Synthesis

Issue 20/2014

Tan, Wei Wen; Hou, Xiaoya; Yoshikai, Naohiko: Pd(II)/Bu₄NBr/DMSO Catalytic System for Practical Synthesis of Indoles and Pyrroles from Imines through Aerobic Dehydrogenative Cyclization

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Issue 17/2014

Danoun, Grégory; Bayarmagnai, Bilguun; Grünberg, Matthias F.; Matheis, Christian; Risto, Eugen; Gooßen, Lukas J.: Sandmeyer Trifluoromethylation

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Issue 16/2014

Wang, Xi; Xu, Yan; Zhou, Yujing; Zhang, Yan; Wang, Jianbo: Conversion of Aromatic Amino into Trifluoromethyl Groups through a Sandmeyer­-Type Transformation

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Issue 15/2014

Schmidt, Anastasia; Maiterth, Elias; Hilt, Gerhard: Cobalt-Catalysed Transformations of 1,3,5-Hexatrienes on a Large Scale

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Issue 14/2014

Santosh Kumar, S. Chandrappa; Vijendra Kumar, Nanjundaswamy; Srinivas, Pullabhatla; Bettadaiah, Bheemanakere Kempaiah: A Convenient Practical Synthesis of Alkyl and Aryl Oxime Esters

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Issue 12/2014

Iwasaki, Takanori; Takagawa, Hiroaki; Okamoto, Kanako; Singh, Surya Prakash; Kuniyasu, Hitoshi; Kambe, Nobuaki: The Cobalt-Catalyzed Cross-Coupling Reaction of Alkyl Halides with Alkyl Grignard Reagents: A New Route to Constructing Quaternary Carbon Centers­

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Issue 11/2014

Hafner, Andreas; Hussal, Christoph; Bräse, Stefan: Preparation of Aromatic Triazenes and Their Application in Silver-Mediated Perfluoroalkylation Reactions

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Issue 10/2014

León, Thierry; Quinio, Pauline; Chen, Quan; Knochel, Paul: BF₃-Mediated Oxidative Cross-Coupling of Pyridines with Alkynyllithium Reagents and Further Reductive Functionalizations of the Pyridine Scaffold

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Issue 09/2014

Theunissen, Cédric; Lecomte, Morgan; Jouvin, Kévin; Laouiti, Anouar; Guissart, Céline; Heimburger, Jérémy; Loire, Estelle; Evano, Gwilherm: Convenient and Practical Alkynylation of Heteronucleophiles with Copper Acetylides

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Issue 08/2014

Wekesa, Francis S.; Phadke, Neha; Jahier, Claire; Cordes, David B.; Findlater, Michael: A Simple and Convenient Method for the Synthesis of N,N-Diaryl Tertiary Amines

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Issue 07/2014

Tsutsumi, Ryosuke; Kim, Seonwoo; Uraguchi, Daisuke; Ooi, Takashi: The Practical Preparation of Chiral N-Sulfonyl Oxaziridines via Catalytic Asymmetric Payne Oxidation

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Issue 06/2014

Soliman, Sameh E.; Kováč, Pavol: Practical Synthesis of Building Blocks for Oligosaccharides Containing the β-d-Galp-(1→3)-β-d-GlcpNAc Motif

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Issue 05/2014

Weseliński, Łukasz J.; Luebke, Ryan; Eddaoudi, Mohamed: A Convenient Preparation of 9H-Carbazole-3,6-dicarbonitrile and 9H-Carbazole-3,6-dicarboxylic Acid

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Issue 04/2014

Zajdlik, Adam; He, Zhi; St Denis, Jeffrey D.; Yudin, Andrei K.: Efficient Preparation of α-Aminoboronic Acid Derivatives via Boroalkyl Group Migration

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Issue 03/2014

Klatt, Thomas; Blümke, Tobias D.; Ganiek, Maximilian A.; Knochel, Paul: Synthesis of 1,2-Dimetallic Compounds via Direct Insertion of Zinc Powder in the Presence of InCl₃: Synthesis of ortho-Bis-functionalized Aromatics

