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Category: Synthesis of Heterocycles

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Issue 05/2024

Spiro-Substituted Dioxetane-Based Chemical Probes with Enhanced Detection and Sensitivity Limits
Palladium-Mediated Diastereoselective Functionalization of Cyrene
Mild Nitrogen-to-Carbon Transmutation of Azaarene N-Oxides
Using Metallaphotoredox Towards the Synthesis of Aryl Nitriles and α-Aryl Nitriles
Access to and Physicochemical Analysis of Fluorinated Saturated Bicyclic Amine Building Blocks
Synthesis of Quinolones from Propargylic Chlorides and Amines
Electrochemical Formal C–H/C–H Regioselective Coupling of Heteroarenes
Copper-Catalyzed Synthesis of N-Heterocyclic Bicycles
Skeletal Editing of Pyridines to Afford 1,2-Diazepines
Electrochemical Cross-Dehydrogenative of Amides and Heteroarenes
Tether-Controlled Regiochemical Access to Complex Polyheterocyclic Molecular Architectures
All PDFs of this category

Issue 04/2024

Efficient Syntheses of Complex Benzoxaboracycles
Late-Stage Selective Functionalization for Bioactive Indole Derivatives
1,3-Dipolar Cycloaddition Approach to Functionalized Tetrahydropyridines
Palladium-Mediated Synthesis of Functionalized Unsaturated Dicarbonyl Compounds
Chemodivergent Cyclization of Propargylamines to Enable Indole and Quinoline Heterocycles
Synthesis of Amides Using Triazine Esters as Stable Acylation Reagents
Selective Synthesis of exo- and endo-3-Azabicyclo[3.1.0]hexane-6-carboxylates
Synthesis of Fused Imidazoles via Iron-Catalyzed C(sp3)–H Amination–Cyclization
Skeletal Editing of Indazoles via Silver-Catalyzed Carbene Insertion
Copper-Catalyzed Synthesis of 4,5,6-Trisubstituted Pyrimidines
Diastereoselective Scandium-Catalyzed Route to Difluorinated Pyrrolidines
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Issue 03/2024

Strained exo-Methylene Heterocycles as Dipolarophiles: Synthesis of Unexplored Spiroisoxazolines
Multicomponent Synthesis of Tetrahydroisoquinolines
Synthesis of 2-Alkylmethyl Pyrroline Derivatives
Sc(OTf)3‑Catalyzed Cycloadditions for the Synthesis of Substituted Indolines
Gram-Scale, Modular Access to C2-Bis(Oxazoline) Ligands
Multicomponent Synthesis of Quinolines via Hydrogen-Transfer Reaction
A Highly Diastereoselective Synthesis of Sulfur-Containing Unnatural Amino Acids
Efficient, Epimerization-Free Solid-Phase Peptide Synthesis
Versatile Synthesis of Tertiary and Heterocyclic and Aromatic Amines
Practical and Efficient Access to Multifunctional BCPs
Synthesis of 2,5-Disubstituted Pyridines via Gold(I)-Catalyzed Cycloisomerization of 1-Bromoalkynes
Nitrogen Atom Insertion into Arenols in the Synthesis of Benzazepines
Palladium-Mediated Synthesis of 3-Methylindoles Under Mild Conditions
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Issue 02/2024

Heteroarene Functionalization Using Solid Gas-MOF Reagents
Ring-Opening the Door to Amination: Nitrobenzene-Derived Azepines as Key Intermediates for N-Arylation
Skeletal Editing of Indoles and Pyrroles by LiHMDS Nitrogen Insertion Reaction
Efficient Access to Novel Vinyl Indomorphan Scaffolds
One-Pot Synthesis of Disubstituted Nicotinonitriles
Copper-Catalyzed Synthesis of Pyrozles from Sydnones and Sydnomines
Photoredox/Cobalt-Catalyzed Cascade Synthesis of 2,5-Disubstituted 1,3,4-Oxadiazoles
Radical-Mediated Synthesis of Isoquinolines
Bi-Catalyzed Trifluoromethylation Using CF3SO2Cl
Intramolecular Diels–Alder Cascade to Access 6- or 7-Aza-Indazoles
Metal-Controlled Regioselective Synthesis of Imidazoles and Pyrroles from 2H-Azirines
Palladium-Catalyzed Asymmetric C–H Functionalization Reactions
sp2–sp3 Coupling of Unprotected Halogenated Anilines with Grignard Reagents
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Issue 01/2024

Reductive Cross-Coupling for C(sp2)–C(sp3) Bond Formation
Regioselective 3-Trifluoromethylated Pyrrole Synthesis Using 2‑Bromo-3,3,3-trifluoropropene (BTP)
Sustainable Approach to 2,5-Disubstituted 1,3,4-Oxadiazoles
Enzyme-Catalyzed Synthesis of Chiral 3,3-Disubstituted Oxindoles
Decarboxylative Coupling to Access Oxetanol Derivatives
Modular, Scalable Synthesis of 1-Aza[3.3]heptanes
One-Pot Conversion of Quinolines into Quinazolines
Modular Synthesis of Isomeric, Spirocyclic Bioactive Scaffolds
The Dual Role of Formic Acid in the Synthesis of N-Arylated Pyrroles from Nitroarenes
Nickel-Catalyzed Synthesis of β-Lactams from Alkenyl Dioxazolones
New Reagents Enable Regioselective Halogenation of Complex, Bioactive Scaffolds
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Issue 12/2023

Regiodivergent C–H Arylation of Thiophenes
Doebner Hydrogen-Transfer Reaction to Access Electron-Deficient Quinolines
Cobalt-Catalyzed Olefin Cyclopropanation via Masked Dialkyl Diazomethanes
TBAI-Mediated Synthesis of Methylsulfonyl Oxazoles from Propargylic Amides
Direct Carbon for Nitrogen Replacement Reaction to Access Functionalized Pyridines
Palladium-Catalyzed C–H Arylation of Functionalized Pyrazoles/Triazoles and Imidazoles
Fused Piperidine Derivatives Featuring Stereogenic CF3 Substitution
Stereoselective Cascade Reaction for the Synthesis of Chiral Fused Diazaheterocycle Scaffolds
Scalable Synthesis of Silacyclohexanones for Silaheterocycles Construction
Modular, Chiral-Auxiliary-Mediated Synthesis of Sterically Constrained β-Amino Acid Derivatives
Synthesis of Functionalized Pyrrolidinones via Smiles–Truce Cascade
Rhodium(III)-Catalyzed Synthesis of Unsymmetrically Substituted 2,2'-Dipyridyl Amines Using 1,2,4-Trizoles
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Issue 11/2023

Ring-Expansion Skeletal Editing of Cycloalkanols through Metal-Free Nitrogen Insertion
Synthesis and Reactivity of a Conformationally Rigid Cubane-Derived Amino Acid
Predictable, Scalable Aliphatic C–H Oxidation of Complex, Drug-Like Molecules
On-DNA Synthesis of Spirocyclic Azetidines via Photocatalyzed [2+2] Cycloaddition
[2+2]-Cycloaddition Approach to Monocyclic Azetidines
P(III)-Directed C(sp2)–H Activation for the Synthesis of Dihydroquinolinones
Synthesis of 3‑Fluoropyrazoles via Radical-Polar Crossover Photoinduced Cyclization
Metal-Free Multicomponent Annulation Cascade for the Synthesis of Pyrimidines
Aza-Bicyclobutanes as Astonishingly Efficient Coupling Partners for Nickel Catalysis
General Approach to Cyclic Arylsulfoximines and their Derivatives
Asymmetric Baeyer–Villiger Oxidation to Access Tetronic Acids
Multigram Access to Functionalized Isoxazolines
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Issue 10/2023

Cu-Mediated Cyclization to Form 1H-Indazoles
Synthesis of Highly Substituted BN-9,1-Naphthalenes from BN-Butafulvenes
Revalorization of Nitrous Oxide for Use as an Oxygen-Transfer Reagent
Cp*Co(III)-Catalyzed Synthesis of Isoquinolones via Regioselective [4+2] Annulation of N-Chlorobenzamides
Secondary Amines from Ammonia Surrogate – Aminopyridinium Salts
Application of Strained Heterocycles as Electrophiles in Ni/Ir-Catalyzed Cross-Couplings
Synthesis of Substituted 2-Oxabicyclo[2.1.1]hexanes via [2π+2σ] Cycloadditions with Bicyclobutanes
Mechanism-Driven Development of a Novel Amide Directing Group for Directed C–H Functionalization
Validation, Development and Execution of an Automated Protocol for C–C Cross-Couplings
Access to Spiro-oxetane Oxindoles via DBU-Catalyzed Activation of Allenoates
General, Direct Ni-Catalyzed Cross-Coupling of Tertiary Synthons with Heteroaryl Halides
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Issue 09/2023

Rh-Catalyzed Asymmetric Carbometallation to Access 3-Substituted Piperidines
Synthesis of Hybrid Scaffolds Featuring 4-Pyridine and 4-Piperidine Moieties
Cu-Mediated C(sp2)–H Elaboration of Benzylic Scaffolds
Copper-Catalyzed Synthesis of Axially Chiral Arylpyrroles via Atroposelective Cyclization of Diyne
One-Pot Synthesis of Pyrazolooxazines from 2,2-Dichlorovinylacetophenones
Efficient Exploration of Reaction Space to Optimize Sustainable Cu-Mediated Ullmann Couplings
Photocatalyzed Formate-Mediated Deoxygenation of Alcohols through Benzoate Ester Intermediates
Synthesis of Polysubstituted Furans via Electrocatalyzed Cyclization
Synthesis of Azabicyclic Systems through [3+2] Cycloaddition of Oxidopyridinium Ions
Versatile Synthesis of 4-Fluoropyrroles
Regioselective Synthesis of Isoxazoles from Ynones
Catalyst-Controlled [3+2] Cycloaddition for the Synthesis of endo- or exo-Substituted Pyrrolidines
Catalytic Asymmetric Synthesis of Morpholinones and Piperazinones via Domino Ring-Opening Cyclization
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Issue 08/2023

Alternative to Ozonolysis for the Oxidative Cleavage of Olefins
General, Scalable Synthesis of 3-Azabicyclo[3.1.1]heptanes
Synthesis and Reactivity of 4H-Dewar Pyridines as Rigid Bioisosteres for 4-Substituted Piperidines
Building Highly Substituted Furyl Boronates via Carbene Boryl Migratory Insertion
Synthesis of P-Heterocycles from Unsaturated Phosphonites with C(sp2)-Electrophiles
Palladium-Catalyzed Synthesis of Indoles from ortho-Nitrostyrene and Formic Acid
Computational Studies on the Reaction Pathways of 1,2-Azaborinine with Unsaturated Organic Compounds
Photocatalyzed Access to Protected Trifluoromethyl Ketones through C–C Bond Formation
Ironing-Out Photodecarboxylation: Cross-Nucleophile Coupling Mediated by Iron Salts
Efficient Ring Opening Kinetic Resolution of 2,3-Aziridinyl Alcohols with Dinuclear Zinc Complexes
Sustainable Syntheses of Pyridines and Quinolines
Radical Ring Expansion of Hemiketal Hydroperoxides to Macrolactones
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Issue 07/2023

Aryl Radicals as XAT Promotors Enable Modular Alkyl Iodide Functionalization
Synthesis of Azabicyclic Cores of the Izidine Alkaloids
Ion-Paired Rhodium-Catalyzed Enantioselective Aziridination of Alkenyl Alcohols
Three-Component Reaction for the Synthesis of Isoxazoles
Stereoselective Synthesis of Six-to Eight-Membered Cyclic Ethers through Homologation/Metathesis
A Magical Rearrangement of Aryl Peroxyoxindoles to 1,3-Benzooxazin-4-ones
Cascade Reaction with Preservation of Stereochemistry for the Synthesis of Fused Cyclic Amine Systems
Synthesis of Functionalized Bicyclic Tetrahydrocyclopentafuran Derivatives
Operationally Simple Dearomatization of Bicyclic Azaarenes
Robust Trifluoromethylation of (Hetero)arylboronic Acid Pinacol Esters
Site Selective C–H Carboxylation of N-Heteroarenes via Electrochemical Reactors
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Issue 06/2023

Sustainable Synthesis of Sym-Triazines
Metal-Free Ring-Opening of Vinylcyclopropanes
Chirality at Oxygen!!
Robust Synthesis of (Hetero)Aryl and Aliphatic Sulfonyl Fluorides
Silver-Catalyzed Synthesis of Phosphorus-Containing Fused-Azepines
First Example of [5,6,5]-Tricyclic Bistetrazole Fused Explosive
Diversity-Oriented Approach to Spirocyclic and Fused Pyrazolopyrrolidines
Synthesis of Aryl Picolyl Sulfones via Formal C–H Activation
Cobalt-Catalyzed Synthesis of Oxetanes and Azetidines
Synthesis of N-Fluoroalkylated Morpholinos – An Application to the New Class of Nucleoside Analogues
Photocatalyzed Synthesis of Multi-Substituted Pyridines from γ-Ketonitriles
Switchable Multipath Cascade Cyclization via Chemodivergent Reaction
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Issue 05/2023

NHC-Mediated Synthesis of γ-Lactams
Organocatalytic Cloke–Wilson Rearrangement to Access Multi-Substituted Furans
Copper-Catalyzed Benzylic sp3 C–H Oxidative Annulation of Ketones and Amines
Robust Synthesis of Functionalized Bicyclic Heteroaromatic Sulfonyl Fluorides
Ruthenium-Catalyzed Synthesis of Piperazines and Diazepanes
Zn-Mediated Synthesis of Pyridines from Alcohols
Practical Arynes from Unfunctionalized Arenes
Versatile Synthesis of 4-Iodopyrrole-2-carbaldehydes
Improved Synthesis of the DLK Inhibitor GDC-0134
Savie: A Biodegradable ‘Drop-In’ Surfactant Replacement for TPGS-750-M
Transformations of Aliphatic Amines and Anilines into Diverse Functionalities
One-Pot Synthesis of N-Functionalized Indoles through a Three-Step Tandem Process
Aerobic Oxidative Cycloaddition Reactions for Pyrazole Synthesis
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Issue 04/2023

Modular Synthesis of Benzimidazoles from Nitroarenes
Oxidant-Free Synthesis of Fully Substituted Pyrroles through Multicomponent Cyclization
Circumventing the Aryldiazonium Salt Isolation in Intramolecular Heck–Matsuda Coupling
Direct and Practical Approach for the Synthesis of δ-Carbolines and Benzofuro[3,2-b]pyridines
Rational Design of a Palladium Catalyst System for C–N Bond Formation of Five-Membered Heteroaryl Halides
Robust Conditions for Nickel-Catalyzed Suzuki–Miyaura Cross-Couplings of Complex Molecules
Palladium-Catalyzed Synthesis of Benzazocines via [6+2] Double Allene Annulation
Catalyst-Free Synthesis of Oxacyclic Spirooxindoles through Oxonium Ylide Mediated Ring Expansion
Scalable Syntheses of Functionalized 2-Oxabicyclo[2.2.2]octanes
Construction of Functionalized Oxazole via Three-Component Cyclization Using a Lewis Acid
Bicyclic Silaazacycles Featuring Silicon at the Ring Junction: Synthesis and Further Transformations
Nickel-Catalyzed One-Pot Cascade Synthesis of N‑Substituted Indoles
Three-Step Modular Synthesis of N-Substituted Bicyclic Systems
Efficient Access to Pharmacologically Relevant 2-Arylpiperazines
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Issue 03/2023

Dearomative Redox-Neutral Strategy for the Selective meta-Functionalization of Pyridines
Ni-Catalyzed Synthesis of 2-Heteroaryl Azetidines
Synthesis of Anilines from Boronic Acids
Rhodium-Catalyzed Cross-Coupling to Form Ketones
Gram-Scale Synthesis and Characterization of HAT
Selective Approach to 1,3-Oxazines via Controlled Amino-Diazidation and Amino-Iodoazidation of Alkenes
Synthesis of Imidazo[1,5-a]pyridines via Anomeric Stereoauxiliary Cleavage of d-Glucosamine
Bench-Stable Reagents for Introduction of Highly Lipophilic Thiofluoroalkyl Fragments
Perfluoroalcohol Solvent-Promoted Inverse Electron Demand Diels–Alder Reactions
Ring Expansion of Isoxazoles using Cu(I) Catalysis
Selective meta-Halogenation of Pyridines
[2+2] Cycloadditions to Access sp3-Rich Spirocycles
Synthesis of Pyrazolo[5,1-c][1,4]oxazine Derivatives from 2,2-Dichlorovinylacetophenones
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Issue 02/2023

Multigram Synthesis of pivZPhos Ligand
Asymmetric Reductive Transamination for the Synthesis of Chiral Piperidines
Room Temperature Metal-Free Heteroaryl Hydrogenation
Ru(II)-Catalyzed Synthesis of Bridged Tetracycles via C–H Allylation and [3+2] Dipolar Cycloaddition
Synthesis and Application in Ni-Mediated C–C Cross-Couplings of a Modular Series of Novel Ligands
Scalable Synthesis of Enantiopure Bicyclic Fluorinated Pyrrolidinol
Enantioselective Transannular Reaction of Macrocyclic Sulfonamides
Two-Step Regioselective Trifluoropropylation of Azoles
Pyrimidines to Pyrazoles Under Mild Conditions
Merging Known Pharmacophores: Synthesis of Substituted N-Indolizines
Building 3-Borylated Pyrrolidines via 1,3-Dipolar Cycloaddition
Efficient Ni-Mediated Cyanation of (Hetero)Aryl Halides under Homogeneous Conditions
Three-Step, One-Pot Regioselective C-3 Trifluoromethylation of Quinolines
Elemental Sulfur-Mediated Annulation of Enaminones to Access 2-Aminofurans and 2-Aminthiophenes
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Issue 01/2023

Synthesis and Biological Activity of Bicyclic Nitroimidazole Derivatives
Synthesis and Characterization of Spiro-Tetrahydro­tetrazines as Energetic Materials
Preparation of 4-Iodo-1-tosylpyrazoles via Iodocyclization of N-Propargyl-N′-tosylhydrazines
Rh(I)-Catalyzed Synthesis of 3-Substituted Oxindoles
One-Pot Synthesis of N-Aryl Tetrahydroquinolines
Iron-Catalyzed Stereo-Convergent Cyclization with E/Z-Mixed Internal Olefines
A Grignard-Free 1,2-Arylation of Isatins
Nickel-Catalyzed Synthesis of chiral N-Heterocycles via C(sp3)–H Activation of Formamides
An Aza-Baeyer–Villiger Reaction for Nitrogen Insertion into Cyclobutanones
Decarboxylative Asymmetric Allylic Alkylation for the Synthesis of α‑Difunctionalized Cyclic Sulfones
Multicomponent Reaction for the Synthesis of Quinoxalin-2-Thiones and Quinoxalines
Catalyst-Free Synthesis of CF3-Containing 2-Pyrazolines via [3+2] Cycloadditions
Pd-Catalyzed Suzuki Coupling of Nitroarenes and Heteroarylboronate Esters
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Issue 12/2022

Silver-Free Chemoselective O-Benzylation of 2‑Quinolinones
Phase Dependent Tautomerism of 1,3-Thiazine Derivatives
Synthesis of N-Heterocycles via Photoredox Catalysis using Bifunctional Sulfilimines and Alkenes
Skeletal Editing through Nitrogen Atom Insertion to Indoles
Synthesis of Cyclic Enecarbamates through Dehydrogenation
Pd-Catalyzed Synthesis of 2,4-Diarylthiazoles
Synthesis of Nβ‑Substituted 1,2-Diazetidin-3-ones
Metal- and Photocatalyst-Free Switchable Redox Photoexcited Annulation of 2-Nitroarylethanols to NHCs
Oxidative Nucleophilic Substitution of Hydrogen for the Synthesis of Aminated Nitro-Substituted Heteroarenes
One-Pot Multicomponent Protocol To Access Sulfenylimidazo[1,5‑a]pyridines
Synthesis of Aziridines by Reaction of Free Amines with Alkenylthianthrenium Salts
Oxidative Condensation to Access Quinoxalines
Diastereoselective Synthesis of THF Derivatives
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Issue 11/2022

Selective N2-Alkylation of 1H-Azaindazoles
Synthesis of 6-Phenanthridines by Photocatalytic Deoxygenation of Alcohols
Synthesis of Versatile Enantiopure Morpholine Fragments from Chiral-Pool Starting Materials
Multicomponent-Reaction-Triggered Cascade Approach to Functionalized Fused 2,6-Diketopiperazines
Design and Synthesis of Azaborine-Based Steroid Mimics
Silver-Catalyzed Synthesis of Densely Functionalized gem-Difluorinated Molecules
Mechanistic Insights into Light-Mediated C–H Functionalization of 2-Phenylpyridines
Furans by Rhodium-Catalyzed Tandem Cyclization of Acrylic Acids
Microwave-Assisted Synthesis of Tertiary Amines from Carbamates
Synthesis of Spiro[furan-2,1′-isoindolin]-3′-ones by Intramolecular Sequential Prins and Ritter Reactions
Nickel-Mediated C(sp2)–C(sp3) Cross-Couplings
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Issue 10/2022

Copper-Catalyzed Isoxazole Synthesis
TEMPO-Mediated Convergent Synthesis of Benzoxazoles from Primary Amines and Cyclohexanones
Photoredox Cross-Coupling for Propellane-Curious Chemists
One-Pot Cascade Synthesis of 2‑Azafluorenones Mediated by Generation of Ammonia in situ
A Mild and Site-Selective Protocol for N1-Carboxylation of 2-Alkynylindoles
NHC-Alcohol Adduct-Mediated Photocatalytic Deoxygenation for the Synthesis of 6-Phenanthridine Derivatives
Carbonyl Compounds through Photochemical Olefin Cleavage
α-C–H Functionalization of Alcohols Delivers C6-Hydroxyalkylated Purines and Purine Nucleosides
Copper-Catalyzed Synthesis of Trifluoromethylated 4H-Pyrans
Manganese(III) Acetate-Promoted Mild Sulfonation of (Het)arenes
Facile Rearrangement of Oxetane-Carboxylic Acids to Lactones
Multicomponent Approach to Functionalized Isoquinolines
Synthesis of Pyrazoloimidazoquinazolinones and COVID-19 Protease Docking Studies
Synthesis of 7-[(Arylsulfanyl)methyl]dibenzo[b,d]azepines
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Issue 09/2022

Three-Step Sequence to Pyrrolizidinones
Access to Azaindolines through a Palladium-Catalyzed Heck Cyclization/Carbonylation Cascade
(Arylethyl)amine Synthesis through Intramolecular Radical Cyclization of Sulfonamides and Alkenes
One-Step Synthesis of Congested γ-Lactam-Based Polyheterocyclic Compounds
Asymmetric Synthesis via Chlorine Radicals to Access Chiral α‑(Het)aryl Amines
Base-Catalyzed Approach to Spirocyclic Oxazole Derivatives by a [3+2]-Cycloaddition Reaction
Visible-Light-Promoted Metal-Free Couplings for Pyridine-Derived Small Molecules and DNA Derivatives
Preparing Sulfonates by a Clauson–Kaas-Type Formation of Sulfonyl Pyrroles from Sulfonamides
Rhodium-Catalyzed Approach to Seven- and Eight-Membered Lactams
Rearrangement of 4-Alkenylisoxazol-5-ones to Pyrrole Analogues
Hexafluoroisopropanol-Promoted Nitrogen-Insertion into S/Se,N-Heterocycles
2,4,5-Trisubstituted 1,3-Oxazoles by [2+2+1]-Cycloaddition of Aldehydes and Nitriles
Multicomponent Reaction to Synthesize Functionalized Spirocyclic 1,4-Diazaheterocycles
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Issue 08/2022

Efficient Functionalization of Aminocyclopropanes
Precious-Metal-Free One-Pot Synthesis of Imidazopyridines and Thiazoles
Highly Regioselective Cross-Coupling of Dihalohetarenes
Ruthenium-Catalyzed Synthesis of Isoquinolinones from Allenylphosphine Oxides and Aromatic Amides
Diastereo- and Enantioselective trans-Hydrogenation of Isoquinolines
Brønsted Acid Mediated Synthesis of 1,4-Dioxanes
Ketoreductase-Mediated Dynamic Kinetic Resolution
Sustainable and Scalable Approach to 5-Substituted-1H-Tetrazoles
ortho-Selective C(sp2)–H Borylation of Pyridines with an Yttrocene Catalyst
Preparation of Diazacyclobutenes by a Lewis Acid Catalyzed [2+2] Cycloaddition
Efficient Synthesis of Versatile Furopyridines from Acyclic Precursors
Photochemical Metal-Free Coupling Reactions for Pyridine-Derived Small Molecules and DNA Conjugates
Synthesis of 2-Benzoxazoles by DMF-Assisted Radical Cyclization of o-Isocyanodiaryl Ethers
Efficient Merging of Proven Pharmacophores
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Issue 07/2022

Preparation of 2-Aminopyridines and 2-Aminoazines by a Zincke Reaction
Expeditious Robust Elaboration of Bicyclic N-Heterocycles
Gram-Scale Synthesis of Fluorinated Pyrazoles and Pyridines
Regioselective Functionalization of in situ Generated Heteroaryl Grignards with Tosyl Aziridines
Gold/Iridium-Catalyzed Enantioselective Synthesis of Spiroketals and Spiroaminals
Gold-Catalyzed Asymmetric Annulations of Enynone Derivatives and Nitrones Generated In Situ
TEMPO Salt Mediated Oxidative Ugi–Azide Approach to Direct Functionalization of N-Heterocycles
BINOL-Mediated Asymmetric Synthesis of Ammonium Salts
Photocatalytic Conversion of Indoles into Spirocyclic Indolines
Organophotoredox-Catalyzed Synthesis of Benzazepine Derivatives under Benign Conditions
Tertiary Amines by Palladium-Mediated Allylic C–H Amination
Copper-Catalyzed Borylation of (Het)aryl Carboxylic Acids
Construction of Silicon Heterocycles by Cobalt-Catalyzed Hydrosilylation of Enynes
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Issue 06/2022

Cross-Coupling Approach to Partially Saturated Heterocycles
Non-Radical-Mediated C–H Alkylation of Pyridines
Regioselective Functionalization of Azoles
C2-Selective SNH Amination of Pyrimidines through Selective Iminium Formation
Robust Difluoromethylation of Nonactivated Ketones
Synthesis of 5-Fluoroindolizines by Photocatalytic Defluorinative Coupling and SNV Cyclization
2-Amino-3,3-difluoro-2,3-dihydrofurans from Difluorocarbenes and Enaminones
Nickel-Mediated Allylation of Heterocycles
Oxindole Synthesis through a Polar–Radical Crossover
Naphthyridinone Formation through Palladium-Catalyzed Annulation of 1,6-Enynes and 2-Iodoanilines
Synthesis of 2-Pyridones by Ring Expansion of Furans or γ-Lactams
Gold and N-Heterocyclic Carbene Relay Catalyzed Synthesis of Pyrrole-Fused Lactones
Selective Synthesis of Pyridines and Pyrimidines Using Isopropene Derivatives
Synthesis of β-Aryl-γ-lactams and 2-Oxo-1,2-dihydroquinolines
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Issue 05/2022

New Silaazacycles: Syntheses of 1,3,5-Diazasilinan-2-ones and 1,3,5-Thiazasilinan-2-imines
Synthesis of Fluoroalkylated Benzimidazole- or Indole-Fused Benzoxazines
One-Pot Transition-Metal-Free Synthesis of Thiadiazine 1-Oxides
Modular Access to Functionalized Pyrroles
Copper Photocatalyzed Synthesis of Heterocycles
Synthesis of Bioactive Fluoropyrrolidines through 1,3-Dipolar Cycloadditions of Azomethine Ylides
Stereoselective Synthesis of Sulfinate Esters via a Chiral Ion Pair
Synthesis of 1,2,4-Thiadiazoles in Ethanol at Room Temperature by Using Hydrogen Peroxide
Synthesis of Novel Isoxazoloazaborines from 4-N-Propargylaminoisoxazoles
Enhanced Potency and Properties by Exploiting Substituted Oxetane as a Cyclobutane Bioisostere
Synthesis of Triazolopyridines with Nitrous Oxide
Electrochemical Syntheses of Substituted Morpholine Derivatives
Heteroaromatic C–H Etherification by Using (Benzo)thiophene-Based Halogen-Transfer Reagents
Access to Densely Substituted Furans by a Tsuji–Wacker-Type Cyclization
Expanding Substrate Scope of the Chemoenzymatic Functionalization of Tetrahydroisoquinolines
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Issue 04/2022

Metal-Free Reduction of Aromatic Nitro Compounds
Synthesis of Trifluoromethylated Azaheterocycles by Radical Chemistry
Synthesis of 1,2,4-Triazepines by a Base-Induced Formal [4+3] Cycloaddition
Access to Dibenzo[c,e]azonines by Iron-Catalyzed Alkyne–Carbonyl Metathesis
Convergent Synthesis of Isoindolines from Cyclic Imines and Organolithium Intermediates
A Solution to Nickel-Catalyzed Cross-Electrophile-Coupling Woes
Facile Halogenation of Aminoheterocycles for Rapid Diversification
Multicomponent Synthesis of Fluorescent Indolizine Tetracycles
Large-Scale Synthesis of 3-Fluoro-6-methoxyquinoline
Transition-Metal-Free One-Pot Synthesis of 3-Acylisoxazoles
TfOH-Promoted Selective C2–N1 Ring-Expansion Reaction of Indazoles
Organophosphorus-Catalyzed Cyclization of N-(2-Hydroxyethyl)amides
Visible-Light-Induced Transition-Metal-Free C(sp2)–H Difluoromethylation of Hetarenes
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Issue 03/2022

Enantioselective Synthesis of 1,4-Benzodiazepinones and 1,4-Benzoazepinones
Enantioselective Synthesis of Bispiro[Oxindole-Pyrrolidine-Pyrazolone] Derivatives
Skeletal Editing through Nitrogen Deletion: Synthesis of Complex Cyclobutanes from Pyrrolidines
Metal-Catalyzed Synthesis of Benzomorpholines
Rhodium-Catalyzed Synthesis of N-Arylaziridines
Solvent-Free Synthesis of 3-Trifluoromethyl-1,2,6-Thiadiazine 1-Oxides
Bronsted Acid-Catalyzed Synthesis of Spirolactams by Dearomatization of (Het)arenes
Annulation Reaction To Construct 2-Aryl-5-Amino- 2H-Tetrazoles
Increased 3D Character of Heterocyclic Systems through Efficient C(sp3)–C(sp3) Bond Formation
Homogeneous Stable Organic Reductants for Cross-Electrophile Coupling Reactions
Synthesis of Allocolchicine Analogues through Construction and Removal of P-centered Radicals
One-Pot Access to Spiropyrrolidines from Azidoboronic Acids and N-Sulfonylhydrazones
Transition-Metal-Free Cross-Coupling To Form 2-Pyridyl Derivatives
Synthesis of Heterocycle-Fused Pyrazoles via Cascade Wolff Rearrangement/Acylation
Sulfur-Mediated Benzoxazole/Benzothiazole Synthesis from Olefins and Aminophenols or Iodoanilines
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Issue 02/2022

Aziridination of Alkenes via Electrochemically Generated Thianthrenium Salts
Synthesis of Isoindolinones from Isoxazoles by a Ring-Opening-and-Closing Cascade Reaction
Synthesis of Complex Guanidines by [4+2]-Cycloaddition Indoles with N-Amidinyliminium Ions
Palladium/Norbornene Cooperative Difunctionalization of Five-Membered Arenes
One-Pot Diastereoselective Preparation of N-Alkenyl-2-Pyridones from 2-Halopyridinium Salts and Aldehydes
Three-Dimensional Five-Membered Nitrogen- and Sulfur-Containing Heterocycles
Direct C–H Functionalization of Azines by Electrochemical Manganese Catalysis
Synthesis of Phenanthridinones by a Cascade Reaction under Mechanochemical Conditions
Synthesis of Cyclobuta-Fused Tetrahydroquinolines
Bridged Bicyclic Lactone Synthesis by Brønsted Acid-Promoted Formation of O-Acyloxocarbenium Ions
Dihydroquinazolinones by a Base-Promoted Intermolecular Cyclization
Acid-Catalyzed Ring Fragmentation to Access Functionalized Pyrroles
C–H Activation To Form 2-Quinolin-8-ylisoquinolin-1(2H)-one Derivatives
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Issue 01/2022

Synthesis of Halogenated Azidopyridines
Pd(II)-Catalyzed Synthesis of Functionalized Dihydrobenzoxazines and a Functionalized Tricyclic System
Machine-Learning-Based Approach to Expanding SAR Exploration
Single-Electron Reduction of Sulfonium Salts for the Generation of Nonstabilized Alkyl Radicals
Regioselective Late-Stage Alkylation of Complex Molecules
Sulfonium-Salt Based Trifluoromethylating Reagent Permits Multiple Reactivity Paradigms
One-Step Synthesis of Pyrazolo[1,5-a]pyrimidines by a Copper-Catalyzed Dehydrogenation/[3+3] Annulation
Gold-Catalyzed Synthesis of Versatile Heterospirocycles
Synthesis of Seven-Membered N,O-Heterocycles by Using a Palladium(sulfoxide) White-Type Catalyst
Indole Synthesis through Reductive Cyclization of 2-Nitrostyrenes with Phenyl Formate as a CO Surrogate
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Issue 12/2021

Demonstrated 6-endo-tet Cyclizations!
Silver-Catalyzed Synthesis of Optically Active Pyrrolo[3,4-b]indoles
7-Alkylidene-Containing Bridged Azabicycles by Tandem Palladium and Copper Catalysis
4-(Perfluoralkyl)triazole-5-Carboxylates
5-Substituted 2-Alkyl-1H-Tetrazoles
Screening Platform for Optimizing Nickel-Catalyzed Suzuki–Miyaura Reactions
Chemoselective N- and O‑Difluoromethylation of 2‑Pyridones, Isoquinolinones, and Quinolinones
Oxazolines, Pyrrolidines, and Dihydrooxazines by Photochemical C(sp3)–H Functionalization
Hydrosilane-Facilitated Reduction of Pyridines through Borenium Catalysis
Versatile 7-Azaindole Intermediates
Nickel-Mediated Enantioselective Piperidine Synthesis
Metal-Free Synthesis of 4‑Aryl-1,2,3-triazoles by Iodine‑Promoted Cyclization
Access to Nonsymmetrical Tri- and Tetraoxanes with Silica Sulfuric Acid
Deoxidative Amination of Azine N-Oxides
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Issue 11/2021

Nitrogen Deletion of Secondary Amines
Molecular Editing through Ring Expansion of Pyrroles and Indoles
Multicomponent Approach to Functionalized Pyrazoles
Sustainable Oxidative Rearrangement of Furan Derivatives
Mild Synthesis of Polysubstituted Functionalized Pyrroles
Enantioselective Approach to β-Amino Acid Derivatives
Copper-Catalyzed Synthesis of β-Lactams from Oximes and Methyl Propiolate
Palladium-Catalyzed Approach to Arylquinolin-2(1H)-ones
Direct Synthesis of Functionalized Benzofurans from Phenols
Nonsymmetrical Trisubstituted s-Triazines: A Scalable Synthesis
Synthesis of Tricyclic Indoles by Enantioconvergent Substitution of Alcohols
Gram-Scale Access to Orthogonally Protected (Aza)spiro[2.3]Hexane Diamines
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Issue 10/2021

Synthesis of Silazacycles from the Elusive 3-Silaazetidine
Synthesis of 2,1-Benzisoxazoles via Decyanative Cyclization
Direct Preparation of N-Substituted Pyrazoles from Primary Aliphatic or Aromatic Amines
Dithioesters as Thiocarbonyl Precursors in Thorpe–Ziegler-Type Cyclization
Regiospecific Three-Component Synthesis of 2-Aminothiophenes
Rh-Catalyzed Synthesis of Thienoacenes from Thiophenes
Direct C–H Functionalization of N-Heteroaromatics with Cyclic Ethers
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Issue 09/2021

Radical Azidation of Cyclopropenes
One-Pot, Two-Step Synthesis of Indole-Fused Diazepanones
Regioselective C–H Borylation via Minisci-Type Reaction
Synthesis of Fluoroalkylated Isoquinolinones via Cobalt-Catalyzed C–H Activation/Annulation
Synthesis of Multisubstituted Pyridines via Nickel Catalysis
One-Pot Knoevenagel Condensation–Reduction Reaction of 2,4-Dihydroxy Quinolines and Pyridines
Umpolung Strategy to Functionalize Pyridines/Quinolines via Phosphonium Intermediates
Rhodium(III)-Catalyzed Synthesis of Functionalized Dihydrobenzofurans
Catalyst-Free Amination of Quinoxalin-2-ones and Benzo[1,4]oxazin-2-ones by Visible Light
Heterogeneous Nickel Catalyst Promotes Indole Formation via Dehydrogenative Coupling
Eight-Membered Cyclic Amines via Morpholine Intermediates
Room-Temperature C–N Coupling with Aryl Chlorides
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Issue 08/2021

Pictet–Spengler Reaction of Ketonitrones
Solvent Synthons: DMSO as an Active Methylene to Synthesize of Benzoxazines from Phenols and Nitriles
Synthesis of Benzazepines through Rhodium-Catalyzed Electrocyclization
Synthesis of Eight-Membered Lactams via Spiroindolines
Carbon Dioxide Incorporation Catalyzed by Nickel
An Elegant Synthetic Avenue to Azetidine-Containing Spirocycles
Synthesis and Evaluation of Novel Nucleotide Analogues Containing Dioxane and Morpholine Rings
Organocatalytic Approach to Chiral Spiro-Dihydropyranones
Phosphine-Catalyzed Synthesis of Functionalized 3-Alkenyl benzofurans
Synthesis of 3‑Aroylimidazo[1,2‑a]‑N‑heterocycles by Using DMSO as a One-Carbon Synthon
Iron-Catalyzed Synthesis of 4-Aryl pyrrolo[1,2-a]quinoxalines from Nonactivated Methyl Arenes
Fluorocyclization of Allylic Alcohols and Amines to Access 3-Functionalized Oxetanes and Azetidines
Gold- and Palladium-Catalyzed Synthesis of Multifunctionalized Nine-Membered Heterocycles
Selective Catalytic C-2 C–H Functionalization of Azoles
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Issue 07/2021

One-Pot Stepwise Synthesis of γ-Lactams through Cycloadditions with Ketenes
Palladium-Catalyzed Synthesis of Benzoxepines from Vinyl-Substituted Cyclopropanes and Salicylaldehydes
Mild Regioselective Reduction of Pyridines to Dihydropyridines
Rhenium-Mediated Synthesis of Five- and Six-Membered Nitrogen-Containing Heterocycles
Sequential Palladium-Catalyzed Synthesis of Benzosultams
Regioselective Synthesis of Indoles form Azoarenes or Azoxyarenes with Ketones
Copper-Catalyzed Synthesis of Quinazolines and 1,2,4-Oxadiazoles
Iridium-Photocatalyzed Synthesis of Bioactive Tetracyclic Nitrogen-Containing Products
2-Pyridones from Enamides through Ni–Al Bimetallic Catalysis
Synthesis of Functionalized Benzimidazoles through C(sp3)–H Amination/C–N Bond Cleavage
Palladium-Catalyzed Synthesis of Enantiopure Eight-Membered Nitrogen Heterocycles
One-Pot Construction of 2,3-Dialkyl-Substituted Quinazolinones from Secondary Amides and Isocyanate
Iridium-Catalyzed Approach to Polycyclic Nitrogen-Containing Systems
Selectfluor-Promoted Synthesis of Functionalized Isothiazolones
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Issue 06/2021

Gold-Catalyzed Synthesis of 2H‑Azirines from Alkynyl N-Sulfinylimines
Visible-Light-Promoted Intramolecular Aminoiodination of Alkynes
Enantioenriched Tetrahydropyridines from Racemic Allyltriflamides through Kinetic Resolution
Synthesis of Triarylethanes by 1,6-Conjugate Addition
Synthesis of Azacycles through a 1,2-Metalate Shift
General Solid-Phase Protocol for Modular Oligonucleotide Synthesis
Multigram Electrosynthesis of Enecarbamates and Related Building Blocks
Indolylcyclopentenes through an Enantioselective Aminopalladation–Heck Reaction
Synthesis of Enantiopure Piperidines by an Asymmetric Aza-Prins Reaction
5-(Trifluoromethyl)pyrazoles by a Regioselective [3+2] Cycloaddition
Trityl-Cation-Initiated Cycloaddition of Benzyl-Substituted Vinylcyclopropanes with Hydrosilanes
Protein-Templated Assembly of Heterodimeric Tryptase Inhibitors
Generation and Regioselective 3,4-Difunctionalization of Pyridynes
Protecting-Group-Free Asymmetric Synthesis of Pyroglutamic Acid Esters
Disaccharide Synthesis through Regioselective O-Glycosylation under Boronic Acid Catalysis
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Issue 05/2021

Synthesis of Indolyl Cyclobutanones by Brønsted Acid Catalysis
Synthesis of 2-Fluoro-1-benzofurans from β,β-Difluoro-o-hydroxystyrenes by 5-endo-trig Cyclization
Explore Three-Dimensional Chemical Space with Triazolobenzodiazepines
Rhodium(III)-Catalyzed Synthesis of Thiobenzofurans
Atroposelective Synthesis of 2-Arylquinazolinones
Nickel-Catalyzed Electrochemical Cross-Coupling of Alcohols and Aryl Halides
Environmentally Friendly Achmatowicz Rearrangement
Synthesis of 2,4,6-Trisubstituted Pyridines from Methyl Ketones and Alkynones
Synthesis of Five-Membered Cyclic Sulfonamide (γ-Sultam) 4,4-Spirocycles
Synthesis of Bi(1,2,3-triazoles) by a Three-Component Reaction
One-Pot Synthesis of 2-Azaaryl Tetrahydroquinolines by a Base-Promoted Reaction
Synthesis of Heterocycles from Potassium Trifluoro(pyrimidin-4-yl)borate Salts
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Issue 04/2021

Rhodium(III)-Catalyzed C–H Activation/Annulation To Form Isoquinolone Scaffolds
Chiral Phosphoric Acid Catalyzed Enantioselective Synthesis of 8-Azabicyclo[4.3.1]decanes
Preparation of Imidazolidine-2-ones from N-Benzoyloxyureas by C–H Amination
Nickel/Copper-Catalyzed Amidation of 2-Iodoglycals to Access Glycosamine Analogues
Palladium-Catalyzed Synthesis of Azepines from Pyrrolidines
Three-Component Approach to Indoles
Synthesis of N-Fused Hetarenes from Alkenes
N-Containing Bicyclic Heterocycles by Annulation of 2H-Azirines with 2-Chloropyridine Derivatives
Et3N-Direct Cycloaddition of Allenoates with Acceptor Diazo-Compounds
Diastereoselective Synthesis of 2,3-Dihydrofurans from Silver Allenes
Synthesis of Enantiomerically Enriched Chiral 1-Pyrrolines
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Issue 03/2021

Thermally Promoted Synthesis of β-Lactam Derivatives
Rhodium-Catalyzed Synthesis of 1H‑Indole-2,3-dicarboxylates from Arylhydrazines and Maleates
Enzymatic Syntheses of Tryptophan Analogues and Incorporation in Biocatalytic Cascades
Increasing the 3D-Character of Heterocyclic Systems through Hydrogenation
Diastereoselective Atom-Economical Synthesis of Dihydropyrans
Rhodium-Catalyzed Synthesis of Chiral Hydrophenanthridinones
Rhodium-Catalyzed Synthesis of Chiral 3,4-Fused Tricyclic Indoles
Rhodium-Catalyzed Synthesis of 1,3-Benzodiazepines
One-Pot Condensation to Tricyclic Azepines
Synthesis of 1,2,4-Triazoles by Annulation of Nitriles with Hydrazines
Cascade Reaction for the Enantioselective Synthesis of Pyrrolizidones
Rhodium-Catalyzed C–H Activation To Form Macrolactams
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Issue 02/2021

Regioselective Scalable Approaches to Trifluoromethylated Pyrazoles
FIavin–Iodine-Coupled Organocatalyzed Synthesis of Imidazo[1,2-a]pyridines
Bridgehead Hydroxylation in the Annulation of Cyclic Aldimines
Palladium-Catalyzed Synthesis of Dibenzothiazines from Aryl Sulfoximines and Arynes
Nickel-Catalyzed C–N Coupling of Heterocycles
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Issue 01/2021

C–H Functionalization of Quinolines, Isoquinolines, and Pyridines by N-Alkenoxyhetareniums
Synthesis of 2-Arylindoles by Iridium(III)-Catalyzed Sequential Annulations
N-Alkylation of Hetarenes through Electrochemical Oxidation of Carboxylic Acids
Gram-Scale Synthesis of Cyclopropane-Fused Saturated Heterocycles Featuring a Trifluoroborate Moiety
Decarboxylative Heteroannulation Route to Phenanthridin-6-ones
Synthesis of Angular and Linear Heteroannulated Furochromenopyridines
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Issue 12/2020

Iodine/Trifluoroacetic Acid-Assisted Multicomponent Synthesis of 4(3H)-Quinazolinones
Electrocatalytic Decarboxylative Synthesis of 1,3,4-Oxadiazoles
Tuning Redox Properties of Bistetronates through Spacer Selection
Stereoselective Synthesis of Cyclopenta[c]pyrazoles by an Interrupted Ohira–Bestmann Reaction
Hypervalent Iodine(III)-Mediated Synthesis of Spirooxazolines
Regioselective C–H Arylation of Quinolone Derivatives
Synthesis of Oxygen-Rich Polycyclic Scaffolds
[4+1]-Spiroannulation of Bromophenols with α,β-Unsaturated Imines: Synthesis of Azaspirocycles
Cobalt-Catalyzed Synthesis of Pyrroles from Nitroarenes
Synthesis of 1,3,4,11-Tetrahydrooxocino[3,4-b]indoles
Synthesis of 1,2,3-Benzothiazaphosphole 1,1-Dioxides
Diverse Syntheses of Furochromone-Based Antimicrobial Agents
Asymmetric Synthesis of Spiro-Benzofurans and Fused Benzopyrans
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Issue 11/2020

