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Synthesis 2005(1): 25-27
DOI: 10.1055/s-2004-834935
DOI: 10.1055/s-2004-834935
SHORTPAPER
© Georg Thieme Verlag Stuttgart · New York
An Expeditious Synthesis of 2,4-Disubstituted 2-Imidazolin-5-ones
Further Information
Received
19 July 2004
Publication Date:
03 December 2004 (online)
Publication History
Publication Date:
03 December 2004 (online)
Abstract
2-Thiomethylimidazolin-5-one undergoes efficient palladium-catalyzed cross-coupling with boronic acids and organostannanes mediated by copper(I) thiophene-2-carboxylate.
Key words
imidazolones - palladium - boronic acids - organostannanes - copper(I) thiophene carboxylate
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