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Issue 02/2014

Woydziak, Zachary R.; Fu, Liqiang; Peterson, Blake R.: Efficient and Scalable Synthesis of 4-Carboxy-Pennsylvania Green Methyl Ester: A Hydrophobic Building Block for Fluorescent Molecular Probes

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Nolla-Saltiel, Roberto; Carrillo-Arcos, Ulises Alonso; Porcel, Susana: Silver Acetate Mediated Acetoxylations of Alkyl Halides

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Issue 01/2014

Jiao, Lei; Bach, Thorsten: Regioselective Direct C–H Alkylation of NH Indoles and Pyrroles by a Palladium/Norbornene-Cocatalyzed Process

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Issue 24/2013

Koch, Niklas; Mazik, Monika: Synthesis of Tripodal and Hexapodal Pyrazole- and Benzimidazole-Bearing Compounds

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Issue 23/2013

Miersch, Anne; Kohlmeyer, Corinna; Hilt, Gerhard: Zinc-Mediated Regiodiverse Synthesis of Vinyl Bromide Derivatives and Their in situ Palladium-Catalysed Cross-Coupling Reactions

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Issue 22/2013

Buonomo, Joseph A.; Everson, Daniel A.; Weix, Daniel J.: Substituted 2,2′-Bipyridines by Nickel Catalysis: 4,4′-Di-tert-butyl-2,2′-bipyridine

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Issue 21/2013

Matsukawa, Satoru; Tsukamoto, Kumiko; Yasuda, Shiori; Harada, Takeru: An Efficient Method for Opening N-Tosylaziridines with Silylated Nucleo­philes by Using Polystyrene-Supported 1,5,7-Triazabicyclo[4.4.0]dec-5-ene as a Reusable Organocatalyst

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Issue 20/2013

Roseblade, Stephen J.; Casas-Arcé, Eva; Nettekoven, Ulrike; Gazić Smilović, Ivana; Zanotti-Gerosa, Antonio; Časar, Zdenko: A Practical Synthetic Approach to Chiral (α-Chloroalkyl)boronic Esters via Iridium-Catalyzed Chemoselective Hydrogenation of Chloro-Substituted Alkenyl Boronates

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Issue 19/2013

Maksymowicz, Rebecca M.; Sidera, Mireia; Roth, Philippe M. C.; Fletcher, Stephen P.: A Convenient Catalytic Asymmetric Conjugate Addition Reaction to Enones Using Alkylzirconium Reagents

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Issue 18/2013

Noole, Artur; Malkov, Andrei V.; Kanger, Tõnis: Asymmetric Organocatalytic Synthesis of Spiro-cyclopropaneoxindoles

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Issue 17/2013

Bhadra, Sukalyan; Dzik, Wojciech I.; Gooßen, Lukas J.: Synthesis of Aryl Ethers from Aromatic Carboxylic Acids

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Issue 16/2013

Lu, Wenbin; Liang, Zhuye; Zhang, Yuwei; Wu, Fan; Qian, Qun; Gong, Hegui: Gram-Scale Ketone Synthesis by Direct Reductive Coupling of Alkyl Iodides with Acid Chlorides

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Issue 15/2013

Darses, Benjamin; Jarvis, Amanda G.; Mafroud, Abdel-Kader; Estenne-Bouhtou, Geneviève; Dargazanli, Gihad; Dauban, Philippe: Asymmetric Synthesis of Amines through Rhodium-Catalyzed C–H Amination with Sulfonimidoylnitrenes

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Issue 14/2013

Lu, Xiaowei; Sail, Deepak; Kováč, Pavol: 4′,6′-O-Benzylidene- and 4′,6′-O-p-Methoxybenzylidene-α,β-cellobiose and Their Hexa-O-β-benzoyl Derivatives

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Issue 12/2013

Liu, Jinxian; Ma, Shengming: Aerobic Oxidation of Propargyl Alcohol: A Convenient Method for the Synthesis of Propiolaldehyde