Isolation and Structural Characterization of Three New Benzazepines
Chiral Hemiketal Formation by Organocatalytic Desymmetrization of gem-Diols
Synthesis of Spirocyclic Pyrrolidones from Diazobutyrolactams
Scalable Synthesis of Functionalized gem-Difluorocyclopropanes
C–H Bond Functionalization of Alicyclic Amines
Synthesis of 2-Formylpyrroles from Pyridinium Iodide Salts
Minisci Reaction of N-Hetarenes with Cyclopropanols as the Radical Source
Synthesis and Derivatization of N-Trifluoromethylated Indoles
Mild Regioselective Halogenation of Anilines, Anilides, and Indoles
Pd-Catalyzed Asymmetric [8+2]-Dipolar Cycloadditions: Synthesis of Ten-Membered Ring Heterocycles
Cobalt(III)-Catalyzed Synthesis of Isoquinolinones and Pyridinones by Annulative Vinylene Transfer
Chiral N,O-Acetals by Asymmetric Hydrogenation of Cationic Intermediates
Metal-Free [5+1]-Cycloaddition Route to Pyrazine 1-Oxides and Pyrazines
Two-Step Synthesis of Functionalized Benzoxazoles
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Issue 10/2020

Modular Syntheses of 5- and 6-Azaindoles
Modular Synthesis of 2,5-Diaryltetrazoles
Synthesis of C2-Substituted Imidazolones
Nickel-Catalyzed Enantioselective Synthesis of 3,3-Disubstituted Oxindoles
Cine-Substitutions of Five-Membered Hetarenes via Sulfonium Salts
Synthesis of Indoles through C–C and C–N Bond Formation of Aliphatic Amines and Nitrosoarenes
One-Pot Synthesis of Polycyclic Indolones by Photocatalytic Annulation of Redox-Active Esters
Bismuth(III)-Catalyzed Synthesis of 2-(Fluoroalkyl)imidazole-5-carbaldehydes
A Sequential C–H Activation–Annulation Route to Fused Phthalimides
Copper-Catalyzed Three-Component Synthesis of γ-Lactams
Synthesis of Chiral γ-Lactams through Pd(II)-Catalyzed Cascade Alkenylation/Aza-Wacker Cyclization
Indium-Catalyzed Synthesis of 1,2-Dihydroquinolines through Rearrangement of Oxetanes
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Issue 09/2020

Electrochemical Alkylation of Hetarenes with Carbazates as Radical Precursors
Photocatalytically Triggered Radical Smiles Rearrangement
Synthesis of Medium-Sized Lactones from Siloxy Alkynes and Lactols by Ring Expansion
Synthesis of Spiro[cyclohexane-1,12′-isoindolo-[1,2‑b]quinazolin]-10′-one Derivatives
Catalyst-Controlled Regioselective C-5 Hetarene Olefination
1,4-Benzoxazepines and Tetrahydroquinolines by Pd-Catalyzed [4+2] and [5+2] Annulations
Rh(III)-Catalyzed Synthesis of 6H-Benzo[c]chromen-6-ones from Sulfoxonium Ylides and Quinones
Automated Photoredox 18F-Difluoromethylation of Acyclovir
Titanium-Mediated Synthesis of Polysubstituted Pyrazoles
Safe and Efficient Synthesis of 4-Aminofurazan-3-Carboxylic Acid and its Ethyl Ester
Rhodium(III)-Catalyzed Synthesis of 1,2-Diaminobenzenes and Benzimidazoles
Ruthenium-Mediated ortho-Selective C–H (Per)fluoroalkylation of Anilines and Indoles
C–H Hydroxymethylation of N-Arylazaindoles with Paraformaldehyde
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Issue 08/2020

Selective C2-H Amination
NHC-Catalyzed Chemo- and Enantioselective Synthesis of 3,4‑2H‑Pyridin-2-ones
Potassium Carbonate-Catalyzed Synthesis of Highly Functionalized Indoles
Rhodium-Catalyzed Synthesis of Enantioenriched Phthalides
Copper-Catalyzed Synthesis of Highly Functionalized Pyrroles from Allenoates
A Mild Skraup Quinoline Synthesis from Anilines and Epoxides
Synthesis of Benzodiazepines from Benzimidazolium Salts
Combined Chemoenzymatic Sequence for the Synthesis of γ-Lactones
Efficient Electrochemical Synthesis of 2-Aryl-1,2,3-Benzotriazoles and their N-Oxides
Benzyne-Mediated Ring Opening of DABCO: Synthesis of 1,4-Disubstituted Piperazines and Piperidines
Synthesis of Tricyclic Indoles from Iodoalkynes and an N-Tosyl Hydroxylamine
Silver(I)-Catalyzed 1,3-Dipolar Cycloaddition Route to Fully Substituted Pyrrolidines
Intramolecular N-Halovinylation to Synthesize Cyclic β-Haloenamides
Asymmetric Synthesis of α-Carboline Derivatives
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Issue 07/2020

Automated Approach to the Modular Synthesis of Drug-Like Molecules
Transition-Metal-Free Synthesis of 3,4-Disubstituted 2-Piperidinones
Synthesis of Oxazolidines, Pyrrolidines and Mannich Bases from Aliphatic Aldehydes
A Scalable Route to N-Difluoromethylated Heterocycles
Modular Rhodium-Catalyzed Synthesis of Quinolines from Anthranils and Acrylic Acids
Reactions of Epoxides, Thiiranes, Aziridines and Azirines with Cyanoform
Synthesis of Alkene Carbonates by Carbon Dioxide Fixation Using Perfluorinated Triol Catalysts
Palladium-Catalyzed β-Cycloalkenylation of Saturated Cyclic Ketones
Palladium-Catalyzed Enantioselective Synthesis of Isoxazolines
Rhodium-Catalyzed Synthesis of Isoquinolines from Aryl Ketones and Alkynes
Ruthenium-Catalyzed Diastereoselective Synthesis of Tetrasubstituted Pyrrolidines
One-Pot Synthesis of 2-Trifluoromethyl-6-azaindoles
Copper-Mediated Synthesis of N2-Aryl-1,2,3-Triazoles
Mild Synthesis of 3H-Indoles and Benzazepinones from Nonactivated Anilines
Asymmetric Synthesis of Cyclopropane-Fused Pyrrolidines
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Issue 06/2020

Synthesis of Alkene Carbonates through Carbon Dioxide Fixation Using Perfluorinated Triol Catalysts
Triazapentalene Synthesis by N–N Bond Formation
Sulfinylation of Indoles, Pyrroles, and Thiophenes
Ligand-Free Palladium(II)-Mediated Synthesis of 2,4-Disubstituted 1,3-Thiazoles
Determination of Basicities and Nucleophilicities of a Series of Organocatalysts
Direct C-2 Carboxylation of Electron-Deficient Indoles
Iridium-Catalyzed Synthesis of Indoles and Indolines
Synthesis of β-Lactams by a Kharasch–Sosnovsky Reaction
Nickel(0)-Catalyzed Enantioselective Synthesis of Butenolides and Lactams
Synthesis of Seven- and Nine-Membered Heteroatom-Containing Rings
Synthesis of 1,2,4-Oxadiazoles from Alkynes and Nitriles
Silver Acetate-Catalyzed Groebke-Blackburn-Bienayme Reaction to Synthesize Imidazo[1,2-a]Pyridines
Synthesis of [6,5]-Spirocycles through Redox-Neutral Cyclizations of Aurones
Stereoselective C–H Cyclopropanation of N-Phenoxysulfonamides
Access to Functionalized Chromanes by Asymmetric [4+2]-Cycloaddition
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Issue 05/2020

SNAr Reaction of Aminooxetanes with Quinazolines: Synthesis of Imidazo[1,2-c]quinazolines
Synthesis of Five-Membered Heterocycles by H3PO2-Catalyzed Cyclization of Stereodefined Alcohols
Pyrylium Reagent for the Radical C–N Borylation of Aromatic Amines
Iridium-Catalyzed Synthesis of Fused Isoquinolines
Photochemical Electrocyclization Synthesis of Azaanthraquinones
AuCl3-Catalyzed Synthesis of Cyclopentenes, Polycycles, Benzocarbocycles, and N-Heterocycles
Copper(I) Chloride-Catalyzed Synthesis of Benzo[4,5]thieno[2,3‑d]thiazoles
Enantioselective Synthesis of Functionalized 1,3-Thiazin-4-ones
Synthesis of 1,2,4-Thiadiazoles and Fused Analogues by Electrochemical S–N Bond Formation
Synthesis of Ethyl 3-Fluoro-1-Pyrrole-2-Carboxylate
Synthesis of Spiropyrazoline Oxindoles and Spiropyrazoline Indanones
Phosphorus-free Reagent for the Chlorination of Aza-Arenes
Dirhodium(II)-Catalyzed C(sp2)–H Azidation for the Synthesis of Azidobenzaldehydes
Three-Component Synthesis of Morpholine Derivatives
Copper-Mediated Synthesis of N-Arylpyrazoles from Cyclopropanols and Aryl Diazonium Salts
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Issue 04/2020

2-Arylpiperidines by Palladium-Catalyzed Addition of Arylboronic Acids to Acylated 2-Hydroxypiperidines
Synthesis of Phosphorylpyrroloindoles by Photocatalytic Phosphinoylation/Cyclization Reactions
Synthesis of Thiochromenes by Palladium-Catalyzed Ring Opening of Cyclopropyl Thioethers
Regioselective Synthesis of Polyfluorinated o-Hydroxyacetophenones
Chemodivergent and Enantiospecific Synthesis of Benzazepines and Allyl Fluorides
Organocatalyzed Synthesis of Fully Substituted Furans from Ynamides and Quinoxaline N-Oxides
Diastereoselective De Novo Synthesis of Functionalized Piperidines
Construction of Highly Substituted Furans and Thiophenes with Sulfur Ylides
C(sp3)–H Functionalization of Aliphatic Acids through β-Lactonization
Asymmetric Copper-Catalyzed Synthesis of Dihydrobenzofuran-3-ols
Palladium(II)-Catalyzed Synthesis of Tribenzo[b,d,f]azepines
Three-Component Synthesis of 3-(Trifluoromethyl)pyrazoles
Base-Promoted Annulations in the Synthesis of Ring-Fused N-Substituted-4-Quinolinones
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Issue 03/2020

One-Step Synthesis of 4-Fluoropyrimidines
Synthesis of Benzofuroindolines through Biocatalytic Oxidative Phenol–Indole [3+2] Reactions
Palladium-Catalyzed Ring Expansion for the Synthesis of 12-Membered Heterocycles
Synthesis of Butenolides from Functionalized Cyclopropenones
Electrochemical Synthesis of trans-2,3-Disubstituted Aziridines
Regioselective Synthesis of CF2H-Containing Pyrazoles
Enantioenriched Dihydroquinolines by NHC Catalysis
Diastereoselective Cyclization of Oxime-Tethered Cyclopropanes to Pyrrolooxazines
Light-Mediated Dehydrogenative Povarov Reaction of Indoles and Benzofurans
Stereoselective and Regioselective Functionalization of Piperidines through C–H Activation
The N-Oxide Moiety as a Traceless Directing Group for Pyridine 2-C(O)–C Bond Activation
Asymmetric Palladium-Catalyzed Synthesis of Fluoropiperidines
Modified Pomeranz–Fritsch Reaction for the Synthesis of 1,2-Dihydroisoquinolines
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Issue 02/2020

Sweet Ligand: Use of Galacturonic Acid in Copper-Catalyzed N-Arylation of Heteroarenes
Oxazoline Synthesis by Using the XtalFluor-E Reagent
Organocatalytic Approach to Spirooxindoles
Synthesis of Sulfonylpyrroloindoles via Photocatalytic Sulfonylation/Cyclization Reactions
Synthesis of Fused Pyridines through a Rhodium-Catalyzed Rearrangement of Furan-Linked Triazoles
Difluoromethylation of 1,2,4-Triazinones by a Copper-Catalyzed Interrupted Click Reaction
Biaryls from Anilines and Aryl Sulfoxides through Sigmatropic Rearrangement
Three-Component Synthesis of Thienothiazoles from Acetophenones
Synthesis of Benzothiophenes by a Twofold C–H Functionalization
Metal-Free Synthesis of Aza-Fused Heteroaromatics
Asymmetric Synthesis of 3,6-Dihydropyridinones
Three-Component Synthesis of Tetrazoles Utilizing ZSM-5 Heterogeneous Catalysis
Pyridotriazole as Carbene Precursor in Rhodium-Catalyzed Synthesis of 3H-Indoles
Copper-Catalyzed C–H Activation Approach to Benzofurans by Using a Traceless Directing Group
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Issue 01/2020

Asymmetric Synthesis of Indolines via a Transient Chiral Directing Group Intermediate
[3+2] Cycloadditions of 3-Nitroindoles with Substituted γ-Allenoates
Rongalite-Catalyzed Synthesis of Polysubstituted Pyrazoles
Protecting Group Controlled Regiodivergent Syntheses of N-Bridged Heterocycles
Asymmetric Synthesis of γ- and δ-Lactone-Fused Tetralin Derivatives
Oxepinocoumarins by Ring-Closing Metathesis
First Synthesis of a Monocyclic Aromatic 1,2,3,5-Tetrazine
Multicomponent Mannich Reaction through C–H Activation of Azabiaryls
Synthesis of Cyclic Sulfoximines through 5-endo-dig Cyclization of N-Propargylsulfinamides
Synthesis of Fluoroalkylated Isoxazoles from Ynones
One-Step Syntheses of Morpholinones and 1,4-Oxazepane-3-ones
Biocatalytic Asymmetric Synthesis of N-Arylated β-Amino Acids and Pyrazolidinones
Synthesis of Pyridone-Fused Phenanthridines through Multistep Radical Addition/Cyclization Reactions
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Issue 12/2019

Divergent Formation of Flavones or Benzofurans from a Common Tyrosine-Based Oxa-Michael Precursor
Synthesis of Bis(pyrroloquinoline) Derivatives from Isatins and β-Keto Amides
Synthesis of Tetracyclic Dihydroquinolinones by a Knoevenagel/Hetero-Diels–Alder Reaction
Conversion of N-Sulfonyl Triazoles into Triazole-Fused Isoindolines
Preparation of Thietane, Thiolane, and Thiane Perfluorinated Diels–Alder Products
Rhodium(II)-Catalyzed Synthesis of Indoloindolones
Decarboxylative Cross-Coupling of Aryls and Hetaryls
Cobalt(II)-Catalyzed Synthesis of Perfluoroalkyl Isoxazoles
Selective Synthesis of Thio-Substituted Cyclotriphosphazene Derivatives
Stereoselective Synthesis of α- and β-l-Rhamnopyranosides
Isoquinolinediones and Isocoumarins by Rhodium(III)-Catalyzed C–H Activation of N-Tosylbenzamides
Synthesis of Di- and Trisubstituted Imidazoles from Methyl Ketones and Aldehydes
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Issue 11/2019

Copper-Catalyzed Synthesis of Di(het)arylamines
Synthesis of Enaminones and Thiazoles Using Iodonium Ylides as Carbene Equivalents
Cooperative Catalysis for the Asymmetric Synthesis of Piperidines
Selective C-2 Directed-Carbonylation of Indoles and Pyrroles
Synthesis of Substituted Morpholines by Fragmentation of Tetrazoles
Rhodium-Catalyzed Synthesis of 2‑Arylindoles from N‑Aryl-2-aminopyridines
Synthesis of Benzazepinones Involving an Unexpected Intramolecular Cyclization
Electrocatalytic Synthesis of Imidazo[1,5-a]quinoline-3-carbonitriles
Asymmetric Radical C–H Amination for the Synthesis of Azoles
Three-Component Assembly of 3,4-Dihydroquinazolines
Synthesis of Phosphinolines and Phosphepines
Buchwald–Hartwig Coupling of Piperidines with Hetaryl Bromides
Synthesis of 3-Phenylimidazo[1,2-a]pyridines by Annulation of Tetrazoles with Phenylacetylenes
Copper-Catalyzed Cyclization of Enaminones to Polycyclic N-Fused Indoles
An Illuminating Synthesis of Benzimidazoles
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Issue 10/2019

Enantioselective Synthesis of Cyclic Dipeptides by Iridium-Catalyzed Hydrogenation
Rhodium-Catalyzed Synthesis of Chiral Sulfoximines and 1,2-Benzothiazines
Pyridine Synthesis by 6π-3-Azatriene Electrocyclization
Copper-Catalyzed Iodine-Mediated Synthesis of Indolizines
Palladium–NHC Catalyzed Coupling of Organolithium Reagents at Low Temperatures
N-Acetyl-Directed Cyclopropanation of Indoles
Synthesis of Spirocyclic Thiadiazino Quinazolinones
3-Aroylquinolines by a Three-Component Reaction of Anilines, Enaminones, and DMSO
Palladium(II)-Catalyzed Synthesis of Pyrroles from Alkynylimines and Isocyanides
Brønsted Acid Catalyzed Synthesis of α-(3-Indolyl) Ketones
Enantioselective Cyclization of Alkenyl Amides to Polycyclic Dihydroindoles
Photoredox Approach to Fluorinated Pyrrolo[1,2-a][1,5]benzodiazepines
Photoredox-Mediated Pyridonation of (Het)Arenes
Decarboxylative Cross-Coupling of α-Amino Acids and α-Oxy Acids with Aryl Nitriles
Cobalt-Catalyzed Synthesis of Benzoindol-2-ones from Naphthylamides
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Issue 09/2019

Photoredox Fischer Indole Synthesis
Three-Component Synthesis of Diazacycles
Photocatalytic Synthesis of N-Heterospirocycles
Synthesis of (5+5)-Annulated Heteroaromatics
Electrochemical C–H Amination of Quinoxalinones
Stereoselective Synthesis of Chiral Isoxazole-dispirobisoxindoles
Triflic Acid-Mediated Synthesis of (Z)-β-Enamido Triflates and Fluorosulfonates
Synthesis of Indolizines from 2-(Propargyloxy)pyridines and Methyl Ketones
Directing-Group-Free C7-Alkylations of N-Alkylindoles by Zirconium Complexes
2,2-Disubstituted Tetrahydrofurans through [4+1] Cyclization
1,3-Dipolar Cycloaddition to Access Spirocyclic Nitrochromene Derivatives
Heteroarenes by Regioselective C–H Activation of Phenol and Aniline Derivatives
Semisaturated Diazoheterocycles through N–N Bond Formation
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Issue 08/2019

Synthesis of Two Azaborine Building Blocks
Phosphonium-Salt-Catalyzed Synthesis of Fused Aziridines by an Aza-Darzens Reaction
Chemoselective Demethylation of Methoxypyridines over Anisoles
Catalytic Azole Acylation with Acyl Fluorides
Acridone Synthesis by Double Amination of Dibromobenzophenones
Enantioselective Catalytic Aryl-Alkenylation To Give Dihydrobenzofurans
Synthesis of 1,2-Benzothiazine 1-Imines as New Heterocyclic Scaffolds
Selective C–H Alkenylation of Isoxazoles
Gold(III)-Catalyzed Synthesis of 4-Aminooxazoles
Synthesis of 1,4-Benzothiazines by Iodide-Catalyzed Alkene Sulfenoamination
Copper-Catalyzed Synthesis of 3,4-Dihydroquinazolines from Anthranils
Silver-Catalyzed Synthesis of Trifluoromethylated Triazines and Pyridines
Asymmetric Synthesis of Dihydrobenzofurans by an Organocatalytic [4+1] Cyclization
DBU-Mediated Synthesis of Bicyclic Heterocycles
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Issue 07/2019

Bithiophenes as a New Class of Organic Photoredox Catalysts
Programable Synthesis of Polyspirocyclic Heterocycles
Combined Electrochemical and Photochemical Syntheses of Pyrrolidines and Oxazolines
Synthesis of 1,3,4-Thiadiazines from Fluorinated Nitrile Imines and Thiols
Synthesis of Pyrazoles by a Silver-Mediated [3+2]-Cycloaddition Reaction
Rhodium(III)-Catalyzed Synthesis of (2H)-Indazoles from Azobenzenes
Synthesis of Fused Indoline–Cyclobutanone Derivatives
Decarboxylative Fluorination of Pyridin-2-ylacetates
Synthesis of 5,5-Disubstituted Hydantoins
Copper-Catalyzed Synthesis of Substituted Indoles and Benzoindoles
Base-Catalyzed Annulation for the Synthesis of Pterocarpene Analogues
Azepines by Palladium-Catalyzed C–H Activation and Isocyanide Insertion
Silver-Catalyzed Synthesis of 4-Trifluoromethyl-1,2,3-triazolines
Manganese-Catalyzed Selective C–H Alkylation of Imidazopyridines
Thiomorpholine Synthesis by a Copper-Catalyzed Three-Component Reaction
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Issue 06/2019

Electrochemical Reduction of Arenes
CuH-Mediated Regiodivergent Synthesis of Chiral Alkylated Indoles
Enantioselective Synthesis of Pentacyclic Spirooxindoles
Synthesis of γ-Arylated Butenolides by Palladium or Copper Catalysis
A C–H Bond Alkenylation/Aza-Michael Route to Benzoisothiazole 1-Oxides
Synthesis of Substituted Benzimidazoles by C–H Imination
Nitrene C–H Bond Insertion Strategy for Synthesis of γ-Lactams
Photoredox Radical/Polar Crossover Synthesis of Nitrogen Heterocycles
Synthesis of α- and β-C-Glycosyl Arenes by Direct Iridium-Catalyzed Hydroarylation
Cobalt-Catalyzed Synthesis of Isoquinolines by Using a Traceless Directing Group
Intramolecular Radical Cyclization of 2-Azaallyls to Benzofuran Derivatives
Rhodium(II)-Catalyzed Enantioselective Synthesis of N-Substituted 2-Pyridones
Hexahydro-1H-cyclopenta[c]pyrazolo[1,2-a]pyrazole-1,5(2H)-diones
9a,10,12,12a-Tetrahydrobenzo[b]cyclopenta[f]pyrrolo[1,2-d][1,4]diazepinones
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Issue 05/2019

Vanadium-Catalyzed Pyrrole Synthesis
Synthesis of Pyrimidine Nucleobases under Prebiotic Conditions
Transannular C–H Arylation of the Azabicyclo[3.1.0]hexane Core
Catalytic Enantioselective Synthesis of 2-Pyrazolines
Gold-Catalyzed Decarboxylative Benzylation of Indoles
Quinolines by Hydride Abstraction Induced Electrocyclization
1H-Pyrrolo[2,3-d]carbazoles by Brønsted Acid Catalyzed Cyclization of Ynamides
Palladium-Catalyzed Synthesis of Polycyclics from Aryl Iodides and Alkynes
Enantioselective Aza-Heck Approach to N-Heterocycles
Palladium-Catalyzed Synthesis of Dihydropyrido-[1,2-a]indolones
Palladium-Catalyzed Asymmetric Allylation of α-Amidopyridinium Salts
Benzoxazoles and Benzoxazines by Intramolecular Aryl Azide Insertion
Nickel-Catalyzed Michael Reaction of Malonates and Nitroalkenes
Minisci Reaction with Organotrifluoroborates: Merging Photo- and Electrochemistry
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Issue 04/2019

Three-Component Synthesis of Quinazolinones
New Biocatalytic Synthesis of Caprolactone by Oxidative Lactonization
Organocatalytic Synthesis of Enantioenriched Five- and Six-Membered Cyclic Ureas
Synthesis of Indolo[1,2-α]indole Derivatives by Gold(I)-Catalyzed Cycloisomerization
Gold Carbene Route to Several Classes of Azaheterocycles
Photodecarboxylative Azidation of Cyclic Amino Acids with Rhodamine 6G
Palladium(II)-Catalyzed Activation for Nucleophilic Substitution Reactions
Cobalt-Catalyzed Synthesis of Quinolines and Acridines from Anthranils
Spiroindolines by Visible-Light-Mediated Intramolecular Cycloadditions
Synthesis of Pyrrolophenanthridine Alkaloids by the Schmidt Reaction
Synthesis of 2-Aminopyrroles and Quinoline-Based Polyazaheterocycles
Titanocene-Catalyzed Synthesis of Functionalized Ring-Fused Piperidines
Electrochemical Synthesis of Fluorinated 2-Oxazolines
Synthesis of Carbazoles and Indolines by Gold-Catalyzed Diels–Alder Reactions
Synthesis of (5E)-5-(Iodomethylene)-1,3-selenazolidin-2-ones
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Issue 03/2019

Synthesis of Spiroazetidinimine Oxindoles
Synthesis of Benzodithiazines by an ortho-Metalation–Oxidative Cyclization Route
Visible-Light-Promoted Decarboxylative C–H Adamantylation of Azoles
Palladium-Catalyzed Synthesis of Indolin-2-ones and Dihydroquinolin-2-ones
Syntheses of Highly Substituted Dihydropyridine Derivatives from Hantzsch Esters
Chemodivergent Approach to Lactones and Lactams
Synthesis of Spirobarbiturate–Cyclopropanes
Cycloaddition Reaction of Alkynyltrifluoroborates with Azetidinones and Oxetanones
Synthesis of N-Heterocyclic Carbene–Boralactone Complexes from Alkenylboranes
A Short Route to 3-Fluoroalkyl-5-Pyrazolecarboxylates
Visible-Light-Mediated Cyclopropane Construction
Reaction of 2-Mercaptopyridine with Nitroallylic Acetates to Form Indolizines
Direct Carbamoylation of Heterocycles through a Minisci Reaction
Iridium-Catalyzed Synthesis of Fluorinated Benzothiazoles
6-exo-dig Iodocyclization Route to Dihydro-1,3-oxazines
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Issue 02/2019

Photochemical Cyclopropanation of Indoles
Visible-Light-Mediated Minisci C–H Alkylation with Dioxygen as Oxidant
Orthogonal Cross-Coupling of a Trifluoromethylated Chromenone Framework
N-Heterocyclic Carbene Catalyzed Synthesis of Substituted Oxetanes
Photocatalytic γ-Lactam Synthesis by Using Carbon Dioxide Activated Amines
Iron-Catalyzed Synthesis of Fluoroalkylated 2H-Azirines from Alkynes
Synthesis of Trifluoromethylated Pyrroles from Azirines
Stereoselective Synthesis of Tetrahydro-1-benzazepines through [4+3] Annulation
Synthesis of Azepines from 1,2,3-Triazoles and 1,3-Dienes
[3+2]-Cycloaddition Route to Imidazoles and Imidazolines
Annulation of Sulfoximines with Diazo Compounds
Enantioselective Synthesis of 4,9-Dihydrothiopyrano[2,3-b]indol-2(3H)-ones
Carbene-Catalyzed Synthesis of Pyrrolo[3,2-c]quinolines
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Issue 01/2019

Synthesis of N-Doped Polycyclic Aromatic Hydrocarbons
Organocatalytic Approach to cis-Octahydroacridines
Synthesis of Perfluoroalkylated Spirobarbiturates
Iridium-Catalyzed C–H Alkenylations: Synthesis of 3-Alkylisobenzofuran-1(3H)-ones
Reaction of Cyclobutanones with Allenylsilanes to form Oxabicyclo[3.2.1]octanes
Photocatalytic Synthesis of 8- to 11-Membered Lactams by C–C Bond Cleavage
Multicomponent Reaction Approach to Aza Analogues of Tropane Alkaloids
Functionalized 2H-Isoindoles by Rhodium-Catalyzed C–H Activation
Metallophotoredox-Catalyzed C–H Arylation of C(sp3)–H Bonds
Ionic-Liquid-Mediated Syntheses of Fused Pyrimidines and Quinazolines
Carbocyclization through an Interrupted Carbonyl–Olefin Metathesis
Synthesis of Pyrrolopyrazinones from N-Substituted 2-Cyanopyrroles
Synthesis of 2‑Aminoquinolines from N‑Acyl‑o‑alkynylanilines
Borane-Catalyzed Synthesis of Azasilaheterocycles
One-Pot Synthesis of Isoquinolinones by Rhodium-Catalyzed C–H Activation
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Issue 12/2018

Stereoselective Synthesis of Phosphorothioate Nucleotides
Chan–Lam Coupling/Friedel–Crafts Reaction Sequence to Acridines
Reductive Isoxazoline-to-Pyrrolidone Ring Interconversion
Rhodium(III)-Catalyzed Synthesis of 1,4-Dihydroisoquinolin-3(2H)-ones
1-Phenylsulfonyl-3-Oxabicyclo[3.1.0]hexan-2-one for the Synthesis of Spirocycles
Organocatalytic Route to Tetrahydrochromeno[4,3-b]pyrrol-4(1H)-ones
Ru-Catalyzed Synthesis of Pyrazines and Pyrroles from Ammonia and Diols
Synthesis of Indoloquinolines by a Dinitrogen-Extrusion/Cyclization Method
Electrochemical Coupling of Benzothiophenes with Phenols
Modified Paal–Knorr Cyclization Route to Substituted Pyrrolodiazepinones
Enantioselective Synthesis of Pyrimidinones by the Biginelli Reaction
Diastereoselective Cyclopropanation of Unsaturated Pyrazolones
Palladium-Catalyzed Synthesis of Indolo[3,2-a]Carbazoles from Indoles
Iron(III)-Catalyzed Asymmetric Synthesis of Tetrahydroindolizines
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Issue 11/2018

One-Step Synthesis of 2-Substituted Indazolones
Synthesis of Quinolines by a Photoredox Catalytic Three-Component Reaction
Copper-Catalyzed Trifluoromethylation via Aryl Radicals
Cobalt-Catalyzed Hydroboration/Cyclization Synthesis of γ-Lactams
SNAr Reaction of Pyridinium Salts with N-, O-, or S-Nucleophiles
Rhodium-Catalyzed Synthesis of Carbazoles from Biarylboronic Acids
Photochemical C–H Functionalization of N-Heterocycles with Carboxylic Acids
Synthesis of Oxazol-2(3H)-ones and Fused Oxazolidones from Ynamides
C–C and C–N Coupling Strategy for the Synthesis of Aminoisoquinolines
Synthesis of Tetrahydroisoquinolines through a Catellani/Heck Reaction
Stereo- and Enantioselective Synthesis of Tetrahydrofurans via Oxocarbenium Ions
Synthesis of 1,2-Annulated Aryl Glycosides
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Issue 10/2018

Synthesis of Enantioenriched 1H/3H-Pyrroles and Pyrroloimidazoles
Indolo[3,2-c]coumarins and Benzofuro[3,2-c]quinolinones
Synthesis of Trifluoromethylated Pyrrolidine and Piperidine Amino Acids
Hypervalent Iodine Reagent for the Synthesis of 2-Substituted Indoles
Phosphonium Salts as Surrogates for Aromatic Carbon–Heteroatom Bond Formation
Scalable Synthesis of an exo-Triazolylazabicycle
Synthesis of Cyclic Ureas by a Cross-Metathesis/Aza-Michael Sequence
Synthesis of Quinolines through Double-Oxidative Dehydrogenative Cyclization
C5 Alkenylation of Imidazoles and the Synthesis of Benzimidazoles
Palladium-Mediated Stereoselective Synthesis of 3,4-Fused Indolines
Samarium(II) Iodide Mediated Synthesis of Five- and Six-Membered N-Heterocycles
Silver-Mediated Synthesis of Fluorinated Oxazolidinones
C4-Activated Arylation of Pyrrolidines and Piperidines
Pyranopyrimidine–Triazole Hybrid Molecules
Quinoline-4-carboxylic Acids and Esters from N,N-Dimethylenaminones and Isatins
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Issue 09/2018

Flow Photochemical Synthesis of Bicyclic Aziridines from Pyridinium Salts
Synergistic Catalysis: Enhanced Regio-selectivity in the Synthesis of 1,2,3-Triazoles
Azaheterocycles by Ring-Closing Metathesis of Enynamides
Transition-Metal-Free Synthesis of 3-Carbonylated Benzofurans
Asymmetric Synthesis of 5,6-Dihydropyran-2-ones
N-Heterocyclic Carbene Catalyzed Enantio-selective Synthesis of 1,5-Benzodiazepines
Synthesis of Functionalized Heteroaromatics from ortho-Ester Protected Pyruvates
Visible-Light-Mediated Synthesis of Trifluoromethylated Coumarins
Synthesis of 2,5-trans-Tetrahydrofuran-2-ylacetonitriles
Cs2CO3-Mediated Synthesis of 2,3-Diaryl-2H-azirines from Ketoxime Acetates
Manganese-Catalyzed Synthesis of peri-Condensed Heterocycles
3-Acylisoquinolines by Cobalt-Catalyzed Annulation of Benzohydrazides
Indolines by Rhodium(III)-Catalyzed Annulation of 2-Alkenylanilides with Alkynes
Carbene-Mediated Benzodioxole Synthesis
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Issue 08/2018

Selective N-Alkylation of 2-Pyridones
A Halocyclization Approach to Enantioenriched Lactones
NHC-Catalyzed Asymmetric Synthesis of Cyclopentene-Fused Tetrahydroquinolines
Ferrocene-Catalyzed Electrosynthesis of Oxindoles and Dihydroquinolin-2-ones
Synthesis of Chromenopyridopyrazines and -diazepines
One-Catalyst, One-Pot, Two C–H Bond Activations
Double C–H Activation Approach to Chromenes
Stereoconserved Synthesis of Triazole-Fused Ketopiperazines
Enantioselective Syntheses of Indolines, Indoles, and Dihydro-2-quinolones
Zinc-Catalyzed Four-Component Synthesis of Highly Substituted Pyridines
Regiocontrolled Synthesis of Pentasubstituted Pyrroles
Rhodium-Catalyzed Indole/Pyrrole Cascade Synthesis
Tetrahydropyrans by an Enantioselective Cross-Dehydrogenative Coupling
Synthesis of Quinoline-4-carboxamides from Ketoxime Acetates and Isatins
Synthesis of Fused Benzothiophenes, Indoles, and Other Heterocycles
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Issue 07/2018

Dihydrobenzofuran Synthesis by Palladium/Norbornene Cooperative Catalysis
Copper-Catalyzed Three-Component Synthesis of Thiazoles
Synthesis of 2-Substituted Indolines via Allyl Boronic Acids Generated in situ
Dioxines and Oxathiines from Epoxides and Episulfides
Gram-Scale Synthesis of Cyclobutane-Fused Pyrrolidines and Piperidines
Regioselective Synthesis of 3-Halopyrazoles
Synthesis of Azolopyrimidines through Rhodium-Catalyzed C–H Functionalization
Flipping a Switch to Access Aziridines
One-Pot Synthesis of Fluoroindenones
Nickel-Mediated C(sp2)–H Amination: Synthesis of Anthranilic Amides
Preparation of Quinazolines from Alkynes and 2-Aryldihydrophthalazinediones
Copper-Catalyzed Synthesis of 5-Arylindazolo[3,2-b]quinazolinones
Synthesis of Imidazolidin-5-ones from Azlactones and β-Carbolines
Copper-Catalyzed Synthesis of Azole-Fused Quinazolines
Synthesis of 2-Aroylbenzofurans from Arynes and Sulfur Ylides
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Issue 06/2018

Heterocycles by NHC-Catalyzed Aerobic Oxidative Annulation
Ligand-Free Catalytic Synthesis of Heterocyclic Sulfones
Vanadium-Promoted Stereoselective Radical Cyclizations to Tetrahydrofurans
Photocatalyzed Synthesis of Sulfonated Isoindolinones
Enantioselective [5+2] Annulations with a Cooperative Catalytic System
Transition-Metal-Free Synthesis of 1,3,5-Triazines
Enantioselective Friedel–Crafts Alkylation of Indoles
Cobalt–Carbene-Catalyzed Synthesis of Indolines
Ruthenium-Catalyzed Remote C–H Activation of Purines
N2-Selective CuO-Catalyzed Coupling of 1H-Indazoles with Diaryliodonium Salts
One-Step Syntheses of 1,4-Diazo Hetero-cycles by Formal [n+2] Cyclizations (n = 4–6)
Dibenzo[f,h]quinolines by Palladium-Catalyzed Decarboxylative Annulation
Michael Addition/[1,2]-Stevens Rearrangement Approach to Piperidines
Synthesis of Oxindolylidene Acetates and Spirooxindolopyrrolidones
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Issue 05/2018

Azepines by a Carbonylative Rhodium-Catalyzed Reaction of Aminocyclopropanes
Xanthates for Radical-Mediated Alkylations of Heteroarenes
Synthesis of 2-(Trifluoromethyl)indoles from 2-Alkynylanilines
Synergistic Rhodium/Gold-Catalysis Approach to Spiroethers
Regioselective Deuterium and Tritium Labeling of Azaarenes
Copper-Catalyzed Synthesis of Fluoroalkylated Isoxazoles
Gold-Catalyzed Synthesis of 4H-Azepines and Pyridines
Iridium-Catalyzed C–H Intramolecular Amidation To Give γ-Lactams
Reactions of a Fluorosulfuryl Cation Donor with Phenols or Amines
Synthesis of Indolizines by Reaction of Pyridines with Allenoates
N-Ring Annelated Furanones by Iron-Catalyzed Cyclic Amine Functionalization
Chiral 3,4-Dihydro-2H-1,4-benzoxazines by Aminohydroxylation of 1,3-Dienes
Synthesis of 2-Azabicyclo[3.2.0]heptanes by [2+2] Photocycloaddition
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Issue 04/2018

Cooperative Amine–Copper Catalysis
Gold-Catalyzed Synthesis of Isoxazole-Fused Heterocycles
Benzannulated Heterocycles by Aza-Claisen Rearrangement
Palladium-Catalyzed Amination of Chloroheteroarenes with Secondary Amines
Dehydrogenative Cyclization of 8-Amido-quinolines
Minisci Alkylation of Heteroarenes with Boronic Acids
Catalytic Pummerer Reaction Approach to 3-Thiofurans and 3-Thiobenzofurans
Synthesis of γ-Lactams by Radical-Induced 1,6-Enyne Cyclization
3,4-Dihydroisoquinolines by Photooxidative Annulation of Imines with Alkenes
α-Functionalization of Unprotected Cyclic Amines by Hydride Abstraction
Facile Access to Dihydrocoumarins through Catalytic Hydroarylation
Electrochemical Synthesis of Imidazo-Fused Heterocycles
Tetrahydropyridines from Condensation of Sulfonamidoenones with N-Sulfonylimines
Synthesis of Spirocyclic Pyrido- and Pyrroloquinolines from an Isatin Derivative
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Issue 03/2018

Synthesis of Fused Indoles from Sulfonamides
One-Pot Rhodium-Catalyzed Synthesis of Highly Substituted Quinolines
Rhodium-Catalyzed Annulation of N-Methoxy-amides: Synthesis of Isoquinolones
Copper-Catalyzed Synthesis of Fluorinated 2,2-Disubstituted Indolin-3-ones
Continuous-Flow Electrosynthesis of Benzothiazoles and Thiazolopyridines
Synthesis of Pyrrolidinones and Piperidinones by Using a Chiral Ammonia Equivalent
Difluoromethoxylation of N-Heteroaromatics
Rhodium(II)-Catalyzed Annulation Route to 5H-Pyrazino[2,3-b]indoles
Synthesis of Fluoropyrrolidines by [3+2] Cycloaddition
Cyclopentaquinolines by Palladium-Catalyzed Reaction of 2-Vinylanilines with Alkynes
Enantioselective Synthesis of Heterocycle-Fused β-Lactones
Hexafluoroisopropanol as a Solvent for Halogenation of (Het)aromatics
Stereoselective Synthesis of Cyclic Ethers by Reductive Cyclization of Alkynols
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Issue 02/2018

[8+2] Cycloannulation: Synthesis of Dihydrocyclohepta[b]pyrrol-2(1H)-ones
Copper-Catalyzed Aerobic Indole Synthesis through Nitrogen Radical Cyclization
Oxidative Cross-Coupling of Nonactivated Substrates to Yield 1-Benzazepines
Cobalt-Catalyzed Synthesis of 5-Aminooxazoles
Palladium-Catalyzed Enantioselective Synthesis of Fused Benzofurans
Synthesis of β-(Hetero)Aryl Ketones through sp3 C–H Activation
Photochemical Synthesis of Chloromethylated Pyrrolidines
Synthesis of Heteroaryl Amino Acids
Copper-Catalyzed Synthesis of 1-(2-Hydroxyaryl)-1H-indazoles
N-Heterocyclic Carbene Catalyzed Synthesis of Substituted Pyridines
Synthesis of Functionalized Spiro-Oxetanes for Combinatorial Chemistry
Manganese-Catalyzed Minisci Alkylation of Heteroarenes
Copper-Catalyzed Synthesis of Dihydropyrroles and Pyrroles
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Issue 01/2018

Phosphinoboration of Pyridines and Related N-Heteroaromatic Systems
Organocatalytic Synthesis of Cyclopenta[b]benzofurans
Synthesis of Substituted Aziridines by Michael Addition Triggered Cyclization
Synthesis of 2,3-Disubstituted Indoles by C–H Functionalization of Azobenzenes
Synthesis of Fluorinated Oxazolines from Allylamides
Iodine-Mediated Intramolecular C–H Ami-nation Route to 1H-Indazoles and 1H-Pyrazoles
Phosphine-Catalyzed Synthesis of Chiral Spiro[cyclopentene-indole]ones
Synthesis of Fluorocoumarins by a Photoredox Reaction
Synthesis of Pyrrolidinoazepines and Pyrrolidinooxazoles by Cycloaddition
Gold Catalysis in an Asymmetric Synthesis of Tetrahydrofurans
Synthesis of Lactones and Lactams by Nickel-Catalyzed Transfer Hydrogenation
Three Rings in One Shot: Diastereo- and Enantioselective Ring-System Synthesis
Spirocyclic Pyrazoles by Ring Expansion of Cyclic Ketones
Practical Synthesis of Azaheterocycles Con-taining a gem-Difluorocyclopropane Moiety
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Issue 12/2017

Synthesis of β-Lactams through Cyclization of Amide Dianions with Diiodomethane
Multicomponent Coupling Reaction for the Synthesis of Fused Furans
β-Enaminones in the Synthesis of Heterocycles
Visible Light-Mediated Trifluoromethyl Group Installation in Flow
Rhodium-Catalyzed C2-Alkylation of Benzimidazoles
Regioselective Metalation of 1,5-Naphthyridine
Copper-Catalyzed Difluoro- and Perfluoroalkylations of Heterocycles
Palladium-Mediated Synthesis of 3,4-Dihydroisoquinoline N-Oxides
Synthesis of 2-Pyridinimines
Benzannulated Heterocycles by Nucleophilic Amination of Methoxyarenes
Tetrahydropyrans by a Rhodium-Catalyzed Metathesis Cascade
Proline Derivatives through a Radical Redox Strategy
Palladium-Catalyzed Synthesis of 1,2-Disubstituted Azaindole Isomers
trans-Selective Alkynylboration of Alkynes to 4-Alkynyl-1,2-oxaborol-2(5H)-ols
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Issue 11/2017

Oxidative C–H Sulfenylation of Carbonyls
Difluoromethylation of Aryl- or Hetarylboronic Acids and Esters
Enantioselective Modular Approach to 3-Azabicyclohexanes
Synthesis of Pyrrolocoumarins and Substituted Pyrroles
Oxetanones and Azetidinones for the Synthesis of 6-Azaspiro[4.3]octanes
Synthesis of Indoles by Ruthenium-Catalyzed C–H Activation
Synthesis of 2-Allyl-3-oxazolin-5-ones and Trisubstituted Pyridines
Ethyl Tertiary Amines as a Carbon Source in Imidazopyridines Synthesis
Rhodium-Catalyzed Cyclizations of Enoldiazoacetamides with Nitrosoarenes
2′-Homoazanucleosides by Ring-Closing Metathesis
Selective N-Methylation of Pyrimidone with Chloro(chloromethyl)dimethylsilane–KF
Synthesis of Trifluoromethylated Pyrido[2,3-d]pyrimidinediones
Synthesis of Trifluoromethylated Heterocycles from N-Carbamoyl Imines
Synthesis of Quinazoline-2,4(1H,3H)-diones from 2-Iodoanilines
Three-Component Synthesis of Benzopyrans from δ-Acetoxy Allenoates
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Issue 10/2017

Rhodium(III)-Catalyzed Indoline C–H Alkylation with Enones
Synthesis of Iodoquinolines from N-Tosyl-2-propynylamines
Borylketenimines in the Synthesis of Borylated Heterocycles
Synthesis of 1-Substituted 2-Azaspiro[3.3]-heptanes
Synthesis of Oxindoles Containing Trifluoromethyl Quaternary Carbon Centers
Synthesis of Fluoropyrrolidines by Using an Iodine/Hydrogen Fluoride Reagent
Click Synthesis of 1-Aza-2,3,4-triphospholenes
Synthesis of 3-Substituted Phthalides by Reductive Hydroiodination
Synthesis of the Tetracyclic Core of Secoyohimbane Alkaloids
Silver-Catalyzed Oxidative Decarboxylation Route to Difluorooxindoles
Synthesis of Furan and Pyrrole Derivatives by Oxetane Ring Opening
One-Pot Synthesis of Thieno[3,2-b]pyridines
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Issue 09/2017

Catalytic C(sp3)–CF3 Bond Formation
Scalable Synthesis of Haloquinolin-2(1H)-ones and Quinolines
Synthesis of 2-Spiropiperidines by the Aza-Maitland–Japp Reaction
Conversion of Endoperoxides into Furans by the Appel Reaction
Synthesis of Tetrahydropyridines by Enantioselective Cyclization of 1,6-Dienes
Visible Light Assisted Synthesis of Imidazoles by Intramolecular C–H Imination
Synthesis of Isoquinolinones by Amide Umpolung
Copper-Catalyzed Annulation of Tetronic Acids with Azirines: Scope and Mechanism
Chiral Binaphthylsulfonate Cluster Catalyst for Cycloaddition Reaction
Diastereoselective Synthesis of Difluoromethylated Spirooxindoles
Synthesis of Dihydrophenanthridines by Dehydrogenative Coupling
Asymmetric Synthesis of Chiral 3,4-Dihydro-2H-pyrancarbonitriles
One-Pot Synthesis of 1,2-Disubstituted Benzimidazoles
Rhodium(III)-Catalyzed Synthesis of Pyrano[2,3,4-de]-quinolines
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Issue 08/2017

