyaura Coupling Between Arylborates and Alkyl Halides
1291
Sequeira, F. C.; Turnpenny, B. W.; Chemler, S. R.: Copper-Mediated Intermolecular Alkene Diamination
1292
Shimizu, M.; Kawanishi, M.; Mizota, I.; Hachiya, I.: N-Allylidene-1,1-diphenylethanamine as Acrolein Synthon
1293
Prinsell, M. R.; Everson, D. A.; Weix, D. J.: Nickel-Catalyzed Reductive Dimerization of Alkyl Halides
1294
Kim, H.; Lee, K.; Kim, S.; Lee, P. H.: Preparation of Indolizines via Palladium-Catalyzed Cycloisomerization
1295
D’Souza, D. M.; Muschelknautz, C.; Rominger, F.; Müller, T. J. J.: Luminescent Push-Pull Indolones in a One-Pot Approach
1296
Gao, F.; Hoveyda, A. H.: α-Selective Nickel-Catalyzed Hydroalumination of Terminal Alkynes
1297
Begouin, J.-M.; Rivard, M.; Gosmini, C.: Cobalt-Catalyzed C-SMe Bond Activation of Heteroaromatic Thioethers

Organo- and Biocatalysis

z1299
All PDFs of this category
1299
Bencivenni, G.; Galzerano, P.; Mazzanti, A.; Bartoli, G.; Melchiorre, P.: Organocatalytic Vinylogous Michael Additions
1300
Uraguchi, D.; Kinoshita, N.; Ooi, T.: Catalytic Asymmetric Protonation of Ketene Disilyl Acetals
1301
Dai, L.; Wang, S.-X.; Chen, F.-E.: Cinchona Alkaloid Squaramide Catalyzed Sulfa-Michael Addition
1302
Qiao, Z.; Shafiq, Z.; Liu, L.; Yu, Z.-B.; Zheng, Q.-Y.; Wang, D.; Chen, Y.-J.: Unexpected δ-Substitution Products
1303
Sohtome, Y.; Shin, B.; Horitsugi, N.; Takagi, R.; Noguchi, K.; Nagasawa, K.: Entropy-Controlled Asymmetric Catalysis
1304
Shiina, I.; Nakata, K.; Ono, K.; Onda, Y.-s.; Itagaki, M.: Highly Efficient Kinetic Resolution of Racemic Carboxylic Acids
1305
Zhu, Q.; Lu, Y.: Bi- and Trifunctional Catalysts for Oxindoles with Quaternary Stereocenters
1306
Mahé, O.; Dez, I.; Levacher, V.; Brière, J.-F.: Phase-Transfer Catalysis in the Asymmetric Synthesis of Pyrazolines
1307
Hashimoto, T.; Kimura, H.; Maruoka, K.: Axially Chiral Dicarboxylic Acid Catalyzed Formal Alkenylations of Imines
1308
Kang, Y. K.; Kim, S. M.; Kim, D. Y.: Organocatalytic Intramolecular 1,5-Hydride Transfer-Ring-Closure Cascade
1309
Uraguchi, D.; Nakamura, S.; Ooi, T.: Asymmetric Direct Henry Reaction of Ynals Catalyzed by Iminophosphorane
1310
Veitch, G. E.; Jacobsen, E. N.: Highly Enantioselective Iodolactonization

Polymer-Supported Synthesis

z1311
All PDFs of this category
1311
Proulx, C.; Lubell, W. D.: 1,3-Dipolar Cycloaddition of Aza-Propargylglycine with Aryl Azides
1312
Liu, Z.; Nefzi, A.: Synthesis of N-Substituted Pyrrolidinone Derivatives via the Ugi Reaction
1313
Wegner, J.; Ceylan, S.; Friese, C.; Kirschning, A.: Facile Oxidations under Flow Conditions in Fixed-Bed Reactors
1314
Corma, A.; Iglesias, M.; Xamena, F. X. Llabrés i; Sánchez, F.: Cyclopropanation of Alkenes with [Cu3(BTC)2] and IRMOF-3-SI-Au
1315
Singh, D.; Deobald, A. M.; Camargo, L. R. S.; Tabarelli, G.; Rodrigues, O. E. D.; Braga, A. L.: Synthesis of Diselenides or Ditellurides with CuO Nanopowder
1316
Hashimoto, N.; Takahashi, Y.; Hara, T.; Shimazu, S.; Mitsudome, T.; Mizugaki, T.; Jitsukawa, K.; Kaneda, K.: Hydrogenation of Quinolines Using Pd0 Nanoparticles on Hydroxyapatite
1317
Mejías, N.; Pleixats, R.; Shafir, A.; Medio-Simón, M.; Asensio, G.: Water-Soluble Palladium Nanoparticles for the Suzuki Cross-Coupling
1318
Haldar, S.; Koner, S.: Hydroarylation of Styrenes with Phenols Catalyzed by Fe-Al-MCM-41
1319
Ottesen, L. K.; Jaroszewski, J. W.; Franzyk, H.: Ring Opening of a Resin-Bound Chiral Aziridine with Phenols
1320
Rajpara, V.; Banerjee, S.; Sereda, G.: Alkylation of Arenes with Fe3O4 Nanoparticles on Oxidized Graphite
1321
Joucla, L.; Cusati, G.; Pinel, C.; Djakovitch, L.: Sequential Suzuki-Miyaura/Heck Reaction Using Pd/SiO2
1322
Xiang, Y.; Meng, Q.; Li, X.; Wang, J.: Imine Formation via Hydrogen-Transfer Nitroarene Reduction
1323
Hirai, Y.; Uozumi, Y.: Buchwald-Hartwig Reaction with Amphiphilic Resin-Supported Palladium
1324
Lei, M.; Ma, L.; Hu, L.: Synthesis of β-Amido Ketones with VB1-Al2O3

Addenda and Errata

1325
New Ligand for Asymmetric Arylation of Aldehydes
1326
Diastereoselective Hydrogenation of Imines
e1
Synform