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Issue 11/2013

Kazmaier, Uli; Bayer, Anton; Deska, Jan: Palladium-Catalyzed Allylic Alkylations as Versatile Tool for Amino Acid and Peptide Modifications

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Issue 09/2013

Trosien, Simon; Schollmeyer, Dieter; Waldvogel, Siegfried R.: Modular Access to 9,9-Spirobifluorenes by Oxidative Coupling Using Molybdenum Pentachloride

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Issue 08/2013

Takeda, Youhei; Okumura, Sota; Minakata, Satoshi: A Practical Synthesis of Azobenzenes through Oxidative Dimerization of Aromatic Amines Using tert-Butyl Hypoiodite

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Issue 07/2013

Wu, Haotian; Hintermann, Lukas: Transfer Hydrogenations of Alkenes with Formate on Pd/C: Synthesis of Dihydrocinchona Alkaloids

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Issue 06/2013

Böse, Dietrich; Lübcke, Marvin; Pietruszka, Jörg: A Mild PPTS-Catalyzed Acetalization of α,β-Unsaturated Aldehydes: The First Single-Step Protocol towards Benzylic Acetals

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Issue 05/2013

Kuang, Jinqiang; Xie, Xi; Ma, Shengming: A General Approach to Terminal Allenols

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Issue 04/2013

Jakubkiene, Virginija; Zurba, Justinas; Cikotiene, Inga: N-Nitroso Group-Assisted Nucleophilic Aromatic Substitution of 6-Chloro­pyrimidines: A Facile and Efficient Synthesis of Pyrimidine-4,6- and -2,4-­diamines

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Issue 03/2013

J. Tilley, Leon; Bobbitt, James M.; Murray, Stephanie A.; Camire, Casey E.; Eddy, Nicholas A.: A Revised Preparation of (4-Acetamido-2,2,6,6-tetramethylpiperidin-1-yl)oxyl and 4-Acetamido-2,2,6,6-tetramethyl-1-oxopiperidinium Tetrafluoroborate: Reagents for Stoichiometric Oxidations of Alcohols

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Issue 02/2013

Messik, Frauke; Oberthür, Markus: An Expedient Access to Still–Gennari Phosphonates

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Issue 01/2013

Monguchi, Yasunari; Yanase, Takayoshi; Mori, Shigeki; Sajiki, Hironao: A Practical Protocol for the Hiyama Cross-Coupling Reaction Catalyzed by Palladium on Carbon

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Issue 24/2012

Boultadakis-Arapinis, Mélissa; Lescot, Camille; Micouin, Laurent; Lecourt, Thomas: Gram-Scale Quaternarization of the Anomeric Position of Carbohydrates: Dramatic Effects of Molecular Sieves on Rhodium(II)-Mediated Decomposi­tion of Diazo Sugars

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Issue 23/2012

Blay, Gonzalo; Fernández, Isabel; Pedro, José R.; Vila, Carlos: Enantioselective Synthesis of Substituted Indoles Through Zirconium(IV)-Catalyzed Friedel–Crafts Alkylation

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Issue 22/2012

Wei, Shengwei; Weiß, Katharina M.; Tsogoeva, Svetlana B.: Convenient One-Pot Two-Step Synthesis of 1,3-Thiazoles via Organocatalyzed Epoxidation of Nitroolefins

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Issue 21/2012

Varela-Fernández, Alejandro; Varela, Jesús A.; Saá, Carlos: Formation of Indoles, Dihydroisoquinolines, and Dihydroquinolines by Ruthenium-Catalyzed Heterocyclizations

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Issue 20/2012

Ichibakase, Tomonori; Nakajima, Makoto: Efficient Preparation of 1,3-Diol Derivatives with Three Contiguous Stereocenters by an Enantioselective Direct Aldol–Tishchenko Reaction