Synthesis of C-Aryl Glycosides by Glycosyl C(sp3)–C(sp2) Stille Cross-Coupling
Niobium-Catalyzed Intramolecular Hydrofunctionalization of Alkenes
Lewis Acid Catalyzed Stereoselective Synthesis of Trisubstituted Tetrahydrofurans
Dibenzoxazepinones and -thiazepinones by Dual Copper-Catalyzed Coupling Reactions
Platinum-Catalyzed Synthesis of 2,3-Dihydro-pyrroles and Polyheterocyclic Compounds
Organocatalytic Approach to Functionalized Furans
Stereoselective Synthesis of Pyrrolidine-2,3-diones by a Claisen Rearrangement
Iron-Catalyzed Spirocyclization–Arylation
Synthesis of Pyridoimidazo-β-carbolines
Visible-Light-Induced Iron-Catalyzed Synthesis of 3,3-Disubstituted Oxindoles
Perhydroindolic Acid Catalyzed Synthesis of Chiral Tricyclic γ-Lactams
Radical Cyclization Approach to Borylated Piperidines
Synthesis of Oxazolidinones by a C–H Amination Reaction
Pyrimidines and Pyridines by Ring Expansion of Cyclobutanones
Alkylation of Amines under Mitsunobu Conditions
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Issue 07/2017

Palladium-Mediated Synthesis of Spiro-Fused Dihydrobenzofurans and Indolines
Synthesis of Active 2-Aminothiophenes through the Gewald Reaction
Enantioselective [3+2] Cycloaddition Route to Pyrrolidines
Copper-Catalyzed Enantioselective [1,3]-Rearrangement to Chiral Propargylic Amines
Tetrahydroquinolines by Sulfenoamination of Alkenes
Highly Diastereoselective Ozonolysis Route to Ozonides with Antimalarial Activity
Palladium-Catalyzed α-Arylation of Ketones in Aqueous Media
Synthesis of C3-Fluorinated Oxindoles by Electrochemical Cross-Coupling
Photocatalytic Deoxygenative Cyclization to Chiral Tetrahydrofurans and Pyrrolidines
Enantioselective Synthesis of 3,4-Dihydroquinolin-2-ones
Carbolithiation in the Synthesis of Heterofused Indolizidines and Pyrroloazepines
Enantioselective Synthesis of Pyrrolidines with Vicinal Stereocenters
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Issue 06/2017

Pyridols by Cyclization and Rearrangement of Alkynyl Oximes
Pyrrolidine Synthesis through C(sp3)–H Alkenylation of Aliphatic Amines
Synthesis of Trifluoromethylated Piperazines from Aziridines
Synthesis of Polysubstituted Furans
Catalytic C–H Activation of Heterocycles
Synthesis of 6-Aminopurines by an Ugi–Smiles Multicomponent Reaction
Synthesis of 2,3-Dihydroimidazo[1,2-a]-pyridines by a Formal [4+2] Cyclization
Synthesis of Quinolines From o-Alkenylaryl Isonitriles
α-Imino Rhodium Carbenoid-Catalyzed Synthesis of Substituted Pyrroles
Synthesis of Kealiinine Alkaloids from Propargylguanidines
Tetrahydroisoquinolines by Intramolecular Asymmetric Reductive Amination
Fused Pyrrolidine β-Lactones by an NHC-Catalyzed Cascade Reaction
Nickel-Catalyzed Synthesis of Benzoisoselenazolones
4-Diazoisochroman-3-imines and 3,5-Dihydroisochromeno-[3,4-d][1,2,3]triazoles
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Issue 05/2017

Functionalized Propellanes, Azetidines, Cyclobutanes, and Chiral Cyclopentanes
Synthesis of 2,5-Disubstituted Oxazoles
De Novo Synthesis of Polyaryl Salicyl Esters
Indole Synthesis by an Intramolecular aza-Stetter Reaction
Synthesis of 2,3-Disubstituted Pyridines by Transition-Metal-Free Amination
Cobalt-Mediated Synthesis of Quinolin-2(1H)-ones
Palladium-Catalyzed Synthesis of 4-(2-Haloaryl)-1,2,3-triazoles
Homonucleosides by Amination/Cyclization of Sulfanyl 1,6-Diynes
1,2,4-Triazines by the Reaction of N-Tosylhydrazones with Aziridines
Intramolecular 2-Aminoimidazole Synthesis from Guanidine
Synthesis of Lactams from Imines and Homophthalic Anhydride
Electroorganic Synthesis of Pyrimido-[4,5-b]indole Derivatives
Copper-Catalyzed Route to Indazolo-[3,2-b]quinazolinones
Photoredox-Promoted Anti-Markovnikov Hydroamination of Nonactivated Olefins
Fused Heterocycles by an Amine-Catalyzed aza-Diels–Alder Reaction
Carbonylative Benzannulation Route to Substituted Benzofurans
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Issue 04/2017

Thioketones in an Asymmetric Thia-Diels–Alder Reaction
Iron-Mediated Synthesis of Pyrroles, Pyrrolines, and Imidazolines
1,3-Dioxane Synthesis by Catalytic Prins Reaction
Synthesis of Morpholines and Piperazines by an Ugi Multicomponent Reaction
Diverse Heterocycles by Pd-Catalyzed Cyclization of Unsaturated N-Sulfonylamides
Rhodium-Catalyzed Synthesis of 1,2,4-Triazines
Reversed Regiochemistry in Halo-lactonizations of Olefins to Lactones
Asymmetric Paal–Knorr Pyrrole Synthesis
Asymmetric α-Arylation of Thioamides
Lewis Acid Catalyzed Synthesis of Azidocyclopentane and Tetrahydropyridines
Synthesis of Pyrroloisoxazole-Based Ring Systems
Silver-Catalyzed Synthesis of Trifluoromethylated Heterocycles
Enantioselective [2+2] Cycloaddition of N-Allenamides with N-Sulfonylketimines
Aza Analogues of Benzyl Isoquinoline Alkaloids
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Issue 03/2017

Photoredox Nitroso-Diels–Alder Reactions
Acridones by Double C–H Carbonylation of Diphenylamines
A New Class of Enantiopure Oxathiazines
Photochemical Stereoselective Synthesis of Azetidines
Multicomponent Synthesis of Substituted 3H-1,4-Benzodiazepines
Synthesis of Hexahydropyrazolo[1,5-a]-pyridines
Palladium-Catalyzed Benzazetidine Synthesis with a Rationally Designed Oxidant
Synthesis of Imidazo[1,5-a]pyrazin-8(7H)-ones
Indole Synthesis through Dizincioindole Formation
Squaramide-Catalyzed Synthesis of 3-Chroman Derivatives
Chromones and Benzofurans by a Divergent Rhodium-Catalyzed Annulation
An Aza-Prins Reaction in the Synthesis of Tricyclic Benzazocines
Synthesis of Indazoles and Indoles from Azobenzenes through C–H Activation
Trifluoromethylated 1,3,4-Thiadiazoles by [2+3] Cycloaddition
Substituted Oxindoles and Dibenzoazepinones through Aryne Insertion
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Issue 02/2017

Palladium-Catalyzed Synthesis of Six- and Seven-Membered-Ring Heterocycles
Enantioselective Organocatalytic Synthesis of Benzo-Fused Acetals
Palladium-Catalyzed Carbonylation of Aliphatic Amines To Form β-Lactams
Stereodivergent Diels–Alder Route to Bicyclic Lactones
Lewis-Acid-Mediated Multistep Synthesis of (–)-Mersicarpine
Direct Nickel-Catalyzed Synthesis of Oxaborins from Benzofurans
Palladium-Catalyzed Synthesis of Cyclopropyl-Fused Azacycles
Synthesis of Pyrrolopyridinones by the Ugi Reaction
Synthesis of Acylated Benzimidazoles with Copper Catalysts
Synthesis of 3-Cyano-1H-indolo-2′-deoxy-ribonucleosides
Synthesis of Polyhydroxyindolizidines from Carbohydrates
Nickel-Catalyzed Trifluoromethylation of Electron-Rich Heteroarenes
Synthesis of 3,4-Dihydroquinazolinones from 2-Aminobenzaldehydes
Synthesis of 6-Phosphorylated Phenanthridines
Synthesis of Pyrroloquinolinones from Donor–Acceptor Cyclopropanes
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Issue 01/2017

Synthesis of 3,3-Diaryloxetanes from Oxetanols by a Friedel–Crafts Reaction
Selective Functionalization of Pyridines via Their Phosphonium Salts
Synthesis of Epoxides by a Darzens Reaction and Vicarious Nucleophilic Substitution
Ytterbium(III)-Catalyzed Synthesis of Epiminodibenzo[b,f][1,5]diazocines
Synthesis of Pyrrolidines, Pyrroles, and Carbazoles by Iridium Catalysis
Enantiospecific Access to Bicyclic Morpholines and Piperazines
Rhodium(III)-Catalyzed Synthesis of Benzo[a]carbazoles
Synthesis of Azetidines by Ring Opening and Closing of Cyclopropanes
Synthesis of Substituted Pyrroles from α-Iminodiazoacetates
Enantioselective Synthesis of Spirooxindole 2H-Azirines
Photochemical [2+2]-Cycloaddition Route to Enantiomerically Pure Oxetins
Synthesis of Polyfunctional Pyrrolidines, Pyrrolines, and Thioxopyrrolidines
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Issue 12/2016

Organocatalytic Approaches to Highly Functionalized Piperidines
Copper-Catalyzed Synthesis of Quinazolinones
Aza-Annulation by C–H Arene Amination with O-Sulfonylhydroxyamines
Interrupted Ugi Reaction in the Synthesis of Spiroindolines
Synthesis of Iodo(trifluoromethyl)isoxazoles from Terminal Alkynes
Modular Assembly of Fused Polycyclic Pyridines
Nickel/Iridium Co-photocatalyzed C(sp3)–H Arylation
Rh-Catalyzed Synthesis of Cinnolines from Phenylhydrazines and Diazo Keto Esters
Photochemical C–H Amidation of Heteroarenes with N-Centered Radicals
Stereoselective Preparation of Substituted Oxetanes
Scandium(III)-Catalyzed Enantioselective Synthesis of Benzimidazoles
Synthesis of Phenanthridinone Derivatives by C–H Arylation
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Issue 11/2016

Isochromanone Synthesis by NHC-Catalyzed Annulation of o-Quinodimethanes
Cobalt(III)-Catalyzed Synthesis of Quina-zolines from Benzimidates and Dioxazolones
Nitro Epoxide Based Synthesis of Morpholines and Benzoxazines
Copper-Catalyzed Synthesis of Isoxazoles from Nitroalkanes and Alkynes
Palladium-Catalyzed Synthesis of Quinazolinone-Fused Phenanthridines
Selective sp2–sp3 Suzuki–Miyaura Coupling of Heteroaryl Chlorides
Gold-Catalyzed Synthesis of Imidazolidines and Tetrahydro-1H-1,3-diazepines
Lewis Acid Catalyzed Synthesis of Azepines from Oxiranes and Alkynes
Synthesis of Indolizidine Lactams by Reductive Cyclization of Cyclic Imides
Synthesis of 1-Aryl-1,2,3,4-tetrahydroiso-quinolines via Aryne Intermediates
Copper-Catalyzed Synthesis of Benzofuran[3,2-c]quinolin-6[5H]-ones
Synthesis of Hetaryluracils
Asymmetric Synthesis of Pyrrolizines
Photocatalytic Synthesis of (Trifluoromethyl)phenanthridines
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Issue 10/2016

Photocatalytic Azolylation of (Het)arenes
C2-Alkylation of Pyridine N-Oxides with 1,1-Diborylalkanes
Photoredox-Catalyzed Aryl Aminations with Ligand-Free Nickel(II) Salts
Rhodium(III)-Catalyzed C–H Activation Route to 1H-Isoindoles
Cobalt-Catalyzed Cross-Coupling Route to Homoallylic Alcohols and Amines
Enantioselective Synthesis of Pyrrolidines by Aminotrifluoromethylation of Alkenes
Directed Decarboxylative Cross-Coupling Route to Piperidines and Pyrrolidines
Synthesis of Perfluorinated Isochromene Derivatives by Ring Expansion
Synthesis of 3-Aminofurans from 1,2,3-Triazoles and Propargylic Alcohols
Sulfonated β-Cyclodextrin-Catalyzed Synthesis of Imidazopyridinamines
Gold-Catalyzed Synthesis of 1,5-Benzodiazepines
Synthesis of Fused and Spiro Dihydrobenzofurans
Synthesis of Isoquinolones and Isocoumarins by a Suzuki–Miyaura Coupling
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Issue 09/2016

Synthesis of Palbociclib: An SNAr Reaction on a Kilogram Scale
Pyrimido[4,5-d]pyridazines by the Reaction of Pyrimidines with Tetrazines
Four-Component Synthesis of 1-Pyrimidin-2-yl-3,4-dihydropyridin-2(1H)-ones
Synthesis of Trifluoromethylated Isoxazoles by [2+3] Cycloaddition
Synthesis of Azabicycloalkanes by Gold(I)-Catalyzed Amination of Ynones
Microwave-Assisted Synthesis of 1-Arylnaphtho[2,1-b]furans
Regiocontrolled Synthesis of Benzo-Fused (Hetero)aromatics from Dihydrofuran Acetals
Copper(I)-Promoted Synthesis of Halogenated Tetrahydrothiophenes
Synthesis of Pyrrolidines and Piperidines with Tin Amine Reagents
Synthesis of Oxindoles from α,β-Unsaturated Amides and Aldehydes
Rhodium-Catalyzed Synthesis of Fused Heterocycles
Synthesis of Functionalized 1,4-Oxazines by Activation of Diazoenals
Functionalized Isoquinolines by Rh(III)-Catalyzed C–H Conjugate Addition
Synthesis of 2-Quinolinones by Lactamization of 2-Alkenylanilines with CO2
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Issue 08/2016

Minisci-Type Reaction of Nonactivated Ethers with Heterocycles
Fluorinated Triazoles by Using a Heterobifunctional Fluoroalkylation Reagent
1,3-Dipolar Cycloaddition of Azomethine Imines with Enecarbamates
Synthesis of Chiral Piperazinones from Aziridine Aldehyde Dimers
[3+2] Cycloaddition Route to Imidazopyrrolo-Fused Isoxazoles
Synthesis of Enantiomerically Enriched Isoquinoline Derivatives
Synthesis of Pyrroles by Rhodium-Catalyzed Hydroacylation of Alkynylamines
Synthesis of 3-Bromoquinoline-2(1H)-thiones
Functionalized Arynes from Aryl Iodonium Salts
Four-Component Palladium-Catalyzed Synthesis of Pyrroles
Palladium-Catalyzed Synthesis of (Spiro)polyheterocycles by Domino Post-Ugi Route
Halogenated Piperidines and Tetrahydropyrans by the Prins Reaction
Palladium-Catalyzed Synthesis of Phenanthridinones by Dual C–H Activation
Heteroannulation Route to Fluorinated Purine Derivatives
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Issue 07/2016

Synthesis of 6-Amino-2,3-dihydro-4-pyridones from Homoallylamines
O-Benzoylhydroxylamine-Promoted Electrophilic Amination of Alkenes
Azaarenes by Palladium-Catalyzed α-Arylation of Ketimines with Aryl Sulfides
Three-Component Aryne-Mediated Synthesis of Dibenzooxazonines
Regioselective Preparation of Tetrazoles without the Use of Azides
Pd-Catalyzed Selective 2-Amination of 2,4-Dichloro-5-(trimethylsilyl)pyrimidine
Three-Component Synthesis of Benzo[e]pyrazolo[1,5-c][1,3]thiazines
Pyrrolidines by Coupling of Olefins with β-Aminoethyl Trifluoroborates
Regiodivergent Synthesis of Dihydroquinolines and Chromenes
Synthesis of 6-Perfluoroalkylated Bicyclic 1,2,3-Triazolo-1,4-oxazines
Tricyclic Indoles by Sequential Friedel–Crafts/Allylic Amination Reactions
Synthesis of 2H-Indazole-Fused Tetrahydroisoquinolinoquinoxalines
Ir-Mediated Cascade Approach to Chiral Indole-Annulated Medium-Sized Rings
Polyfunctional Alkenyl Organometallic Reagents for Heterocycle Synthesis
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Issue 06/2016

Benzofurans from β-Pyrones and Phenols
4-Bromo-1,2-dihydroisoquinolines from ortho-Triazolylbenzyl Bromides
Lewis Base-Catalyzed Dynamic Kinetic Resolution of Azole Esters
Synthesis of Indazoles by Oxidative N–N Bond Formation
Benzoxazocindiones from Phthalic Acids and Cyclic Sulfamidates
Palladium-Catalyzed Three-Component Synthesis of 2-Aroylbenzofurans
Tetrahydronaphthyridines by a Radical Pictet–Spengler Reaction
Pyrrolizidines and Indolizidines by Photooxidation of Furylalkylamines
Enantioselective Synthesis of Piperidines from Pyridines
Three-Component Synthesis of Pyrazolo [3,4-d]thiazolo[3,2-a]pyrimidines
Triazole–Gold Catalyzed Approach to Substituted 2,3-Dihydrooxepines
Copper-Catalyzed C–N Coupling/Madelung Synthesis of Indoles
Direct Ketone Synthesis by Hetaryl Grignard Addition to Carboxylic Acids
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Issue 05/2016

Multicomponent Diastereoselective Synthesis of Tetrahydropyridines in Aqueous Micelles
Reductive Fischer Indole Synthesis from N-Aryl Conjugated Hydrazones
Stereocontrolled Late-Stage Remote Arylation of Bioactive Saturated N-Heterocycles
Imidazopyridines by SNAr Addition of Metalated Isonitriles to 2-Chloro Heterocycles
Synthesis of Fluorinated Indoles by Oxidative Dearomatization of Anilines
DDQ-Promoted C–H Activation Approach to Pyrrolidine Alkaloids
SN2′/SNV Reactions in the Synthesis of 2-Fluoro-2-pyrrolines
Synthesis of Medium-Ring S,N-Heterocycles Using a Dithiadiazocane
Synthesis of Strained Heterocycles by Flow Photochemistry
Rhodium-Catalyzed Synthesis of Indoles from Imidamides and Diazo Keto Esters
Palladium-Catalyzed Synthesis of Difluoromethylthiolated Heterocycles
Photoredox Synthesis of 3,3-Difluoroindol-2-ones
Ligand-Free Palladium-Catalyzed Synthesis of Carbazoles
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Issue 04/2016

Copper-Catalyzed Synthesis of Substituted 1,4-Oxathianes
Piperazines by Palladium-Catalyzed Reactions of Propargylic Alcohols
Tetrafluoroimidazopyridines by Radical-Mediated Annulation
Synthesis of Pyridinyl and Quinolinyl Triflates or Tosylates by Diazotization
Biomimetic Photocatalytic C–H Activation Route to Coumarins
γ-Lactams by Palladium-Catalyzed Intramolecular C(sp3)−H Alkenylation
Iodine-Mediated Synthesis of Pyrido[1,2-a]benzimidazoles
Synthesis of (Aminoalkyl)boronates from Cyclic Sulfamidates
Spiropyrazolones by Sequential Michael and Conia–ene Reactions
Isoquinolinium, Cinnolinium, and Quinolizinium Salts by Oxidative Annulation
Synthesis of 3-Fluoropyrroles by Ring-Closing Metathesis
Synthesis of Propellane, Azetidine, and Cyclobutane Amines
Synthesis of Indolines by an Iron-Catalyzed (4+1) Cycloaddition
Fluorinated 4H-1,4-Thiazine 1,1-Dioxides
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Issue 03/2016

Synthesis of Dihydrofurans from β-Ketocarbonyl Compounds and Olefins
Synthesis of Oxazinanones from β-Lactams by Amide Bond Activation
Tetrahydroquinolines by Michael Addition/Nitro-Mannich Reaction
Palladium-Catalyzed Heteroannulation Route to (E)-Oxindolylideneacetates
Aldehyde Allylation/Cyclization with Isocyanato Allylboronic Esters
Enantiopure α-Substituted Piperazines by Asymmetric Lithiation−Trapping
Gold-Catalyzed Synthesis of 7-Acylindoles from Anthranils
Synthesis of Fluorinated Thiophenes by Ring Contraction of Thiopyrans
Synthesis of 1-Benzyl- or 1-Benzoyliso-quinolines by Dehydrogenative Coupling
Palladium-Catalyzed Synthesis of Difluoroalkylated Phenanthridines
Pd-Catalyzed Arylation/[1,2]-Wittig Rearrangement of Pyridylmethyl Ethers
Synthesis of Imidazo[1,2-a]pyridines by 1,3-Dipolar Cycloaddition
Synthesis of Pyrrolopyridines from 3-Aminopyrrole
Synthesis of Benzoxazoles by Copper/Palladium Catalysis
Three-Component Synthesis of Oxazolidin-2-ones
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Issue 02/2016

Multicomponent Reaction/Staudinger/aza-Wittig Synthesis of 2H-Pyrrolo[3,4-c]quinolines
Palladium-Catalyzed Carbonylative C–H Functionalization of Heterocycles
Synthesis of Cyclic Amino Boronates from Boryl Sulfamate Esters
Synthesis of N-Methyliminodiacetic Acid Boryl Heteroaryls
Synthesis of α,β-Epoxy Ketones by Ruthenium-Catalyzed Oxidative Coupling
Triarylantimony-Catalyzed Heteroannulation Route to 2-Arylquinoxalines
Stereoselective Synthesis of Tetrahydro-benzofuranones with Lewis-Base Catalysis
Rhodium/Scandium-Catalyzed Synthesis of Dihydronaphthofurans
Synthesis of Substituted Isatogens and Oxindoles
C–H Activation Route to Isoxazolinones and β-Lactams
[3+2] Cycloaddition Route to Spiropyrrolidin-2-ones
Palladium-Catalyzed Synthesis of 2-Alkenyl-3-arylindoles
Heteroannulation Route to Imidazo[1,2-a]pyridines
Synthesis of Tetrahydrofurans and Pyrrolidines from β-Hydroxy or β-Amino Ketones
Palladium-Catalyzed Benzylic Arylation of Azaarylmethylamines
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Issue 01/2016

Synthesis of Benzo[1,3]oxathiins from Benzobisthietes
Enantioselective Propargylation of Cyclic N-Sulfonylketimines
Palladium-Catalyzed Synthesis of Ring-Fused Benzosultams and Benzosultones
Oxidative Cross-Dehydrogenative Coupling of N-Heterocycles with Aldehydes
Rhodium-Catalyzed C-7 Functionalization of Indoles
Three-Component Synthesis of Dihydropyridopyrimidines
Synthesis of Substituted Isoquinolines from Aryl 1,2,3-Triazoles
Cobalt(III)-Catalyzed Synthesis of Isoquino-lines from O-Acyl Oximes and Alkynes
Ruthenium-Catalyzed Synthesis of Hydroxybutenolides
Convenient Access to Sulfinyl Derivatives of Heterocycles
Palladium-Catalyzed Enantioselective Synthesis of Benzoxazinoindoles
Silver-Catalyzed Heteroannulation Route to Benzofuro- and Benzothienopyridines
Substituted 1,2,3-Triazoles by Copper-Catalyzed Cycloaddition/N-Alkylation
Enantioselective Synthesis of 1,2-Dihydro-pyridines by Formal [4+2] Cycloaddition
Synthesis of Oxazoles from Methyl Ketones and Amino Acids
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Issue 12/2015

Synthesis of Highly Functionalized Oxetanes
Acid-Catalyzed Synthesis of Carbazoles from Indoles and 2-Amidodihydrofurans
Synthesis of Six- and Seven-Membered Heterocycles
Synthesis of 2-Aminoindoles and 5-Amino-indolo[1,2-a]quinazolines
Nickel-Catalyzed Anti-Markovnikov Hydroheteroarylation of Nonactivated Alkenes
Synthesis of Cyclic Ethers by Alkoxylation of Nonactivated sp3 C–H Bonds
Manganese(I)-Catalyzed C–H Bond Amidation of Heteroarenes
Silver-Catalyzed Synthesis of 2-Aryl-5-(trifluoromethyl)tetrazoles
Imidazotetrazolodiazepinones by a Ugi–Azide Multicomponent Reaction
Rhodium Carbenoid-Catalyzed Synthesis of 2,5-Epoxybenzo[f][1,4]oxazepines
Potassium Persulfate Mediated Synthesis of Dihydrofurans
Oxidative Radical Decarboxylation Route to 6-Alkyl- or 6-Arylphenanthridines
Radical-Mediated Difluoromethylenephosphonation
Highly Substituted Pyrimidines by Multicomponent Reactions
Synthesis of Tetrasubstituted Furopyridazinones from Nitrile Imines
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Issue 11/2015

Synthesis of Spiroxindoles by Enantioselective [3+2] Annulation
Efficient Synthesis of 5-Nitro-7-azaindole on a Kilogram Scale
Substituted 7-Azaindoles by Directed Ortho Metalation/Nucleophilic Aromatic Substitution
Synthesis of Polyfunctionalized 1,4,2-Oxathiazoles by Oxidative Cyclization
Dihydroisocoumarin Synthesis by C–H ortho-Alkylation of Benzoic Acids
Copper-Catalyzed Asymmetric Synthesis of Thiazolidine-2-imines
Synthesis of Oxazoles from 2H-Azirines and Aldehydes by Photoredox Catalysis
Synthesis of Indoles by Reductive Cyclization of ortho-Nitrostyrenes
Ylidenemalononitrile Enamines in the Synthesis of Pyridines and Pyrones
Synthesis of Azetidin-3-ones from Allenes by Oxidative Amination
Synthesis of α-Hetaryl Nitriles by Asymmetric Reductive Cross-Coupling
Synthesis of Borazaroquinolines and Borazaroisoquinolines
Synthesis of Tetrasubstituted Furans by the Morita–Baylis–Hillman Reaction
Substrate-Controlled C-2 Amination of Dichloropyrimidines with Tertiary Amines
Asymmetric Synthesis of Heterocycle-Fused Butyrolactones
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Issue 10/2015

Synthesis of Fused Imidazobenzodiazepinones by Ugi Reaction
Oxabicycles from Gold-Catalyzed Prins-Type Cyclization of Enynols
Nickel-Catalyzed Asymmetric Synthesis of Axially Chiral Isoquinolones
Enantioselective Synthesis of Chiral Fluorinated Isoindolinones
Synthesis of Oligocyclic Dienes by anti-Carbopalladation–Heck Reaction
Copper-Catalyzed Synthesis of Phosphonylated Quinoline-2,4-diones
Synthesis of Pyrazolo-triazolo[1,4]oxazepines by [2+3] Cycloaddition
Palladium-Catalyzed Synthesis of Dibenzofurans from 2-Iododiaryl Ethers
Synthesis of Pyrazoles from N-Propargyl Hydrazones Mediated by tert-BuOK
Four-Component Reaction Approach to Uracil Analogues
Lewis Acid Catalyzed Synthesis of Di/Trifluoromethyl-1,2,3,4-Tetrahydroquinazolines
Gold-Catalyzed Synthesis of 2-Aminoindoles and β-Carbolines
New Biocatalysts for the Efficient Synthesis of Enantiopure N-Heterocycles
Synthesis of 2-Azabicyclo[3.2.0]hept-2-enes and Pyrroles from Aza-enynes
Synthesis of Trisubstituted Isoxazoles from Morita–Baylis–Hillman Acetates
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Issue 09/2015

Synthesis of Isoxazolino Phenanthridines
Morpholines and Spirocyclic Dihydrofurans from Oxetanyl N,O-Acetals
Synthesis of Dihydro-1H-benzothiazolopyridines by NHC Catalysis
Azaquinolizinium Salts by Ring-Closing Metathesis
Formal Hydroamination of Alkenes with Nitro- and Heteroarenes
Radical-Mediated Annulations of Benzene-Linked 1,n-Enynes
Optimized Process Route to a Benzoxazepine-Derived Kinase Inhibitor
Metal-Free Synthesis of Perfluorinated Oxindoles
Selective Synthesis of 3- or 5-Substituted Aminopyrazoles
7-Azaindoles via Rhodium(III)-Catalyzed C–H Activation–Annulative Coupling
Aminodifluoromethylation of Unactivated Alkenes
Stereodivergent Synthesis of Substituted Tetrahydrofurans
Pyrroles and Oxazines via Cycloaddition of Borodienes with Nitrosoarenes
A Radical Oxidative Annulation Route to Dihydrofurans and Indolizines
Synthesis of Benzazoles Catalyzed by Sodium tert-Butoxide
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Issue 08/2015

Synthesis of Cyclic Imines from Acetals/Ketal and Cyclic Sulfamidates
Copper-Catalyzed Synthesis of Imidazopyridines
Synthesis of Phenanthridines by Reaction of 2-Acetylbiphenyls with TMSN3
Stereoselective Cascade Reactions to Fused Heterocycles from Allenes
Synthesis of Pyrazole-Fused Coumarin Derivatives using Copper Catalysis
Copper-Catalyzed Synthesis of 2-Imidazolidinones from Biaziridines
1,2-Oxazetidines: Synthesis, Characterization, and Synthetic Applications
Snieckus, Victor; Gomes, Sara: Hydrazones as Dienophiles in Inverse Electron Demand Diels–Alder Reactions
Palladium(II)-Catalyzed Synthesis of Polyheterocycles
Cobalt-Catalyzed Synthesis of Indenoisoquinolinones
Enyne Cross-Metathesis Approach to 1,2,3-Trisubstituted Pyrroles
Synthesis of Oxygen-Bridged Bicyclic Ethers by Prins Cyclization
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Issue 07/2015

Rhodium(III)-Catalyzed Synthesis of 1,2-Benzothiazines
Enantioselective Copper(I)-Catalyzed Construction of Spiroketals
6-endo-dig versus 5-exo-dig. The Profound Effects of Acetonitrile
Synthesis of Dihydropyridin-2-ones via an Ugi–Aldol Reaction
Minisci-Type Synthesis of Tetrahydropyridopyridazines
Single-Step Synthesis of Isoindolinones
Synthesis of Fluorinated Diphenylpyrazole
Four New Bonds in One Pot: Isoxazolines from Olefins and 2-Ethylquinolines
Pyrido[2,3-c]coumarins via an Intramolecular Povarov Reaction
Synthesis of 1,2-Borazaronaphthalenes
Benzyne Route to Benzothiazoles
Copper-Catalyzed Oxidative Annulation Approach to Oxadiazoles
Enamide Umpolung for the Synthesis of Heterocycles
Oxabicycles via Sequential Prins–Wagner–Ritter Processes
Synthesis of Hexahydropyrano[3,4-c]chromenes via Prins Bicyclization
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Issue 06/2015

Pd-Catalyzed Ortho-Amination/ipso-Functionalization of Aryl Iodides
Catalytic Enantioselective Piperidine Synthesis by [4+2] Cyclization
Stereoselective Intramolecular [3+2] Annulations to Fused Heterocycles
Synthesis of Fluorine-Containing 3-Hydroxypyridin-4-ones
Quinoxalines from Pyrroloarylisocyanide by Photoredox Catalysis
Synthesis of Heteroring-Annulated 1,4-Oxazepines
Chirality Transfer in the Synthesis of Pyrrolidines
Thia-Prins Cyclization Approach to Tetrahydrothiophenes and -furans
Three-Component Synthesis of Fluorinated Pyrazoles
2-Picolylamines and Imidazopyridines from Pyridotriazoles by Rh(II) Catalysis
Palladium-Catalyzed Route to Ortholactones from Cyclic Enol Ethers
Synthesis of Benzo[b]thiophenes by Sequential Cyclization Reactions
Multicomponent Synthesis of Benzopyrans
In Situ Generation of Difluoromethyl Diazomethane. Synthesis of Pyrazoles
Iron-Catalyzed Synthesis of Isoxazoles from Homopropargylic Alcohols
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Issue 05/2015

Modular Assembly of Imidazoles by 1,3-Dipolar Cycloaddition
Construction of Aza/Oxa-Spirocyclic Skeletons. Formal Synthesis of (±)-Halichlorine
Polycyclic Spiroindolines from Asymmetric Dearomatization of Indoles
1,4-Benzothiazines by Copper-Catalyzed Ring Expansion of Benzothiazoles
Synthesis of Dibenzothiazepine Dioxides by Reductive Heck Cyclization
Synthesis of Pyrroles and Dihydropyrazines from Azirines and 1,2,3-Triazoles
One-Pot Cycloaddition–Strecker Cascade to Imidazo[1,2-a]heterocycles
Trifluoromethylthiolation of Indoles
Synthesis of F5C2-Substituted Pyrazoles
Carbonylated Benzofurans by Metal-Free Radical Cyclizations of 1,6-Enynes
Synthesis of Substituted Pyrroles and 1,2-Oxazinanes
An Unexpected Route to Pyrrolo[2,3-c]pyridazin-6-ones
A Photoredox Approach for the Synthesis of Pyrrolidine-2-ones
Functionalized Azides for the Synthesis of Pyrrolidin-2-ones and Pyrroles
Copper-Mediated Synthesis of 3-Chloro-4-iodoisoxazoles
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Issue 04/2015

Atom-Efficient Organolanthanide 1,2-Dearomatization of Pyridines
Arene–Ynamide Cyclization Approach to Pyrroloquinolines
Imidazoles and Imidazoliums from Propargylamines and Isonitriles
Diastereoselective Synthesis of Fluorinated Amino-Sugars
Synthesis of Fused Indoles and Pyridin-2-ones by Radical Cyclization Cascades
Synthesis of Polyfluoro-1,3-thiazine Derivatives
Preparation of Pyrido[3,4-d]azepines by Pyridine Ring Heteroannulation
Synthesis of Dihydropyrazines from N-Sulfonyl-1,2,3-triazoles and Aziridines
Palladium-Catalyzed Heteroannulation Route to Azaindoles
Rhodium-Catalyzed Directed Halogenation of π-Excessive Heterocycles
Sultams by Arylation of Cyclic N-Sulfonyl Aryl Alkyl Ketimines
Ruthenium-Catalyzed Synthesis of 1,4-Benzodiazepines
Seven-Membered Heterocycles by Chlorosilane-Catalyzed Heteroannulation
Synthesis of Enantioriched δ-Lactones from β-Halo-α-keto Esters
Rhodium-Catalyzed Oxidative Annulation Route to 1-Aminoindolenines
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Issue 03/2015

Palladium-Catalyzed Synthesis of Isatins from Anilines by Double Carbonylation
Microwave-Assisted Synthesis of Pyrazolotriazines
Multicomponent Synthesis of 3-Arylmethyl-2,5-diarylthiophenes
Benzimidazole-Fused Thiadiazoles From ortho-Phenylenediamine Dithioureas
Preparation of Spirocyclic N-Heterocycles Utilizing Stannyl Amine Reagents
Difluoro-oxindoles by C–H Bond Difluoro-alkylation of Chlorodifluoroacetanilides
Aminoindolines and -indoles by Rhodium-Catalyzed C–H Bond Activation
Synthesis of Fused Pyridines by a ZnCl2-Promoted Three-Component Reaction
Spiro[indene-1,2′-pyrrolidene] by [3+2] Annulation of Pyrroles with Alkynes
Asymmetric Synthesis of Dihydropyridinones and Derivatization
A Hydroheteroarylation Route to 2-Substituted Benzoxazoles
Metal-Free Tandem Oxidative Acylation–Cyclization to Coumarins
6-Trifluoroethylphenanthridines by Photoredox Reaction
Highly Substituted Pyrazoles from N-Propargyl Hydrazones
Indium-Catalyzed Intramolecular Hydroarylation Route to 2H-Chromenes
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Issue 02/2015

Copper-Promoted Synthesis of Pyrimidines by Dimerization of Amino Esters
Indolines by Heck Reaction, C–H Activation, and Amination with Diaziridinones
Synthesis of 1,6-Annulated 2-Pyridones by Nickel-Catalyzed Hydroarylation
Rhodium(II)-Catalyzed Synthesis of Fused Azepine Derivatives
Preparation of 2,5-Dihydroazepines from Dienyltriazoles by [4+3] Cycloaddition
Dihydrofurans and Dihydroindoles by Annulation of Tethered Triazoles
Rhodium(III)-Catalyzed Synthesis of 2H-Chromenes
Prins Reaction–Pinacol Rearrangement Route to Oxaspiro[4.5]decan-1-one
Quinolines from the Reaction of o-Halo N-Arylhydroxylamines with Olefins
Cu(I)- and Pd(II)-Catalyzed Synthesis of Functionalized Imidazo[1,2-a]pyridines
Copper/NHC-Catalyzed Synthesis of 1,4-Diarylimidazoles from Isocyanides
Palladium-Catalyzed Synthesis of Oxazoles and Thiazoles
Synthesis of 7-Trifluoromethylpyrazolo[1,5-a]pyrimidines
Synthesis of Octahydro-2H-chromenes via Prins Reaction–Arylthiolation
Stereoselective Synthesis of l-Rhamnose-Derived Fused Triazoles
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Issue 01/2015

Pd-Catalyzed Synthesis of N-Aryl Indoles
Direct Cyclization–Trifluoromethylthiolation to 4H-Chromen-4-ones
Rhodium(I)-Catalyzed [4+2]-Cycloaddition Route to 1,2-Dihydropyridines
One-Pot Diastereoselective Synthesis of Azabicyclo[2.2.2]octanes
Aziridine and β-Lactam Synthesis by Amination and Carbonylation Reactions
Tetrahydrofurans and Pyrrolidines from N-Tosylhydrazones via C–H Insertion
Copper(I)-Catalyzed Synthesis of 3-Amino-2-pyrones and 2,5-Dihydrofurans
Auto-Oxidation–Povarov Annulation Approach to Quinolines
Synthesis of Indoles, Pyrazoles, and Pyridazinones
NHCs in Rhodium-Catalyzed C–H Activation–Annulation to Fused Imidazolium Salts
Iron-Mediated Synthesis of Pyrroles from Cyclopropanes
Synthesis of 2-Aminothiophenes from Alkynoates and Thioamides
An Improved Procedure for a Pd-Catalyzed Amidation Approach to Imidazopyridines
Enantioselective Synthesis of 3,4-Dihydrothiacarbazol-2(9H)-ones
Copper-Catalyzed Amidation of π-Excessive Heterocycles
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Issue 12/2014

Synthesis of Imidazo-Fuzed Heterocycles via Gold-Catalyzed Cycloaddition
Inverse-Electron-Demand Diels–Alder Reaction of Asymmetric 1,2,3-Triazines
Pyridazines via an Organophosphorus-Catalyzed Diaza-Wittig Reaction
Palladium-Catalyzed Synthesis of Quinolines From Cyclopropanols
Catalyst-free Synthesis of 1-Aryltetrazoles
Synthesis of Phenanthridines from Diaryliodonium Salts and Nitriles
Synthesis of Oxazinoindoles and Pyrrolooxazines by Sc(III) Catalysis
Amidation–Oxidative Cyclization Route to 2-Aryl-2H-benzotriazoles
Fused Isoquinolones by Aryne/Alkyne Insertion into C–H/N–H Bonds
ArI-Catalyzed Synthesis of Benzolactones
Copper-Catalyzed Synthesis of 1-Bromoindolizines from Pyridines
Enantioselective Synthesis of Pyrrolidinones and Dihydropyridinones
A Photocatalytic Hydroamination Route to Dihydropyrazoles
Synthesis of 1,4-Thiazepin-5(4H)-ones without Transition Metals
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Issue 11/2014

Spirocyclic and Ring-Expanded Fused Pyrazoles
Synthesis of Aminotriazoloazepinone-Containing Di- and Tripeptides
N-Aryl Heterocycles by Catalytic Photoredox Olefin Hydroamination
Synthesis of the SF5 Analogue of Umemoto Salt
An Organocatalytic Cascade Route to Functionalized Azepines
Iron-Catalyzed Synthesis of Difluoromethylsulfonylated Oxindoles
Quinoxaline N-Oxides by Dehydrogenative N-Incorporation of Imines
Synthesis of Spiroaminals by Au/Sc Relay Catalysis
NHC-Promoted Annulation Approach to Pyranyl Aldehydes
C-8 Alkylation and Alkynylation of Quinoline N-Oxides by Rhodium Catalysis
Copper-Catalyzed Synthesis of Dibenzodiazepinones
Copper-Catalyzed Synthesis of Sulfonylated Oxindoles
Synthesis of Benzotriazoles from 2-(Arylamino)aryliminophosphoranes
Synthesis of Heterocycles by Palladium-Catalyzed Intramolecular C–H Amination
Three-Component Reaction Approach to Aminopyrazoles and Iminopyrimidines
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Issue 10/2014

Stereoselective Synthesis of trans-Oxazolidinones via C–H Oxidation
CF3-Substituted Pyrazolines and Pyrazoles via Huisgen Cycloaddition
Manganese-Mediated Coupling Approach to Fused Lactone-Pyrrolidinones
1,3-Carbonyl Transposition of Ynones in the Context of Heterocyclic Chemistry
Synthesis of 1,3-Disubstituted Pyrimido-pyrimidinedithiones
Pyrrolideines via Cycloaddition of Silyl Ketene Acetals to Metallocarbene Precursors
Mild C–H Activation of Tethered Alkynes for the Synthesis of 3,4-Fused Indoles
Pyrroloquinolinones by Cascade Nitration–Cyclization of 1,7-Enynes
Bisheterocycles via Rh(III)-Catalyzed C–H Activation–1,3-Diyne Coupling Route
Isoindoloquinazolinones by Palladium Catalysis
Synthesis of Various Thia-2H-indazoles via the Davis–Beirut Reaction
One-Pot Synthesis of Fluorinated Thiadiazolo[3,2-a]pyrimidin-7-ones
Safe and Scalable Preparation of 2-Nitropyrroles
Phenanthridinones via Benzyne Intermediates Using Palladium Catalysis
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Issue 09/2014

Synthesis of Bioactive Nucleoside Analogues
2,3-Dihydro-1H-indazoles by Rhodium Catalysis
C–H Fluorination and Nucleophilic Aromatic Substitution of Nitrogen Heterocycles
2H‑Indazoles by Condensation−Cadogan Reductive Cyclization
Pd/C-Catalyzed Synthesis of 2-Substituted Benzothiazoles
Diastereoselective Preparation of Enantioenriched Polycyclic Oxoquinolines
Intramolecular Aryl–Aryl Coupling of 2-Substituted N-Phenylbenzamides
Synthesis of 1,3-Oxathiolan-2-ylidenes from α-Enolic Dithioesters and Epoxides
Synthesis of Oxepines by Cycloisomerization of 1,7-Oxadienes
Biomimetic Synthesis of Symmetrical Tetrasubstituted Pyrroles
Three-Component Synthesis of Fully Substituted Triazoles
Synthesis of Pyrroles by Photocatalyzed Cycloaddition of Alkynes to Azirines
C(sp2)–C(sp3) Bonds by Intramolecular Reductive Cross-Coupling
Fused Heterocycles via C–H Activation and Cyclization of Indoles and Pyrroles
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Issue 08/2014

Pyrrolo- and Pyrazolopiperidines by Stereoselective Organocatalysis
Synthesis of Benzofuro[2,3-c]pyridines
Multicomponent Synthesis of Thiazepines
Synthesis of 3-Substituted Isoxazole Derivatives Using Copper(II) Nitrate
Synthesis of Dihydropyrroles via Sequential Heck–Suzuki Reaction
Asymmetric Synthesis of 1,3-Oxathiolan-5-ones
Synthesis of Polysubstituted Benzofurans from 2-Alkynylphenols
Three-Component Synthesis of Fully Substituted Pyrazoles
Pyridoquinazolinones by Palladium-Catalyzed C–H Bond Activation
Copper-Mediated Synthesis of Fused Cyclopropylpyrrolidines
Three-Step Synthesis of 3-Phosphonopyrroles via Hydroamination
Regioselective Synthesis of Linear and Angular Pyridoquinazolones
Michael Addition–Reductive Lactamization Route to 5-Alkyl-5-aryl-γ-lactams
Isoquinolines by Manganese-Catalyzed Annulation of Aryl Imines with Alkynes
Synthesis of Perfluoroalkyl Pyrroles and Thiophenes from Cyclopropanes
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Issue 07/2014

Synthesis of Azepines by HSbF6-Catalyzed Cycloaddition of Aziridines with Acetylenes
F3C-Containing Phenanthridines by Palladium-Catalyzed Intramolecular Cyclization
Azoloquinazolines from ortho-Triazoloanilines Using an Isocyanide Linchpin
Asymmetric Arylative Cyclization of 5-Alkynones with Arylboronic Acids
Synthesis of β-Lactones via Intramolecular Rhodium-Catalyzed Cyclization
Synthesis of 4-Alkyl-2,3-difluorobut-2-enolides by Cyclization
Dihydro-oxazinones from Salicylamides
3-Methylene-1-pyrrolines from N-Propargylic β-Enaminones
Gold-Catalyzed Synthesis of Thiazoles via Methanesulfonyloxymethyl Ketones
Palladium-Controlled Regioseletive Arylative Cyclization of Alkynols to Cyclic Ethers
Hydroisoquinolines via Organocatalytic Diels–Alder/Nucleophilic Ring Closure
Heterocyclic-Fused Benzopyrans by Heck-Type Reaction
Synthesis of Trifluoromethyl-Containing Imidazoles
Transition-Metal-Free Synthesis of Indazoles and Azaindazoles
Triazolopyridines by Metal-Free Heteroannulation
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Issue 06/2014