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Bahnck, Kevin B.; Shavnya, Andrei; Tao, Yong; Lilley, Susan C.; Andrews, Melissa P.; Aspnes, Gary E.; Bernhardson, David J.; Bill, David R.; Bundesmann, Mark W.; Dow, Robert L.; Karki, Kapil; Le, Tung; Li, Qifang; Munchhof, Michael J.; Nematalla, Asaad; Nihlawi, Mohammed; Patel, Leena; Perreault, Christian; Waldo, Michael: Efficient Synthesis of 4-Amino-2-methoxy-7,8-dihydropyrido[4,3-d]pyrimidin-5-ones: Practical Access to a Novel Chemotype in the Development of DGAT-1 Inhibitors

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Issue 19/2012

Kinuta, Hirotaka; Kita, Yusuke; Rémond, Emmanuelle; Tobisu, Mamoru; Chatani, Naoto: Novel Synthetic Approach to Arylboronates via Rhodium-Catalyzed Carbon–Cyano Bond Cleavage of Nitriles

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Kraus, George A.; Riley, Sean: A Large-Scale Synthesis of α-Olefins and α,ω-Dienes

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Issue 18/2012

Csuk, René; Vasileva, Galina; Barthel, Alexander: Towards an Efficient Preparation of Hydromorphone

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Issue 17/2012

Stecko, Sebastian; Michalak, Michał; Stodulski, Maciej; Mucha, Łukasz; Parda, Kamil; Furman, Bartłomiej; Chmielewski, Marek: Practical One-Pot Synthesis of Protected l-Glyceraldehyde Derivatives

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Issue 16/2012

Aitken, R. Alan; Collett, Chris J.; Mesher, Shaun T. E.: Convenient Preparation of Long-Chain Dialkyl Phosphates: Synthesis of Dialkyl Phosphates

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Issue 15/2012

Mori, Takamichi; Nakamura, Toshiyuki; Onodera, Gen; Kimura, Masanari: Regio- and Stereoselective Multicomponent Coupling Reaction of Alkynes and Dimethylzinc Involving Allylnickelacycles

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Issue 14/2012

Miyata, Kengo; Kitamura, Masato: Asymmetric Dehydrative C-, N-, and O-Allylation Using Naph-diPIM-dioxo-i-Pr–CpRu/p-TsOH Combined Catalyst

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Issue 13/2012

Trofymchuk, Sergii; Bezdudny, Andrii V.; Pustovit, Yurii M.; Lukin, Oleg; Boyko, Alexander N.; Chekotylo, Alexey; Tolmachev, Andrei A.; Mykhailiuk, Pavel K.: A Facile Synthesis of Isomeric C-(2,2,2-Trifluoroethyl)anilines

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Issue 12/2012

Matsuda, Naoki; Hirano, Koji; Satoh, Tetsuya; Miura, Masahiro: Copper-Catalyzed Direct Amination of Polyfluoroarenes and Azoles with Hydroxylamines and Its Application to the Synthesis of 3-Aminobenzoheteroles

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Issue 11/2012

Modha, Sachin G.; Trivedi, Jalpa C.; Mehta, Vaibhav P.; Ermolat’ev, Denis S.; Van der Eycken, Erik V.: Efficient Preparation of Tetrasubstituted Pyrazines Starting from Pyrazin-2(1H)-ones

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Issue 10/2012

Zhao, Peng; Wang, Fei; Xi, Chanjuan: A Convenient Metal-Free Method for the Synthesis of Benzothiazolethiones from o-Haloanilines and Carbon Disulfide

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Issue 09/2012

Li, Dong; Ohmiya, Hirohisa; Sawamura, Masaya: Efficient Preparation of β-Branched γ,δ-Unsaturated Esters through Copper-Catalyzed Allylic Alkylation of Ketene Silyl Acetal

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Issue 08/2012

Yarmolchuk, Vladimir S.; Bezdudny, Andrii V.; Tolmacheva, Nataliya A.; Lukin, Oleg; Boyko, Alexander N.; Chekotylo, Alexey; Tolmachev, Andrei A.; Mykhailiuk, Pavel K.: An Efficient and Safe Method for the Multigram Synthesis of trans-2-(Trifluoromethyl)cyclopropylamine