Synthesis of N-Heterocycles via Rhodium(III)-Catalyzed C–H Activation
Cu- and Pd-Catalyzed Heteroannulation Route to Imidazo[4,5-c]pyridines
Benzofurans via Gold-Catalyzed Intramolecular Alkoxyboration of Alkynes
Synthesis of β-Lactams via Intramolecular Oxidative Amidation
Isoindolones via Intramolecular Amination of Benzylic C–H Bonds
Synthesis of Isoindolin-1-ones by sp3 C–H Bond Activation–Cyclization
Synthesis of Quinolinones via Aryne Insertion into C–S Bonds
Oxidative Coupling of Acrylic Acids and Amides with Alkynes
Two-Stage Chemoselective Methylation Method for Heteroarenes
Allylation–Radical Cyclization to Difluoromethylated Dihydrobenzoheteroles
Pyrroles from Terminal Alkynes, N-Sulfonyl Azides, and Alkenyl Alkyl Ethers
Palladium-Catalyzed One-Pot Synthesis of Oxazolopyrazines by Heteroannulation
One-Pot Four-Step Regioselective Preparation of Pyrazoles and Isoxazoles
Copper-Catalyzed Route to Azido-Substituted Isoxazolines
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Issue 05/2014

[3+2] Cycloaddition Route to Spirooxindoles
Synthesis of 1,2-Benzisoxazoles by Palladium-Catalyzed [4+1] Annulation
Synthesis of Trisubstituted Oxazoles via a Three-Component, One-Pot Reaction
Efficient C–C Aryl–Heteroaryl Bond Formation by Photoredox Direct Arylation
Pyrroles via Copper-Promoted Oxidative Coupling of Enamides with Alkynes
Construction of Fused Pyrroles from 1,3-Diones and N-Alkynylhydroxyamines
Rhodium-Catalyzed Synthesis of Polysubstituted Indoles from Styryl Azides
Synthesis of Functionalized Pyrroles by a Multi-Component Reaction
One-Pot Asymmetric Synthesis of 2,3-Dihydropyrroles
Ruthenium-Catalyzed Synthesis of Lactams from Cyclic Amines and Water
Rhodium-Catalyzed Synthesis of β-Naphthols and Indenes
Synthesis of Spiromorpholinotetra-hydropyrans Through a Prins Bicyclization
Oxa- versus Thia-Selectivity in the Prins Cyclization
Transition-Metal-Free Synthesis of 1,4-Benzodiazepinones
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Issue 04/2014

New Route for the Construction of Indoles from Anilines and Epoxides
Synthesis of Benzisoxazolones by Ruthenium and Copper Catalysis
Transition-Metal-Free Synthesis of Carbazoles from 2-Nitrobiaryls
Synthesis of Annulated P-Heterocycles
One-Pot Synthesis of Carbazole-1,4-quinones
Asymmetric Synthesis of Highly Substituted Pyrrolidines via [3+2] Cycloaddition
Two-Step Synthesis of Benzimidazoles from Nitrosoaromatics
Palladium-Catalyzed C–H Activation Route to β‑Lactams
Synthesis of Pyrrolooxazoles by a [3+2] Cycloaddition Route
Synthesis of 3,4-Carbocycle-Fused Indoles by Rhodium Catalysis
Functionalization of Imidazoles via Metalation and Sulfoxide–Magnesium Exchange
β-Lactams from N-Allylamines Using Palladium Catalysis
One-Step Synthesis of 2-Sulfonylbenzofurans
Synthesis of Pyrazolopyrimidines from 1,2-Allenic Ketones and Aminopyrazoles
Multicomponent and Solvent-Free Synthesis of Pyrimidines From Ketones
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Issue 03/2014

Intramolecular Ene Synthesis of 3-Pyrrolines
Spiroaminals and Spiroketals via Au/La and Au/Y Relay Catalysis
Synthesis of Pyrazoles via Nickel-Catalyzed Cyclotrimerization
Synthesis of Oxazolones by a β-Selective Oxidative Heck Coupling
Iridium-Catalyzed Route to Enantioenriched Tertiary Alcohols and Thioethers
Synthesis of Dihydroimidazoles and Quinazolinones via C–H Amination
Multicomponent Synthesis of Aza-Dibenzazepines Catalyzed by Rh/Pd
Synthesis of 3,5-Diphenyl-1H-pyrazoles by Mechanochemical Ball Milling
Synthesis of 1,3-Oxazin-6-ones from Enamides Catalyzed by Palladium
1,3-Cycloaddition Route to 1,2,3-Triazoles Catalyzed by Copper
Variation of the Pictet–Spengler Synthesis of Tetrahydrocarbolines
Gold-Catalyzed Synthesis of Tetrazoles from Alkynes
Synthesis of 3H-Pyrrolo[2,3-c]quinolin-4(5H)-ones Using ToSMIC Derivatives
Substituted α-Amino-β-Lactams via Sequential C–H Arylation/C–H Amidation
Diastereoselective Synthesis of Dibenzo[c,e]azepines
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Issue 02/2014

Heteroannulation Route to Benzofurans
Three-Component Synthesis of Rhodanines on Nanoporous Silica
Synthesis of Benzofuranones from Alkynyl Aryl Ethers
Transformation of Sulfonylpyrroles into 6-Azaindoles
Iron(III) Chloride Catalyzed Synthesis of Spirocyclic Pyrimidinones
Ir(III)/Bi(OTf)3-Catalyzed Prins Route to Pyran-Fused Indoles
Synthesis of Substituted Thiophenes from Polyhalogenated Nitrobutadienes
Palladium-Catalyzed Heteroannulation Route to 3-Trifluoromethylbenzofurans
Rhodium-Catalyzed Synthesis of Furo[2,3-b]pyran-6-ones
Synthesis of 2,5-Dihydrofurans via a Petasis Borono-Mannich Reaction
Rhodium-Catalyzed ortho-C–H Acylation Route to 3-Alkylidenephthalides
Synthesis of 1,3-Thiazin-2-ones via an Asymmetric Hetero-Diels–Alder Reaction
Asymmetric Organocatalytic Synthesis of 2,6-Diazabicyclo[2.2.2]octanones
C4-Alkenylation of 3-Formyl Indoles via Ruthenium(II)-Catalyzed C–H Activation
Synthesis of Piperazines via Gold-Catalyzed Cyclization of Propynyl Diamines
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Issue 01/2014

Synthesis of 2-Trifluoromethylquinolines via a [2+3] Cycloaddition
Iodine-Mediated 1,3-Dipolar Cycloaddition to Benzo(f)isoindole-4,9-diones
Three-Component Synthesis of (Pyrrolo)quinazolines
Synthesis of 6-Trifluoromethyl-Phenanthridines from Diaryl Isonitriles
Synthesis of Fused Imidazole–Chromenone and –Quinolone Derivatives
C2-Substituted Indoles via Ruthenium-Catalyzed C–H Bond Functionalization
Synthesis of 1,2,3-Triazoles from N-Tosylhydrazones and Anilines
Synthesis of 5-Arylfuranones via a Carbonylative Heck Reaction
Hydroarylation Approach to Phosphacoumarins
Asymmetric Organocatalytic Synthesis of Lactams and Lactones
Polycyclic Imines via Radical Cyclization of Ene Sulfonamides
Synthesis of Phosphaisocoumarins via Ruthenium Catalysis
Three-Component Route for the Regioselective Construction of N-Arylbenzimidazoles
Construction of Spirocyclic Oxindoles for Indole Alkaloid Synthesis
Aza-Morita–Baylis–Hillman Synthesis of Benzoxazepines
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Issue 12/2013

Diels–Alder Reaction–Fragmentation of Pyridinium Salts and Alkynes
Synthesis of 2-Fluoropyrroles from gem-Difluorocyclopropyl Ketones
Gold-Catalyzed Synthesis of Furan-3-ones via [2,3]-Sigmatropic Rearrangement
Synthesis of Imidazoquinolone Carbonitriles from Tetracyanoethylene
Rh(III)-Catalyzed Regioselective C–H Activation Route to Naphthyridinones
Metalation of 7-Azaindoles
Silver-Catalyzed Synthesis of Oxindoles
Radical Spirocyclization Route to Spirooxindoles
Pyrrolo[2,3-d]pyrimidines Through Activation of N-Benzyl Groups by Distal Amides
Pd-Catalyzed C–H Activation Route to Hydroxy Isoindolones
Synthesis of Pyrido[1,2-b]indazoles from the Reaction of 2-Arylpyridines with NaN3
Ag-Catalyzed [5+2]-Cycloaddition Route to Dihydroazepines
Synthesis of Substituted Coumarins from Propargyl Vinyl Ethers
Rhodium-Catalyzed Synthesis of Benzazepinones
Efficient Heteroannulation Route to 2-Trifluoromethyl Quinolines
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Issue 11/2013

Organocatalytic Route to 2,3,4,6-Tetra- and 2,3,4,5,6-Pentasubstituted Pyridines
Synthesis of 6H-Benzo[c]chromen-6-ones via Carbonylative C–H Cyclization
C–H Activation Route to C-4 Substituted Isoquinolones
Rh/Pd-Catalyzed Synthesis of Aza-Dihydrodibenzoxepines
Efficient Borane-Catalyzed cis-Selective Reduction of 2,6-Disubstituted Pyridines
1,3-Dipolar Cycloaddition Route to Pyrrolo-[3,4-c]pyrrole-1,3-diones
General Strategy for the Synthesis of Cyclopropane-Fused Heterocycles
Heteroannulation Route to 2-Hetarylbenzo-thiazoles through Redox Coupling
Asymmetric α-Arylation Route to 5,5-Disubstituted Hydantoins
Ionic Liquid Promoted Synthesis of Substituted Benzofurans
Pd(II)-Catalyzed C–H Activation Route to Indolines
Synthesis of Cytotoxic Fluorinated 1,2,4-Triazoles
Intramolecular Acylative Coupling Approach to Dibenzo[b,e]azepin-11-ones
Synthesis of Pyridazines and Their Fused Derivatives from 1,3-Diketones
Synthesis of Dihydropyrimidin-4-ones from Propargyl Amides and Sulfonyl Azides
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Issue 10/2013

Biginelli Synthesis of Pyrimidones Using Terminal Alkenes as Precursors
Synthesis of Isoxazolines and Pyrazolines via Radical C–H Oxidation
Synthesis of 1-Aryl 1,2,4-Triazoles by a Three-Component Condensation
Coumarin Synthesis by Carbonylation of 2-Hydroxystyrenes
Synthesis of Pyrazolines via a Catalytic Asymmetric 1,3-Dipolar Cycloaddition
Synthesis of Functionalized Cyclazines in One Pot Using Palladium Catalysis
Carbamoylation–Bromolactamization Route to Five- and Six-Membered Lactams
Palladium-Catalyzed Oxidative Annulation Route to Benzo[b]furans
Regioselective Synthesis of 3,4,5- and 1,3,5-Trisubstituted Pyrazoles
Oxidative Cyclization–Dehydrogenation Route to 2-Aminobenzothiazoles
Palladium-Catalyzed Synthesis of 4-Aminophthalazinones
Diarylpyridazines through Sequential Regioselective Suzuki Coupling
Synthesis of 6H-Benzo[c]chromen-6-ones via C–H Activation–Lactonization
Synthesis of Benzo[b]furans Using 2-(2-Hydroxyphenyl)acetonitriles
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Issue 09/2013

Palladium(II)-Catalyzed Dehydrogenative Heck Route to Pyrroles
Synthesis of Homobenzotetramisole Organocatalysts by Heteroannulation
Iron-Catalyzed Synthesis of Pyrrolidines via C–H Bond Amination
A One-Pot Amine-Catalyzed de novo Synthesis of Highly Substituted Pyridines
Synthesis of Perimidines and 1,5-Benzodiazepines
Regioselective Functionalization of Pyrimidines and Pyrazines via Metalation
One-Pot, Three-Component Sonogashira–Heterocyclization–Heck Reactions
Benzimidazoisoquinoline Synthesis by Ru-Catalyzed Oxidative C–C and C–N Coupling
Synthesis of Pyrazoloisoquinolines from Alkynes and Pyrazoles
Benzyne-Mediated Heteroannulation Route to Indolines and Carbazoles
Cu-Catalyzed C–N Cross-Coupling of Iodopyridines with Nitrogen Heterocycles
Ag-Catalyzed Isocyanide-Alkyne Cycloaddition Route to Pyrroles
Ru-Catalyzed Heteroannulation Route to Isoquinolines and Thienopyridines
Pyrido[1,2-a]benzimidazoles via Iodine(III)-Mediated Demethylenation
Gold-Catalyzed Synthesis of (Z)-1,2-Dihydro-1-tosylbenzo[b]azepin-3-ones
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Issue 08/2013

SNAr Route to Pyrazolo[3,4-d]pyrimidines
Regioselective C–H Activated Alkylation of Pyrroles
Furoxan Synthesis From Styrenes Under Non-Acidic Conditions
18F-Labeled Heterocycles by Huisgen 1,3-Dipolar Cycloaddition
Synthesis of [1,2]Oxazino[5,4-b]indoles by Intermolecular [3+3] Cycloaddition
Synthesis of Quinazolinones via Radical Skeletal Rearrangement
Synthesis of Fluorinated Azabicycles
Efficient Chelation-Controlled Synthesis of Aza-Sugars from Aziridines
Pd/In-Catalyzed Synthesis of Furans from β-Methoxystyrene and Dicarbonyls
Au(I)/Ag(I)-Heteroannulation Approach to Heterocycles with a Very Long Name
Synthesis of Benzo and Fused Heterocyclic Imidazoles from Nitroaminoaryls
Rhodium(III)-Catalyzed C–H Activation Route to Azepinones
C(sp3)–N Bond Formation for the Synthesis of Five- to Seven-Membered Azacycles
Synthesis of Spiro[indoline]oxindoles from Isatin Ketonitrones and Alkynes
Heteroannulative C–H Activation Route to Pyrazoles and Indazoles
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Issue 07/2013

Aryne-Mediated Route to Substituted Carbazoles
Oxidative Heteroannulation Route to Imidazo[1,5-a]pyridines
Cu-Catalyzed Double C–H Activation–Cyclization Route to Hydrazones
Stereodivergent Oxetan-3-one Syntheses from Allenes
Synthesis of Tricyclic Indoles by an Intramolecular Larock Indole Synthesis
Copper-Mediated Synthesis of Pyrrolo[2,1-f][1,2,4]triazin-4(3H)-ones
Synthesis of Chiral Pyrrolidines via Intra-molecular Thiourea-Catalyzed Cyclization
Heteroannulation Route to 2-Acylindoles and 2-Acylindolines
Benzofuran Synthesis Using a Sonogashira–Larock Heteroannulation Protocol
Phenazine Synthesis Involving Smiles Rearrangement of Intermediate Arynes
Synthesis of Pyrroloindolines via Rh(II)-Catalyzed Annulation of Indoles
Silver(I)-Catalyzed Cycloaddition Route to Pyrroles
Cu-Catalyzed Heteroannulation Route to 2-Substituted Benzo[d]thiazoles
CuBr-Catalyzed C–N Coupling Heteroannulation Route to 3-Aminoindazoles
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Issue 06/2013

Synthesis of Pyrazolo[1,5-a]pyrimidines
Synthesis of Indolizinones via Sequential Ritter and Pictet–Spengler Reactions
Functionalized γ-Lactams via Dess–Martin Periodinane Oxidation of Pyrroles
Intramolecular Cyclization Route to Disubstituted 4-Selenyl Isoxazoles
Palladium-Catalyzed Oxidative Isocyanide Insertion for Heterocyclic Synthesis
Synthesis of Substituted 1,2,4-Triazoles from Formamidrazones and Isocyanides
Iridium-Catalyzed Synthesis of Pyrroles from Secondary Alcohols and β-Amino Alcohols
Expedient Access to Biologically Relevant Furan-Based Scaffolds
Scalable Approach to 4-Aminopyrimidines
A Three-Component Copper-Catalyzed Synthesis of Bicyclic Isoxazolidines
Synthesis of Trisubstituted Imidazoles via Oxidative Diamination of Alkynes
A Copper-Catalyzed [3+2]-Cycloaddition Route to Substituted Imidazoles
C–H Activation Route to Phthalazinones from N′-Methylenebenzohydrazides
2-Aryl-3-fluoro-5-silylthiophenes via a [2,3]-Sigmatropic Rearrangement
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Issue 05/2013

Palladium-Catalyzed Synthesis of 3-Alkynylindoles
Synthesis of Tetrahydroquinazolinediones and Dihydropyrido[2,3-d]pyrimidines
Copper-Catalyzed Synthesis of Furans via (2-Furyl)Carbene Complexes
Interconversion of Benzodiazepinediones into Oxazoloquinolinones
Gold(I)-Catalyzed Synthesis of Pyrrolo[1,2-a]indoles
FeBr3-Catalyzed C–H Activation Route to Indazoles and Pyrazoles
Phenanthridine Derivatives from Intramolecular Diels–Alder Reaction
Rhodium-Catalyzed Synthesis of Phthalides from Benzoic Acids
De Novo Synthesis of 2-Pyridones
Two-Step Synthesis of 2H-Indazoles via C–H Activation of Azobenzenes
One-Pot Synthesis of Benzo[4,5]imidazo[2,1-a]isoquinolines
Zinc Triflate Catalyzed Double Michael Addition Route to Enantioenriched Chromans
Synthesis of Pyrroles and 2H-Pyrrolo[3,4-c]quinolines
Synthesis of 2-Aryl-2H-indazoles Using Silver Catalysis
A Cloke–Wilson Rearrangement Approach to Fused Bromofurans
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Issue 04/2013

Gold(III)-Catalyzed Synthesis of Furans Using Enynones
Pd-Catalyzed Synthesis of Spirooxindoles
Phosphine-Catalyzed γ-Addition of N-Nucleophiles to Allenoates and Alkynoates
2-(Phenylsulfinyl)acetamide as a Two-Carbon Unit for 2-Pyridone Synthesis
Regioselective Synthesis of Oxa- and Thiadiazoles from Thiosemicarbazides
Diels–Alder Cycloaddition Approach to Indoles from Alkynol-Furans
Piperidines and Azepines via Asymmetric Aminofluorination of Olefins
Stereoselective Synthesis of Chiral 1,4-Oxazepanes
Condensation of Vinyl Azides with Stabilized Acetonitriles to 2-Aminopyrroles
Synthesis of Carbazolones via PIFA-Mediated Annulation of 2-Aryl Enaminones
Synthesis of 1H-Imidazo[1,2-a]imidazol-5-amines from 2-Aminoimidazoles
Synthesis of Benzofuranones via C–H Activation–Lactonization
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Issue 03/2013

Iodine-Mediated Synthesis of Oxazoles
One-Pot Synthesis of Benzimidazoles from 2-Nitroanilines and Aldehydes
Synthesis of 3-Nitroindoles via an Intramolecular α-Selective Heck Reaction
Copper-Catalyzed MCR to Pyrido[1,2-a]-pyrimidin-4-imines
Synthesis of Pyrroles from Cyclopropanes and Nitrones via Oxazine Intermediates
Synthesis of 1,4-Benzodiazepines via a Double SNAr Reaction
Gold-Catalyzed de novo Synthesis of Highly Substituted N-Alkoxypyrroles
N-Heterocyclic Carbene Catalyzed Synthesis of Enantioenriched Lactones
Rhodium-Catalyzed Annulation Route to Heterocyclic MIDA Boronates
One-Pot Synthesis of Isoxazolines
Synthesis of Tetrasubstituted Pyrimidine Sulfonamides
Copper-Catalyzed Synthesis of Acridones from 2-Aminobenzophenones
Three-Component Synthesis of Functionalized Cyclazines
Synthesis of Cyclic Aryl Sulfonic Acid Derivatives
Silver Triflate Catalyzed Synthesis of Imidazo[1,2-a]pyridines
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Issue 02/2013

Concise Synthesis of Complex Polycyclic Lactams
Copper-Catalyzed Heteroannulation to Tetrahydroxanthen-1-ones
Palladium-Catalyzed Asymmetric Synthesis of Cyclopropane-Fused Quinoline Derivatives
Iron(II) Chloride-Catalyzed Synthesis of Imidazo[1,2-a]pyridines
Palladium-Catalyzed Carbonylative Annulation to Flavones
Domino Staudinger–Aza-Wittig Synthesis of 1H-Pyrazolo[1,5-b]indazoles
Robust Nickel-Mediated Methodology for the Cross-Coupling of Heterocycles
Synthesis of Dipyrido[1,2-a:3′,4′-d]imidazole Salts from 2-Aminopyridine
Palladium-Catalyzed Intramolecular C(sp3)–H Alkenylation Route to Hexahydroindoles
PIDA-Mediated Intramolecular Oxidative Cyclization of Enamides to Oxazoles
Synthesis of Benzimidazoles and Quinazolinones via Pd-Catalyzed Heteroannulation
Synthesis of Benzazoles Using S8 as the Oxidizing Agent
Snieckus, Victor; Zhao, Yigang: Synthesis of Phenanthridinones via C–H Activation of N-Methoxybenzamides
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Issue 01/2013

Isatoic Anhydrides via C–H Activation
Access to Quaternary Amino Acids via Dynamic Kinetic Resolution of Azlactones
Synthesis of 3-Fluoropyrazoles from 2-Trifluoromethyl-1-alkenes
A C–O/C–N Coupling Route to 1,4-Benzoxazines
Organocatalytic Synthesis of Chromans and Benzopyrano[3,4-c]pyrrolidine
De Novo Synthesis of Pyridones From Enaminones and Alkynes
Synthesis of Pyrimidines from Propargylic Hydroxylamines
Palladium-Catalyzed C–N/C–C Coupling Route to Substituted Indoles
Iridium-Catalyzed Synthesis of Substituted Piperazines
Iron-Catalyzed Synthesis of Pyrazoles from Hydrazones
Phenyliodine(III) Diacetate-Promoted Synthesis of Benzimidazoles
Palladium-Catalyzed Synthesis of Benzo[b][1,4]oxazepines
Pd-Catalyzed Synthesis of Indeno[1,2-c]chromenes from 2-Alkynylhalobenzenes
Palladium-Catalyzed Three-Component Synthesis of Oxazolines and Oxazines
Synthesis of Heterocyclic Triquinanes via Sequential Radical Cyclizations
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Issue 12/2012

Palladium-Catalyzed Cyclization of Electron-Deficient Enynes
A Palladium-Catalyzed Multicomponent Heteroannulation Route to Indoles
A Pd-Catalyzed C–H Activation Route to Benzisoxazolones
Rhodium-Catalyzed Synthesis of 3-Aryl Indoles from 1-Sulfonyl 1,2,3-Triazoles
Synthesis of Sultams via Rh(III)-Catalyzed Directed C–H Activation
Synthesis of Imidazopyridines by Cu(II)/Fe(III) Co-catalyzed C–N Coupling
Synthesis of 5-Acyl-2-amino-1,3,4-thiadiazoles From Acid Chlorides
Synthesis of Functionalized Azaindolines and Azatetrahydroquinolines
Stereoselective Access to Quaternary Carbon Atoms via SN2 Cleavage of Azetidinium Ions
Ru-Catalyzed Synthesis of Polysubstituted Pyrazoles
Copper–Silver Cocatalyzed Synthesis of Pyrazoloisoquinolines
Synthesis of 3-Aminoindolizines Enabled by Flow Technology
Synthesis of Cyclic Azomethine Imines as Precursors to β-Aminocarbonyl Scaffolds
Copper-Catalyzed Synthesis of 1,4-Dihydroazete Derivatives
Cu- and Ni-Catalyzed Regioselective Synthesis of Disubstituted Pyrroles
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Issue 11/2012

Rhodium/Lewis Acid Catalyzed Cascade Synthesis of Tetrahydropyridazines
Heterocycles via Use of 2-Heteroaryl-2-(tetrahydrofuranyliden)acetonitriles
Practical Brønsted Acid Mediated Synthesis of Coumarins from Allenes
Cu-Catalyzed Synthesis of Furoindolines from Tryptophols
Synthesis of Isoindolinones by an Asymmetric Aza-Wacker-type Cyclization
Silver-Catalyzed Heteroannulation Route to 1-Aminoisoquinolines
One-Pot Gold-Catalyzed Synthesis of Azepino[1,2-a]indoles
Cascade Synthesis of 3-Pyrrolines by a Heck–Aza-Michael Reaction
Expedient Route to Complex Alkaloids through Pd(II)-Catalyzed Indole C-2 Alkylation
Synthesis of Iodotriazoles Using in Situ Generated Electrophilic Triiodide
One-Pot Asymmetric Synthesis of 4-Hydroxypyrazolidines from Aldehydes
Direct C-2 Pyridine C–H Olefination
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Issue 10/2012

Gold-Catalyzed Intramolecular Annulation Route to 2,3-Dihydro-1H-pyrrolizines
Au(I)-Catalyzed Synthesis of Indole- and Arene-Fused Hexahydroquinolizinones
Synthesis of Benzoxazepines from Epoxides and Anthranilic Acids
A Palladium-Catalyzed Enantioselective Hydroamination Route to Pyrrolidines
Copper-Catalyzed Oxytrifluoromethylation of Alkenes to Oxygenated Heterocycles
Cu-Catalyzed Carboetherification Approach to Polycyclic Tetrahydrofurans
An Aryne Condensation–P-Cyclization Sequence to Dibenzophosphole-Boranes
Synthesis of Aminopyrimidinethiones from α-Azidovinyl Ketones and Thiourea
Pd-Catalyzed Synthesis of Indolines via Intramolecular Aryl C–H Amination
Cu-Catalyzed Synthesis of Cinnolines from N-Methyl-N-phenylhydrazones
Synthesis of Fluorinated (4-Aminoquinolinyl)phosphonates
syn-1,2-Diamines and Arylpiperazines via [3,3]-Diaza-Cope Rearrangement
Pd-Catalyzed Heteroannulation Route to Phthalazinones
Iodine-Catalyzed Three-Component Reaction to 4-Arylfuro[2,3-a][4,7]phenanthrolines
A C–H Activation Route to Indoloquinolines and Pyrroloquinoxalines
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Issue 09/2012

Palladium-Catalyzed Synthesis of Quinolines
Synthesis of Benzoxazoles by an Asymmetric Ugi-Type Reaction
Ni-Catalyzed Synthesis of 3-Piperidones from 3-Azetidinones and Alkynes
Regioselective, Modular C–N and Suzuki Coupling Route to Triazoles
Piperidines and Tetrahydroisoquinolines via Hydride Transfer Cyclization
Gold-Catalyzed Cyclizations Leading to Indenoazepines and Strained Bicycles
Metal-Free Aziridine Synthesis from Unfunctionalized Olefins
Iodocyclization Route to Pyrroles and Furans in PEG
Organocatalytic Synthesis of Quinolines and Chiral 1,4-Dihydroquinolines
Synthesis of Isoxazoles from 1,3-Dialkynes and Hydroxylamine
Synthesis of Azetidines by Epoxide Ring-Opening–Ring-Closure Procedure
Cu-Catalyzed Regioselective Synthesis of 1,2,3- or 1,2,4-Triaryltriazoles
Isoindolinols and Dihydroisobenzofuranols via Combined Au–Pd Catalysis
Sonogashira Coupling–Heteroannulation Route to Substituted 5-Azaindoles
3,1-Benzoxazines from N-Acyl-o-Toluidines via Cu-Catalyzed Heteroannulation
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Issue 08/2012

Au-Catalyzed Carbonyl Migration for the Synthesis of Azepinoindol-1-ones
One-Pot Pd-Catalyzed Synthesis of Isoquinolines and Furo/Thienopyridines
Synthesis of Isoquinolin-1(2H)-ones via Pd-Catalyzed Isocyanide Coupling
Synthesis of Piperazine-2,5-diones via a Convenient Dieckmann Cyclization
A Cu-Catalyzed Double C–N Coupling Approach to Cinnolines
Functionalized Enantioenriched Dihydropyrans by [4+2] Cycloaddition
DABCO-Mediated [4+2] Annulation Approach to 2,3-Dihydropyran-4-ones
Selectivity in Palladium-Catalyzed Carboesterification – Amides versus Esters
Synthesis of Benzofuro[3,2-d]pyrimidines from 3-Chlorochromones
Synthesis and Suzuki Coupling of 2-Aryl-Trisubstituted Oxazoles
Indoloazocines via a Sequential Ugi–Gold-Catalyzed Hydroarylation
Polysubstituted Pyridines via Re-Catalyzed Alkyne Insertion
Synthesis of 3-Carboxylated Indoles from 2-Ethynylanilines and CO2
Iron-Catalyzed Substitution of Benzoxazoles and Benzothiazoles
Palladium-Catalyzed Synthesis of Indoles via Oxidative C–H Activation
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Issue 07/2012

Synthesis of Trifluoromethylated Aziridines from Trifluoromethyl Diazomethane
A Catalytic Multicomponent Synthesis of cis-4,5-Disubstituted Pyrrolidinones
Ruthenium-Catalyzed Dehydrative Benzofuran Synthesis via C–H Activation
Gold-Catalyzed Synthesis of 2,4-Disubstituted Furans
Nickel-Mediated, Regioselective Syntheses of Substituted Piperidines
Synthesis of 1H-Indazoles by the Reaction of Arynes with Hydrazones
Synthesis of Azetidines from Glycine Esters and a Vinylsulfonium Salt
Bicyclic Furans via Ru-Catalyzed Transfer Oxygenative Cyclization of Diynes
Enantioselective Synthesis of γ-Butyro-lactones via Dynamic Kinetic Resolution
TiCl4-Mediated Cyclocondensation Reaction to Indolizines
Oxygen Heterocycles via Divergent Reactivity of a π-Allylpalladium Species
Pd-Catalyzed Heteroannulation Route to Imidazo[4,5-b]pyridines and -pyrazines
Copper-Catalyzed Heteroannulation Route to Indoles
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Issue 06/2012

Isoquinoline-Catalyzed Synthesis of Azirines
Oxadiazoles: Synthesis, Properties and Significance in Medicinal Chemistry
Synthesis of Tetrahydrothiopyrans via Thiocarbenium Ion Cyclization
Cu-Promoted Oxidative Heteroannulation Approach to Benzofurans
Synthesis of 4-Aryl-2-quinolinone by a Tandem Heck/C–H Amidation Approach
Cu-Catalyzed Heteroannulation Route to [1,2,3]Triazolo[1,5-a]quinoxalin-4(5H)-ones
Sonogashira-Mediated Route to Benzo[c]chromen-6-ones
Copper Oxide Catalyzed Synthesis of Benzo[e][1,2,4]triazines
Synthesis of Pyridazino[1,2-a]indazoliums by N–N Bond Forming
Pyrrolobenzoxazoles via Three-Component [3+2] Heterocycloannulation
Rh-Catalyzed De Novo Synthesis of Pyridines from Terminal Alkynes and Ketoximes
Silver-Mediated Dual C–H/C–H Activation for the Synthesis of 3-Acyl Furans
Synthesis of Furans by Au-Catalyzed Cyclization of (E)-1-Aryloxy-1-en-3-ynes
Diverse Heterocycles from a Naphthofuran Hydroxypropenone Sodium Salt Synthon
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Issue 05/2012

Cu-Catalyzed Synthesis of Indolizines
Pd-Catalyzed Heteroannulative Route to Isocoumarins
Synthesis of Oxindoles via Intramolecular Enantioselective α-Arylation
Efficient Stereoselective Synthesis of Tricyclic Chromenoisoxazolines
Diastereoselective Rh-Catalyzed Cascade Affording Piperidine Derivatives
Dearomatizative Intramolecular 1,3-Dipolar Cycloaddition of Nitrile N-Oxides
Gold-Catalyzed Asymmetric Heteroannulation Route to Isochromenes
Convergent Domino Oxidation for Oxazole Synthesis
Cu-Catalyzed Synthesis of Imidazopyridines from 2-Aminopyridines and Nitroolefins
Substituted Pyrroles via Rh-Catalyzed Rearrangement of α-Diazo Oxime Ethers
Five-, Six- and Seven-Membered N-Hetero-cycles via Pd(II)-Catalyzed Hydroamination
Three-Component Synthesis of Pyrido[2,1-d]-[1,2,5]triazepines
Pd-Catalyzed C(sp3)–H Activation Route to Oxindoles
Rhodium-Catalyzed Intramolecular [2+2+2] Cycloaddition to Planar-Chiral Cyclophanes
Pd-Catalyzed C–H Activation–Carboamination Route to Phenanthridines
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Issue 04/2012

One-Pot Synthesis of Cannabinoids via In-verse-Electron-Demand Diels–Alder Reaction
Ru-Catalyzed Synthesis of Isocoumarins from Benzoic Acids and Alkynes
Modular Access to 2-Substituted Pyridines via Suzuki Cross-Coupling of MIDA Boronates
Synthesis of Benzo[a]quinolizines by a MCR/Allylation/Heck Sequence
Indoloquinolizines from a One-Pot, 12-Step, Three-Component Cascade Reaction
Heterocyclo[3.3.1.0]nonanes by Pt-Catalyzed Cycloisomerization of Allyl Alkynes
Synthesis of Isochromanones and Isoquinolines via Friedel–Crafts Cyclization
Pd-Catalyzed Synthesis of Indolo[1,2-a]-Quinoxalines
Catalytic Oxidative Synthesis of Quinazolines and Benzoxazines
Cyclocarbonylation of Enynes Using Glyceraldehyde as a Carbonyl Source
A Domino Radical Smiles Rearrangement Approach to Indolin-2-ones
Annulation–Electrophilic Amination Approach to 3-Aminobenzofurans and -indoles
Oxidative Rearrangement Approach to Fused Imidazolines and Quinazolines
Polysubstituted Oxazoles via Cerium(III)-Promoted Cyclization of Propargyl Amides
Synthesis of Thieno[3,2-c]pyridinones by Cyclopropyl Thione Rearrangement
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Issue 03/2012

One-Pot Heteroannulative Synthesis of α-Carbolines from 2-Aminoindoles
Diastereoselective Narasaka–Heck Route to Bicyclic N-Heterocycles
Organocatalytic Enantioselective Friedel–Crafts Approach to 2,3-Dihydrobenzofurans
Pd-Catalyzed Multicomponent Synthesis of 4-Aminophthalazin-1(2H)-ones
Pd-Catalyzed Synthesis of Dibenzoazepines from 2-Bromoanilines
Multicomponent Synthesis of Benzo[a]pyrano[2,3-c]phenazines
Regiospecific Synthesis of Polysubstituted Pyridines
Regioselective Arylation of Pyridine N-Oxides via Silver-Catalyzed C–H Activation
Concise Synthesis of Tetrahydro-5H-indolo[3,2-c]quinolines
Synthesis of Nitrated Triazoles as Potentially New Explosives
Oxidative Expansion of Oxiranes and Oxetanes via Copper Catalysis
Azetidines, Pyrrolidines, and Indolines via C(sp3)–H and C(sp2)–H Bond Amination
Tetrahydro-1,4-benzodiazepin-2-ones from Ugi MCR Intermediates
Fused Pyridazino[4,5-b]oxazepine-diones via Smiles Rearrangement
Copper-Catalyzed Synthesis of 2H-Isoindole-1-Carboxylates
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Issue 02/2012

(Pyrazolo)pyrimidines/Purines via a Three- Component Reaction
A Tandem Amination–Cycloisomerization Approach to Imidazo[1,2-a]pyridines
Rh-Catalyzed Alkyne Hydroacylation Route to Highly Substituted Furans
Copper-Catalyzed Oxacyclization to Fused Heteroaryl Pyranones
Highly Substituted Pyridines via C–H Rhodation of Unsaturated Ketoximes
Pd-Catalyzed Three-Component Synthesis of Oxazolines and Benzoxazoles
Synthesis of Quinolines from N-Alkyl Anilines and Olefins
Pd-Catalyzed Intramolecular C–H-Activation Approach to Phenanthridines
PhI(OCOCF3)2-Mediated Synthesis of 2-(Trifluoromethyl)oxazoles
Modular Synthesis of Unsymmetrically Polysubstituted and Fused Pyridines
Multicomponent Synthesis of 5-Carboxamide Oxazolines
Copper/Copperless Synthesis of Tetrazoles via C–H and C–C Bond Cleavages
Radical Cyclization Approach to Piperidyl Benzofuran/Benzopyran Spirocycles
A Three-Component Synthesis of Imidazolines
Three-Component Synthesis of Pyrazoles Using Titanium Catalysis
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Issue 01/2012

Synthesis of Azabicyclo[3.1.1]heptane Derivatives from Cyclobutanones
Ni-Catalyzed Cycloaddition Approach to Fused Pyridine Derivatives
Phthalimide Synthesis via Oxidative Carbonylation of Benzamides
[3+2]-Dipolar Cycloaddition Route to 2H-Indazoles
Organocatalytic [3+2]-Cycloaddition Route to 1,2,3-Triazoles
Pd-Catalyzed Cross-Coupling–Lactonization Route to Dibenzopyranones
Concise Synthesis of Trifluoromethyl-Substituted Benzofuranols
Quinolines and Tetrahydroquinolines via Pd(0)-Catalyzed C–H Bond Functionalization
Intramolecular Heck-Type Synthesis of Piperideines and Pyridines
Synthesis of 3,4-Diaryl-3-pyrrolin-2-ones from Pyrrole Weinreb Amides
Pd-Catalyzed Synthesis of Furans from 1,3-Dicarbonyls and Propargylic Alcohols
Mitsunobu-Based Synthesis of Four-Membered Cyclic Oxaphosphetanes
Organocatalytic Enantioselective Synthesis of Functionalized Piperidines
One-Pot Synthesis of Benzo[b]furans from Phenols and Bromoalkynes
Stannous Chloride Mediated Synthesis of Spiroindolinone Quinazolines
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Issue 12/2011

Karthikeyan, J.; Cheng, C.-H.: Pd-Catalyzed Synthesis of Phenanthridinones by Double C-H Activation
Shintani, R.; Moriya, K.; Hayashi, T.: Palladium-Catalyzed Enantioselective Synthesis of Silacyles
Denmark, S. E.; Kornfilt, D. J. P.; Vogler, T.: Ethers via Catalytic Asymmetric Thiofunctionalization of Alkenyl Alcohols
Estrada, A. A.; Lyssikatos, J. P.; St-Jean, F.; Bergeron, P.: Synthesis of Pyrimidines via N-Vinyl Tertiary Enamides
Anas, S.; Cordi, A.; Kagan, H. B.: Pd-Catalyzed Enantioselective Synthesis of 2-Methyl Indolines
Wang, Y.; Luo, Y.-C.; Hu, X.-Q.; Xu, P.-F.: Metal-Free Synthesis of 2-Trifluoromethyl Furans
Chai, G.; Qiu, Y.; Fu, C.; Ma, S.: Synthesis of Chromones from 2,3-Allenoic Acids and Benzynes
Patil, S. S.; Patil, S. V.; Bobade, V. D.: Iron-Catalyzed Synthesis of Aminoindolizines and Quinolines
Reddy, C. R.; Reddy, M. D.; Srikanth, B.; Prasad, K. R.: Metal-Free Synthesis of Pyrroles From Morita-Baylis-Hillman Acetates
Li, Y.; Hong, D.; Zhu, Y.; Lu, P.; Wang, Y.: Copper-Catalyzed One-Pot Synthesis of 5-Sulfonamidopyrazoles
Yamagishi, M.; Nishigai, K.; Hata, T.; Urabe, H.: Two-Step Heck-Mediated Synthesis of Pyrroles from Sulfonamides and Bromoacetylenes
Nandi, G. C.; Samai, S.; Singh, M. S.: Cycloaddition Approach to Substituted Thiophenes
Sun, L.-L.; Deng, C.-L.; Tang, R.-Y.; Zhang, X.-G.: Heteroannulation Route to Benzothiophenes from 2-Bromo Alkynylbenzenes
Panteleev, J.; Zhang, L.; Lautens, M.: A Multicatalytic Domino Heteroannulation Approach to Dihydroquinolines
Kuninobu, Y.; Yoshida, T.; Takai, K.: Pd-Catalyzed C-H Activation Route to Dibenzophosphole Oxides
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Issue 11/2011

Tsvelikhovsky, D.; Buchwald, S. L.: Concise Palladium-Catalyzed Synthesis of Dibenzodiazepines
Zheng, D.; Wang, Z.; Wu, J.: Synthesis of 1-Aroxyisoquinolines from Phenols and 2-Alkynylbenzaldoximes
Varela-Fernández, A.; Varela, J. A.; Saá, C.: Ru-Catalyzed Heteroannulation to Indoles, Dihydroisoquinolines, and Dihydroquinolines
Zhao, J.; Wu, C.; Li, P.; Ai, W.; Chen, H.; Wang, C.; Larock, R. C.; Shi, F.: [3+2] Cycloaddition to Pyrido[1,2-b]indazoles
Ackermann, L.; Pospech, J.: Ruthenium-Catalyzed Synthesis of Phthalides in Water via C-H Alkenylation
Wu, Z.; Huang, Q.; Zhou, X.; Yu, L.; Li, Z.; Wu, D.: One-Pot Cu-Catalyzed C-N Coupling Approach to Pyrido[1,2-a]benzimidazoles
Pews-Davtyan, A.; Beller, M.: Efficient Zinc-Mediated Heteroannulation Route to 3-Amidoindoles
Candito, D. A.; Panteleev, J.; Lautens, M.: Base-Mediated Intramolecular Aryne-Ene Cyclization
Ylijoki, K. E. O; Kündig, E. P.: Synthesis of Benzoxazinones via Palladium-Catalyzed Intramolecular C-O Coupling
Hong, D.; Zhu, Y.; Li, Y.; Lin, X.; Lu, P.; Wang, Y.: Copper-Catalyzed Three-Component Synthesis of Polysubstituted Pyrroles
Zhu, D.; Zhao, J.; Wei, Y.; Zhou, H.: Sonogashira-Hydroamination Route to 1,2,4-Trisubstituted Pyrroles
Davies, P. W.; Cremonesi, A.; Dumitrescu, L.: Gold-Catalyzed [3+2]-Cycloaddition Approach to 2,4,5-Trisubstituted Oxazoles
Radi, M.; Casaluce, G.; Botta, M.: Microwave-Facilitated Synthesis of Pyrimidinones
Sperança, A.; Godoi, B.; Pinton, S.; Back, D. F.; Menezes, P. H.; Zeni, G.: Iron-Mediated Heteroannulation Route to Isochromenones
Wang, Y.; Wang, H.; Peng, J.; Zhu, Q.: Pd-Catalyzed Heteroannulation Route to 4-Aminoquinazolines via C-H Amidination
All PDFs of this category

Issue 10/2011

Pace, V.; Hoyos, P.; Sinisterra, J. V.; Alcántara, A. R.; Holzer, W.: Synthesis of 2-Aminoepoxides from Aminohalohydrins Using KF on Celite
Ma, B.; Wang, Y.; Peng, J.; Zhu, Q.: Pd-Catalyzed Synthesis of Quinazolin-4(3H)-ones from N-Aryl Amidines
Jiang, H.; Ji, X.; Li, Y.; Chen, Z.; Wang, A.: Pd-Catalyzed Synthesis of 1,4-Dihydro-pyridines via a Multicomponent Reaction
Lopchuck, J. M.; Gribble, G. W.: A Convenient 1,3-Dipolar Cycloaddition Approach to Pyridylpyrroles
Szatmári, I.; Fülöp, F.: Oxazinoisoquinoline Synthesis via the Unusual Reactivity of Aminomethylnaphthols
Babinski, D. J.; Aguilar, H. R.; Still, R.; Frantz, D. E.: Pericyclic Approach to Synthesis of Substituted Pyrazoles
Wetzel, A.; Gagosz, F.: Gold-Catalyzed Heteroannulation Route to Indolin-3-ones and Indoles
Yu, X.; Lu, X.: 1-Benzoxepines from 2-Acylmethoxyaryl Boronic Acids and Allenoates
Chen, L.; Fu, H.; Qiao, R.: Intramolecular Ullmann Cross-Coupling Route to Fused Pyridoquinazolinones
Kumar, R.; Namboothiri, I. N. N.: Sulfonylpyrazoles via Base-Mediated Reaction of Diazosulfone with Nitroalkenes
Li, W.; Li, X.; Wu, W.; Liang, X.; Ye, J.: One-Pot Enantioselective Michael-Aldol Approach to Imidazole Derivatives
Jarvis, S. B. D.; Charette, A. B.: Synthesis of Enantiopure Piperidines via an Aziridinium Ring Expansion Reaction
Nakanishi, M.; Katayev, M.; Besnard, C.; Kündig, E. P.: Palladium-Catalyzed C-H Activation Induced Enantioselective Route to Fused Indolines
Nishino, M.; Hirano, K.; Satoh, T.; Miura, M.: Cu-Catalyzed Oxidative Synthesis of Tetrahydroquinolines from N-Methylanilines
Nakai, K.; Kurahashi, T.; Matsubara, S.: Ni-Catalyzed Cycloaddition Approach to Coumarins by C-C σ-Bond Cleavage
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Issue 09/2011