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Issue 07/2012

Grubb, Alan M.; Schmidt, Michael J.; Seed, Alexander J.; Sampson, Paul: Convenient Preparation of Halo-1,3-thiazoles: Important Building Blocks for Materials and Pharmaceutical Synthesis

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Issue 06/2012

Oh, Ken; Fuchibe, Kohei; Yokota, Misaki; Ichikawa, Junji: Facile Synthesis of Substituted 1,1-Difluoroallenes via Carbonyl Difluorovinylidenation

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Issue 05/2012

Rendina, Victor L.; Kaplan, Hilan Z.; Kingsbury, Jason S.: Highly Efficient and Enantioselective α-Arylation of Cycloalkanones by Scandium-Catalyzed Diazoalkane-Carbonyl Homologation

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Issue 04/2012

Shirinian, Valerii Z.; Shimkin, Alexey A.; Lonshakov, Dmitry V.; Mailyan, Artur K.; Lvov, Andrey G.; Krayushkin, Michail M.: An Environmentally Friendly Synthesis of Michler’s Ketone Analogues in Water

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Issue 03/2012

Rassadin, Valentin A.; Sokolov, Viktor V.; Khlebnikov, Alexander F.; Ulin, Nikolay V.; Kozhushkov, Sergei I.; de Meijere, Armin: Convenient Synthesis of Ethenylcyclopropane and Some 2-Cyclopropylcyclopropane Derivatives

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Issue 02/2012

Mita, Tsuyoshi; Higuchi, Yuki; Sato, Yoshihiro: Convenient and Practical Synthesis of α-Amido Stannanes

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Issue 01/2012

Rossy, Cybille; Fouquet, Eric; Felpin, François-Xavier: A Sustainable Procedure Combining the Advantages of Both Homogeneous and Heterogeneous Catalysis for the Heck-Matsuda Reaction

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Issue 24/2011

Lach, Slawomir; Witt, Dariusz: A New and Convenient Method for the Preparation of Functionalized Phosphorothioates

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Issue 23/2011

Cadu, Alban; Paptchikhine, Alexander; Andersson, Pher G.: Birch Reaction Followed by Asymmetric Iridium-Catalysed Hydrogenation

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Issue 22/2011

Ladouceur, Sébastien; Soliman, Ahmed M.; Zysman-Colman, Eli: One-Pot Click Synthesis of 1N-Alkyl-4-aryl-1,2,3-triazoles from Protected Arylalkynes and Alkyl Bromides

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Issue 21/2011

Rassukana, Yuliya V.: Methyl α-Iminotrifluoropropionate: A Novel Convenient Building Block for the Preparation of Functionalized Derivatives Bearing a Trifluoroalanine Residue

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Issue 18/2011

Felpin, François-Xavier; Fouquet, Eric: Reliable and Safe, Gram-Scale Hydrogenation and Hydrogenolysis of O-Benzyl Ether Groups with In Situ Pd⁰/C Catalyst

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Issue 17/2011

Romer, Duane R.: Convenient Laboratory Method for the Synthesis of Symmetrical 1,3-Diphenylacetone Derivatives

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Issue 16/2011

Presset, Marc; Mailhol, Damien; Coquerel, Yoann; Rodriguez, Jean: Diazo-Transfer Reactions to 1,3-Dicarbonyl Compounds with Tosyl Azide

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Issue 15/2011

Saget, Tanguy; Cramer, Nicolai: Convenient Preparation of Tri-tert-butylphosphonium Tetrafluoroborate

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Issue 14/2011

Hruszkewycz, Damian P.; Cavanaugh, Kathryn R.; Takamura, Kathryn T.; Wayman, Lora M.; Curley Jr., Robert W.: Efficient, Low-Cost Synthesis of Retinal (Vitamin A Aldehyde)