Rogress, D. C.; Larock, R. C.: Arynes in the Synthesis of N-Arylisatins
Li, P.; Zhao, J.; Wu, C.; Larock, R. C.; Shi, F.: Synthesis of NH-Free 3-Substituted Indazoles
McAusland, D.; Seo, S.; Pintori, D. G.; Finlayson, J.; Greaney, M. F.: The Benzyne Fischer Indole Reaction
Teller, H.; Fürstner, A.: Enyne Cycloisomerization Route to an Anti-depressant Drug Candidate, GSK1360707
Xiao, B.; Gong, T.-J.; Liu, Z.-J.; Liu, J.-H.; Luo, D.-F.; Xu, J.; Liu, L.: Pd-Catalyzed Synthesis of Dibenzofurans by Phenol-Directed C-H Activation
Han, B.; Wang, C.; Han, R.-F.; Yu, W.; Duan, X.-Y.; Fang, R.; Yang, X.-L.: (4-Hydroxy-TEMPO)-Catalyzed Synthesis of 2-Aryl Quinazolines
Zhou, F.; Liu, J.; Ding, K.; Liu, J.; Cai, Q.: Copper-Catalyzed Synthesis of Pyrrolo[3,2-c]quinolin-4-nones
Zheng, D.; Chen, Z.; Liu, J.; Wu, J.: Synthesis of 1-Aminoisoquinolines from 2-Alkynylbenzaldoximines
Burkhard, J. A.; Tchitchanov, B. H.; Carreira, E. M.: Synthesis of Isoxazoles from the Reaction of Nitroalkanes with Oxetanes
Wu, X.; Li, L.; Zhang, J.: Nickel-Catalyzed Diastereoselective Synthesis of Oxazolidines
Neo, A. G.; Carrillo, R. M.; Marcos, C. F.: Conversion of Anilines into 2-Aminobenzo-thiazoles via Herz Compounds
Kumar, M. R.; Park, A.; Park, N.; Lee, S.: Copper-Catalyzed Three-Component Synthesis of 2H-Indazoles
Ryabukhin, S. V.; Naumchik, V. S.; Plaskon, A. S.; Grygorenko, O. O.; Tolmachev, A. A.: Synthesis of 3-Haloquinolines via the Friedländer Reaction
Jepsen, T. H.; Larsen, M.; Jørgensen, M.; Nielsen, M. B.: An Efficient Protocol for the Synthesis of Dibenzodithiapentalene
Verma, A. K.; Shukla, S. P.; Singh, J.; Rustagi, V.: Iodocyclization Route to Indolo- and Pyrroloquinolines
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Issue 08/2011

Churchill, G. H.; Raw, S. A.; Powell, L.: Effects of Addition Rate on the Synthesis of Pyridopyrimidinediones
Zheng, Z.; Tang, L.; Fan, Y.; Qi, X.; Du, Y.; Zhang-Negrerie, D.: FeBr3-Mediated Heteroannulation Route to Yield N-Amino-3-Nitrile-Indoles
Zhang, G.; Luo, Y.; Wang, Y.; Zhang, L.: Gold-Catalyzed Heteroannulation Route of N-Allyl Ureas to Tricyclic Indolines
Wang, F.; Cai, S.; Wang, Z.; Xi, C.: Synthesis of 2-Mercaptobenzothiazoles via Metal-Free Heteroannulation
Shi, L.; Liu, X.; Zhang, H.; Jiang, Y.; Ma, D.: Cu-Mediated Heteroannulation Route to 2-Thio-Substituted Benzothiazoles
Francis, S.; Kiyoi, T.; Reid, M.; Davies, K.; Laats, S.; McArthur, D.; Feilden, H.; Easson, A. M.; Kiyoi, Y.; Wishart, G.; Ray, P.: Sythesis of Serotonin Antagonists Using an Intramolecular Diels-Alder Approach
Neumann, J. J.; Rakshit, S.; Dröge, T.; Würtz, S.; Glorius, F.: Heteroannulation Route to Indoles from N-Aryl Enamines via C-H Activation
Calvet, G.; Livecchi, M.; Schmidt, F.: Pd-Catalyzed Heteroannulation Route to Substituted 5-Azaindoles
He, W.; Li, C.; Zhang, L.: Gold-Catalyzed [2+2+1] Synthesis of 2,5-Disubstituted Oxazoles
Alsabeh, P. G.; Lundgren, R. J.; Longobardi, L. E.; Stradiotto, M.: Pd-Catalyzed Synthesis of Indoles via NH3 Cross-Coupling-Alkyne Cyclization
Paradise, C. L.; Sarkar, P. R.; Razzak, M.; De Brabander, J. K.: AuCl3-Catalyzed Synthesis of 5-Bromomethyl Oxazoles from Amino Acids
Surmont, R.; Verniest, G.; De Schrijver, M.; Thuring, J. W.; Holte, P. ten; Deroose, F.; De Kimpe, N.: Synthesis of 3-Amino-4-fluoropyrazoles Using Selectfluor
Ascic, E.; Jensen, J. F.; Nielsen, T. E.: Ruthenium-Catalyzed Synthesis of Complex Indolizidinones
Samanta, R.; Antonchick, A. P.: Palladium-Catalyzed C-H Activation Route to Dibenzothiophenes
Ackermann, L.; Lygin, A. V.; Hofmann, N.: De Novo Ruthenium-Catalyzed Synthesis of 2-Pyridones
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Issue 07/2011

Mehta, V. P.; Modha, S. G.; Rujiter, E.; Van Hecke, K.; Van Meerwelt, L.; Pannecouque, C.; Balzarini, J.; Orru, R. V. A.; Van der Eycken, E.: Microwave-Assisted Synthesis of Dibenzoazepinones
Ritson, D. J.; Spiteri, C.; Moses, J. E.: Silver-Mediated Synthesis of Oxazoles
Seki, H.; Georg, G. I.: Synthesis of Cyclic Enaminones via Ketene Cyclization
Roux, L.; Charrier, C.; Salomon, E.; Ilhan, M.; Bisseret, P.; Tarnus, C.: Oxazepin-4-ones via Hypervalent Iodine Mediated Ring Expansion
Barber, D. M.; Sanganee, H.; Dixon, D. J.: Synthesis of 2,5-Disubstituted Pyrroles by Nitro-Mannich/Hydroamination Cascades
Zhang, R.; Zhang, D.; Liang, Y.; Zhou, G.; Dong, D.: Synthesis of Pyrimidin-4(3H)-ones via Vilsmeier-Haack Reaction
Wang, F.; Cai, S.; Liao, Q.; Xi, C.: Cu-Catalyzed Synthesis of 2-Aminobenz-imidazoles
Rong, Z.-Q.; Li, Y.; Yang, G.-Q.; You, S.-L.: Camphor-Derived Organocatalytic Synthesis of Chromanones
Meng, T.; Zou, Y.; Khorev, O.; Jin, Y.; Zhou, H.; Zhang, Y.; Hu, D.; Ma, L.; Wang, X.; Shen, J.: Synthesis of 3-Aminocoumarin and Derivatives via Copper Catalysis
Liu, Y.; Jacobs, H. K.; Gopalan, A. S.: Intramolecular Cyclization of Acyloxy Sulfones to Fused Furans and Benzofurans
Zhou, J.; He, J.; Wang, B.; Yang, W.; Ren, H.: Regioselective Synthesis of Benzotriazoles via 1,7-Palladium Migration
Okuma, K.; Matsunaga, N.; Nagahora, N.; Shioji, K.; Yokomori, Y.: Synthesis of Indolinones from Arynes and Amino Acid Esters
Hirano, K.; Satoh, T.; Miura, M.: Synthesis of 3-Aminobenzofurans via Cu-Catalyzed Annulative Amination
Chen, J.; Ni, S.; Ma, S.: Synthesis of 2,3,5-Trisubstituted Furans from Cyclopropenyl-1,1-Dicarboxylates
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Issue 06/2011

Zhang, X.; Chen, D.; Zhao, M.; Zhao, J.; Jia, A.; Li, X.: Rhodium-Catalyzed Synthesis of Isoquinolines from Oximines and Alkynes
Zhao, J.; Zhao, Y.; Fu, H.: Transition-Metal-Free SNAr-Type Synthesis of Chromones
Weiß, K. M.; Wei, S.; Tsogoeva, S. B.: Synthesis of 1,3-Thiazoles from Nitrostyrenes and Aromatic Thioamides
Kumar, R. K.; Ali, Md. A.; Punniyamurthy, T.: Palladium-Catalyzed C-H Activation/C-N Coupling Route to 1-Aryl-1H-benzotriazoles
Hirano, K.; Inaba, Y.; Takahashi, N.; Shimano, M.; Oishi, S.; Fujii, N.; Ohno, H.: Gold-Catalyzed Hydroamination-Hydroarylation Route to Fused Indoles
Lei, M.; Ma, L.; Hu, L.: Tetrahydropyranoquinolinone via a Knoevenagel Reaction
Xu, W.; Jin, Y.; Liu, H.; Jiang, Y.; Fu, H.: Synthesis of Quinazolinones by Combined Ullmann Coupling-Oxidative C-H Amidation
Kim, J. H.; Lee, S.-g.: One-Pot Synthesis of Indoles and N-Fused Indoles from Nitriles
Nakao, Y.; Morita, E.; Idei, H.; Hiyama, T.: Nickel-Catalyzed Dehydrogenative [4+2]-Cycloaddition Route to Dihydropyridones
Xu, J.; Wei, J.; Bian, L.; Zhang, J.; Chen, J.; Deng, H.; Wu, X.; Zhang, H.; Cao, W.: A Catalyst-Free MCR Approach to 1,5-Benzodiazepines
Frutos, R. P.; Tampone, T.; Mulder, J. A.; Xu, Y.; Reeves, D.; Wang, X.-J.; Zhang, L.; Krishnamurthy, D.; Senanayake, C. H.: A Boronic Acid Catalyzed Route to Imidazoles. Synthesis of LFA-1 Antagonists
Blanchot, M.; Candito, D. A.; Larnaud, F.; Lautens, M.: Phenanthridine Synthesis via a Pd-Catalyzed Direct Arylation/N-Arylation Sequence
Attanasi, O. A.; Berretta, S.; De Crescentini, L.; Favi, G.; Giorgi, G.; Mantellini, F.; Nicolini, S.: Zinc(II)-Catalyzed Synthesis of Poly-functionalized Pyrroles
Ng, E. P. J.; Wang, Y.-F.; Chiba, S.: Mn(III)-Catalyzed Synthesis of Pyrroles from Vinyl Azides and β-Keto Acids
Kang, J. Y.; Connell, B. T.: Synthesis of Furans via Indium-Catalyzed Rearrangement of Acetylenic Epoxides
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Issue 05/2011

Salman, G. A.; Hussain, M.; Iaroshenko, V.; Villinger, A.; Langer, P.: Thienopyrroles and Benzothienoquinolines via Palladium-Catalyzed Domino Reactions
Vedachalam, S.; Wong, Q.-L.; Maji, B.; Zeng, J.; Ma, J.; Liu, X.-W.: Synthesis of Chromones via an Intramolecular Hydroacylation
Castanedo, G. M.; Seng, P. S.; Blaquiere, N.; Trapp, S.; Staben, S. T.: Metal-Free Synthesis of 1,3,5-Trisubstituted 1,2,4-Triazoles
Chunavala, K. C.; Joshi, G.; Suresh, E.; Adimurthy, S.: Catalyst- and Solvent-Free Synthesis of Substituted Imidazo[1,2-a]pyridines
Guru, M. M.; Ali, M. A.; Punniyamurthy, T.: Cu(II)-Catalyzed Synthesis of Benzoxazoles from Bisaryloxime Ethers
Wang, Z.-J.; Yang, F.; Lv, X.; Bao, W.: One-Pot Synthesis of Fused Unsymmetrical 2,2′-Biindolyls
Pews-Davtyan, A.; Beller, M.: Zinc-Catalyzed Hydroamination Route to Di- and Trisubstituted Imidazoles
Frolova, L. V.; Evdokimov, N. M.; Hayden, K.; Malik, I.; Rogelj, S.; Kornienko, A.; Magedov, I. V.: Synthesis of Polysubstituted 2-Aminopyrroles via a Multicomponent Reaction
Gurunathan, S.; Perumal, P. T.: Synthesis of Dihydroquinolines via Pd/Cu-Catalyzed Heteroannulation
Chen, Z.; Huang, G.; Jiang, H.; Huang, H.; Pan, X.: Palladium-Catalyzed Sonogashira Coupling and Iodocyclization Route to 3-Iodofurans
Xiong, Z.; Qiu, X.-L.; Huang, Y.; Qing, F.-L.: TBS-Directed 1,3-Dipolar Cycloaddition to 5-Trifluoromethyl-1,2,3-triazoles
Kunzer, A. R.; Wendt, M. D.: Synthesis of 2-Halo-3-carboxyindoles
Gross, U.; Gross, P. J.; Shi, M.; Bräse, S.: NHC-Catalyzed Synthesis of Coumarins
Adib, M.; Ansari, S.; Bijanzadeh, H. R.: Synthesis of N-Amino-Succinimides by a Multicomponent Reaction
Saito, T.; Ogawa, S.; Takei, N.; Kutsumura, N.; Otani, T.: Palladium-Catalyzed Heteroannulation Route to 4-Alkylidene-4H-3,1-benzoxazines
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Issue 04/2011

Balamurugan, K.; Jeyachandran, V.; Perumal, S.; Menéndez, J. C.: One-Pot Synthesis of Tetrahydroisoquinolines via Benzene Ring Annulation
Trost, B. M.; Lumb, J.-P.; Azzarelli, J. M.: Palladium-Catalyzed Atom-Economical Synthesis of Pyrroles
Rai, A.; Singh, A. K.; Singh, S.; Yadav, L. D. S.: Organocatalytic Cascade Synthesis of Decahydroquinolines
Cież, D.; Svetlik, J.: Synthesis of Imidazolin-5-ones by Thermolysis of α-Azido Esters
Lei, Y.; Wang, Z.-Q.; Xie, Y.-X.; Yu, S.-C.; Tang, B.-X.; Li, J.-H.: Base-Mediated Synthesis of 4,5-Disub-stituted Furan-2(5H)-ones
Yu, X.; Pan, X.; Wu, J.: Synthesis of Pyrazoloisoquinolines via a Multicomponent Suzuki Reaction Sequence
Attanasi, O. A.; De Crescentini, L.; Favi, G.; Nicolini, S.; Perrulli, F. R.; Santeusanio, S.: Synthesis of 1,3,5-Trisubstituted Hydantoin via a Three-Component Reaction
Světík, J.; Kettmann, V.: Unexpected Products from the Biginelli Reactions of 3-Amino-1,2,4-triazole
Liang, F.; Lin, S.; Wei, Y.: Synthesis of Furo[3,2-c]pyridinones via an Aza-Oxy-Carbanion Relay Strategy
D’Souza, A. M.; Spiccia, N.; Basutto, J.; Jokisz, P.; Wong, L. S.-M.; Meyer, A. G.; Holmes, A. B.; White, J. M.; Ryan, J. H.: 1,3-Dipolar Cycloaddition Route to 1,3-Benzodiazepinones
Kumar, P. M.; Kumar, K. S.; Poreddy, S. R.; Mohakhud, P. K.; Mukkanti, K.; Pal, M.: Extending the Scope of the Biginelli Reaction Using Palladium Catalysis
Gainer, M. J.; Bennett, N. R.; Takahashi, Y.; Looper, R. E.: Rhodium(II)-Catalyzed Hydroamination of Propargylguanidines
Dell’Acqua, M.; Facoetti, D.; Abbiati, G.; Rossi, E.: Sonogashira-Heteroannulative Route to Dihydroisobenzofurans
Wang, W.; Ollio, S.; Herdtweck, E.; Dömling, A.: Combined Ugi-Pictet-Spengler Synthesis of Polycyclic Ketopiperazines
Jen, T.; Mendelsohn, B. A.; Ciufolini, M. A.: Oxidative Approach to Isoxazolines
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Issue 03/2011

Too, P. C.; Wang, Y.-F.; Chiba, S.: Rhodium(III)-Catalyzed Heteroannulation Route to Isoquinolines
Zhang, X.; Teo, W. T.; Chan, P. W. H.: Ytterbium(III)-Catalyzed Synthesis of 2-Aryloxazoles
Shafi, S.; Kędziorek, M.; Grela, K.: Cross-Metathesis Strategy for Pyrrole Synthesis
Nayak, M.; Batra, S.: Copper-Catalyzed Synthesis of Heterofused Benzoxazepines and -diazepines
Maestri, G.; Larraufie, M.-H.; Derat, E.; Ollivier, C.; Fensterbank, L.; Lacôte, E.; Malacria, M.: Synthesis of Phenanthridines via Palladium/Norbornene Catalysis
Siry, S. A.; Timoshenko, V. M.: Synthesis and Reactivity of 2-Polyfluoroalkyl Thiopyrylium Salts
Halland, N.; Nazaré, M.; Alonso, J.; R’kyek, O.; Lindenschmidt, A.: Domino Approach to 1-Aminoindoles from 2-Halophenylacetylenes
Alonso, J.; Halland, N.; Nazaré, M.; R’kyek, O.; Urmann, M.; Lindenschmidt, A.: Pd-Catalyzed Heteroannulative Synthesis of Benzimidazoles and Imidazopyridines
Bartrum, H. E.; Blakemore, D. C.; Moody, C. J.; Hayes, C. J.: In-Flow Approach to β-Keto Esters and Use in the Synthesis of Pyrimidines
Kazmaier, U.; Persch, A.: Synthesis of 5-Substituted Thiazolyl Peptides via the Thio-Ugi Reaction
Chen, K.-P.; Chen, Y.-J.; Chuang, C.-P.: α-Nitrocinnamate Esters for the Synthesis of Highly Functionalized Isoxazoles
Majumdar, K. C.; Ponra, S.; Ghosh, D.; Taher, A.: Multicomponent Aza-Diels-Alder Synthesis of Phenanthrolines and Pyranoquinolines
Cao, H.; Vieira, T. O.; Alper, H.: Palladium-Catalyzed Heteroannulation Route to Benzazepinones
Hu, H.; Shi, K.; Hou, R.; Zhang, Z.; Zhu, Y.; Zhoua, J.: One-Pot Synthesis of Indolizines from Pyridines, Benzyl Halides, and Alkenes
Ouyang, H.-C.; Tang, R.-Y.; Zhong, P.; Zhang, X.-G.; Li, J.-H.: CuI/I2-Mediated Synthesis of Iodoisoquinoline-Fused Benzimidazoles
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Issue 02/2011

Li, Y.; Wheeler, K. A.; Dembinski, R.: Au/Ag-Catalyzed Synthesis of 3-Fluorofurans
Kurochkin, N. N.; Fesenko, A. A.; Cheshkov, D. A.; Davudi, M. M.; Shutalev, A. D.: Acid-Catalyzed Rearrangement of Ureido-dihydrofurans to N-Pyrrole Ureas
Lin, S.; Zhao, G.-L.; Deiana, L.; Sun, J.; Zhang, Q.; Leijonmarck, H.; Córdova, A.: Enantioselective Synthesis of Dihydrofurans Using Dynamic Kinetic Resolution
Wang, C.; Li, S.; Liu, H.; Jiang, Y.; Fu, H.: Copper-Catalyzed Ullmann-Type Coupling Route to Quinazolines
Jiang, H.; Huang, H.; Cao, H.; Qi, C.: Synthesis of Oxazoles via TBHP/I2-Mediated Reaction of Alkenes with Benzylic Amines
Ermolat’ev, D. S.; Bariwal, J. B.; Steenackers, H. P. L.; De Keersmaecker, S. C. J.; Van der Eycken, E. V.: Silver-Catalyzed Synthesis of 2-Amino-imidazole Alkaloids
De Sarkar, S.; Studer, A.: NHC-Catalyzed Michael Addition for the Synthesis of Dihydropyranones
Ozawa, T.; Horie, H.; Kurahashi, T.; Matsubara, S.: A Nickel-Catalyzed [2+2+1]-Cycloaddition Approach to Lactams
Cioffi, C. L.; Lansing, J. J.; Yüksel, H.: Synthesis of 2-Aminobenzoxazoles from 2-Aminophenols
Cikotiene, I.; Sazinas, R.; Mazeikaite, R.; Labanauskas, L.: Synthesis of Fused Thiophene-Isoxazoles from 2-Alkynyl-3-Nitro-Thiophenes
Zeng, F.; Alper, H.: Synthesis of 1,4-Benzothiazepin-5-ones from N-Tosyl Aziridines and 2-Iodothiophenols
Campbell, J. B.; Dedinas, R. F.; Trumbower-Walsh, S.: Synthesis of Isoindolones from Imines and ortho-Iodobenzoyl Acid Chlorides
Sanz, R.; Guilarte, V.; Hernando, E.; Sanjuán, A. M.: Directed ortho-Metalation-Halocyclization Route to Benzothiophenes
Huang, J.; Macdonald, S. J. F.; Harrity, J. P. A.: Palladium-Catalyzed Heterannulation Synthesis of 3-Borylated Indoles
Li, C.; Zhang, Q.; Tong, X.: Tertiary Amine Catalyzed Annulation Route to Tetrasubstituted Pyrans
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Issue 01/2011

Álvarez, R.; Martínez, C.; Madich, Y.; Denis, J. G.; Aurrecoechea, J. M.; de Lera, Á. R.: Benzofurans, Indoles, and Isoquinolones via Castro-Stephens and Heck Reactions
Dong, C.; Xie, L.; Mou, X.; Zhong, Y.; Su, W.: Palladium-Catalyzed Synthesis of 1,3,4-Benzotriazepines and Indazoles
Li, R.-J.; Pi, S.-F.; Liang, Y.; Wang, Z.-Q.; Song, R.-J.; Chen, G.-X.; Li, J.-H.: Palladium-Catalyzed Annulation Route to 6H-Benzo[c]chromenes
Muthusaravanan, S.; Perumal, S.; Yogeeswari, P.; Sriram, D.: Substituted Indolizines via a Multicomponent 1,3-Dipolar Cycloaddition Strategy
Liu, C.; Zhang, X.; Wang, R.; Wang, W.: Synthesis of 4H-Chromenes by an Enantio-selective Oxa-Michael-Aldol Reaction
Chen, J.; Ma, S.: Regioselective Synthesis of 2-Alkoxyfurans from Cyclopropenyl Carboxylates
Ballini, R.; Gabrielli, S.; Palmieri, A.; Petrini, M.: Metal-Free Synthesis of 1,4-Disubstituted Carbazoles from Sulfonylindoles
Morin, M. S. T.; St-Cyr, D. J.; Arndtsen, B. A.: Horner-Wadsworth-Emmons Reagent as 1,3-Dipolar Cycloaddition Precursor
Ouizem, S.; Cheramy, S.; Botuha, C.; Chemla, F.; Ferreira, F.; Pérez-Luna, A.: Cyclization of Zincated Homoallylamino Nitriles to Methanopyrrolidines
Lourdusamy, E.; Yao, L.; Park, C.-M.: Synthesis of Pyrroles by [3+2] Cycloaddition of α-Diazo Oxime Ethers with Alkenes
Patil, N. T.; Raut, V. S.: Metal/Amine Cooperative Catalysis. Heteroannulation Route to Quinolines
Jacq, J.; Bessières, B.; Einhorn, C.; Einhorn, J.: 1,3-Diaryl Isobenzofurans from Arylboronic Acids and ortho-Keto Aldehydes
Yagoubi, M.; Cruz, A. C. F.; Nichols, P. L.; Elliott, R. L.; Willis, M. C.: Palladium-Catalyzed Heteroannulation Route to Indoles and Benzofurans
Seki, H.; Georg, G. I.: Synthesis of Dihydropyridin-4(1H)-ones via Wolff Rearrangement
Zeng, L.-Y.; Cai, C.: Multicomponent Synthesis of Azaphenanthreneamides
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Issue 12/2010

Desai, A. A.; Wulff, W. D.: Synthesis of Chiral Aziridines from Imines and Diazoacetamides
Shimizu, R.; Egami, H.; Nagi, T.; Chae, J.; Hamashima, Y.; Sodeoka, M.: Direct C2 Indole Trifluoromethylation Using Togni’s Reagent
Baeza, A.; Mendiola, J.; Burgos, C.; Alvares-Builla, J.; Vaquero, J. J.: Synthesis of Pyridopyrrolopyrimidines. Total Synthesis of Varioline B and Deoxyvariolin B
Akkilagunta, V. K.; Reddy, V. P.; Kakulapati, R. R.: Synthesis of Quinoxalines via Ru/C Benzoin Oxidation and Diamine Condensation
Zhang, X.; Teo, W. T.; Sally; Chan, P. W. H.: Facile Acid-Catalyzed Route to Thiazoles from Propargylic Alcohols and Thioamides
Hong, D.; Chen, Z.; Lin, X.; Wang, Y.: Synthesis of Indoles from 2-Azidoacrylate and ortho-Silyl Aryltriflates
Ballini, R.; Gabrielli, S.; Palmieri, A.: Synthesis of Tetrasubstituted Furans by Michael Addition to β-Nitroacrylates
Toyoshima, T.; Mikano, Y.; Miura, T.; Murakami, M.: Palladium-Catalyzed Synthesis of 3,3-Disubstituted Oxindoles
Barluenga, J.; Lonzi, G.; Riesgo, L.; López, L. A.; Tomás, M.: Copper(I)-Catalyzed Annulation Route to Indolizines
Wray, B. C.; Stambuli, J. P.: Synthesis of N-Arylindazoles and Benz-imidazoles from ortho-Aminobenzoximes
Inman, M.; Moody, C. J.: Copper-Mediated Synthesis of Indolequinones from Bromoquinones
Yang, Q.; Cao, H.; Robertson, A.; Alper, H.: Palladium-Catalyzed Cyclocarbonylative Synthesis of Dibenzoxazepinones
Fujita, M.; Yoshida, Y.; Miyata, K.; Wakisaka, A.; Sugimura, T.: Enantioselective Synthesis of Dihydro-isochromanones Using Hypervalent Iodine
Kwok, S. W.; Fotsing, J. R.; Fraser, R. J.; Rodionov, V. O.; Fokin, V. V.: Synthesis of 1,5-Diaryl-1,2,3-triazoles Under Transition-Metal-Free Conditions
Zeghida, W.; Besnard, C.; Lacour, J.: Rhodium(II)-Catalyzed Synthesis of Polyether Macrocyles
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Issue 11/2010

Spergel, S. H.; Okoro, D. R.; Pitts, W.: Palladium-Catalyzed α-Heteroarylation Route to 4-, 5-, 6- and 7-Azaindoles
Yan, R.-L.; Luo, J.; Wang, C.-X.; Ma, C.-W.; Huang, G.-S.; Liang, Y.-M.: Copper-Catalyzed Synthesis of Poly-substituted Pyrroles from Enamino Ketones
Wang, X.; Lu, Y.; Dai, H.-X.; Yu, J.-Q.: Palladium(II)-Catalyzed Heteroannulation Route to Dihydrobenzofurans
Misra, N. C.; Ila, H.: 4-Bis(methylthio)methylene-2-phenyloxazol-5-one: Template for Oxazoles
Kobatake, T.; Fujino, D.; Yoshida, S.; Yorimitsu, H.; Oshima, K.: Synthesis of Trifluoromethylbenzofurans by Extended Pummerer Reaction
Pohjakallio, A.; Pihko, P. M.; Laitinen, U. M.: Synthesis of 2-Isoxazolines via Conjugate Additions
Mai, D. N.; Wolfe, J. P.: Synthesis of Chiral Pyrrolidines by Palladium-Catalyzed Carboamination
Zhang, J.; Senthilkumar, M.; Ghosh, S. C.; Hong, S. H.: Ruthenium-Catalyzed Synthesis of Cyclic Imides
Lin, M.; Hao, L.; Ma, R.-d.; Zhan, Z.-p.: Indium-Mediated Multicomponent Synthesis of Pyrroles
Liu, F.; Qian, D.; Li, L.; Zhao, X.; Zhang, J.: Gold(I)-Catalyzed Synthesis of Furo[3,4-d]-[1,2]oxazines
Zhang, Q.; Fang, T.; Tong, X.: Triphenylphosphine-Catalyzed Synthesis of Dihydropyridines and Pyrans
Jana, S.; Clements, M. D.; Sharp, B. K.; Zheng, N.: Synthesis of 2,3-Disubstituted Indoles by Iron(II)-Catalyzed Aromatic C-H Amination
Crossley, J. A.; Browne, D. L.: Cycloaddition Route to 4-Iodoisoxazoles
Chen, W.; Hu, M.; Wu, J.; Zou, H.; Yu, Y.: Synthesis of Pyrrolo[1,2-a]pyrazines from Vinyl Azides
Kaïm, L. El; Grimaud, L.; Ronsseray, C.: One-Pot Modified Japp-Klingeman-Fischer Indole Synthesis
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Issue 10/2010

Fordyce, E. A. F.; Morrison, A. J.; Sharp, R. D.; Paton, R. M.: Synthesis of 1,2,4-Thiadiazoles and Isothiazoles
Kim, J.; Song, H.; Park, S. B.: Regioselective Synthesis of N-Alkyl-3-substituted Tetrahydroindazolones
Ye, L.; He, W.; Zhang, L.: Gold-Catalyzed Synthesis of Oxetan-3-ones from Propargylic Alcohols
Bonnamour, J.; Piedrafita, M.; Bolm, C.: Effect of Fe and Cu Salts in the Heteroannulative Synthesis of Benzo[b]furans
Awasthi, C.; Yadav, L. D. S.: NHC-Mediated [2+2] Cycloaddition Route to Nitro-β-thiolactams
Yu, H.; Jin, W.; Sun, C.; Chen, J.; Du, W.; He, S.; Yu, Z.: Synthesis of Bicyclic Pyridones from 1,3-Butadienes
Li, S.; Yuan, Y.; Zhu, J.; Xie, H.; Chen, Z.; Wu, Y.: Copper-Catalyzed Annulative Synthesis of 2-Fluoromethylated Quinolines
Liu, C.-C.; Parthasarathy, K.; Cheng, C.-H.: Nickel-Catalyzed Heteroannulative Route to Isoquinolones
Parsons, A. T.; Smith, A. G.; Neel, A. J.; Johnson, J. S.: Mg-Catalyzed Dynamic Asymmetric Synthesis of Chiral Pyrrolidines
Xi, J.; Dong, Q.-L.; Liu, G.-S.; Wang, S.; Chen, L.; Yao, Z.-J.: Bischler-Napieralski Synthesis of Phenanthridines
Tobisu, M.; Fujihara, H.; Koh, K.; Chatani, N.: Copper-Catalyzed Borylative and Silylative Cyclization of Isocyanides to Indoles
Spiteri, C.; Keeling, S.; Moses, J. E.: 1H-Indazoles via Huisgen [3+2] Cycloaddition of Benzynes with Nitrile Imines
Malakar, C. C.; Merisor, E.; Conrad, J.; Beifuss, U.: Molybdenum Complex Catalyzed Reductive Cyclization of ω-Nitro Alkenes
Polivanova, A. G.; Shkavrov, S. V.; Churakov, A. V.; Lermontov, A. S.; Lermontov, S. A.: Synthesis of 1,5-Disubstituted Fluorinated Tetrazoles
Brenzovich Jr., W. E.; Benitez, D.; Lackner, A. D.; Shunatona, H. P.; Tkatchouk, E.; III, W. A. Goddard; Toste, F. D.: Gold-Catalyzed Intramolecular Aminoarylation to Pyrrolidines
All PDFs of this category

Issue 09/2010

He, Z.; Li, H.; Li, Z.: Intramolecular Cyclization of Enamines to 3H-Indoles Mediated by Iodine
Lamandé-Langle, S.; Abarbri, M.; Thibonnet, J.; Duchêne, A.; Parrain, J.-L.: Palladium-Catalyzed Three-Component Synthesis of Pyrroles
Cacchi, S.; Fabrizi, G.; Goggiamani, A.; Perboni, A.; Sferrazza, A.; Stabile, P.: Palladium-Catalyzed Synthesis of 2,3-Di-substituted Indoles from Aryldiazonium Salts
Gong, X.; Yang, H.; Liu, H.; Jiang, Y.; Zhao, Y.; Fu, H.: Copper-Catalyzed Synthesis of 2,4-Disubstituted Imidazolones
Ca’, N. Della; Motti, E.; Mega, A.; Catellani, M.: Palladium-Catalyzed Multicomponent Synthesis of Phenanthridines
Kienle, M.; Unsinn, A.; Knochel, P.: Synthesis of Sulfur Heterocycles from Dithiocarbamates
Turner, M.; Linder, T.; Schnürch, M.; Mihovilovic, M. D.; Stanetty, P.: Concerning the Regioselectivity of the Hurd-Mori Reaction for 1,2,3-Thiadiazoles
Shi, Z.; Cui, Y.; Jiao, N.: Heteroannulation Route to β- and γ-Carbolinones from Indolecarboxamides
Tang, B.-X.; Song, R.-J.; Wu, C.-Y.; Liu, Y.; Zhou, M.-B.; Wei, W.-T.; Deng, G.-B.; Yin, D.-L.; Li, J.-H.: Copper-Catalyzed Synthesis of Isatins from Formyl-N-arylformamides
Gao, X.; Pan, Y.-m.; Lin, M.; Chen, L.; Zhan, Z.-p.: Silver- and Iron-Catalyzed Synthesis of Substituted Thiazoles
Saleem, R. S. Z.; Tepe, J. J.: Heterocyclic Interconversion of Oxazolones into Triazolines and Triazoles
Xin, X.; Wang, Y.; Kumar, S.; Liu, X.; Lin, Y.; Dong, D.: Multicomponent Synthesis of Polysubstituted Pyridines
Guimond, N.; Gouliaras, C.; Fagnou, K.: Rhodium-Catalyzed Synthesis of Isoquinolones
Uyanik, M.; Yasui, T.; Ishihara, K.: Catalytic Hypervalent Iodine Spirolacton-ization Using m-CPBA as Co-Oxidant
Miura, T.; Yamauchi, M.; Kosaka, A.; Murakami, M.: Nickel-Catalyzed Annulative Synthesis of 1,2-Benzothiazine-1,1(2H)-dioxides
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Issue 08/2010

Nakamura, I.; Zhang, D.; Terada, M.: Copper-Catalyzed Synthesis of Pyridine N-Oxides from α,β-Unsaturated Oximes
Lu, J.; Gong, X.; Yang, H.; Fu, H.: Copper-Catalyzed One-Pot Synthesis of Benzimidazo[1,2-b]isoquinolin-11-ones
Gaddam, V.; Ramesh, S.; Nagarajan, R.: CuI/La(OTf)3-Catalyzed Synthesis of Isomeric Ellipticine
Moghaddam, F. M.; Mirjafary, Z.; Saeidian, H.; Taheri, S.; Soltanzadeh, B.: One-Step Synthesis of Annulated Hydroquinolines
Chen, Z.; Zhu, J.; Xie, H.; Li, S.; Wu, Y.; Gong, Y.: Copper-Catalyzed Cascade Synthesis of Triazoloquinoxalines
Varela-Fernández, A.; García-Yebra, C.; Varela, J. A.; Esteruelas, M. A.; Saá, C.: Osmium-Catalyzed Synthesis of 3-Benzoxepines
Ye, Z.; Lv, G.; Wang, W.; Zhang, M.; Cheng, J.: Rhodium-Catalyzed Synthesis of 3-Aryl and 3-Alkenyl Phthalides
Spiteri, C.; Mason, C.; Zhang, F.; Ritson, D. J.; Sharma, P.; Keeling, S.; Moses, J. E.: Synthesis of 1,2-Benzisoxazoles via a 1,3-Dipolar Cycloaddition
Koldobskii, A. B.; Tsvetkov, N. P.; Solodova, E. V.; Kalinin, V. N.: A Lactonization Route to 5-(Trifluoromethyl)-2(5H)-furanones
Liu, Y.; Bao, W.: Synthesis of 1,4-Benzodioxanes via Epoxide Opening and Cyclization
Wahab, B.; Ellames, G.; Passey, S.; Watts, P.: Synthesis of Substituted Indoles Using Flow Microreactors
Wang, H.-Y.; Mueller, D. S.; Sachwani, R. M.; Londino, H. N.; Anderson, L. L.: Synthesis of Pyrroles via [3,3]-Rearrangement and Paal-Knorr Reaction
Volkova, Y. A.; Averina, E. B.; Grishin, Y. K.; Bruheim, P.; Kuznetsova, T. S.; Zefirov, N. S.: One-Step Synthesis 3-Nitroisoxazoles
Wu, C.; Fang, Y.; Larock, R. C.; Shi, F.: Synthesis of 2H-Indazoles via [3+2]-Dipolar Cycloaddition
Ueda, M.; Sato, A.; Ikeda, Y.; Miyoshi, T.; Naito, T.; Miyata, O.: Synthesis of Trisubstituted Isoxazoles via Gold-Catalyzed Domino Reaction
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Issue 07/2010

Reddy, U. C.; Saikia, A. K.: Multicomponent Prins-Friedel-Crafts Synthesis of 4-Aryl-5,6-Dihydropyrans
Zhou, H.; Zhu, D.; Xie, Y.; Huang, H.; Wang, K.: Gallium-Catalyzed Synthesis of 1,3-Dihydrobenzo[c]thiophenes
Yang, X.; Fu, H.; Qiao, R.; Jiang, Y.; Zhao, Y.: α-Arylation-Heteroannulation Route to 2-Amino-1H-indole-3-carboxylates
Zhang, X.; Lu, Z.; Fu, C.; Ma, S.: Synthesis of Polysubstituted Furans by a Sonogashira-Cyclization Route
Chernyak, D.; Chernyak, N.; Gevorgyan, V.: Copper-Catalyzed Three-Component Coupling Synthesis of 3-Aminoindol(in)es
Lu, Y.; Wang, D.-H.; Engle, K. M.; Yu, J.-Q.: Synthesis of Isochromans by Palladium-Catalyzed C-H Olefination
Coy B., E. D.; Jovanovic, L.; Sefkow, M.: trans-Dihydrobenzofurans via Diazotization-Palladium-Catalyzed Oxyarylation
Xing, C.-H.; Liao, Y.-X.; He, P.; Hu, Q.-S.: Rhodium-Catalyzed Synthesis of Chiral 3-Substituted Phthalides
Mohanan, K.; Martin, A. R.; Toupet, L.; Smietana, M.; Vasseur, J.-J.: Regioselective Synthesis of Phosphonyl Pyrazoles
Fuwa, H.; Matsukida, S.; Sasaki, M.: Dihydropyranone Synthesis Using a Sonogashira Coupling
Shen, G.; Bao, W.: Copper(I)-Catalyzed Synthesis of Benzoxazoles and Benzimidazoles
Xin, Y.; Zhao, J.; Han, J.; Zhu, S.: 1,3-Dipolar Cycloaddition Synthesis of 3-Trifluoroacetyl Pyrroles
Yu, X.; Du, B.; Wang, K.; Zhang, J.: Synthesis of 2,3-Dihydroisoxazoles from Enynes and Hydroxylamines
Lefebvre, V.; Cailly, T.; Fabis, F.; Rault, S.: Hydrazone C-N Coupling Route to 3-Aminoindazoles
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Issue 06/2010

Yasmin, N.; Ray, J. K.: Efficient Heteroannulation Route for the Synthesis of Isoindoles and Pyrroles
Lorion, M.; Agouridas, V.; Couture, A.; Deniau, E.; Grandclaudon, P.: Synthesis of Benzosultams from Cyclic Sulfamidates
Ding, C.; Tu, S.; Yao, Q.; Li, F.; Wang, Y.; Hu, W.; Zhang, A.: Radical-Mediated Decarboxylative Route to Naphtho[2,3-a]carbazoles
Guan, Z.-H.; Yan, Z.-Y.; Ren, Z.-H.; Liu, X.-Y.; Liang, Y.-M.: Synthesis of Indoles via Iron-Catalyzed Heteroannulative Oxidative Coupling
Adib, M.; Ansari, S.; Feizi, S.; Bijanzadeh, H. R.: Multicomponent Synthesis of Triazoloquinazolines
Cai, Q.; Li, Z.; Wei, J.; Fu, L.; Ha, C.; Pei, D.; Ding, K.: Copper-Catalyzed Synthesis of Aza-Fused Polycyclic Quinolines
Lu, H.; Tao, J.; Jones, J. E.; Wojtas, L.; Zhang, X. P.: Synthesis of Cyclophosphoramidates by Intramolecular C-H Amination
Kondoh, A.; Yorimitsu, H.; Oshima, K.: Palladium-Catalyzed Heteroannulation Route to 2-Indolylphosphines
Zeng, F.; Alper, H.: Synthesis of 2-Heteroquinazolin-4-(3H)-ones via Palladium Catalysis
Ye, L.; Cui, L.; Zhang, G.; Zhang, L.: Gold-Catalyzed Synthesis of Dihydrofuran-3-ones from Homopropargylic Alcohols
Huo, Z.; Gridnev, I. D.; Yamamoto, Y.: Electrophile-Induced Cyclization of ortho-Azido Propynyl Benzenes to Quinolines
Majumder, S.; Odom, A. L.: Pyrimidine Synthesis via a Titanium-Catalyzed Multicomponent Reaction
Dubrovskiy, A. D.; Larock, R. C.: Synthesis of Benzisoxazoles by [3+2] Cycloaddition of Nitrile Oxides with Arynes
Liu, Y.; Wang, M.; Yuan, H.; Liu, Q.: Copper(II) Bromide/BoronTrifluoride Cocatalyzed Synthesis of Benzofurans
Liu, Y.; Qian, J.; Lou, S.; Zhu, J.; Xu, Z.: Gold(III)-Catalyzed Synthesis of 4H-Chromenes
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Issue 05/2010

Vorobyeva, D. V.; Karimova, N. M.; Vasilyeva, T. P.; Osipov, S. N.; Shchetnikov, G. T.; Odinets, I. L.; Röschenthaler, G.-V.: Copper-Catalyzed Synthesis of Triazolyl-α-CF3-α-Aminophosphonates
Oh, C. H.; Karmakar, S.; Park, H.; Ahn, Y.; Kim, J. W.: Silver-Catalyzed Heteroannulation Route to Indoles
Pews-Davtyan, A.; Tillack, A.; Schmöle, A.-C.; Ortinau, S.; Frech, M. J.; Rolfs, A.; Beller, M.: Zinc Halide Mediated Synthesis of 3-Amidoindoles
Dheur, J.; Sauthier, M.; Castanet, Y.; Mortreux, A.: Rhodium-Catalyzed Carbonylative Addition-Cyclization Approach to Furans
Spiteri, C.; Sharma, P.; Zhang, F.; Macdonald, S. J. F.; Keeling, S.; Moses, J. E.: Synthesis of 1,2-Benzisoxazoles by 1,3-Dipolar Cycloaddition
Devarie-Baez, N. O.; Xian, M.: One-Pot Synthesis of Benzisothiazoles from ortho-Mercaptoacylphenones
Saito, T.; Furukawa, N.; Otani, T.: Pyrrolo[2,3-b]quinolines via a Rhodium-Catalyzed Pauson-Khand-Type Reaction
Reichelt, A.; Falsey, J. R.; Rzasa, R. M.; Thiel, O. R.; Achmatowicz, M. M.; Larsen, R. D.; Zhang, D.: Triazolopyridines via Selective Palladium-Catalyzed Monoarylation of Hydrazides
Meng, T.-j.; Hu, Y.; Wang, S.: Palladium-Catalyzed Synthesis of Five-Membered Heterocycles from 1,6-Enynes
Zhang, Z.; Zhang, Q.; Ni, Z.; Liu, Q.: Silver-Mediated Synthesis of Furo[3,2-b]-β/γ-Lactams
Yang, Q.; Alper, H.: Ligand-Free Cyclocarbonylation of ortho-Iodophenols and Acetylenes to Chromones
Gorugantula, S. P.; Carrero-Martínez, G. M.; Dantale, S. W.; Söderberg, B. C. G.: Palladium-Catalyzed Synthesis of Pyrrolo-Fused Compounds from Nitroarenes
Li, J.; Li, S.; Li, C.; Liu, Y.; Jia, X.: Tandem Conjugate Addition-Cyclization Synthesis of 1,5-Benzodiazepines
Ma, D.; Geng, Q.; Zhang, H.; Jiang, Y.: Copper/l-Proline-Catalyzed Synthesis of Phenothiazines
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Issue 04/2010

Zhang, G.; Cui, L.; Wang, Y.; Zhang, L.: Gold-Catalyzed Synthesis of THFs and Pyrrolidines by Oxidative Coupling
Huang, X.; Zhang, T.: Synthesis of C9-Functionalized Xanthenes and Acridines
Liu, W.; Jiang, H.; Zhang, M.; Qi, C.: Synthesis of Highly Substituted Furans from Alkynoates and 1,3-Dicarbonyls
Zhang, X.; Yao, T.; Campo, M. A.; Larock, R. C.: Halo-Induced Heteroannulation Route to Quinolines
Han, J.; Xu, B.; Hammond, G. B.: Copper-Catalyzed Synthesis of Pyrrolidines and Piperidines
Vovk, M. V.; Golovach, N. M.; Sukach, V. A.: Synthesis of 4-Aryl-4-trifluoromethyl-4H-1,3-oxa(thia)zines
Zeng, X.; Kinjo, R.; Donnadieu, B.; Bertrand, G.: Gold(I)-Catalyzed Hydroammoniumation and Methylamination of Alkynes to Indoles
Matsnev, A.; Noritake, S.; Nomura, Y.; Tokunaga, E.; Nakamura, S.; Shibata, N.: Synthesis of Thiophenium Salts: A Trifluoromethylation Reagent
Peng, C.; Wang, Y.; Liu, L.; Wang, H.; Zhao, J.; Zhu, Q.: Synthesis of Substituted Quinolines from 2-Alkynylanilines
He, Z.-Q.; Han, B.; Li, R.; Wu, L.; Chen, Y.-C.: Enantioselective Synthesis of Lactone-[2,3-b]piperidines
Fontana, F.; Tron, G. C.; Barbero, N.; Ferrini, S.; Thomas, S. P.; Aggarwal, V. K.: Palladium-Catalyzed Synthesis of β-Lactams by Carbonylation of Vinyl Aziridines
Liu, W.; Jiang, H.; Huang, L.: Synthesis of Polysubstituted Pyrroles by Condensation of Acetylenes and Amines
Okitsu, T.; Nakazawa, D.; Kobayashi, A.; Mizohata, M.; In, Y.; Ishida, T.; Wada, A.: Iodocyclization-Based Synthesis of Spiro Heterocycles
Zhao, T.; Xu, B.: Palladium-Catalyzed C-N Coupling-Hydroamination Route to 4-Quinolones
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Issue 03/2010