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Issue 13/2011

Königs, C. David F.; Oestreich, Martin: Shortened Synthesis of a Silicon-Stereogenic Cyclic Silane

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Issue 06/2011

Norberg, A. Monica; Smith III, Milton R.; Maleczka Jr., Robert E.: Practical One-Pot C-H Activation/Borylation/Oxidation: Preparation of 3-Bromo-5-methylphenol on a Multigram Scale

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Issue 04/2011

Bucher, Christoph; Gilmour, Ryan: A Modular Synthesis of Fluorinated, Chiral Polar Lipids

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Issue 02/2011

Gross, Stefan; Heuser, Stefan; Ammer, Carolin; Heckmann, Golo; Bach, Thorsten: 2,4-Disubstituted Thiazoles by Regioselective Cross-Coupling or Bromine-Magnesium Exchange Reactions of 2,4-Dibromothiazole

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Issue 01/2011

Zhang, Zhi-Guang; Haag, Benjamin A.; Li, Jin-Shan; Knochel, Paul: Efficient Preparation of Polyfunctional Indoles via a Zinc Organometallic Variation of the Fischer Indole Synthesis

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Issue 23/2010

Kozhushkov, Sergei I.; Wagner-Gillen, Karsten; Khlebnikov, Alexander F.; de Meijere, Armin: Productive Syntheses of 1-Ethynylcyclopropylamine and 1-Ethynylcyclobutylamine

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Issue 22/2010

Bernhardt, Sebastian; Metzger, Albrecht; Knochel, Paul: Direct Addition of Functionalized Organozinc Reagents to Carbon Dioxide, Ketones, and Aldehydes in the Presence of MgCl₂

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Issue 21/2010

Welschoff, Nina; Waldvogel, Siegfried R.: Practical Synthesis of Optically Pure Menthylamines Starting from Racemic Neomenthol

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Issue 20/2010

Pearson-Long, Morwenna S. M.; Beauseigneur, Alice; Karoyan, Philippe; Szymoniak, Jan; Bertus, Philippe: Titanium-Catalyzed Cyclopropanation of Boc-Protected Cyanohydrins: A Short Access to Aminocyclopropanecarboxylic Acid Derivatives

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Issue 18/2010

Chmielewski, Michał J.: A Short, Multigram Synthesis of 1,8-Diaminocarbazole

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Issue 17/2010

Pandey, Ankur; Bolm, Carsten: Metal-Free Synthesis of N-Cyano-Substituted Sulfilimines and Sulfoximines

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Issue 16/2010

Metzger, Albrecht; Melzig, Laurin; Knochel, Paul: Scaled-Up Transition-Metal-Catalyzed Cross-Coupling Reactions of Thioether-Substituted N-Heterocycles with Organozinc Reagents

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Issue 15/2010

Wunderlich, Stefan H.; Bresser, Tomke; Dunst, Cora; Monzon, Gabriel; Knochel, Paul: Efficient Preparation of Polyfunctional Organometallics via Directed ortho-Metalation

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Issue 14/2010

Yamada, Shigeyuki; Knochel, Paul: Large-Scale Preparation of Aromatic Fluorides via Electrophilic Fluorination with Functionalized Aryl- or Heteroarylmagnesium Reagents

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Issue 13/2010

Hehn, Jörg P.; Gamba-Sánchez, Diego; Kemmler, Michael; Fleck, Martin; Basler, Birte; Bach, Thorsten: [2+2]-Photocycloaddition Reactions of Tetronic Acid Esters and Amides

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Dunst, Cora; Kienle, Marcel; Knochel, Paul: Preparation of Heterocyclic Amines via a Copper(I)-Mediated Oxidative Cross-Coupling of Organozinc Reagents with Lithium Amides

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Issue 12/2010

Desai, Aman A.; Huang, Li; Wulff, William D.; Rowland, Gerald B.; Antilla, Jon C.: Gram-Scale Preparation of VAPOL Hydrogenphosphate: A Structurally Distinct Chiral Brønsted Acid