Tejedor, D.; Méndez-Abt, G.; García-Tellado, F.: Substituted Dihydropyridines from Propargyl Enol Ethers
Wu, T.; Yin, G.; Liu, G.: Pd-Catalyzed Synthesis of Fluoropiperidines
Staben, S. T.; Blaquiere, N.: Pd-Catalyzed Synthesis of 1,2,4-Triazoles
Wong, Y.-C.; Parthasarathy, K.; Cheng, C.-H.: Cobalt-Catalyzed Synthesis of Pyrrolidinones from Nitriles and Acrylamides
Baxendale, I. R.; Schou, S. C.; Sedelmeier, J.; Ley, S. V.: General Syntheses of Heterocycles Using Modular Flow Reactors
Xu, X.; Li, H.; Xie, X.; Li, Y.: Iron-Catalyzed Synthesis of 9-Substituted Xanthenes
Yang, X.; Liu, H.; Fu, H.; Qiao, R.; Jiang, Y.; Zhao, Y.: Copper-Catalyzed Synthesis of Quinazolines From 2-Bromobenzonitriles
Jiang, H.; Mai, R.; Cao, H.; Zhu, Q.; Liu, X.: l-Proline-Catalyzed Synthesis of Highly Substituted 1,4-Dihydropyridines
Okamoto, N.; Miwa, Y.; Minami, H.; Takeda, K.; Yanada, R.: Platinum-Catalyzed Synthesis of Indoles and Isoquinolines from 2-Alkynylarylamides
Chernyak, N.; Tilly, D.; Li, Z.; Gevorgyan, V.: Palladium-Catalyzed Synthesis of Fused Heterocycles
Gao, H.; Zhao, X.; Yu, Y.; Zhang, J.: Gold-Catalyzed Synthesis of Furo[3,4-c]-azepines
Queffélec, C.; Montchamp, J.-L.: Synthesis of Diverse P,N-Containing Heterocycles
Han, X.; Lu, X.: Pd-Catalyzed Synthesis of Dihydrocoumarins
Shen, Z.; Lu, X.: Copper-Mediated Halocyclization Route to 3-Haloindoles
Chouhan, G.; Alper, H.: Synthesis of 1,4-Benzo- and Pyrido-oxazepinones via a Domino Process
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Issue 02/2010

Varela-Fernández, A.; González-Rodrígues, C.; Varela, L. A.; Castedo, L.; Saá, C.: Ruthenium-Catalyzed Heteroannulation Route to Benzofurans and Isochromenes
Morgans, G. L.; Ngidi, E. L.; Madeley, L. G.; Khanye, S. D.; Michael, J. P.; de Koning, C. B.; van Otterlo, W. A. L.: Allylation-Isomerization-RCM Strategy for Benzo-Fused 1,4-Heteroatom Heterocycles
Dumitrascu, F.; Georgescu, E.; Caira, M. R.; Georgescu, F.; Popa, M.; Draghici, B.; Dumitrescu, D. G.: [2+3] Cycloaddition Approach to Multisubstituted N-Arylpyrroles
Chen, Z.; Yu, X.; Su, M.; Yang, X.; Wu, J.: AgOTf/Bi(OTf)3-Catalyzed Synthesis of Isoquinolines
Shen, G.; Lv, X.; Bao, W.: Copper-Catalyzed Synthesis of 2-Amino-benzothiazoles
Fustero, S.; Catalán, S.; Aceña, J. L.; Pozo, C. del: Synthesis of 6-Fluorinated 3,4-Dihydro-pyrimidinones
Tsuchikama, K.; Hashimoto, Y.-k.; Endo, K.; Shibata, T.: Iridium-Catalyzed Heteroannulation Route to Benzofurans and Indoles
Trogu, E.; Cecchi, L.; De Sarlo, F.; Guideri, L.; Ponticelli, F.; Machetti, F.: Copper-Catalyzed Synthesis of Isoxazoles
Jeanty, M.; Blu, J.; Suzenet, F.; Guillaumet, G.: Synthesis of 4- and 6-Azaindoles via the Fischer Indole Reaction
Guo, X.; Yu, R.; Li, H.; Li, Z.: Iron-Catalyzed Synthesis of Polysubstituted Benzofurans
Ishiwata, Y.; Togo, H.: Synthesis of Oxazoles from Alkyl Aryl Ketones and Nitriles Using Oxone
Saha, P.; Ramana, T.; Purkait, N.; Ali, M. A.; Paul, R.; Punniyamurthy, T.: Copper Nanoparticle Catalyzed Synthesis of Benzimidazoles, -oxazoles and -thiazoles
Adib, M.; Ansari, S.; Feizi, S.; Damavandi, J. A.; Mirzaei, P.: Multicomponent Synthesis of Trisubstituted Imidazoles
Yoshikawa, T.; Shindo, M.: Synthesis of 2-Pyrones and Tetronic Acids via Silver(I) Catalysis
Cai, Q.; Li, Z.; Wei, J.; Ha, C.; Pei, D.; Ding, K.: Copper-Catalyzed Synthesis of Indole-2-carboxylates
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Issue 01/2010

Ueda, S.; Nagasawa, H.: Copper-Catalyzed Synthesis of 1,2,4-Triazoles
Liang, Z.; Hou, W.; Du, Y.; Zhang, Y.; Pan, Y.; Mao, D.; Zhao, K.: FeCl3-Mediated Synthesis of Benzo[b]furans from α-Aryl Ketones
Lage, S.; Martínez-Estíbalez, U.; Sotomayor, N.; Lete, E.: Palladium-Catalyzed Synthesis of Pyrroloisoquinolines and Isoindoles
Yasmin, N.; Ray, J. K.: Cs2CO3-Promoted Synthesis of Substituted Oxazoles
Mizuno, A.; Kusama, H.; Iwasawa, N.: Rhodium-Catalyzed Synthesis of Pyrroles by [4+1] Cycloaddition
Qiu, J.-W.; Zhang, X.-G.; Tang, R.-Y.; Zhong, P.; Li, J.-H.: Iron-Catalyzed Synthesis of 2-Aminobenzo-thiazoles
Yadav, J. S.; Reddy, B. V. S.; Narasimhulu, G.; Chandrakanth, D.; Satheesh, G.: Cerium(III)-Catalyzed Synthesis of N-Arylpyrrolidines
Phan, D. H. T.; Kim, B.; Dong, V. M.: Rhodium-Catalyzed Enantioselective Synthesis of Phthalides
Rizk, T.; Bilodeau, E. J.-F.; Beauchemin, A.: Hydroamination Route to Pyridines and Pyrazines
Praveen, C.; Jegatheesan, S.; Perumal, P. T.: Gold-Catalyzed Synthesis of Quinolines
Pi, S.-S.; Zhang, X.-G.; Tang, R.-Y.; Li, J.-H.: CuBr-Catalyzed Synthesis of 2-Aminobenzo-thiazoles
Contiero, F.; Jones, K. M.; Matts, E. A.; Porzelle, A.; Tomkinson, N. C. O.: Acid-Mediated Synthesis of Benzofurans from Arylhydroxylamines
Ahmad, O. K.; Hill, M. D.; Movassaghi, M.: One-Step Synthesis of Polysubstituted Pyrimidines
Parvatkar, P. T.; Parameswaran, P. S.; Tilve, S. G.: Iodine-Catalyzed One-Pot Synthesis of 6H-Indoloquinoline Derivatives
Egi, M.; Azechi, K.: Gold-Catalyzed Synthesis of Pyrroles and Furans
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Issue 12/2009

González-Gómez, Á.; Domínguez, G.; Pérez-Castells, J.: Gold-Catalyzed Synthesis of Benzazepines
Gruit, M.; Michalik, D.; Tillack, A.; Beller, M.: Platinum-Catalyzed Synthesis of Pyrrolo[3,2-c]azepin-4-ones
Gao, L.; Hwang, G.-S.; Lee, M. Y.; Ryu, D. H.: Catalytic Enantioselective Synthesis of 2-Pyrazolines
Li, H.; Hsung, R. P.: Rh-Catalyzed Synthesis of 2-Amido-furans via Cyclopropenation of Ynamides
Wang, J.-Y.; Wang, X.-P.; Yu, Z.-S.; Yu, W.: Lewis Acid Catalyzed Synthesis of Multisubstituted Pyrroles
Ueno, S.; Ohtsubo, M.; Kuwano, R.: Palladium-Catalyzed Synthesis of Tetrahydroisoquinolines
Cantagrel, G.; de Carné-Carnavalet, B.; Meyer, C.; Cossy, J.: FeCl3-Promoted Cyclization of o-Alkylaryl Isocyanates to Oxindoles
Mosslemin, M. H.; Anary-Abbasinejad, M.; Anaraki-Ardakani, H.: Multicomponent Synthesis of 2-Aminofurans
Hodgkinson, R. C.; Schulz, J.; Willis, M. C.: Cascade N-Annulation Route to 7-Azaindoles
Bernini, R.; Fabrizi, G.; Sferrazza, A.; Cacchi, S.: Copper-Catalyzed C-H Activation to Polysubstituted Indoles
Pati, K.; Liu, R.-S.: Ruthenium-Catalyzed Synthesis of Pyridones and Isoquinolones
Yamashita, M.; Horiguchi, H.; Hirano, K.; Satoh, T.; Miura, M.: Construction of Carbazoles via Pd-Catalyzed Oxidative Coupling of Alkynes
Kazmaier, U.; Schmidt, C.: One-Pot Stereoselective Synthesis of Furanoid Amino Acids
Chen, D.; Shen, G.; Bao, W.: Copper-Catalyzed Synthesis of 2H-1,4-Benzoxazin-3-(4H)-ones
Murru, S.; Ghosh, H.; Sahoo, S. K.; Patel, B. K.: Synthesis of Arylthiobenzothiazoles via a Copper(I)-Catalyzed S-Arylation
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Issue 11/2009

Wang, Y.-F.; Chiba, S.: Mn(III)-Mediated Synthesis of Pyridines
Facoetti, D.; Abbiati, G.; d’Avolio, L.; Ackermann, L.; Rossi, E.: TiCl4-Catalyzed Synthesis of Pyrimido[1,6-a]indol-1-ones
Donets, P. A.; van Hecke, K.; van Meervelt, L.; van der Eycken, E. V.: Synthesis of Indoloazocine by Hg(OTf)2-Catalyzed Intramolecular Carbocyclization
Bryan, C. S.; Braunger, J. A.; Lautens, M.: Pd-Catalyzed Synthesis of Benzothiophenes from gem-Dihalovinyl Thiophenols
Duguet, N.; Salwin, A. M. Z.; Smith, A. D.: Asymmetric Synthesis of 3-Alkyl-3-aryl-oxindoles
Savitha, G.; Felix, K.; Perumal, P. T.: Pd-Catalyzed Synthesis of 3-Bromo-2H-Chromenes
Azizi, N.; Khajeh-Amiri, A.; Ghafuri, H.; Bolourtchian, M.; Saidi, M. Reza: FeCl3-Catalyzed Synthesis of N-Substituted Pyrroles in Water
Friedman, R. Keller; Rovis, T.: Rh-Catalyzed Cycloadditions of Unsymmetrical Alkynes with Isocyanates
Allen, C. P.; Benkovics, T.; Turek, A. K.; Yoon, T. P.: Synthesis of Tetrahydroisoquinolines and Tetrahydropyridines from Oxaziridines
Lu, W.; Song, W.; Hong, D.; Lu, P.; Wang, Y.: Cu-Catalyzed Multicomponent Synthesis of 1,2,3,4-Tetrahydropyrimidines
Tang, S.; He, J.; Sun, Y.; He, L.; She, X.: Regioselective One-Pot Straightforward Synthesis of Isoxazoles
Chandra, A.; Singh, B.; Khanna, R. S.; Singh, R. M.: Pd-Catalyzed One-Pot Coupling-Annulation Synthesis of Pyrano[4,3-b]quinolines
Zhao, X.; Zhang, E.; Tu, Y.-Q.; Zhang, Y.-Q.; Yuan, D.-Y.; Cao, K.; Fan, C.-A.; Zhang, F.-M.: Au(I)-Catalyzed Synthesis of Cycloalkene-Fused Pyrroles
Burton, D. J.; Hansen, S. W.: Synthesis of Fluorinated α-Pyrans
Yang, D.; Liu, H.; Yang, H.; Fu, H.; Hu, L.; Jiang, Y.; Zhao, Y.: Efficient Cu-Catalyzed Synthesis of 1,2,4-Benzothiadiazine-1,1-dioxides
All PDFs of this category

Issue 10/2009

Roveda, J.-G.; Clavette, C.; Hunt, A. D.; Gorelsky, S. I.; Whipp, C. J.; Beauchemin, A. M.: Synthesis of Azacarbocycles via Hydroamination and Aminocarbonylation
Mei, T.-S.; Wang, X.; Yu, J.-Q.: Synthesis of Indolines by Pd(II)-Catalyzed Amination of C-H Bond
Henssler, J. T.; Matzger, A. J.: Synthesis of theThieno[3,2-b]thiophene and Thieno[3,2-b]furan Bare Ring Systems
Zhu, W.; Mena, M.; Jnoff, E.; Sun, N.; Pasau, P.; Ghosez, L.: Synthesis of Piperidones by MCR
Shintani, R.; Hayashi, S.-y.; Murakami, M.; Takeda, M.; Hayashi, T.: Stereoselective Synthesis of Spirooxindoles
Yavari, I.; Souri, S.; Sirouspour, M.; Bayat, M. J.: Synthesis of Fused Quinoxalines and Benzoxazines
Anary-Abbasinejad, M.; Poorhassan, E.; Hassanabadi, A.: Synthesis of 2,5-Dihydropyrroles from Acetylene Esters and α-Arylamino Ketones
Reddy, G.; Kumar, P. A.; Anand, R. V.; Mukkanti, K.; Reddy, P. P.: Synthesis of Indolo [1,2,5]-Triazepines and [1,2,5]-Oxadiazines
Chen, Z.; Ding, Q.; Yu, X.; Wu, J.: Cyclization/[3+2]-Cycloaddition Reaction of N′-(2-Alkynylbenzylidene) Hydrazides
Watanabe, T.; Oishi, S.; Fujii, N.; Ohno, H.: Palladium-Catalyzed Direct One-Pot Synthesis of Carbazoles
McQuaid, K. M.; Long, J. Z.; Sames, D.: Synthesis of Dihydrobenzopyrans via Hydride Transfer Cyclization
Khlebnikov, V.; Patel, K.; Zhou, X.; Reddy, M. M.; Su, Z.; Chiacchia, F. S.; Hansen, H. C.: Efficient Synthesis of 2-Aryl-4H-pyrano[2,3-b]pyridine-4-ones
Han, Z.-Y.; Xiao, H.; Chen, X.-H.; Gong, L.-Z.: Synthesis of Chiral Tetrahydroquinolines by Relay Catalysis
Zhong, W.; Guo, B.; Lin, F.; Liu, Y.; Su, W.: Synthesis of Thiazolopyrimidinones under Solvent-Free Conditions
Li, J.; Wang, D.; Zhang, Y.; Chen, B.: Synthesis of N-Unsubstituted 1,2,3-Triazoles by a One-Pot Reaction
All PDFs of this category

Issue 09/2009

Liang, J.; Chen, J.; Du, F.; Zeng, X.; Li, L.; Zhang, H.: Synthesis of Spiro β-Lactams and Oxoindoles by Oxidative Dearomatization
Ñunez, A.; Abarca, B.; Cuadro, A. M.; Alvarez-Builla, J.; Vaquero, J. J.: Ring-Closing Metathesis Approach to Quinolizinium Salts
Han, Z.-G.; Tu, S.-J.; Jiang, B.; Yan, S.; Zhang, X.-H.; Wu, S.-S.; Hao, W.-J.; Cao, X.-D.; Shi, F.; Zhang, G.; Ma, N.: Chemoselective Synthesis of Naphthyridines and Pyrano[3,2-c]pyridines
Budén, M. E.; Vaillard, V. A.; Martin, S. E.; Rossi, R. A.: Photostimulated Intramolecular SRN1 Reaction of Diarylamines to Carbazoles
Ueda, S.; Nagasawa, H.: Copper-Catalyzed C-H Activation for the Synthesis of Benzoxazoles
Suzuki, Y.; Ohta, Y.; Oishi, S.; Fujii, N.; Ohno, H.: Synthesis of Pyrroloindoles and Dipyrrolo-pyridines by a Hydroamination Route
Heydari, A.; Khaksar, S.; Tajbakhsh, M.; Bijanzadeh, H. R.: General Synthesis of Hantzsch Esters in 2,2,2-Trifluoroethanol
Spitz, C.; Lohier, J.-F.; Reboul, V.; Metzner, P.: Synthesis of 1,3-Benzothiazines by Catalytic Generation of Cesium Acetylide
Joyce, L. L.; Batey, R. A.: Synthesis of 2-Aminobenzothiazoles via Oxidative C-H Functionalization
Schuler, M.; Monney, A.; Gouverneur, V.: Synthesis of 4,4-Difluorodihydrofuran-3(2H)-ones
Li, L.; Li, Z.; Wang, Q.: Organocatalytic Synthesis of Benzo[b]thiepines
Gising, J.; Örtqvist, P.; Sandström, A.; Larhed, M.: An Improved Synthesis of Dichloro-pyrazinones
Wender, P. A.; Strand, D.: Silver-Catalyzed Synthesis of 2,3-Dihydro-pyrroles
Han, B.; He, Z.-Q.; Li, J.-L.; Li, R.; Jiang, K.; Liu, T.-Y.; Chen, Y.-C.: Piperidines from Organocatalytic Inverse-Demand Aza-Diels-Alder Reaction
Fukamachi, S.; Konishi, H.; Kobayashi, K.: One-Pot Synthesis of 2-Sulfanylindoles
All PDFs of this category

Issue 08/2009

Yoshino, Y.; Kurahashi, T.; Matsubara, S.: Ni-Catalyzed Synthesis of 4-Quinolones from Alkynes and Isatoic Anhydrides
Heravi, M. M.; Baghernejad, B.; Oskooie, H. A.: Three-Component Synthesis of Benzothiazines
Lechel, T.; Möhl, S.; Reissig, H.-U.: Synthesis of 5-Alkoxy Pyrimidines via Enamides
Ackermann, L.; Barfüßer, S.; Potukuchi, H. K.: Copper-Catalyzed Domino Synthesis of Indoles
Komine, Y.; Kamisawa, A.; Tanaka, K.: Synthesis of Dibenzofurans by Rhodium-Catalyzed [2+2+2] Cycloaddition
Heim-Riether, A.; Gipson, K. R.: One-Pot Synthesis of Imidazo[2,1-a]phthal-azines
Coulter, M. M.; Dornan, P. K.; Dong, V. M.: Rh-Catalyzed Synthesis of Benzoxapinones and Benzothiapinones
Rahanyan, N.; Linden, A.; Baldridge, K. K.; Siegel, J. S.: Diazafluoranthene Derivatives via Diels-Alder Reaction
Rao, R. K.; Naidu, A. B.; Sekar, G.: Synthesis of 1,4-Benzoxazines by Domino SN2 and Goldberg Coupling
Zhang, J.; Zhang, M.; Cao, W.; Song, L.; Qian, Q.; Tan, J.; Shao, M.: Synthesis of Trifluoromethyl-Substituted Tetrahydropyrans
Spitz, C.; Lohier, J.-F.; Santos, J. Sopkova-de Oliveira; Reboul, V.; Metzner, P.: 1,4-Benzothiazepines via Nucleophilic Catalysis
Engstrom, K. M.; Baize, A. L.; Franczyk, T. S.; Kallemeyn, J. M.; Mulhern, M. M.; Rickert, R. C.; Wagaw, S.: Friedel-Crafts, Thermal or Reductive Cyclization Route to Thienopyridines
Merkul, E.; Boersch, C.; Frank, W.; Müller, T. J. J.: Three-Component Synthesis of Substituted N-Boc-4-iodopyrroles
Shi, Z.; Zhang, C.; Li, S.; Pan, D.; Ding, S.; Cui, Y.; Jiao, N.: Dioxygen as Oxidant for the Synthesis of Indoles by Pd-Catalyzed C-H Activation
Greszler, S. N.; Johnson, J. S.: Diastereoselective Synthesis of γ-Butyro-lactones
All PDFs of this category

Issue 07/2009

Yadav, L. D. S.; Kapoor, R.; Garima: One-Pot Synthesis of Thietanes
Muravyova, E. A.; Shishkina, S. V.; Musatov, V. I.; Knyazeva, I. V.; Shishkin, O. V.; Desenko, S. M.; Chebanov, V. A.: Multi-Component Synthesis of Pyrazolopyridopyrimidines
Bernini, R.; Cacchi, S.; Fabrizi, G.; Filisti, E.; Sferrazza, A.: Synthesis of Substituted Quinolines via a Heteroannulation Process
Ackermann, L.; Sandmann, R.; Kaspar, L. T.: Titanium-Catalyzed Intermolecular Hydroamination Route to Pyrroles
Andersson, H.; Gustafsson, M.; Boström, D.; Olsson, R.; Almqvist, F.: Synthesis of trans-2,3-Dihydropyridine
N-Oxides and Piperidines
Khoshkholgh, M. J.; Lotfi, M.; Balalaie, S.; Rominger, F.: Synthesis of Pyrano[2,3-c]coumarins via Intramolecular Domino Reactions
Cao, H.; Jiang, H.; Yao, W.; Liu, X.: Synthesis of Substituted Furans via Copper-Catalyzed Domino Reactions
Xu, D.; Xu, X.; Liu, Z.; Sun, L.-P.; You, Q.: Copper-Catalyzed Synthesis of 2-Substituted Oxazolopyridines
Pokhodylo, N. T.; Matiychuk, V. S.; Obushak, M. D.: Regioselective Cycloaddition Route to 5-Aminotriazoles
Pan, Y.-m.; Zheng, F.-j.; Ling, H.-x.; Zhan, Z.-p.: One-Pot Synthesis of Substituted Oxazoles
Giles, R. L.; Sullivan, J. D.; Steiner, A. M.; Looper, R. E.: Synthesis of Substituted 2-Aminoimidazoles
Ohta, Y.; Oishi, S.; Fujii, N.; Ohno, H.: Copper-Catalyzed Synthesis of Tetrahydro-β-carbolines
Tan, J.; Xu, X.; Zhang, L.; Li, Y.; Liu, Q.: Stereoselective Synthesis of Pyrrolizidines
Loos, P.; Riedrich, M.; Arndt, H.-D.: An Aza-Wittig Route to Imidazolines and Imidazoles
Shimizu, M.; Hirano, K.; Satoh, T.; Miura, M.: Waste-Free Synthesis of Condensed Heterocycles
All PDFs of this category

Issue 06/2009

Sañudo, M.; García-Valverde, M.; Marcaccini, S.; Delgado, J. J.; Rojo, J.; Torroba, T.: Four-Component Ugi Approach to Benzodiazepines
Manarin, F.; Roehrs, J. A.; Gay, R. Mozzaquatro; Brandão, R.; Menezes, P. H.; Nogueira, C. W.; Zeni, G.: Electrophilic Heteroannulation Strategy for the Synthesis of 2-Chalcogenbenzofurans
Fontaine, P.; Masson, G.; Zhu, J.: Synthesis of 2-Aminopyrroles by Sequential MCR/[4+1] Cycloaddition
Liu, X.-Y.; Che, C.-M.: Pt(II)-Catalyzed Synthesis of Indolines and Tetrahydroquinolines
Aureggi, V.; Davoust, M.; Gericke, K. M.; Lautens, M.: Palladium-Catalyzed Cascade Synthesis of Pyrrolobenzazepines
Takenaka, K.; Itoh, N.; Sasai, H.: Enantioselective Synthesis of Spirobilactams by Pd-Catalyzed N-Arylation
Nakamura, I.; Sato, Y.; Terada, M.: Platinum-Catalyzed Cascade Synthesis of Indoloquinazolinones
Zhang, W.; Xu, H.; Tang, W.: Stereoselective Synthesis of Lactones From Conjugated Enynes
Li, L.; Wang, M.; Zhang, X.; Jiang, Y.; Ma, D.: Synthesis of Isoindolin-1-ones via Copper-Catalyzed Intramolecular Cyclization
Shaabani, A.; Sarvary, A.; Rezayan, A. H.; Keshipour, S.: Three-Component Synthesis of Pyrano[2,3-c]pyrazoles
Reyes-Gutiérrez, P. E.; Torres-Ochoa, R. O.; Martínez, R.; Miranda, L. D.: Synthesis of Azepino[4,5-b]indolones via Radical-Mediated Tryptamine Substitution
Cui, L.; Zhang, G.; Peng, Y.; Zhang, L.: Gold-Catalyzed Synthesis of Tetrahydrobenz[b]azepin-4-ones
Schneekloth, J. S.; Kim, J.; Sorensen, E. J.: Preparation of Substituted Indoxyls and Aminoindoles
Xiao, Y.; Zhang, J.: Pd-Catalyzed Domino Reaction of Tetrasubstituted Furans
Barluenga, J.; Jiménez-Aquino, A.; Aznar, F.; Valdés, C.: A Pd-Catalyzed Combined α-Arylation/C-N Coupling Synthesis of Indoles
All PDFs of this category

Issue 05/2009

Hui, B. W.-Q.; Chiba, S.: Synthesis of Isoindoles and Isoquinolines via 1,3-Dipolar Cycloaddition and Electrocyclization
Wen, L.-R.; Ji, C.; Li, M.; Xie, H.-Y.: 2-Chloroaroylthioamides in the Synthesis of Thiochromeno[2,3-b]pyridines
Lu, L.; Cao, W.; Chen, J.; Zhang, H.; Zhang, J.; Chen, H.; Wei, J.; Deng, H.; Shao, M.: Synthesis of 3a,4,5,6-Tetrahydroimidazo-[1,5-b]isoxazoles
Tadd, A. C.; Matsuno, A.; Fielding, M. R.; Willis, M. C.: Palladium-Catalyzed Carbonylative Synthesis of 2-Quinolones
Abbiati, G.; Arcadi, A.; Marinelli, F.; Rossi, E.; Verdecchia, M.: Concise Synthesis of Isoxazolino[4,5-c]-quinolines
Jia, Y.-X.; Kündig, E. P.: Synthesis of Oxindoles by Direct Intramolecular Oxidative Coupling
DeAngelis, A.; Taylor, M. T.; Fox, J. M.: Three-Component Synthesis of Di- and Tetrahydrofurans under Rhodium Catalysis
Beutner, G. L.; Kuethe, J. T.; Kim, M. M.; Yasuda, N.: Synthesis of Pyrazolopyridines
Surmont, R.; Verniest, G.; Colpaert, F.; Macdonald, G.; Thuring, J. W.; Deroose, F.; De Kimpe, N.: Synthesis of 3-Fluoropyrroles
Han, F.-b.; Ge, Z.-m.; Cheng, T.-m.; Li, R.-t.: Four-Component Synthesis of Dithiocarbonyloxazolidines
Parsons, A. T.; Johnson, J. S.: Asymmetric [3+2] Cycloaddition Route to Tetrahydrofurans
Tsuritani, T.; Yamamoto, Y.; Kawasaki, M.; Mase, T.: Synthesis of 3,4-Dihydro-2(¹H)-quinolinone via Ring Expansion
Cernak, T. A.; Lambert, T. H.: Multicatalytic Synthesis of α-Pyrrolidinyl Ketones Under Pd(II)/In(III) Catalysis
Huang, X.-C.; Wang, F.; Liang, Y.; Li, J.-H.: Synthesis of Substituted Benzo-[b]naphtho-[2,1-d]furans via a Domino Process
Wang, L.; Liu, Q.-B.; Wang, D.-S.; Li, X.; Han, X.-W.; Xiao, W.-J.; Zhou, Y.-G.: Synthesis of Dihydroxazines via Opening of Aziridines
All PDFs of this category

Issue 04/2009

Murarka, S.; Zhang, C.; Konieczynska, M. D.; Seidel, D.: Lanthanide Triflate Catalyzed Hetero-annulation Route to Tetrahydroquinolines
Sakakibara, K.; Nozaki, K.: Lithiated Dithiane Ring Opening of N-Protected Aziridines
Petronijevic, F.; Timmons, C.; Cuzzupe, A.; Wipf, P.: Microwave-Assisted Diels-Alder Approach to 4-Substituted Indoles
Lu, Y.; Fu, X.; Chen, H.; Du, X.; Jia, X.; Liu, Y.: Polysubstituted Pyrroles from (Z)-Enynols
Shestopalov, A. M.; Rodinovskaya, L. A.; Fedorov, A. E.; Kalugin, V. E.; Nikishin, K. G.; Gakh, A. A.: Nucleophilic Fluorination of 3-Cyanopyridines
Attanasi, O. A.; Favi, G.; Filippone, P.; Perrulli, F. R.; Santeusanio, S.: Synthesis of Functionalized Pyridazines from 1,2-Diaza-1,3-butadienes
Tan, B.; Shi, Z.; Chua, P. J.; Li, Y.; Zhong, G.: Synthesis of N-Hydroxypyrroles Using N-Selective Nucleophilicity of Oximes
Bellur, E.; Yawer, M. A.; Hussain, I.; Riahi, A.; Fatunsin, O.; Fischer, C.; Langer, P.: Synthesis of Disubstituted Pyrroles from
1,3-Dicarbonyls and Azides
Tejedor, D.; López-Tosco, S.; González-Platas, J.; García-Tellado, F.: Synthesis of Substituted Pyrroles from Skipped Diynes
Tu, S.-J.; Cao, X.-D.; Hao, W.-J.; Zhang, X.-H.; Yan, S.; Wu, S.-S.; Han, Z.-G.; Shi, F.: Multicomponent Synthesis of Benzothiazepinones
Kison, C.; Opatz, T.: Synthesis of Imidazoles and Oxazoles by Aldimine Cross-Coupling
Gimbert, C.; Vallribera, A.: Synthesis of Benzothiazines via an Intramolecular Thioamide S-Michael Addition
Chen, Z.-B.; Hong, D.; Wang, Y.-G.: Synthesis of Multisubstituted Pyridines from α-Diazocarbonyl Derivatives
Agarwal, P. K.; Sharma, S. K.; Sawant, D.; Kundu, B.: Synthesis of Pyrimidoquinolines via the Pictet-Spengler Reaction
All PDFs of this category

Issue 03/2009

Liu, X.-t; Huang, L.; Zheng, F.-j; Zhan, Z.-p: Synthesis of Pyrroles Using InCl3 as a Multifunctional Catalyst
Esquivias, J.; Alonso, I.; Arrayás, R. Gómez; Carretero, J. C.: Asymmetric Synthesis of Tetrahydropyridines via Diels-Alder Reaction
Pfrengle, F.; Dekaris, V.; Schefzig, L.; Zimmer, R.; Reissig, H.-U.: InCl3-Mediated Cleavage of Acetonides on Acid-Sensitive Heterocycles
Teague, S. J.: De Novo Pyridine Ring Synthesis and Methylsulfinyl Displacement by Amines
Kozio, A.; Frelek, J.; Wonica, M.; Furman, B.; Chmielewski, M.: Lewis Acid Mediated Enantioselective Synthesis of Oxacephams
Stuart, D. R.; Bertrand-Laperle, M.; Burgess, K. M. N.; Fagnou, K.: Synthesis of Indoles via Oxidative Coupling of Acetanilides with Acetylenes
Kim, J.; Lee, S. Y.; Lee, J.; Do, Y.; Chang, S.: Utility of Ammonium Salts for the Synthesis of Amidines
Jacq, J.; Einhorn, C.; Einhorn, J.: Regiospecific Synthesis of 1,3-Diaryliso-benzofurans
Yamamoto, Y.; Kirai, N.: Copper-Catalyzed Hydroarylation: Synthesis of 4-Arylcoumarins
Xu, Z.; Hu, W.; Zhang, F.; Li, Q.; Lü, Z.; Zhang, L.; Jia, Y.: Pd-Catalyzed Synthesis of (Aza)Indoles from o-Haloanilines and Aldehydes
Sukach, V. A.; Golovach, N. M.; Melnichenko, N. V.; Tsymbal, I. F.; Vovk, M. V.: Synthesis of Chiral 4-Trifluoromethyl-3,4-dihydroazin-2-ones
Ackermann, L.; Althammer, A.; Fenner, S.: Pd-Catalyzed Direct Arylations of Heteroaromatics using Aryl Sulfonates
Zheng, Z.; Alper, H.: Synthesis of Isoquinolin-1-ones via Pd-Catalyzed Carbonylation-Heteroannulation
Peng, Y.; Yu, M.; Zhang, L.: Gold-Catalyzed Synthesis of Indolizin-7-ones from Enynyl β-Lactams
Xie, C.; Zhang, Y.; Xu, P.: Three-Component Synthesis of Pyrido[2,1-a]isoindoles

Issue 02/2009

Shaabani, A.; Maleki, A.; Mofakham, H.: One-Pot Three-Component Synthesis of Tetrahydro-1H-1,5-benzodiazepines
Shaaban, M. R.: Microwave-Assisted Synthesis of Trifluoromethyl-Containing Heterocycles
Lv, X.; Liu, Y.; Qian, W.; Bao, W.: Cu-Catalyzed Heteroannulation Route to 2-Iminobenzo-1,3-oxathioles
Samanta, S.; Mohapatra, H.; Jana, R.; Ray, J. K.: Intramolecular Heck Route to 5-, 6-, and 7-Membered O-Containing Heterocycles
Fischer, D.; Tomeba, H.; Pahadi, N. K.; Patil, N. T.; Huo, Z.; Yamamoto, Y.: Synthesis of Isoquinolines by I2-Mediated Electrophilic Heteroannulation
Feroci, M.; Chiarotto, I.; Rossi, L.; Inesi, A.: The Gewald Synthesis of 2-Aminothiophenes using Activated Sulfur
Grigg, R.; Sridharan, V.; Shah, M.; Mutton, S.; Kilner, C.; MacPherson, D.; Milner, P.: Pd-Catalyzed Three-Component Synthesis of Isoindolones and Phthalazones
Melkonyan, F.; Topolyan, A.; Yurovskaya, M.; Karchava, A.: Concise Cu-Catalyzed Synthesis of 3-Carboxyl-N-Aminoindoles
Jordan-Hore, J. A.; Johansson, C. C. C.; Gulias, M.; Beck, E. M.; Gaunt, M. J.: Oxidative Pd(II)-Catalyzed C-H Bond Activation Route to Carbazoles
Teimouri, M. B.; Mansouri, F.: One-Pot Three-Component Synthesis of 7H-Phenaleno[1,2-b]furan-7-ones
Wang, Y.-F.; Toh, K. K.; Chiba, S.; Narasaka, K.: Mn(III)-Catalyzed Synthesis of Pyrroles from 1,3-Dicarbonyls and Vinyl Azides
Khankischpur, M.; Kurz, T.: Microwave-Assisted Synthesis of 1,2,4-Triazolium Ylides
Han, B.; Li, J.-L.; Ma, C.; Zhang, S.-J.; Chen, Y.-C.: Organocatalytic Asymmetric Inverse-Electron-Demand Aza-Diels-Alder Reaction
Ghosh, D.; Thander, L.; Ghosh, S. K.; Chattopadhyay, S. K.: Aza-Claisen-RCM Route to 1-Benzazepine Derivatives
Cheng, X.; Vellalath, S.; Goddard, R.; List, B.: Direct Catalytic Asymmetric Synthesis of Cyclic Aminals from Aldehydes

Issue 01/2009

Wipf, P.; Maciejewski, J. P.: Ti-Catalyzed Synthesis of Indolines
Cikotiene, I.; Morkunas, M.; Rudys, S.; Buksnaitiene, R.; Brukstus, A.: Thermal Heteroannulation Route to Pyrido[4,3-d]pyrimidines
Fu, Z.; Wang, M.; Ma, Y.; Liu, Q.; Liu, J.: Ketene Thioacetals in Furan Ring Construction
Hashimoto, T.; Uchiyama, N.; Maruoka, K.: Asymmetric Synthesis of Aziridines from Diazoacetamides and N-Boc Imines
Chan, Y.; Guthmann, H.; Brimble, M. A.; Barker, D.: Diastereoselective Mannich-Based Synthesis of Piperidones
Arnott, G.; Brice, H.; Clayden, J.; Blaney, E.: Synthesis of Spirocyclic Piperidines from
N-Arylisonicotinamides
Kaim, L. El; Gizzi, M.; Grimaud, L.: Synthesis of Highly Substituted Indoles via an Intramolecular Heck Cyclization
Chang, J. H.; Shin, H.: Large Scale One-Pot Synthesis of 4-Substituted-1H-Pyrrole-3-Carboxylates
Wasa, M.; Yu, J.-Q.: Synthesis of β-, γ-, and δ-Lactams via Pd(II)-Catalyzed C-H Activation
Shanthi, G.; Perumal, P. T.: Three-Component Synthesis of Substituted Chromenes
Andersson, H.; Gustafsson, M.; Olsson, R.; Almqvist, F.: Synthesis of 2-Substituted Pyridine N-Oxides via Directed ortho-Metalation
Imase, H.; Noguchi, K.; Hirano, M.; Tanaka, K.: Au-Catalyzed Cycloisomerization of
N-Alkenyl Alkynylamides to 2-Pyridones
Horneff, T.; Chuprakov, S.; Chernyak, N.; Gevorgyan, V.; Fokin, V. V.: Rh(II)-Catalyzed Transannulation of
1,2,3-Triazoles with Nitriles
Yang, D.; Fu, H.; Hu, L.; Jiang, Y.; Zhao, Y.: Cu-Catalyzed Heterannulation Route to Benzimidazoles from ortho-Haloacetanilides
Veitch, G. E.; Bridgwood, K. L.; Rands-Trevor, K.; Ley, S. V.: Magnesium Nitride as a Source of Ammonia for the Paal-Knorr Synthesis of Pyrroles

Issue 12/2008

Grant, D.; Dahl, R.; Cosford, N. D. P.: Microreactor Synthesis of 1,2,4-Oxadiazoles
Paone, D. V.; Shaw, A. W.: Synthesis of Highly Substituted Imidazoles from 1,2-Amino Alcohols and Thioamides
Bray, C. D.: A Diels-Alder Approach to Benzannulated [5,6]-Spiroketals
Willy, B.; Dallos, T.; Rominger, F.; Schönhaber, J.; Müller, T. J. J.: Three-Component Synthesis of 1,5-Benzo-
diazepines
Mamedov, V. A.; Saifina, D. F.; Gubaidullin, A. T.; Saifina, A. F.; Rizvanov, I. K.: One-Pot Synthesis of 2-(Indolizin-2-yl)benz-imidazoles from Quinoxalinones
Barluenga, J.; Riesgo, L.; Vicente, R.; López, L. A.; Tomás, M.: Cu(I)-Catalyzed Synthesis of Polysubstituted Furans
Batchelor, D. V.; Beal, D. M.; Brown, T. B.; Ellis, D.; Gordon, D. W.; Johnson, P. S.; Mason, H. J.; Ralph, M. J.; Underwood, T. J.; Wheeler, S.: Acid-Mediated Synthesis of 3-N,N-Dialkyl-amino-1,2,4-Triazoles
Rudkin, M. E.; Joensuu, P. M.; MacLachlan, W. S.; Lam, H. W.: Synthesis of β-Hydroxylactams via Co-Catalyzed Alkylative Aldol Cyclization
Gasiecki, A. F.; Cross, J. L.; Henry, R. F.; Gracias, V.; Djuric, S. W.: Synthesis of Spiro Pyrrolidines from Tetrahydropyridinium Salts
Gabriele, B.; Mancuso, R.; Salerno, G.: Synthesis of Functionalized Benzofurans via Pd-Catalyzed Cycloisomerization
Sasada, T.; Sakai, N.; Konakahara, T.: Three-Component Synthesis of Tetra-substituted Pyridines
Eidamshaus, C.; Burch, J. D.: Pd-Catalyzed Enolate α-Arylation. Synthesis of Benzofurans
Cui, S.-L.; Wang, J.; Wang, Y.-G.: Synthesis of Indoles from N-Aryl Amides and Ethyl Diazoacetate
Horn, J.; Marsden, S. P.; Nelson, A.; House, D.; Weingarten, G. G.: Rh-Catalyzed Conjugate Addition of o-Amino-arylboronates. Synthesis of Quinolines
Alizadeh, A.; Hosseinpour, R.; Rostamnia, S.: Synthesis of 4-Hydroxy-1H-pyrrole-2,3-dicarboxylic Acids

Issue 11/2008

Iaroshenko, V. O.; Volochnyuk, D. M.; Kryvokhyzha, N. V.; Martyloga, A.; Sevenard, D. V.; Groth, U.; Brand, J.; Chernega, A. N.; Shivanyuk, A. N.; Tolmachev, A. A.: An Undemanding Synthesis of Thiazolo[4,5-d]pyridines
Kokotos, C. G.; McGarrigle, E. M.; Aggarwal, V. K.: Three-Component Synthesis of Epoxides and Aziridines via Sulfur Ylides
Ding, Q.; Wu, J.: Halogen Electrophile Induced Cyclization Route to Isoquinoline N-Oxides
Plaskon, A. S.; Ryabukhin, S. V.; Volochnyuk, D. M.; Gavrilenko, K. S.; Shivanyuk, A. N.; Tolmachev, A. A.: 3-Formylchromone to Quinoline Interconversion
Sniady, A.; Morreale, M. S.; Wheeler, K. A.; Dembinski, R.: Synthesis of 3-Chlorofurans and 5-Chlorofuropyrimidine Nucleosides
Miura, T.; Yamauchi, M.; Murakami, M.: Ni-Catalyzed Conversion of 1,2,3-Benzo-triazin-4-ones into Isoquinolones
Yoshida, M.; Al-Amin, M.; Matsuda, K.; Shishido, K.: Pt-Catalyzed Cyclization of Propargylic Oxiranes to Substituted Furans
Kraus, G. A.; Guo, H.: Intramolecular Aza-Wittig Route to 2-Aryl Indoles
Li, X.; Deng, H.; Luo, S.; Cheng, J.-P.: Synthesis of 2,5-Dihydro-(1H)-pyrrol-2-ones from Pyruvate, Aldehydes and Anilines
Hayes, S. J.; Knight, D. W.; O’Halloran, M.; Pickering, S. R.: AgNO3-Catalyzed 5-endo-dig Cyclizations to Form Pyrazole N-Oxides and Pyrazoles
Wang, F.; Fu, H.; Jiang, Y.; Zhao, Y.: Cu-Catalyzed Huisgen Cycloaddition of Sulfonyl Azides ‘on Water∏
Yadav, J. S.; Reddy, B. V. S.; Maity, T.; Kumar, G. G. K. S. Narayana: Synthesis of 4-Azidotetrahydropyrans via Prins Cyclization
Kishi, Y.; Nagura, H.; Inagi, S.; Fuchigami, T.: Synthesis of Fluorinated Heterocycles via Prins Cyclization in Ionic Liquids
Yadav, L. D. S.; Kapoor, R.: 3-Amino-2(1H)-pyridinones from 1,3-Oxazolon-5-ones by a Multicomponent Reaction
Dehnhardt, C. M.; Espinal, Y.; Venkatesan, A. M.: One-Pot Synthesis of Tetrahydroquinolines by an Imino-Diels-Alder Reaction

Issue 10/2008

Adam, M. S. S.; Kühl, O.; Kindermann, M. K.; Heinicke, J. W.; Jones, P. G.: Synthesis of N-Substituted Pyrido[b]-Anellated Azaphospholes
Clarke, P. W.; Zaytsev, A. V.; Morgan, T. W.; Whitewood, A. C.; Wilson, C.: Synthesis of Piperidinones via a Multicomponent Condensation
Hill, M. D.; Movassaghi, M.: Synthesis of Azaheterocycles by Microwave-Assisted Activation of N-Acylarylamines
Downer-Riley, N. K.; Jackson, Y. A.: Radical-Mediated Cyclization of Thiobenzamides into Benzothiazoles
Crovetto, L.; Rios, R.: Synthesis of Pyrrolidines by a Three-Component Reaction
Shapiro, N. D.; Toste, F. D.: Synthesis of Azepines by a Gold-Catalyzed [4+3] Annulation
Cacchi, S.; Fabrizi, G.; Filisti, E.: Synthesis of Pyrroles and Pyridines by Cyclization of N-Propargylic β-Enaminones
Minatti, A.; Buchwald, S. L.: Cu-Catalyzed Domino Synthesis of Indolines
Ghavtadze, N.; Fröhlich, R.; Würthwein, E.-U.: Aza-Nazarov Synthesis of 2H-Pyrroles
Isobe, A.; Takagi, J.; Katagiri, T.; Uneyama, K.: Synthesis of Polyfluoroalkylquinolines by Pd-Catalyzed Heteroannulation
Marsden, S. P.; Watson, E. L.; Raw, S. A.: 3-Aminooxindoles via Microwave-Assisted Intramolecular Arylation
Fan, R.; Li, W.; Ye, Y.; Wang, L.: One-Pot Oxidative Heteroannulations to 5-Aminocoumaran Derivatives
Carson, M. W.; Giese, M. W.; Coghlan, M. J.: Synthesis of Benzopyridyloxepines Contain-
ing Stereodefined Exocyclic Double Bonds
Watzke, M.; Schulz, K.; Johannes, K.; Ullrich, P.; Martens, J.: Synthesis of Caprolactams from Cyclic Imines by Cross-Metathesis
Sarkar, N.; Banerjee, A.; Nelson, S. G.: Synthesis of Polysubstituted Piperidines by Diels-Alder Reaction of N-Alkenyl Iminiums

Issue 09/2008

Huang, J.; Chen, Y.; King, A. O.; Dilmeghani, M.; Larsen, R. D.; Faul, M. M.: Pd-Catalyzed Synthesis of 4-Quinolones
Karikomi, M.; D’hooghe, M.; Verniest, G.; De Kimpe, N.: Synthesis of 1,5-Benzothiazepines from Aziridines and 2-Aminothiophenol
Pohlhaus, P. D.; Sanders, S. D.; Parsons, A. T.; Li, W.; Johnson, J. S.: Synthesis of Tetrahydrofurans from Aldehydes and Cyclopropanes
Hernández, J. N.; Ramírez, M. A.; Rodríguez, M. L.; Martín, V. S.: Synthesis of 5-Alkynylproline Derivatives via Intramolecular Nicholas Reaction
Seregin, I. V.; Schammel, A. W.; Gevorgyan, V.: Mild Complementary Cycloisomerization Reactions to N-Fused Heterocycles
Manning, J. R.; Davies, H. M. L.: Synthesis of Pyridines via Rh-Catalyzed Ring Expansion of Isoxazoles
Beccalli, E. M.; Borsini, E.; Broggini, G.; Palmisano, G.; Sottocornola, S.: Pd-Catalyzed Cyclization of Propargylamides to Oxazoles
Nakamura, I.; Sato, T.; Terada, M.; Yamamoto, Y.: Gold-Catalyzed Synthesis of Benzothio-phenes with Chirality Transfer
Kobayashi, T.; Hatano, S.; Tsuchikawa, H.; Katsumura, S.: Synthesis of 2-Arylpyridines via Stille Coupling-Azaelectrocyclization
Noël, R.; Fargeau-Bellassoued, M.-C.; Vanucci-Bacqué, C.; Lhommet, G.: Synthesis of Chiral Tetrahydropyridines via a Three-Component Reaction
Shaabani, A.; Soleimani, E.; Rezayan, A. H.; Sarvary, A.; Khavasi, H. R.: Four-Component Synthesis of 3,4-Dihydro-coumarin Derivatives
Chang, W.-R.; Lo, Y.-H.; Lee, C.-Y.; Wu, M.-J.: Pd-Catalyzed Cyclization to Form Benzo-pyranones from Enediynes
Jiang, B.; Dong, J.-j; Jin, Y.; Du, X.-l; Xu, M.: Proline-Catalyzed Friedländer Synthesis of Quinolines
Lee, Y. T.; Chung, Y. K.: Ag-Catalyzed Synthesis of Pyrazoles from Propargyl N-Sulfonylhydrazones

Issue 08/2008

Zidar, N.; Kikelj, D.: Reductive Amination-Annulation Route to N-Substituted Dihydro-1,4-Benzoxazin-2-ones
Mo, W.; Liao, G.; Wang, T.; He, H.: Synthesis of Fluorine-Containing Pyrido[4,3-d]pyrimidines
Liu, H.-L.; Jiang, H.-F.; Zhang, M.; Yao, W.-J.; Zhu, Q.-H.; Tang, Z.: Synthesis of Pyrazoles by Three-Component One-Pot Process
Zuo, H.; Meng, L.; Ghate, M.; Hwang, K.-H.; Cho, Y. K.; Chandrasekhar, S.; Reddy, Ch. R.; Shin, D.-S.: One-Pot Synthesis of Benzoxazinones via Smiles Rearrangement
Attanasi, O. A.; Favi, G.; Filippone, P.; Giorgi, G.; Mantellini, F.; Moscatelli, G.; Spinelli, D.: Synthesis of Pyrroles and Pyrazoles by Mukai-yama-Michael Addition/Heterocyclization
Xia, M.; Xiang, G.-F.; Wu, B.; Han, Y.-F.: Regioselective Synthesis of Chrom-4-ones and Fused Flavones
Hopkin, M. D.; Baxendale, I. R.; Ley, S. V.: Synthesis of Pyrroloisoquinolines via Multicomponent Condensation
Xie, H.; Zu, L.; Oueis, H. R.; Li, H.; Wang, J.; Wang, W.: Inverse Diels-Alder Proline-Catalyzed Route to 1,2,4,5-Tetrazines
Lu, S.-M.; Alper, H.: Pd-Catalyzed Synthesis of Dibenzoxazo-cinones and Related Heterocycles
Samuel, R.; Chandran, P.; Retnamma, S.; Sasikala, K. A.; Sreedevi, N. K.; Anabha, E. R.; Asokan, C. V.: Synthesis of Thiophenes and Annulated Thio-phenes via Alkylation of 3-Oxo-Propanedithioates
Chen, J.; Wu, D.; He, F.; Liu, M.; Wu, H.; Ding, J.; Su, W.: Gallium(III) Triflate Catalyzed Synthesis of Quinazolinones from Isatoic Anhydrides
Zhang, C.-T.; Zhang, X.; Qing, F.-L.: Synthesis of Trifluoromethyltriazoles via 1,3-Dipolar Cycloaddition
Peters, J.-U.; Capuano, T.; Weber, S.; Kritter, S.; Sägesser, M.: Synthesis of 2-Quinolones via Intramolecular Olefination
Filák, L.; Rokob, T. A.; Vaskó, G. Á; Egyed, O.; Gömöry, A.; Riedl, Z.; Hajos, G.: A Tunable Heteroannulation Route to Fused Pyrazoles
Yang, Y.-Y.; Zhou, W.-G.; Chen, Z.-B.; Hong, D.; Wang, Y.-G.: An Aza-Wittig Route to Isoquinolines from Azidoarylacrylates

Issue 07/2008

Ramalingan, C.; Park, Y.-T.: Synthesis of Lactams and Diazepanones via Beckmann Rearrangement
Yadav, J. S.; Reddy, B. V. Subba; Chaya, D. N.; Kumar, G. G. K. S. Narayana; Aravind, S.; Kunwar, A. C.; Madavi, C.: Synthesis of 4-Iodopiperidines via Aza-Prins Cyclization
Garrido, N. M.; García, M.; Díez, D.; Sánchez, M. R.; Sanz, F.; Urones, J. G.: Ireland-Claisen Rearrangement - Michael Addition Sequence to δ-Amino Acids
Viirre, R. D.; Evindar, G.; Batey, R. A.: Copper-Catalyzed Domino Annulation Reaction to Benzoxazoles
Arimitsu, S.; Jacobsen, J. M.; Hammond, G. B.: Iodocyclization-Cross-Coupling Route to Trisubstituted 3-Fluorofurans
Watanabe, T.; Oishi, S.; Fujii, N.; Ohno, H.: Synthesis of Indolines via C-H Activation of N-tert-Butyl-2-bromoanilines
Sudhir, V. Sai; Baig, R. B. Nasir; Chandrasekaran, S.: Huisgen [2+3]-Cycloaddition Route to Triazolopyrazinones
Tang, Q.; Zhang, C.; Luo, M.: ortho Amination of Naphthols by N-N Bond Cleavage of Hydrazines
Huang, X.-C.; Liu, Y.-L.; Liang, Y.; Pi, S.-F.; Wang, F.; Li, J.-H.: Synthesis of Benzofurans via Aryne-Iodonium Ylide Cycloaddition
Butin, A. V.; Tsiunchik, F. A.; Abaev, V. T.; Zavodnik, V. E.: Synthesis of Thioindoles Using an Intramolecular Friedel-Crafts Reaction
Thornton, A. R.; Blakey, S. B.: Synthesis of Cyclic Sulfamates by a Cascade Process
Nandialath, V.; Abhilash, K. G.; Suresh, E.; Nair, V.: Synthesis of Indolo[3,2-a]carbazoles by Reaction of Indoles with 1,2-Diones
Sridharan, V.; Avendaño, C.; Menéndez, J. C.: Synthesis of Tetrahydroquinolines via CAN-Catalyzed Povarov Reaction
Wu, P.; Wan, Y.; Cai, J.: Organocatalytic Michael Addition of Indoles to Activated Alkenes in Water
Wang, K.; Xiang, D.; Liu, J.; Pan, W.; Dong, D.: Substituted 1H-Pyrazoles and Isoxazoles from Cyclopropyl Oximes

Issue 06/2008

Alegret, C.; Ginesta, X.; Riera, A.: Stereoselective Synthesis of Hydroxypipecolic Acids
Elinson, M. N.; Miloserdov, F. M.; Ilovaisky, A. I.; Feducovich, S. K.; Belyakov, P. A.; Nikishin, G. I.; Dorofeev, A. S.; Zelinsky, N. D.: Electrochemically Induced Three-Component Synthesis of Chromenes
Willy, B.; Rominger, F.; Müller, T. J. J.: Three-Component Synthesis of 3,4,5-Trisubstituted Isoxazoles
Murray, R. G.; Whitehead, D. M.; Strat, F. Le; Conway, S. J.: Gallium(III) Triflate Catalyzed Conversion of Aldehydes and Ketones to Hydantoins
Alex, K.; Tillack, A.; Schwarz, N.; Beller, M.: Intermolecular Zinc-Mediated Hydroamination of Alkynes to Indoles
Han, Y.; Xie, Y.-X.; Zhao, L.-B.; Fan, M.-J.; Liang, Y.-M.: Three-Component Synthesis of Highly Substituted 2-Imidazolines
Lee, E. E.; Rovis, T.: Rhodium-Catalyzed Enantioselective Cycloaddition Route to Indolizidines
Morgan, I. R.; Yazici, A.; Pyne, S. G.; Skelton, B. W.: Synthesis of Acylaminopyrrolidines and -piperidines via Diastereoselective Ritter Reaction
Deng, X.; Mani, N. S.: Regioselective Two-Component Synthesis of Polysubstituted Pyrazoles
Yeom, H.-S.; Kim, S.; Shin, S.: Gold(I)- and Silver(I)-Catalyzed Heteroannulation Route to Isoquinoline-N-Oxides
Pohjakallio, A.; Pihko, P. M.: Acid-Base Catalyzed Formation of 2-Isoxazolines
Yoo, E. J.; Chang, S.: Copper-Catalyzed Heteroannulation Route to Indolines
Zeghida, W.; Debray, J.; Chierici, S.; Dumy, P.; Demeunynck, M.: Synthesis of Quinazolinones by a Friedel-Crafts Heteroannulation Route
Counceller, C. M.; Eichman, C. C.; Wray, B. C.; Stambuli, J. P.: Metal-Free N-N Bond-Forming Route to Indazoles

Issue 05/2008

Chan, A.; Scheidt, K. A.: Pyrazolidinones via Amination of Homoenolates Catalyzed by N-Heterocyclic Carbenes
Arcadi, A.; Bianchi, G.; Inesi, A.; Marinelli, F.; Rossi, L.: Electrochemical Cyclization of 2-Alkynylanilines to Indole Derivatives
Zheng, Z.; Alper, H.: Palladium-Catalyzed Carbonylative 3-Component Synthesis of Quinazolinones
Rammah, M. M.; Othman, M.; Ciamala, K.; Strohmann, C.; Rammah, M. B.: Silver-Catalyzed Synthesis of Spiroisoindole-butyrolactones
Huang, W.; Shen, Q.; Wang, J.; Zhou, X.: Iron-Catalyzed Friedel-Crafts Synthesis of Dihydro- and Tetrahydroisoquinolines
Dahl, T.; Tornøe, C. W.; Bang-Andersen, B.; Nielsen, P.; Jørgensen, M.: Palladium-Catalyzed Three-Component Synthesis of Phenothiazines
Wang, J.-Y.; Guo, X.-F.; Wang, D.-X.; Huang, Z.-T.; Wang, M.-X.: Aziridines in Heteroannulation. Synthesis of 1,4-Benzodiazepines
Ruano, J. L. G.; de Haro, T.; Singh, R.; Cid, M. B.: Diastereoselective Synthesis of Nitropiperidones from N-p-Tolylsulfinyl β-Nitroamines
Loska, R.; MĄkosza, M.: Synthesis of Fluorinated Heteroaromatics by [3+2] Cycloaddition of N-Oxides with Hexafluoropropene
Hosokawa, T.; Matsumura, A.; Katagiri, T.; Uneyama, K.: Synthesis of Fluorinated Quinolines and a Pyrazoloquinoline
Alcaide, B.; Almendros, P.; Luna, A.; Campo, T. Martínez del: Synthesis of 4-Hydroxypipecolic Acid β-Lactam Analogues from Oxoazetidines

Issue 04/2008

Donohoe, T. J.; Fishlock, L. P.; Procopiou, P. A.: Construction of 2-Pyridones and Pyridines via Ring-Closing Metathesis
Liu, Z.; Shi, F.; Martinez, P. D. G.; Raminelli, C.; Larock, R. C.: Synthesis of Indazoles by Cycloaddition of Diazo Acetates with Arynes
Sripada, L.; Teske, J. A.; Deiters, A.: A Microwave-Assisted Cyclotrimerization Route to Phenanthridines
Aliyenne, A. O.; Kraïem, J.; Kacem, Y.; Hassine, B. B.: A Lateral Metallation Strategy for 1,2-Benzothiazin-3-one 1,1-Dioxides
Parhasarathy, K.; Jeganmohan, M.; Cheng, C.-H.: Synthesis of Multisubstituted Pyridines from Ketoximes and Alkynes
Wang, Z.; Wu, J.: Synthesis of Indolylquinolin-2-ones via a Cross-Coupling-Cyclization Sequence
AlajarÍn, M.; Bonillo, B.; Vidal, A.; Bautista, D.: A Biradical Cylization Route to Axially Chiral Biheteroaryls
Keith, J. M.: One-Step Synthesis of Imidazolo-Heteroarenes from Heteroarene N-Oxides
Zhang, Z.; Tan, J.; Wang, Z.: Synthesis of 2-Methylquinolines via Oxidative Aza-Wacker Cyclization
Alcaide, B.; Almendros, P.; Cabrero, G.; Ruiz, M. P.: Iodine-Catalyzed Enantioselective Synthesis of Pyrrolidin-2-ones from β-Lactams
Ackermann, L.; Sandmann, R.; Villar, A.; Kaspar, L. T.: Hydroamination-Heck Annulation Route to 3-Substituted Indoles
Onizawa, Y.; Kusama, H.; Iwasawa, N.: W(CO)5-Catalyzed Synthesis of 2- and 3-Azabicyclo[3.3.0]octanes
Siamaki, A. R.; Black, D. A.; Arndtsen, B. A.: A Palladium-Catalyzed Carbonylative Cross-Coupling Route to Imidazolones
Praveen, C.; Kumar, K. Hemanth; Muralidharan, D.; Perumal, P. T.: Oxidative Cyclization of ortho-Phenolic and Thiophenolic Imines
Barluenga, J.; Jiménez-Aquino, A.; Fernández, M. A.; Aznar, F.; Valdés, C.: Three-Component Synthesis of 2,3,5-Triaryl Pyridines

Issue 03/2008

Heller, B.; Redkin, D.; Gutnov, A.; Fischer, C.; Bonrath, W.; Karge, R.; Hapke, M.: Synthesis of Chiral Pyridyl Alcohols by Cyclotrimerization
Cui, S.-L.; Wang, J.; Wang, Y.-G.: Copper-Catalyzed Synthesis of 2-Imino-1,2-dihydroquinolines and -thiochromenes
Martín, R.; Cuenca, A.; Buchwald, S. L.: Copper-Catalyzed C-N Bond Coupling Approach to Highly Substituted Oxazoles
Hurst, T. E.; Miles, T. J.; Moody, C. J.: [c]-Annelated Pyridines via Intramolecular Diels-Alder Reaction
Voskressensky, L. G.; Listratova, A. V.; Borisova, T. N.; Alexandrov, G. G.; Varlamov, A. V.: Ring Expansion of Tetrahydroisoquinolines to Form Benzoazocines
Szabo, R.; Crozet, M. D.; Vanelle, P.: Double Suzuki-Miyaura Coupling in the Synthesis of Imidazo[1,2-a]pyridine Derivatives
Alcaide, B.; Almendros, P.; Carrascosa, R.; Redondo, M. C.: Synthesis of Substituted Pyrroles from 2-Azetidinone Allenols
Adriaenssens, L. V.; Hartley, R. C.: Synthesis of Piperidinones from β-Amino Acids by Petasis Methylenation
Fuller, P. H.; Chemler, S. R.: Polycyclic Lactams via Cu(II)-Mediated Intramolecular Alkene Carboamination
Leogane, O.; Lebel, H.: Curtius-Rearrangement Approach to 2,3-Substituted Indoles
Dash, J.; Lechel, T.; Reissig, H.-U.: Three-Component Synthesis of Functionalized Pyridines
Zhao, L.-B.; Guan, Z.-H.; Han, Y.; Xie, Y.-X.; He, S.; Liang, Y.-M.: Synthesis of Furans via Copper-Catalyzed [4+1] Cycloaddition
Han, Y.; Xie, Y.-X.; Zhao, L.-B.; Fan, L.-J.; Liang, Y.-M.: Synthesis of Imidazolines from N-Imidoylaziridines
Otani, T.; Kunimatsu, S.; Nihei, H.; Abe, Y.; Saito, T.: In-Mediated Conversion of 2-Alkynylphenyl Isothiocyanates to Quinoline-2-thiones
Butler, J. D.; Solano, D. M.; Robins, L. I.; Haddadin, M. J.; Kurth, M. J.: Substituted Indazolobenzoxazines via One-Pot Intramolecular Bis-Heterocyclizations

Issue 02/2008

Zhao, B.; Yuan, W.; Du, H.; Shi, Y.: Copper(I)-Catalyzed Diamination of Terminal Olefins to Vicinal Diamines
Heller, S. T.; Natarajan, S. R.: Nickel-Catalyzed Synthesis of Pyrazolo[3,4-c]pyridines via Alkyne Annulation
Kim, I.; Won, H. K.; Choi, J.; Lee, G. H.: Synthesis of Indolizines via Iodocyclization of Pyridine Allylic Acetates
Dubbaka, S. R.; Kienle, M.; Mayr, H.; Knochel, P.: Pyridine Ring Heterannulation via Imine-eneyne Ring Closure
Delain-Bioton, L.; Villemin, D.; Lohier, J.-F.; Sopkova, J.; Jaffres, P.-A.: Copper-Catalyzed Synthesis of Triazolyl-alkylphosphonates
Sugiyama, M.; Hong, Z.; Liang, P.-H.; Dean, S. M.; Whalen, L. J.; Greenberg, W. A.; Wong, C.-H.: Enzymatic One-Pot Synthesis of Iminocyclitols
Chen, Y.; Xie, X.; Ma, D.: Cascade Process from Anilines to Indoles Involving a Copper-Catalyzed Arylation
Solé, D.; Serrano, O.: Pd-Catalyzed Intramolecular Cyclization of 2-Iodoanilino Esters to Dihydroquinolin-4-ones
Cui, S.-L.; Wang, J.; Wang, Y.-G.: Copper-Catalyzed Three-Component Reaction to Imino-pyrrolines
Miura, T.; Takahashi, Y.; Murakami, M.: Rh-Catalyzed Synthesis of 3-Alkylideneoxindoles from 2-Alkynylisocyanates and Arylboronic Acids
Browne, D. L.; Helm, M. D.; Plant, A.; Harrity, J. P. A.: [2+3]-Cycloaddition Route to Pyrazole Boronic Esters from Sydnones and Alkynylboronates
Ding, Q.; Wu, J.: Combined Ag- and Proline-Catalyzed Three-Com-ponent Synthesis of 1,2-Dihydroisoquinolines
Wang, Z.; Wan, W.; Jiang, H.; Hao, J.: One-Pot Synthesis of N-Acyl Indolines from 2-Aminophenethyl Alcohols
Chen, L.; Zhao, Y.-L.; Liu, Q.; Cheng, C.; Piao, C.-R.: Pyridinones from Reaction of Vilsmeier-Haack Reagents with Ketene Dithioacetals
Gabriele, B.; Mancuso, R.; Salerno, G.; Costa, M.: 2-Benzofuran-2-acetamides via Sequential Pd(0)-Pd(II) Catalysis

Issue 01/2008

Bodtke, A.; Pfeiffer, W.-D.; Görls, H.; Dollinger, H.; Langer, P.: Synthesis of Imidazo[1,2-c]quinazolines from Isothiocyanatobenzonitriles
Ding, Q.; Wang, B.; Wu, J.: Dihydroisoquinolin-1-ylphosphonates via a Copper-Catalyzed Three-Component Reaction
Sriramurthy, V.; Barcan, G. A.; Kwon, O.: Asymmetric Synthesis of Oxazolidines, Thiazolidines, and Pyrrolidines
Devarie-Baez, N. O.; Shuhler, B. J.; Wang, H.; Xian, M.: One-Pot Synthesis of 2,3-Disubstituted Thiophenes via a [1,4]-Silyl Migration Reaction
Bonnamour, J.; Legros, J.; Crousee, B.; Bonnet-Delpon, D.: Synthesis of 1,2,3-Triazoles via Huisgen 1,3-Dipolar Cycloaddition
Gabillet, S.; Lecerclé, D.; Loreau, O.; Carboni, M.; Dézard, S.; Gomis, J.-M.; Taran, F.: Synthesis of 5- and 6-Membered S,O- and S,N-Heterocycles
Nakamura, I.; Sato, T.; Terada, M.; Yamamoto, Y.: Gold-Catalyzed Synthesis of Benzo[b]thiophenes from Alkynylphenylthiosilanes
Bellina, F.; Cauteruccio, S.; Rossi, R.: Diarylated Imidazoles via Sequential Metal-Catalyzed Suzuki and C-H Activation Reactions
John, O. R. S.; Killeen, N. M.; Knowles, D. A.; Yau, S. C.; Bagley, M. C.; Tomkinson, N. C. O.: α-Oxytosylation of Ketones: Synthesis of Thiazoles and Imidazoles
Handy, S. T.; Wilson, T.; Muth, A.: One-Pot Double Suzuki Cross-Coupling: Synthesis of Diarylated Pyridines
Yan, B.; Liu, Y.: Gold-Catalyzed Three-Component Synthesis of Aminoindolizines
Zheng, N.; Anderson, K. W.; Huang, X.; Nguyen, H. N.; Buchwald, S. L.: Synthesis of N-Aryl Benzimidazoles by Pd-Catalyzed Amination-Heteroannulation
Teimouri, M. B.; Khavasi, H. R.: Synthesis of Naphthofuroquinones by a Three-Component Reaction
Fujiwara, S.-i; Asanuma, Y.; Shin-ike, T.; Kambe, N.: Cu-Catalyzed Three-Component Synthesis of 1,3-Benzoselena- and -tellurazoles
Dénès, F.; Beaufils, F.; Renaud, P.: Synthesis of Pyrrolizidines and Indolizidines via Radical 1,5-Hydrogen Transfer

Issue 12/2007

Tanimori, S.; Ura, H.; Kirihata, M.: Copper-Catalyzed α-Enolate Arylation Route to 2,3-Disubstituted Indoles
Korotkov, V. S.; Larionov, O. V.; Hofmeister, A.; Magull, J.; de Meijere, A.: Synthesis of Pyrazolidines via GaCl3-Catalyzed Insertion of Diazines into Cyclopropanes
Sayyed, I. A.; Alex, K.; Tillack, A.; Schwarz, N.; Michalik, D.; Beller, M.: Sequential Hydroamination-Fischer Cyclization Route to Indoles
Farran, D.; Parrot, I.; Martinez, J.; Dewynter, G.: Stereoselective Ring Contraction of Diketopiperazines into Pyrrolidine-2,4-diones
Li, Y.; Zou, H.; Gong, J.; Xiang, J.; Luo, T.; Quan, J.; Wang, G.; Yang, Z.: Zinc Triflate Catalyzed Synthesis of Condensed Maleimides and Carbazoles
Itoh, T.; Mase, T.: Palladium-Catalyzed Synthesis of Benzothiazoles Using a Thiol Surrogate
Shabashov, D.; Daugulis, O.: C-H-Activated ortho-Arylation of Anilides and Their Cyclization to Phenanthridines
Downer-Riley, N. K.; Jackson, Y. A.: Synthesis of Benzothiazoles and Benzoxazoles from Thiobenzamides
Barbero, N.; Carril, M.; SanMartin, R.; Domínguez, E.: Copper-Catalyzed Intramolecular Cyclization of 2-Haloacetanilines to Benzo[d]oxazoles
Wang, Z.; Fan, R.; Wu, J.: Regioselective Suzuki Cross-Coupling Route to 3,4-Disubstituted Quinolin-2(1H)-ones
Yan, B.; Zhou, Y.; Zhang, H.; Chen, J.; Liu, Y.: Copper-Catalyzed Heteroannulation of Propargylic Pyridines to Indolizines
Hayes, S. J.; Menzies, M. D.; O’Halloran, M.; Tan, W.; Knight, D. W.: Synthesis of Substituted Furans via Silica-Supported Silver Catalysis
Yadav, J. S.; Reddy, B. V. Subba; Rao, Y. Gopal; Srinivas, M.; Narsaiah, A. V.: Cu-Catalyzed Synthesis of Imidazo[1,2-a]pyridines from α-Diazoketones and 2-Aminopyridines
Babudri, F.; Cicco, S. R.; Farinola, G. M.; Lopez, L. C.; Naso, F.; Pinto, V.: AlCl3-Mediated Synthesis of Furans from Acid Chlorides and bis-Silylated Butadiene
Alizadeh, A.; Oskueyan, Q.; Rostamnia, S.: Three-Component Synthesis of Furylnicotinamides and Isonicotinamides

Issue 11/2007

Yang, X.-J.; Zhang, L.-S.; Liu, J.-T.: Preparation of Perfluoroalkylated 1,2-Dihydropyrimidines and Pyrimidines
Zu, L.; Xie, H.; Li, H.; Wang, J.; Jiang, W.; Wang, W.: Organocatalytic Domino Michael-Aldol Reaction to Chiral Benzothiopyrans
Braibante, M. E. F.; Braibante, H. T. S.; de Tavares, L. Carvalho; Rohte, S. F.; Costa, C. C.; Morel, A. F.; Stüker, C. Z.; Burrow, R. A.: Regioselective Synthesis of Pyrazoles from β-Oxo Thioxoesters and α-Oxoketene O,N-Acetals
Gabriele, B.; Mancuso, R.; Salerno, G.; Ruffolo, G.; Plastina, P.: Synthesis of Quinolines by Catalyzed Cyclodehydration of Aminoaryl-2-yn-1-ols
Liu, G.-B.; Zhao, H.-Y.; Yang, H.-J.; Gao, X.; Li, M.-K.; Thiemann, T.: Reductive Cyclization of o-Nitrophenylazophenols to Benzotriazoles
Nakhla, J. S.; Wolfe, J. P.: Asymmetric Synthesis of Chiral Piperazines
Bajtos, B.; Yu, M.; Zhao, H.; Pagenkopf, B. L.: Synthesis of 2,3-Fused Indoles
Hill, G. B.; Mortlock, A. A.: Synthetic Routes to 4-Amino-Pyrazoles from Vinamidinium Salts
Patil, N. T.; Wu, H.; Yamamoto, Y.: Palladium-Catalyzed Hydroamination Route to 2-Substituted Tetrahydroquinolines
Palacios, F.; Herrán, E.; Rubiales, G.; Alonso, C.: Pyridine Derivatives from Vinylic Phosphazenes via an aza-Wittig Reaction
Schwier, T.; Sromek, A. W.; Yap, D. M. L.; Chernyak, D.; Gevorgyan, V.: Cycloisomerization of Alkynyl Ketones to Multisubstituted Furans
Saha, B.; Sharma, S.; Sawant, D.; Kundu, B.: One-Pot Three-Component Synthesis of Triazoles in Water
Fuwa, H.; Sasaki, M.: Synthesis of Indoles and Indolines from α-Phosphoryloxy Enecarbamates
Landge, S. M.; Schmidt, A.; Outerbridge, V.; Török, B.: (Pd/C/K-10)-Catalyzed One-Pot Synthesis of Substituted Pyrazoles
Henry, C. E.; Kwon, O.: Synthesis of Fused Coumarins via Cycloaddition Reactions

Issue 10/2007

Suzuki, H.; Sakai, N.; Iwahara, R.; Fujiwaka, T.; Satoh, M.; Kakehi, A.; Konakahara, T.: Synthesis of Fluorinated Pyridines and Their Conversion into Naphthyridines
Loska, R.; Majcher, M.; Makosza, M.: Synthesis of Trifluoromethylated Pyridines and Quinolines Using Me3SiCF3
Sun, Z.; Yu, S.; Ding, Z.; Ma, D.: Copper-Catalyzed Asymmetric Synthesis of Dihydropyridines
Mancheño, O. G.; Bolm, C.: Synthesis of Tetrazole and Oxadiazole Sulfoximines
Donets, P. A.; Van der Eycken, E. V.: Synthesis of 3-Benzazepines via an Intramolecular Reductive Heck Reaction
KaÏm, L. El; Grimaud, L.; Oble, J.: Ugi-Smiles Metathesis Approach to Pyrimido Azepines
Fuwa, H.; Sasaki, M.: Heck/Diels-Alder Cascade Route to Tetrahydrocarbazoles
Cortez, G. A.; Baxter, C. A.; Schrock, R. R.; Hoveyda, A. H.: Ru- and Mo-Catalyzed Asymmetric Synthesis of Pyrans and Piperidines
Clarke, P. A.; Zaytzev, A. V.; Whitwood, A. C.: One-Pot Synthesis of Highly Functionalized Piperidines
Song, J.; Shen, Q.; Xu, F.; Lu, X.: Palladium-Catalyzed Enantioselective Synthesis of γ-Butyrolactones
Xia, Y.; Li, W.; Qu, F.; Fan, Z.; Liu, X.; Berro, C.; Rauzy, E.; Peng, L.: Synthesis of Bitriazolyl Nucleosides via Huisgen [2+3] Cycloaddition
Przewloka, T.; Chen, S.; Xia, Z.; Li, H.; Zhang, S.; Chimmanamada, D.; Kostik, E.; James, D.; Koya, K.; Sun, L.: Regioselective Synthesis Of 3-Acylated Indolizines Using a Brederick-Type Reagent
Fattuoni, C.; Usai, M.; Cabiddu, M. G.; Cadoni, E.; Montis, S. De; Cabiddu, S.: Synthesis of Thieno[3,2-b]thiophene 1,1-Dioxide Derivatives
Kang, S. B.; Clercq, E. De; Lakshman, M. K.: Pd-Catalyzed Synthesis of C4-Aryl Pyrimidinone Nucleoside Analogues
Ding, Q.; Ye, Y.; Fan, R.; Wu, J.: Metal-Tuned Synthesis of Isoindolyl and Isoquinolinyl Phosphonates

Issue 09/2007

Zhang, L.; Wu, J.: Improved Friedländer Synthesis of Quinolines
Yoshida, H.; Fukushima, H.; Morishita, T.; Ohshita, J.; Kunai, A.: Three-Component Coupling Strategy to Benzoannulated N- or O-Heterocycles
Fischer, D.; Tomeba, H.; Pahadi, N. K.; Patil, N. T.; Yamamoto, Y.: Transition-Metal-Free Synthesis of Isoquinolines
Rueping, M.; Antonchick, A. P.: Enantioselective Reduction of Pyridines via Brønsted Acid Catalysis
Melo, T. M. V. D. Pinhoe; Nunes, C. M.; Soares, M. I. L.; Paixão, J. A.; Beja, A. M.; Silva, M. R.: Diazafulvenium Methides in Synthesis of Functionalized Pyrazoles
Zhang, X.; Hsung, R. P.; Li, H.: Synthesis of Fused Triazoles via Azide-[3+2] Cycloaddition and Ring-Closing Metathesis
Young, D. D.; Deiters, A.: Synthesis of Fused Pyridines via Solid-Supported Cyclotrimerization Reaction
Fattuoni, C.; Usai, M.; Cabiddu, M. G.; Cadoni, E.; Montis, S. De; Cabiddu, S.: Synthesis of Thieno[3,2-b]thiophene 1,1-Dioxide Derivatives
Pridmore, S. J.; Slatford, P. A.; Daniel, A.; Whittlesey, M. K.; Williams, J. M. J.: Ruthenium-Catalyzed Pyrrole Synthesis from 1,4-Alkynediols
Bonne, D.; Dekhane, M.; Zhu, J.: Multicomponent Synthesis of Oxazoles and Furopyrrolones
Belskaia, N. P.: Synthesis of 2H-[1,2,3]thiadiazolo[5,4-b]indoles from Isatin-Derived Hydrazines
Berseneva, V. S.; Bakulev, V. A.; Dehaen, W.; Toppet, S.; Borovkova, M.: De Novo Synthesis of 4-Thio- and 4-Aminopyrrole[3,4-c]pyridines
Newman, C. A.; Antilla, J. C.; Chen, P.; Predeus, A. V.; Fielding, L.; Wulff, W. D.: Asymmetric Synthesis of Dihydropyridinones
Basnet, A.; Thapa, P.; Karki, R.; Na, Y.; Jahng, Y.; Jeong, B.-S.; Jeong, T. C.; Lee, C.-S.; Lee, E.-S.: The Synthesis of Trisubstituted Pyridines via Kröhnke Reaction
Chuprakov, S.; Hwang, F. W.; Gevorgyan, V.: Rhodium-Catalyzed Synthesis of Indolizines and Imidazopyridines
Shafiq, Z.; Liu, L.; Liu, Z.; Wang, D.; Chen, Y.-J.: Ag(I)-Catalyzed Nucleophilic Substitution of Baylis-Hillman Adduct with Indoles

Issue 08/2007

Bonin, M.-A.; GiguÈre, D.; Roy, R.: Synthesis of N-Arylimidazoles by Catalytic Cross-Cycloaddition of Isocyanides
Littke, A.; Soumeillant, M.; III, R. F. Kaltenbach; Cherney, R. J.; Tarby, C. M.; Kiau, S.: Palladium-Catalyzed Cyanation of Aryl and Heteroaryl Chlorides
Shindo, M.; Yoshimura, Y.; Hayashi, M.; Soejima, H.; Yoshikawa, T.; Matsumoto, K.; Shishido, K.: Synthesis of Furans, Pyrroles and Thiophenes Using Ynolate Building Blocks
Qi, X.; Ready, J. M.: Cu-Mediated Synthesis of Pyrazoles via 1,3-Dipolar Cycloaddition
Garner, P.; Hu, J.; Parker, C. G.; Youngs, W. J.; Medvetz, D.: Asymmetric, exo-Selective Synthesis of trans-4,5-Disubstituted Pyrrolidines
Stroup, B. W.; Szklennik, P. V.; Forster, C. J.; Serrano-Wu, M. H.: Selective Amination of Trihalopyridines
Chuprakov, S.; Chernyak, N.; Dudnik, A. S.; Gevorgyan, V.: Direct Pd-Catalyzed Arylation of Triazoles
Oikawa, M.; Takeda, Y.; Naito, S.; Hashizume, D.; Koshino, H.; Sasaki, M.: Synthesis of Isoquinolines via 1,3-Dipolar Cycloaddition-Heck Coupling
Yin, J.; Xiang, B.; Huffman, M. A.; Raab, C. E.; Davies, I. W.: Synthesis of 2-Aminopyridines and 2-Amino-Quinolines from Their N-Oxides
Lewis, J. C.; Bergman, R. G.; Ellman, J. A.: Rh-Catalyzed C-H Activation Route to 2-Alkylpyridines and 2-Alkylquinolines
Lu, J.-Y.; Arndt, H.-D.: Regioselective Synthesis of Functionalized 3-Hydroxypyridines
Milgram, B. C.; Eskildsen, K.; Richter, S. M.; Scheidt, W. R.; Scheidt, K. A.: Symmetric 3,4-Disubstituted Pyrroles via Piloty-Robinson Synthesis
Pisani, L.; Prokopcov, H.; Kremsner, J. M.; Kappe, C. O.: Microwave-Assisted Biginelli Synthesis of Dihydropyrimidine-2-ones
Solovyev, A. Y.; Androsov, D. A.; Neckers, D. C.: One-Pot Synthesis of Substituted 2-Aminobenzo[b]thiophenes

Issue 07/2007

Chebanov, V. A.; Saraev, V. E.; Desenko, S. M.; Chernenko, V. N.; Shishkina, S. V.; Shishkin, O. V.; Kobzar, K. M.; Kappe, C. O.: Synthesis of Pyrazoloquinolizinones via a Three-Component Reaction
Reeves, J. T.; Song, J. J.; Tan, Z.; Lee, H.; Yee, N. K.; Senanayake, C. H.: Synthesis of 2-Formylpyrroles via Heterocyclic Interconversion
Masdeu, C.; GÓmez, E.; Williams, N. A. O.; Lavilla, R.: Benzimidazolium Salts from Dihydropyridines and Isocyanides
Zhou, C.-Y.; Che, C.-M.: Gold-Catalyzed Synthesis of Pyrrolidones by an 5- and 6-exo-trig Cycloaddition Reaction
Hulcoop, D. G.; Lautens, M.: Two-Carbon Annulation of N-Arylpyrroles to Benzoindoles and Pyrroloquinolines
Sridharan, V.; Perumal, P. T.; Avendaño, C.; Menéndez, J. C.: Synthesis of Tetrahydroquinolines via a Vinylogous Aza-Povarov Reaction
Pinto, A.; Neuville, L.; Zhu, J.: Palladium-Catalyzed Synthesis of 3-(Diarylmethylene)oxindoles
Someya, H.; Ohmiya, H.; Yorimitsu, H.; Oshima, K.: Synthesis of Pyrrolidines by Cobalt-Catalyzed Intramolecular Cyclization
Peng, L.; Zhang, X.; Ma, J.; Zhong, Z.; Wang, J.: Synthesis of Pyrroles from Allenic Aldehydes and Amines
Dang, T. T.; Langer, P.: One-Pot Regioselective Synthesis of Pyrazole-5-Carboxylates
Wang, X. L.; Zheng, X. F.; Liu, R. H.; Reiner, J.; Chang, J. B.: Pictet-Spengler Synthesis of Naphthoquino[b]-benzo[e][1,4]diazepines
Dai, L.-Z.; Shi, Y.-L.; Zhao, G.-L.; Shi, M.: Base-Catalyzed 2H-Chromene Synthesis from Salicylaldehydes and Allenes
Szlosek-Pinaud, M.; Diaz, P.; Martinez, J.; Lamaty, F.: Synthesis of 2,3-Dihydrobenzofuran by Tandem Palladium-Catalyzed Reactions
Vik, A.; Gundersen, L.-L.: Synthesis of Tetrahydrodiazepinopurines by Ring-Closing Metathesis
Tu, S.; Zhang, J.; Jia, R.; Jiang, B.; Zhang, Y.; Jiang, H.: Synthesis of a New Class of Pyrido[2,3-d]pyrimidine Derivatives

Issue 06/2007

Nair, V.; Mathew, S.; Biju, A.; Suresh, E.: Zwitterion-Induced Synthesis of Pyrazines and Pyrazolopyridazines
Nakamura, I.; Yamagishi, U.; Song, D.; Konta, S.; Yamamoto, Y.: Au- and In-Catalyzed Synthesis of 3- and 6-Sulfonylindoles
Worlikar, S. A.; Kesharwani, T.; Yao, T.; Larock, R. C.: Synthesis of 2H-Benzopyran via Electrophilic Cyclization
Zhang, Z.; Zhang, Q.; Sun, S.; Xiong, T.; Liu, Q.: Highly Regioselective Synthesis of Furoquinoline Derivatives
Viña, D.; Olmo, E. del; López-Pérez, J. L.; Feliciano, A. San: One-Pot Cu-Catalyzed Synthesis of 3-Substituted Indazoles
Schomaker, J. M.; Bhattacharjee, S.; Yan, J.; Borhan, B.: Stereoselective Synthesis of Pyrrolidines from Aziridinols
Savitha, G.; Niveditha, S. K.; Muralidharan, D.; Perumal, P. T.: Spiro Hydrofuran Oxindole Derivatives by Oxidative Cyclization
Oh, C. H.; Park, H. M.; Park, D. I.: Pd-Catalyzed Reductive Double Cyclization of Yne-enynals to Furans
Ghorai, M. K.; Das, K.; Kumar, A.: Enantiopure N-Tosylazetidines from α-Amino Acids
Ackermann, L.; Althammer, A.: Pd-Catalyzed Synthesis of Carbazoles and α-Carbolines via C-H Activation
Li, H.; Wang, J.; Xie, H.; Zu, L.; Jiang, W.; Duesler, E. N.; Wang, W.: Organo-Catalyzed Synthesis of 1,2-Dihydroquinolines
Hajra, S.; Sinha, D.; Bhowmick, M.: Zn-Catalyzed Synthesis of 1,5-Disubstituted Tetrazoles
Saito, T.; Sugizaki, K.; Otani, T.; Suyama, T.: Rhodium-Catalyzed Intramolecular Hetero-Pauson-Khand Reaction
Battistuzzi, G.; Bernini, R.; Cacchi, S.; Salve, I. De; Fabrizi, G.: 4-Aryl-2-quinolones Through Heck and Buchwald-Hartwig Reaction

Issue 05/2007

Barluenga, J.; Jiménez-Aquino, A.; Valdés, C.; Aznar, F.: Synthesis of Indoles by Domino C/N-Arylation of Azaallylic Anions
Liu, Y.; Song, Z.; Yan, B.: Synthesis of 3-Aminoindolizines via Pd/Cu-Catalyzed Reactions
Jiménez-González, L.; García-Muñoz, S.; Álvarez-Corral, M.; Muñoz-Dorado, M.; Rodríguez-García, I.: A Diastereoselective Sakurai-Metathesis Route to Dihydrobenzofurans
Cyr, D. J. St; Martin, N.; Arndtsen, B. A.: Four-Component Synthesis of Highly Substituted Pyrroles
Yerushalmi, S.; Lemcoff, N. G.; Bittner, S.: Synthesis of Large Heterocyclic-Ring Fused Naphthoquinones
Zhou, Y.; Jr, J. A. Porco; Snyder, J. K.: Microwave-Assisted, Co-Catalyzed Synthesis of Naphthyridines
Kang, Q.; Zhao, Z.-A.; You, S.-L.: Asymmetric Synthesis of 3-Indolyl Methylamines (Gramines)
Rech, J. C.; Yato, M.; Duckett, D.; Ember, B.; LoGrasso, P. V.; Bergman, R. G.; Ellman, J. A.: Rh-Catalyzed C-H Activation Route to Bicyclic Imidazoles
Ando, K.; Akai, Y.; Kunitomo, J.-i; Yokomizo, T.; Nakajima, H.; Takeuchi, T.; Yamashita, M.; Ohta, S.; Ohishi, T.; Ohishi, Y.: Synthesis of Furobenzazepinones by an Intramolecular Heck Reaction
Galliford, C. V.; Scheidt, K. A.: Rh-Catalyzed Synthesis of N-Aryl Trisubstituted Pyrroles
Wang, X.; Gribkov, D. V.; Sames, D.: Pd-Catalyzed C-H Activation Route to Aryl Indoles and Pyrroles
Chassaing, S.; Kumarraja, M.; Sido, A. S. S.; Pale, P.; Sommer, J.: Regioselective Cu(I)-Zeolite-Catalyzed Synthesis of Triazoles
Roy, U. K.; Jana, P. K.; Roy, S.: Pd/Sn Mediated Multicomponent Synthesis of Tetrahydropyrans
Sridharan, V.; Avendaño, C.; Menéndez, J. C.: Three-Component Synthesis of Tetrahydroquinolines
DiMauro, E. F.; Kennedy, J. M.: 3-Amino-Imidazopyridines by a Microwave-Assisted Synthesis

Issue 04/2007

Dadiboyena, S.; Xu, J.; II, A. T. Hamme: Synthesis of Isoxazoles via [2+3]-Dipolar Cycloaddition Using Alkyne Surrogates
Zhao, B.; Lu, X.: Benzofurans via Pd(II)-Catalyzed Arylboronic Acid Addition to Nitriles
Ferrer, C.; Amijs, C. H. M.; Echavarren, A. M.: Gold-Catalyzed Synthesis of Azepino[4,5-b]indoles and Indoloazocines
Viña, D.; Olmo, E. del; López-Pérez, J. L.; Feliciano, A. San: A Cu-Catalyzed C-N Bond Coupling Route to Substituted Indazoles
Galliford, C. V.; Martenson, J. S.; Stern, C.; Scheidt, K. A.: Spirooxindoles from a 3-CR of Imines, Diazoesters, and Olefin Dipolarophiles
Sundén, H.; Ibrahem, I.; Zaho, G.-L.; Eriksson, L.; Córdova, A.: Organocatalytic Synthesis of Benzopyrans
Tang, W.-J.; Zhu, S.-F.; Xu, L.-J.; Zhou, Q.-L.; Fan, Q.-H.; Zhou, H.-F.; Lam, K.; Chan, A. S. C.: Asymmetric Hydrogenation of Quinolines
Servais, A.; Azzouz, M.; Lopes, D.; Courillon, C.; Malacria, M.: Radical Cyclization of N-Acylcyanamides to Pyrroloquinazolines
Teimouri, M. B.: One-Pot Synthesis of Pyrazolo[1,2-b]phthalazinediones
Xie, F.; Li, S.; Bai, D.; Lou, L.; Hu, Y.: Synthesis of Substituted Pyrimidines from Chromones
Cadierno, V.; Gimeno, J.; Nebra, N.: Fully Substituted Furans by One-Pot Propargylation-Cycloisomerization
Paul, S.; Chotana, G. A.; Holmes, D.; Reichle, R. C.; Jr, R. E. Maleczka; III, M. R. Smith: Ir-Catalyzed Selective C-7 Borylation of 2-Substituted Indoles
Wood, M. C.; Leitch, D. C.; Yeung, C. S.; Kozak, J. A.; Schafer, L. L.: Zirconium-Catalyzed Asymmetric Cyclohydroamination of Alkenes
Lingaiah, B. V.; Ezikiel, G.; Yakaiah, T.; Reddy, G. V.; Rao, P. S.: Synthesis of 4-Quinazolinones under Green Conditions
Conreaux, D.; Bossharth, E.; Monteiro, N.; Desbordes, P.; Vors, J.-P.; Balme, G.: Regioselective Cross-Coupling Route to 3,5-Disubstituted 2-Pyridones

Issue 03/2007

Raju, S.; Batchu, V. R.; Swamy, N. K.; Dev, R. V.; Sreekanth, B. R.; Babu, J. M.; Vyas, K.; Kumar, P. R.; Mukkanti, K.; Annamalai, P.; Pal, M.: Fused Thienopyranones via Sonogashira-Based Heteroannulation
Parks, B. W.; Gilbertson, R. D.; Domaille, D. W.; Hutchison, J. E.: Metathesis-Mediated Route to 6,6-Bicyclic Malonamides
Chaume, G.; Van Severen, M.-C.; Marinkovic, S.; Brigaud, T.: Synthesis of Enantiopure (S)- and (R)-α-Trifluoromethyl Proline
Kearney, A. M.; Vanderwal, C. D.: Heterocyclic Interconversion. Pyridinium Salts to Indole-3-propenals
García-Cuadrado, D.; Cuadro, A. M.; Alvarez-Builla, J.; Sancho, U.; Castano, O.; Vaquero, J. J.: Synthesis of Biquinolizinium Salts
Blanco, G.; Seguí, N.; Quintela, J. M.; Peinador, C.; Chas, M.; Toba, R.: One-Pot Synthesis of Pyrazinothienopyrimidinones
Zheng, Z.; Yu, Z.; Luo, N.; Han, X.: Synthesis of Bicyclic Pyrazolinones Using Fischer Carbene Complexes
Fuchibe, K.; Hatemata, R.; Akiyama, T.: Chiral Proline Derivatives via One-Pot [3+2] Cycloaddition-Cross-Coupling
Silva, F.; Reiter, M.; Mills-Webb, R.; Sawicki, M.; Klär, D.; Bensel, N.; Wagner, A.; Gouverneur, V.: Palladium-Catalyzed Wacker-Heck Reactions
Leclerc, J.-P.; Fagnou, K.: Cross-Coupling Reactions of DiazineN-Oxides with Aryl Halides
Ponnala, S.; Sahu, D. P.: Oxidative Heteroannulation Route to Benzoxazoles and Benzimidazoles
Sezer, S.; Özdemirhan, D.; Şahin, E.; Tanyelia, C.: Cyclopentenone-Fused Perhydroperans via Pauson-Khand Reaction
Majireck, M. M.; Weinreb, S. M.: Ru-Catalyzed [3+2] Cycloaddition of Azides with Alkynes to form Triazoles
Wu, Z.; Huang, X.: Synthesis of Furan-2(5H)-ones via Oxidative Free-Radical Cyclization
Kondo, T.; Nomura, M.; Ura, Y.; Wada, K.; Mitsudo, T.: Ruthenium-Catalyzed Pauson-Khand Synthesis of Maleimides

Issue 02/2007

Barluenga, J.; Valdes, C.; BeltrÁn, G.; Escribano, M.; Aznar, F.: Palladium-Catalyzed Synthesis of 1H-1,2,3-Triazoles
Pinto, A.; Neuville, L.; Retailleau, P.; Zhu, J.: Pd-Catalyzed C-H Activation Route to 3-(Methylenyl)indolinones
Motti, E.; Faccini, F.; Ferrari, I.; Catellani, M.; Ferraccioli, R.: Synthesis of 6H-Dibenzopyrans via an Unsymmetrical Aryl-Aryl Cross-Coupling
Tang, W.; Ding, Y.-X.: Palladium-Catalyzed Hydroaminative Route to Phosphaisoquinolin-1-ones
Movassaghi, M.; Hill, M. D.: Quinazolines and Pyrimidines by Electrophilic Activation of Amides
Qacemi, M. El; Ricard, L.; Zard, S. Z.: Radical-Mediated Synthesis of Imidazopyridinones
Merkul, E.; Müller, T. J. J.: One-Pot Synthesis of 2,5-Disubstituted Oxazoles
Willis, M. C.; Snell, R. H.; Fletcher, A. J.; Woodward, R. L.: Pd-Catalyzed C-N Coupling. Synthesis of 2,4-Quinazolinediones
Schmidt, D.; Conrad, J.; Klaiber, I.; Beifuss, U.: Pyranones from Potassium Salts of Acyclic Tricarbonyl Compounds
DÍez-GonzÁlez, S.; Correa, A.; Cavallo, L.; Nolan, S. P.: 1,2,3-Triazoles by a [3+2] Cycloaddition of Azides and Alkynes
Demir, A. S.; Subasi, N. T.; Sahin, E.: Stereoselective Cyclization Routes to Fused Pyrrole-Pyrazine-Oxazoles
Vugts, D. J.; Koningstein, M. M.; Schmitz, R. F.; de Kanter, F. J. J.; Groen, M. B.; Orru, R. V. A.: Synthesis of Dihydropyrimidones and Thiazines by a Multicomponent Reaction
Ye, F.; Alper, H.: Palladium-Catalyzed Synthesis of Lactones and Lactams in Ionic Liquids
Ma, C.; Ding, H.; Zhang, Y.; Bian, M.: Synthesis of Polysubstituted Furan-Fused 1,4-Thiazepine Derivatives
Zhou, Z.-Z.; Ji, F.-Q.; Cao, M.; Yang, G.-F.: Microwave-Assisted Intramolecular Stetter Reaction in Ionic Liquids

Issue 01/2007

Fayol, A.; Fang, Y.-Q.; Lautens, M.: Pd-Catalyzed Sequential C-N and C-C Coupling Route to 2-Vinylindoles
Lebeuf, R.; Robert, F.; Schenk, K.; Landais, Y.: Diastereoselective Hydroamination Route to Hexahydroindoles
Martín, R.; Rivero, M. R.; Buchwald, S. L.: Pyrroles and Pyrazoles by a C-N Coupling-Hydroamination Sequence
Reddy, R. P.; Davies, H. M. L.: Enantioselective Synthesis of Oxazolidinones
Correa, A.; Tellitu, I.; Domínguez, E.; SanMartin, R.: Synthesis of Benzothiazol-3-ones
Lamer, A.-C. Le; Gouault, N.; David, M.; Boustie, J.; Uriac, P.: Fluorous-Phase Synthesis of α-Methyleneγ-lactones
Ichikawa, J.; Nadano, R.; Ito, N.: 4-Difluoromethylene-1-Pyrrolines by Intramolecular Heck Cyclization
Alajarín, M.; Ortín, M.-M.; Sánchez-Andrada, P.; Vidal, Á: Pericyclic Ring Closure of Ketenimines to Quinolinones
Guastavino, J. F.; Barolo, S. M.; Rossi, R. A.: An SRN1 Route to 3-Substituted and Fused Isoquinolin-1-(2H)-ones
Seregin, I. V.; Gevorgyan, V.: Gold-Catalyzed Synthesis of Pyrrole-Fused Heterocycles
Rassukana, Y. V.; Khomenko, E. A.; Onys’ko, P. P.; Sinitsa, A. D.: Synthesis of 1,3-Oxathiolan-5-ones and Benzoxathian-4-ones
Rios, R.; Sundén, H.; Ibrahem, I.; Zhao, G.-L.; Eriksson, L.; CÓrdova, A.: Chiral Benzothiopyrans by Organocatalysis
Correa, A.; Tellitu, I.; Domínguez, E.; SanMartin, R.: Metal-Free Synthesis of Indolines
Mross, G.; Holtz, E.; Langer, P.: 2-Alkenylfurans via Feist-Benary and Wittig Reactions
Li, Y.; Liang, F.; Bi, X.; Liu, Q.: Substituted Thiophenes via Intramolecular Thia-anti-Michael Addition

Issue 12/2006

Yu, R. T.; Rovis, T.: Indolizinone and Quinolizinone via Asymmetric [2+2+2] Cycloaddition
Chang, S.; Lee, M.; Jung, D. Y.; Yoo, E. J.; Cho, S. H.; Han, S. K.: Synthesis of Cyclic Amidines via Ru-Catalyzed Hydroamination
Dai, W.; Petersen, J. L.; Wang, K. K.: Synthesis of Tetracyclic ABCD Ring Cores of Camptothecins
Crowley, P. J.; Russell, S. E.; Reynolds, L. G.: Pyridazines by Acetylenic 1,2,4-Triazole Cyclization/Fragmentation
Kuninobu, Y.; Nishina, Y.; Nakagawa, C.; Takai, K.: Rhenium-Catalyzed Synthesis of Isobenzofurans
Bennasar, M. L.; Roca, T.; Monerris, M.; García-Díaz, D.: Heteroring Annulation Using TandemN-Acylamide Methylenation-RCM
Chen, W.; Yuan, X.-H.; Li, R.; Du, W.; Y, Wu; Ding, L.-S.; Cheng, Y.-C.: Organocatalytic and Stereoselective Synthesis of Bipyrazolidin-3-ones
Zanatta, N.; Schneider, J. M. F. M.; Schneider, P. H.; Wouters, A. D.; Bonacorso, H. G.; Martins, M. A. P.; Wessjohann, L. A.: Synthesis of Trifluoromethyl Pyrroles
Wan, X.; Xing, D.; Fang, Z.; Li, B.; Zhao, F.; K Zhang; Yang, L.; Shi, Z.: Phenethylamine Trimerization to Pyrroles
Deng, X.; Mani, N. S.: A Regioselective Cycloaddition Route to Pyrazoles
Ermolat’ev, D. S.; Giménez, V. N.; Babaev, E. V.; Van der Eycken, E.: Regiospecific 3-Arylation of Imidazo[1,2-a]pyrimidines
Banaszak, E.; Comoy, C.; Fort, Y.: Pyrano- and Oxepinopyridines by RCM
Yoshida, H.; Fukushima, H.; Ohshita, J.; Kunai, A.: Benzyne-Mediated Route to Benzoxazinones
Ichikawa, J.; Kaneko, M.; Yokota, M.; Itonaga, M.; Yokoyama, T.: Synthesis of Dihydrobenzoindazoles and Dihydrobenzoquinazolines
Ohkubo, M.; Hayashi, D.; Oikawa, D.; Fukuhara, K.; Okamoto, S.; Sato, F.: Titanium-Mediated Synthesis of N-Substituted 2-Arylpyrroles

Issue 11/2006

Blaszykowski, C.; Aktoudianakis, E.; Bressy, C.; Alberico, D.; Lautens, M.: Synthesis of Annulated N-Containing Heterocycles via C-H Activation
Morton, D.; Pearson, D.; Field, R. A.; Stockman, R. A.: Sulfur Ylide Mediated Asymmetric Synthesis of Aziridines from Sulfinylketimines
Asao, N.; Iso, K.; S, Yudha: Three-Component Synthesis of 1,2-Dihydroisoquinolines
Bhattacharya, A.; Cherukuri, S.; Plata, R. E.; Patel, N.; Tamez, V. Jr; Grosso, J. A.; Peddicord, M.; Palaniswamy, V. A.: One-Pot Synthesis of 3,4-Disubstituted Pyrrole-2-Esters
Aparicio, D.; Attanasi, A.; Filippone, P.; Ignacio, R.; Lillini, S.; Mantellini, F.; Palacios, F.; de Santos, J. Mlos: Synthesis of Pyrazines from Diaza-butadienes and 1,2-Diamines
Heller, S. T.; Natarajan, S. R.: A Classical but Short One-Pot Synthesis of Pyrazoles
Komeyama, K.; Morimoto, T.; Takaki, K.: Synthesis of Pyrrolidines from Aminoolefins by Hydroamination
McLaughlin, M.; Palucki, M.; Davies, I. W.: One-Pot Synthesis of Azaindoles and Indoles
Muhuhi, J.; Spaller, M. R.: Synthesis of Tetrahydroquinolines via an Intramolecular Aza-Diels-Alder Reaction
Kunetsky, R. A.; Dilman, A. D.; Struchkova, M. I.; Belyakov, P. A.; Tartakovsky, V. A.; Ioffe, S. L.: 1,3-Dipolar Cycloaddition Route to Isoxazoline N-Oxides
Lu, B. Z.; Zhao, W.; Wei, H.-X.; Dufour, M.; Farina, V.; Senanayake, C. H.: One-Pot Synthesis of 2,3-Disubstituted Indoles
Gwiazda, M.; Reissig, H.-U.: Synthesis of Highly Substituted Imidazoles from Lithiated Methoxyallene
Kanazawa, C.; Kamijo, S.; Yamamoto, Y.: Cross-Cycloaddition of Two Different Isocyanides to Imidazoles
Liu, J.; Shen, M.; Zhang, Y.; Li, G.; Khodabocus, A.; Rodriguez, S.; Qu, B.; Farina, V.; Senanayake, C. H.; Lu, B. Z.: Pd-Catalyzed Heteroannulation Route to Polycyclic Indoles
Sanz, R.; Fernández, Y.; Castroviejo, M. P.; Pérez, A.; Fañanás, F. J.: Synthesis of Carbazoles, Dibenzofurans and -thiophenes via Benzynes

Issue 10/2006

Harrison, T. J.; Kozak, J. A.; Corbella-Pané, M.; Dake, G. R.: Silver- and Gold-Catalyzed Pyrrole Synthesis
Zhang, Z.; Liu, C.; Kinder, R. E.; Han, X.; Qian, H.; Widenhoefer, R. A.: Synthesis of O- and N-Heterocycles by Au(I)-Catalyzed Allene Cyclizations
Wittmann, U.; Tranel, F.; Fröhlich, R.; Haufe, G.: Synthesis of Fluoropyridines from 4-(2-Fluoroallyl)oxazolones
Bellina, F.; Cauteruccio, S.; Rossi, R.: Palladium- and Copper-Catalyzed Arylation of Azoles
D’hooghe, M.; Vanlangendonck, T.; Törnroos, K. W.; De Kimpe, N.: Synthesis of cis-3,5-Disubstituted Morpholines from Aziridines
Herrera, A.; Martínez-Alvarez, R.; Chioua, R.; Almy, J.: Synthesis of Tetrahydropyrido[4,3-d]pyrimidines from 4-Piperidinone
Beccalli, E. M.; Broggini, G.; Martinelli, M.; Paladino, G.; Rossi, E.: Synthesis of Indolo-Fused Nitrogen Heterocycles
Yuan, Q.; Jian, S.-Z.; Wang, Y.-G.: Enantioselective Synthesis of β-Lactams Using Menthone Auxiliary Induction
Lin, Y.; Liu, J.-T.: α-Difluoromethylenephostones by Iodocyclization
Demydchuk, B. A.; Brovarets, V. S.; Chernega, A. N.; Rusanov, E. B.; Drach, B. S.: Synthesis of Benzimidazole-Fused Triazepines, Triazocines, and Triazonines
Zhu, Y.; Huang, S.; Wan, J.; Yan, L.; Pan, Y.; Wu, A.: Diastereoselective Routes to Thiazines, Oxazines and Pyranopyrimidines
Turunen, B. J.; Georg, G. I.: Synthesis of Cyclic and Bicyclic Enaminones from β-Amino Acids
Liu, X.-Y.; Li, C.-H.; Che, C.-M.: Synthesis of Thiazinanes and Pyrrolidinones via Au(I)-Catalyzed Hydroamination
Fritz, J. A.; Nakhla, J. S.; Wolfe, J. P.: Carboaminative Route to Imidazolidin-2-ones
Sañudo, M.; Marcaccini, S.; Basurto, S.; Torroba, T.: Synthesis of Cyclic Dipeptidyl Ureas via Ugi Three-Component Reaction

Issue 09/2006

de Figueiredo, R. M.; Fröhlich, R.; Christmann, M.: Synthesis of Chiral Azetidines
Inada, Y.; Yoshikawa, M.; Milton, M. D.; Nishibayashi, Y.; Uemura, S.: Ru-Catalyzed Propargylation of Aromatics and Heteroaromatics
Karpov, A. S.; Merkul, E.; Oeser, T.; Müller, T. J. J.: Multicomponent Synthesis of Substituted 3-Halofurans
Kim, H.; Lee, C.: Synthesis of Fused Piperidines by Rhodium-Catalyzed Cyclization
Oh, C. H.; Reddy, V. R.; Kim, A.; Rhim, C. Y.: Synthesis of Substituted Furans by Pt-Catalyzed Cyclization of Enynones
Ambrogio, I.; Cacchi, S.; Fabrizi, G.: Pd-Catalyzed Synthesis of 2-(Aminomethyl)indoles
Natarajan, S. R.; Chen, M.-H.; Heller, S. T.; Tynebor, R. M.; Crawford, E. M.; Minxiang, C.; Kaizheng, H.; Dong, J.; Hu, B.; Hao, W.; Chen, S.-H.: Lateral Metallation-Cycloannulation Synthesis of 2H-quinolizin-2-ones
Jurík, V.; Wilhelm, R.: Chiral Imidazolinium Salts: Lewis Acids, Shift Reagents and Ionic Liquids
Sakai, N.; Ridder, A.; Hartwig, J. F.: Synthesis of Tropenes by Pd-Catalyzed Double Hydroamination
De Benassuti, L.; Buttero, P. Del; Molteni, G.: Stereoselective Synthesis of Enantiopure Pyrrolo[3,4-c]pyrazoles
Smith III, A. B.; Kürti, L.; Davulcu, A. H.: Modular Synthesis of Fused Indole Derivatives
Lin, L.; Fan, Q.; Qin, B.; Feng, X.: Enantioselective Cu-Catalyzed Hetero-Diels-Alder Synthesis of δ-Lactones
Rosiak, A.; Christoffers, J.: A Short Synthesis of Unsymmetrical 2,3-Dihydrothiopyran-4-ones
Patil, N. T.; Lutete, L. M.; Wu, H.; Pahadi, N. K.; Gridnev, I. D.; Yamamoto, Y.: Asymmetric Synthesis of O- and N-Heterocycles by Intramolecular Hydroamination and -alkoxylation
Stanislawski, P. C.; Willis, A. C.; Banwell, M. G.: Synthesis of 1,1-Spirocyclic Tetrahydroisoquinoline Systems

Issue 08/2006

Lagisetty, P.; Russon, L. M.; Lakshman, M. K.: Synthesis of C6-Azolyl Purine Nucleosides
Barluenga, J.; Garciá-Rodrígez, J.; Martínez, S.; Suárez-Sobrino, A. L.; Tomás, M.: Synthesis of Fused Imidazoles from Fischer Carbenes and 1,4-Diazafulvenes
Binder, J. T.; Kirsch, S. F.: Silver- and Gold-Catalyzed Synthesis of Highly Substituted Pyrroles
Yu, Y.; Stephenson, G. A.; Mitchell, D.: Synthesis of 3-Benzazepinones via Palladium-Catalyzed Hydroamination
Burke, P. J.; Rigby, J. H.: Synthesis of Pyrroloindoles from Indole Isocyanates
Ren, H.; Knochel, P.: C-H Activation Approach to Condensed N-Heterocycles
Trost, B. M.; Machacek, M. R.; Faulk, B. D.: Asymmetric Synthesis of N- and O-Heterocycles Using Sequential Ru-Pd Catalysis
Chen, W.; Su, C.; Huang, X.: A New Approach to Substituted Pyrrolotriazoles
More, S. V.; Sastry, M. N. V.; Yao, C.-F.: Three-Component Synthesis of Pyrano- and Furanoquinolines
Zhou, W.-J.; Ji, S.-J.; Shen, Z.-L.: Synthesis of Ferrocenyl Pyridines
Wang, Y.; Burton, D. J.: Synthesis of Fluorinated Pyrones
DiMauro, E. F.; Vitullo, J. R.: Synthesis and Transformations of Fused Bicyclic Heteroaryl Borates
Ludek, O. R.; Meier, C.: Regioselective O- and N-Alkylation of Pyrimidine Nucleosides via the Mitsunobu Reaction
Handy, S. T.; Sabatini, J. J.: Regioselective Double Suzuki Cross Coupling of Dibromopyrroles
Moonen, K.; Dieltiens, N.; Stevens, C. V.: Synthesis of 2-Phosphonopyrroles

Issue 07/2006

Yang, X.; Luo, S.; Fang, F.; Liu, P.; Lu, Y.; He, M.; Zhai, H.: Intramolecular [3+2] Cycloaddition Approach to Nicotine Analogues
Neogi, A.; Majhi, T. P.; Mukhopadhyay, R.; Chattopadhyay, P.: Benzoxazocines by Palladium-Catalyzed Intramolecular Amination
Toffano, M.; Dobrota, C.; Fiaud, J.-C.: Catalytic Pd-Mediated Approach to Enantiopure Phosphorus Ligands
Couty, S.; Meyer, C.; Cossy, J.: Combined Heck-Suzuki Reactions in a Synthesis of Lennoxamine
Zhoa, A.; Njogu, M. N.; Pittman, C. U.: Synthesis of Chiral Oxazolo and Thiazolo Isoquinolinones
Deprez, N. R.; Kalyani, D.; Krause, A.; Sanford, M. S.: 2-Arylation of Indoles using Diaryliodonium Salts
IJsselstijn, M.; Cintrat, J. C.: Synthesis of 4-Amino Triazoles by Huisgen [3+2] Cycloaddition
Lee, C. K. Y.; Herlt, A. J.; Simpson, G. W.; Willis, A. C.; Easton, C. J.: Asymmetric Synthesis of Δ2-Isoxazolines
Williams, J. T.; Bahia, P. S.; Kariuki, B. M.; Spencer, N.; Philp, D.; Snaith, J. S.: Synthesis of cis- or trans-3,4-Disubstituted Piperidines
Lesma, G.; Danieli, B.; Saccheti, A.; Silvani, A.: Synthesis of Cyclic β-Amino Acids by RCM
Denmark, S. E.; Fan, Y.: Diastereoselective Approach to Non-racemic Bipyridine bis-N-Oxides
Movassaghi, M.; Hill, M. D.: Pyridine and Quinoline Derivatives via Ru-Catalyzed Cyclization of Azadienynes
Langlois, N.; Nguyen, B. K. Le; Retailleau, P.; Tarnus, C.; Salomon, E.: Synthesis of Indolizidines Bearing Quaternary Stereocenters
Pastre, J. C.; Correia, C. R. D.: Heck Reaction of Acrylates with Arenediazonium Tetrafluoroborates
Herrera, A.; Martínez-Alvarez, R.; Ramiro, P.; Molero, D.; Almy, J.: Synthesis of 2,5- and 2,4,5-Substituted 1,3-Oxazoles

Issue 06/2006

Youn, S. W.: Gold-Catalyzed Pictet-Spengler Reactions
Kong, A.; Han, X.; Lu, X.: Palladium(II)-Catalyzed Cyclization of 3-(3′-Alkenyl)indoles to Carbazoles
Pigge, F. C.; Coniglio, J. J.; Dalvi, R.: Dearomatization Route to Cyclohexadienone Spirolactams
Reddy, L. R.; Corey, E. J.: Synthesis of a Fused β-Lactone via Pyridine-Assisted [2+2] Cycloaddition
Taylor, A. M.; Schreiber, S. L.: Asymmetric Alkynylation of Isoquinoline Iminium Salts
Duggineni, S.; Sawant, D.; Saha, B.; Kundu, B.: Pictet-Spengler Synthesis of Thiazolo- and Pyrazolo-quinolines
Sawant, D.; Kumar, R.; Maulik, P. R.; Kundu, B.: Synthesis of Indazole Derivatives Involving Aryl Nitrene Species
Parenty, A. D. C.; Guthrie, K. M.; Song, Y.-F.; Smith, L. V.; Burkholder, E.; Cronin, L.: One-Pot Synthesis of Imidazophenanthridinium Salts
Kusama, H.; Miyashita, Y.; Takaya, J.; Iwasawa, N.: Metal-Mediated Heterocyclic Annulation to Indolopyrrolidines
Peng, Z.-H.; Journet, M.; Humphrey, G.: Palladium-Catalyzed C-N Bond Coupling Reactions. Aminopyrimidine Synthesis
Liu, C.; Widenhoefer, R. A.: Pd(II)-Catalyzed Synthesis of Tetrahydrocarbazoles and 3-Substituted Indoles
Liu, Z.; Rainier, J. D.: Synthesis of Perhydroindolines by Ring-Opening/Ring-Closing Metathesis
Adib, M.; Sheibani, E.; Mostofi, M.; Ghanbary, K.; Bijanzadeh, H. R.: Three-Component Diastereoselective Synthesis of Imidazooxazines
Evans, P. A.; Lai, K. W.; Zhang, H.-R.; Huffman, J. C.: Rhodium-Catalyzed N-Allylation of Thymine
Park, D. Y.; Lee, M. J.; Kim, T. H.; Kim, J. N.: Synthesis of 3,4,5-Trisubstituted Pyridines from Baylis-Hillman Adducts

Issue 05/2006

Nakamura, M.; Ilies, L.; Otsubo, S.; Nakamura, E.: Transformations of 3-Zinciobenzofurans and 3-Zincioindoles
Cropper, E. L.; White, A. J. P.; Ford, A.; Hii, K. K(M): Regioselective Synthesis of Dihydrophenanthridines, Benzazepinones and Benzoazocinones
Maulide, N.; Markó, I. E.: Stereoselective Synthesis of Bicyclic Lactones from Furans
Evindar, G.; Batey, R. A.: Copper-Catalyzed C-O and C-S Cross-Coupling Routes to Benzoxazoles and -thiazoles
White, J. D.; Ihle, D. C.: Synthesis of Spiropyrrolines via Photocycloaddition-Retro-Mannich Reactions
Wiedemann, S. H.; Ellman, J. A.; Bergman, R. G.: Rh-Catalyzed C-H Addition of Quinazolines to Alkenes
Ferrer, C.; Echavarren, A. M.: Gold-Catalyzed Synthesis of 6-, 7- and 8-Membered Heteroannulated Indoles
Zhang, J.; Zhang, Y.; Schnatter, W. F. K.; Herndon, J. W.: Fischer Carbene Complexes in Annulation Reactions to Heterocyclic Enyne Aldehydes
Lee, S. J.; Beak, P.: (-)-Sparteine-Mediated Asymmetric Synthesis of Polysubstituted Azepanes
Voskressensky, L. G.; Borisova, T. N.; Kostenev, I. S.; Kulikova, L. N.; Varlamov, A. V.: Tetrahydropyridine to Azocine Ring-Expansion Reactions
Zhao, L.; Liang, F.; Bi, X.; Sun, S.; Liu, Q.: Dihydropyrido[2,3-d]pyrimidines by Double [5+1] Annulation
Zulys, A.; Dochnahl, M.; Hollmann, D.; Löhnwitz, K.; Herrmann, J.-S.; Roesky, P. W.; Blechert, S.: Intramolecular Hydroamination Route to Heterocycles
Lee, J. M.; Chang, S.: Lactone Heteroannulation by Intramolecular C-H Bond Activation
Kiselyov, A. S.: Synthesis of Fluoro Isoquinolines via Quinodimethide (QM) Intermediates
Comins, D. L.; Smith, E. D.: C-5 Functionalization of (S)-Nicotine via 1-Acyl-1,4-dihydronicotine

Issue 04/2006

Chowdhury, C.; Mandal, S. B.; Achari, B.: Synthesis of Triazoles (I): Sequential Sonogashira Coupling and [2+3] Cycloaddition
Gracias, V.; Darczak, D.; Gasiecki, A. F.; Djuric, S. W.: Synthesis of Triazoles (II): van Leusen Imidazole Synthesis-Intramolecular [2+3] Cycloaddition
Yanai, H.; Taguchi, T.: Synthesis of Triazoles (III): Azidation of Dialkoxyacetylenes-Intramolecular [2+3] Cycloaddition
Rossi, E.; Abbiati, G.; Canevari, V.; Celentano, G.; Magri, E.: Synthesis of 2-Substituted Indoles by Cross-Coupling Reactions
Kuninobu, Y.; Tokunaga, Y.; Kawata, A.; Takai, K.: Synthesis of Phthalimidines via C-H Bond Activation
Linnepe, P.; Schmidt, A. M.; Eilbracht, P.: Synthesis of Indoles by a Combined Hydroformylation-Fischer Indolization Route
Handy, S. T.; Zhang, Y.: Predicting Regioselectivity in Cross-Coupling of Polyhaloheteroaromatics
Young, D. W.; Comins, D. L.: Synthesis of Dihydropyridones Involving Directed ortho-Metallation
Moonen, K.; Stevens, C. V.: Synthesis of Phosphono-β-Lactams
Tanaka, S.; Yasuda, M.; Baba, A.: Synthesis of Substituted Quinolines under Aerobic Conditions
Deng, X.; Mani, N. S.: Sonogashira-Mediated Synthesis of 4-Aryl-5-Pyrimidinylimidazoles
Wardrop, D. J.; Burge, M. S.: Stereocontrolled Synthesis of 4-6-Ring Lactams
Kuninobu, Y.; Nishimura, S.; Takai, K.: Synthesis of 4H-Pyrido[1,2-a]pyrimidin-4-ones
Mkhalid, I. A. I.; Coventry, D. N.; Albesa-Jove, D.; Batsanov, A. S.; Howard, J. A. K.; Perutz, R. N.; Marder, T. B.: Synthesis of Pyridyl and Pyridazyl Boropinacolates by Ir-Catalyzed C-H activation

Issue 03/2006

Dondas, H. A.; Fishwick, C. W. G.; Gai, X.; Grigg, R.; Kilner, C.; Dumrongchai, N.; Kongkathip, B.; Kongkathip, N.; Polysuk, C.; Sridharan, V.: Synthesis of Pyrrolidinyl, Pyrazolidinyl, and Isoxazolidinyl Isoquinolines
Korivi, R. P.; Cheng, C.-H.: Synthesis of Isoquinolines by Nickel-Catalyzed Heteroannulation
Lefoix, M.; Daillant, J.-P.; Mérour, J.-Y.; Gillaizeau, I.; Coudert, G.: Regioselective Metallative Functionalization of 5-Azaindole
Calvet, G.; Blanchard, N.; Kouklovsky, C.: Synthesis of Polysubstituted Pyrroles via Dihydro-1,2-oxazines
Tanaka, K.; Kitamura, M.; Narasaka, K.: Synthesis of α-Carbolines
Huynh, M. H. V.; Hiskey, M. A.; Chavez, D. E.; Gilardi, R. D.: Tetraazapentalenes: Formation and Rearrangement
Strat, F. Le; Vallette, H.; Toupet, L.; Maddaluno, J.: Synthesis of Complex Condensed Heterocycles by Diels-Alder Reactions
Lu, K.; Luo, T.; Xiang, Z.; You, Z.; Fathi, R.; Chen, J.; Yang, Z.: Multi-Component Synthesis of 5H-Furoisoindole and Pyrrolo[3,4-f]indole Derivatives
Hamasaki, A.; Ducray, R.; Boger, D. L.: Synthesis of Pyridazines by a Diels-Alder Strategy
Kuznetsov, N. Y.; Khrustalev, V. N.; Godovikov, I. A.; Bubnov, Y. N.: Bridged Azabicycles by Ring-Closing Metathesis
Garner, P.; Kaniskan, H. Ü: Synthesis of 1H-Furo- and Pyrrolo[3,4-c]pyrrole Derivatives by Multicomponent Reactions
Loones, K. T. J.; Maes, B. U. W.; Meyers, C.; Deruytter, J.: Synthesis of Imidazoles by Pd- and Cu-Catalyzed C-N Bond Formation
Dunne, K. S.; Bisaro, F.; Odell, B.; Paris, J.-M.; Gouverneur, V.: Synthesis of P-Stereogenic Oxaphosphacyclohexene-1-oxides by Ring-Closing Metathesis
Mukai, C.; Takahashi, Y.: 2,3-Disubstituted Indoles by Stille Cross- Coupling Reaction
McElhinney, A. D.; Marsden, S. P.: Synthesis of Indolizines as Illustrated in Alkaloid Construction

Issue 02/2006

Xu, H.-W.; Li, G.-Y.; Wong, M.-K.; Che, C.-M.: Chiral Pyrrolines via Asymmetric 1,3-Dipolar Cycloaddition Reactions
Tsang, W. C. P.; Zheng, N.; Buchwald, S. L.: Synthesis of Carbazoles by Tandem C-H Activation and Buchwald-Hartwig Amination
Feldman, A. K.; Colasson, B.; Sharpless, K. B.; Fokin, V. V.: A Concept for the Regioselective Synthesis of 1,2,3-Triazoles
Konno, T.; Chae, J.; Miyabe, T.; Ishihara, T.: Regioselective Synthesis of 4-Fluoroalkyl Isoquinolines
Duvelleroy, D.; Perrio, C.; Parisel, O.; Lasne, M.-C.: Indium(III)-Mediated Synthesis of Quinoline-4-carboxylic Acid Derivatives
Ohno, H.; Yamamoto, M.; Iuchi, M.; Tanaka, T.: Aromatizing Route to Benzo-, Benzofuranyl-, and N-Tosylindolenyl-isoindolines
Corey, E. J.; Tian, Y.: Synthesis of Azabiaryls by a non-Cross-Coupling Method
Bressy, C.; Alberico, D.; Lautens, M.: A C-H Insertion Route to Fused Indoles
Waldo, J. P.; Larock, R. C.: Convenient Synthesis of Isoxazoles
Kazmaier, U.; Ackermann, S.: Synthesis of Endothiopeptides via Ugi Reaction and their Conversion to Thiazoles
Zhang, L.: Synthesis of Functionalized 2,3-Indoline-Fused Cyclobutanes
Sainz, Y. F.; Raw, S. A.; Taylor, R. J. K.: Multisubstituted Pyridines from 1,2,4-Triazines by Diels-Alder Chemistry
Berkessel, A.; Cleemann, F.; Mukherjee, S.: Oxazinones as Synthetic Intermediates for Enantiomerically Pure β-Amino Acids
Février, F. C.; Smith, E. D.; Comins, D. L.: Regioselective Lithiation of (S)-Nicotine

Issue 01/2006

Zhao, J.; Larock, R. C.: A Benzyne Route to Xanthones and Thioxanthones
González-Vera, J. A.; García-López, M. T.; Herranz, R.: Synthesis of Pyrrolo-imidazoindoles from Tryptophan Methyl Ester
Ney, J. E.; Hay, M. B.; Yang, Q.; Wolfe, J.-P.: Palladium-Catalyzed Stereoselective Synthesis of 2-Allylpyrrolidines
Clochard, M.; Grundy, J.; Donnadieu, B.; Mathey, F.: Synthesis of 3-Acylphospholes
Yanada, R.; Obika, S.; Kobayashi, Y.; Inokuma, T.; Oyama, M.; Yanada, K.; Takemoto, Y.: Synthesis of 3-Benzylideneoxindoles
Larquetoux, L.; Ouhamou, N.; Chiaroni, A.; Six, Y.: Titanium(IV)-Catalyzed Synthesis of 3-Azabicyclo[3.1.0]hexane Derivatives
Rosas, N.; Sharma, P.; Arellano, I.; Ramírez, M.; Pérez, D.; Hernández, S.; Cabera, A.: Fe(II)-Mediated Synthesis of 5-Carboxy-3-pyrrolin-2-ones
Frisch, K.; Landa, A.; Saaby, S.; Jørgensen, K. A.: Enantioselective Synthesis of 1,2-Dihydroisoquinolines and 1,2-Dihydrophthalazines
Kaloko Jr, J.; Hayford, A.: Synthesis of Indolizine Derivatives by Electrocyclization
Hiramatsu, N.; Takahashi, N.; Noyori, R.; Mori, Y.: Stereoselective Synthesis of Fused Tetrahydropyrans
Markgraf, J. H.; Dowst, A. A.; Hensley, L. A.; Jakobsche, C. E.; Kaltner, C. J.; Webb, P. J.; Zimmerman, P. W.: A Versatile Synthesis of Benzacanthinones by Intramolecular Radical Coupling
Ahmed, M. S. Mohamed; Kobayashi, K.; Mori, A.: Palladium-Catalyzed Multicomponent Synthesis of Pyrazoles and Isoxazoles
Welter, C.; Moreno, R. M.; Streiff, S.; Helmchen, G.: Synthesis of (+)(R)- and (-)(S)-Nicotine via Enantioselective Ir-Catalyzed Allylic Amination
Dziedzic, M.; Lipner, G.; Illangua, J. M.; Furman, B.: Synthesis of Dihydropyridinones and Hexahydroindolizin-7(1H)-one Derivatives
Adamo, M. F. A.; Donati, D.; Duffy, E. F.; Sarti-Fantoni, P.: Diastereoselective Synthesis of Spiroisoxazolines

Issue 03/2005

Khedkar, V.; Tillack, A.; Michalik, M.; Beller, M.: New Synthesis of Fischer Indole Hydrazone Intermediates
Nakano, H.; Tsugawa, N.; Fujita, R.: Enantioselective Diels-Alder Route to Isoquinuclidines
Arcadi, A.; Cacchi, S.; Fabrizi, G.; Marinelli, F.; Parisi, L. M.: Regioselective Synthesis of 2-Substituted 3-Acylindoles
Rudler, H.; Denise, B.; Xu, Y.; Parlier, A.; Vaissermann, J.: Synthesis of Bridged Bicyclic Lactones of Dihydroheteroaromatics
Fiorelli, C.; Marchioro, C.; Martelli, G.; Monari, M.; Savoia, D.: Stereoselective Iodine-Mediated Synthesis of Diazabicyclo[2.2.1]heptanes
Sakoda, K.; Mihara, J.; Ichikawa, J.: Synthesis of Fluoropyrroles
Sromek, A. W.; Rubina, M.; Gevorgyan, V.: Au(III)-Catalyzed Synthesis of Polysubstituted Halofurans
Rejzek, M.; Stockman, R. A.; van Maarseveen, J. H.; Hughes, D. L.: A Cascade Azide Formation, Cycloaddition and Michael Addition to a Quinolizidine
Revesz, L.; Blum, E.; Wicki, R.: Synthesis of Bicyclic O- and N-Bridged Piperazines
Al-Harrasi, A.; Reissig, H.-U.: [3+3] Cycloaddition Approach to the Synthesis of Substituted Pyrans and Oxapanes
Saaby, S.; Baxendale, I. R.; Ley, S. V.: [2+2+2] Cyclotrimerization to Benzofurans, Benzothiophenes and Isoindoles
Hughes, C. C.; Miller, A. K.; Trauner, D.: Electrochemical Synthesis of Oxygenated Dihydrofurans
Pan, Y.; Holmes, C. P.; Tumelty, D.: Negishi Cross Coupling Route to N-Unsubstituted α,α-Difluorohomophthalimides
Alcaide, B.; Almendros, P.; Rodríquez-Acebes, R.: Synthesis of Oxindole and β-Lactam Spiro-ethers
Laitar, D. S.; Müller, P.; Gray, T. G.; Sadighi, P.: The Synthesis of an N-Heterocyclic Carbene-Stabilized Gold(I) Fluoride

Issue 02/2005

Nicolaou, K. C.; Lee, S. H.; Estrada, A. A.; Zak, M.: Construction of Substituted N-Hydroxyindoles
Land, E. J.; Perona, A.; Ramsden, C. A.; Riley, P. A.: Synthesis of Spiroheterocyclic Cyclohexadienones of Biological Interest
Gorin, D. J.; Davis, N. R.; Toste, F. D.: Regiospecific Substituted Pyrroles Synthesis
Moore, J. E.; Davis, M. W.; Goodenough, K. M.; Wybrow, R. A. J.; York, M.; Johnson, C. N.; Harrity, J. P. A.: Isoxazole Boronic Esters
Ye, M.-C.; Li, B.; Zhou, J.; Sun, X.-L.; Tang, Y.: Modular Synthesis of Tris(oxazolines)
Langer, P.; Bodtke, A.; Saleh, N. N. R.; Görls, H.; Schreiner, P. R.: Synthesis and Physiochemical Properties of a New Heterocyclic System
Abbiati, G.; Arcadi, A.; Canevari, V.; Capezzuto, L.; Rossi, E.: Carbonylative Sonogashira Synthesis of Quinolines and Naphthyridines
Yamamoto, Y.; Hayashi, H.; Saigoku, T.; Nishiyama, H.: Polycyclic Pyrrole Derivatives
Taguchi, K.; Sakaguchi, S.; Ishii, Y.: Green Chemistry: Synthesis of Quinolines
Zabawa, T. P.; Kasi, D.; Chemler, S. R.: Intramolecular Hydroamination Route to Thiazolidine-1,1-dioxides
Shabashov, D.; Daugulis, O.: Aryl-Aryl and Aryl-Alkyl Coupling via N-Heterocycle C-H Activation
Charles, M. D.; Schultz, P.; Buchwald, S. L.: Synthesis of Heteroaromatic Amines by C-N Cross-Coupling
Oi, S.; Sakai, K.; Inoue, Y.: (Z)-β-Arylation of 2-Alkenylpyridines by C-H Activation Process
Fukada, T.; Akashima, H.; Iwao, M.: Benzene Ring Functionalization of Indoles by Iterative Directed peri and ortho Lithiation
Stroh, C.; Mayor, M.; von Hänisch, C.: Synthesis of Stable Organic Radicals by Suzuki-Miyaura Cross-Coupling

Issue 01/2005

Chung, J. Y. L.; Cvetovich, R.; Amato, J.; McWilliams, J. C.; Reamer, R.; DiMichele, L.: Enantioselective Pyrrolidine Synthesis
Cutri, S.; Diez, A.; Bonin, M.; Micouin, L.; Husson, H.-P.: Regio- and Stereoselective Synthesis of Structurally Diverse Polycyclic Indolyldiamines
Yi, C. S.; Yun, S. Y.; Guzei, I. A.: Regioselective Hydroamination for the Synthesis of Tricyclic Quinolines
Denmark, S. E.; Montgomery, J. I.: Synthesis of a Highly Strained Heterocycle Involving a Nitro Acetal to Aminal Rearrangement
Lin, Y. S.; Liu, C. W.; Tsai, T. Y. R.: A Heterocyclic N-Oxide-Mediated Morita-Baylis-Hillman Reaction
Ohno, H.; Miyamura, K.; Mizutani, T.; Kadoh, Y.; Takeoka, Y.; Hamaguchi, H.; Tanaka, T.: Tandem Cyclization of Allenenes to Tri- and Tetracyclic Heterocycles
Grimster, N. P.; Gauntlett, C.; Godfrey, C. R. A.; Gaunt, M. J.: Palladium-Catalyzed Regioselective Direct C-2 and C-3 Functionalization of Indoles
Wang, Z.; Bao, W.; Jiang, Y.: Synthesis of Aza-Stilbenes via an Ullmann C-N Coupling Reaction in Ionic Liquids
Cottineau, B.; O’Shea, D. F.: Carbolithiation of Vinyl Pyridines as a Route to 7-Azaindoles
Soderberg, B. C. G.; Hubbard, J. W.; Rector, S. R.; O’Neil, S. N.: Synthesis of Fused Indoles by Sequential Heck Reaction and N-Heteroannulation
Kim, M. S.; Kim, Y.-W.; Hahm, H. S.; Jang, J. W.; Lee, W. K.; Ha, H.-J.: A Stereospecific Synthesis of Imidazolidin-2-ones from Aziridine-2-carboxylates and Isocyanates
Zhao, J.; Hartwig, J. F.: Ruthenium-Catalyzed Cyclization of Diols to Lactones
Sommen, G. L.; Linden, A.; Heimgartner, H.: Cycloaddition of Carbodiimides to Selenazetidines
Zhuang, W.; Hazell, R. G.; Jørgensen, K. A.: Enantioselective Synthesis of Tryptamines and Tetrahydro-β-carbolines
Nakao, Y.; Imanaka, H.; Sahoo, A. K.; Yada, A.; Hiyama, T.: Tetraorganosilicon Reagents for Cross-Coupling Reactions

Issue 00/2005

Padwa, A.; Lynch, S.; Mejìa-Oneto, J.; Zhang, H.: Cycloaddition Chemistry of 2-Vinyl-Substi­-tuted Indoles and Related Heteroaromatics
Piechaczyk, O.; Doux, M.; Ricard, L.; Floch, P. le: Synthesis of 1-Phosphabarrelene Phosphine Sulfide Substituted Palladium(II) Complexes
Kawasaki, T.; Ogawa, A.; Terashima, R.; Saheki, T.; Ban, N.; Sekiguchi, H.; Sakaguchi, K.; Sakamoto, M.: Synthesis of Diversely Functionalized Hexa­­-hydropyrrolo[2,3-b]indoles
Jacquot, D. E. N.; Zöllinger, M.; Lindel, T.: Total Synthesis of the Marine Natural Product rac-Dibromophakellstatin
Jezek, E.; Schall, A.; Kreitmeier, P.; Resier, O.: Radical-Mediated Synthesis of Sesquiterpene Lactones
Smitrovich, J. H.; Davies, I. W.: Catalytic C-H Functionalization Driven by CO as a Stoichiometric Reductant - Application to Carbazole Synthesis
Iwasaki, T.; Kohinata, Y.; Nishide, H.: Poly(thiaheterohelicene): A Stiff Conjugated Helical Polymer Comprised of Fused Benzothiophene Rings
Ishida, S.; Nishinaga, T.; West, R.; Komatsu, K.: Generation and Aromaticity of 2-Silaimidazo-lium Ion, a New π-Conjugated Silylium Ion
Capito, E.; Brown, J.; Ricci, A.: Directed Palladation: Fine Tuning Permits the Catalytic 2-Alkenylation of Indols
D’hooghe, M.; Rottier, M.; Jolie, R.; De Kimpe, N.: Coupling of 1-Alkyl-2-(bromomethyl)aziri­-dines with Lithium Dialkylcuprates towards 1,2-Dialkylaziridines
Klumpp, D. A.; Kindelin, P. J.; Li, A.: Superacid-Promoted Reactions of Pyrazole­-carboxaldehydes and the Role of Dicationic Electrophiles
Adamo, M. F. A.; Baldwin, J. E.; Adlington, R. M.: Bis-acetylenic Ketones for the Synthesis of 1,2,4-Triazepine and Oxatriazaindenone Cores
Ma, S.; Yu, Z.; Gu, Z.: An Efficient Synthesis of Bibutenolides from 2,3-Allenoic Acids
Oi, S.; Aizawa, E.; Ogino, Y.; Inoue, Y.: Ru-Catalyzed ortho-Selective Direct Cross-Coupling Reaction of 2-Aryloxazolines and 2-Arylimidazolines
Martin, D.; Baceiredo, A.; Gornitzka, H.; Schoeller, W.; Bertrand, G.: A Stable P-Heterocyclic Carbene