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Issue 11/2010

Kemme, Susanne T.; Schmidt, Yvonne; Grünanger, Christian U.; Laungani, Andy C.; Herber, Christian; Breit, Bernhard: Economic Large-Scale Synthesis of o- and m-Diphenylphosphinobenzoic Acids

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Issue 10/2010

Delaunay, Thierry; Conreaux, David; Bossharth, Emmanuel; Desbordes, Philippe; Monteiro, Nuno; Balme, Geneviève: Practical One-Pot Syntheses of Regioisomeric Furan-Fused Pyridinones (and Quinolinones) from Common Precursors

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Issue 09/2010

Wiesner, Markus; Wennemers, Helma: Peptide-Catalyzed Conjugate Addition Reactions of Aldehydes to Nitroolefins

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Issue 08/2010

Sparr, Christof; Tanzer, Eva-Maria; Bachmann, Julia; Gilmour, Ryan: A Concise Synthesis of (S)-2-(Fluorodiphenylmethyl)pyrrolidine: A Novel Organocatalyst for the Stereoselective Epoxidation of α,β-Unsaturated Aldehydes

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Issue 07/2010

Rousseau, Géraldine; Robert, Frédéric; Landais, Yannick: Synthesis of (1-Allylcyclohexa-2,5-dienyl)arenes

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Issue 06/2010

Sridharan, Vellaisamy; Ruiz, Miriam; Menéndez, J. Carlos: Mild and High-Yielding Synthesis of β-Keto Esters and β-Ketoamides

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Issue 05/2010

Metzger, Albrecht; Argyo, Christian; Knochel, Paul: Large-Scale Preparation of Polyfunctional Benzylic Zinc Reagents by Direct Insertion of Zinc Dust into Benzylic Chlorides in the Presence of Lithium Chloride

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Issue 04/2010

Phillips, James G.; Jaworska, Maria; Lew, Willard: A Practical Synthesis of 1-N-SEM-Protected 3-Iodo-7-methyl-2-piperidin-3-ylindole

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Issue 03/2010

Schur, Christine; Groß, Andreas; Hartung, Jens: A Practical Method for O-Acylation of N-Hydroxythiazole-2(3H)-thiones

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Issue 02/2010

da Silva Prado, Viviana; Burtoloso, Antonio Carlos B.: An Improved Procedure for the Preparation of [Bis(2,2,2-trifluoroethyl)phosphono]acetic Acid

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Issue 01/2010

Geoffroy, Philippe; Ballet, Marie-Paule; Finck, Sidonie; Marchioni, Eric; Marcic, Christophe; Miesch, Michel: Synthesis of Racemic and Enantiomerically Pure Acetylenic ω-Keto Esters Derived from 2-Methyl-1,3-cycloalkanediones and 2-Methylcycloalkanones Respectively

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Issue 24/2009

Vogt, Florian; Jödicke, Kai; Schröder, Jürgen; Bach, Thorsten: Paternò-Büchi Reactions of Silyl Enol Ethers and Enamides

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Issue 23/2009

Procuranti, Barbara; Myles, Lauren; Gathergood, Nicholas; Connon, Stephen J.: Pyridinium Ion Catalysis of Carbonyl Protection Reactions

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Issue 22/2009

Steel, Patrick G.; Woods, Tom M.: Enol Phosphinates and Phosphonates: Practical Electrophiles for Cross-Coupling Strategies

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Issue 21/2009

Brunner, Gerhard; Eberhard, Laura; Oetiker, Jürg; Schröder, Fridtjof: Cyclopropanation with Dibromomethane under Grignard and Barbier Conditions

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Issue 20/2009

Lőrincz, Krisztián; Kele, Péter; Novák, Zoltán: The Sequential Sonogashira-Click Reaction: A Versatile Route to 4-Aryl-1,2,3-triazoles

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Issue 19/2009

Zhou, Guoqiang; Lim, Daniel; Fang, Fang; Coltart, Don M.: A Practical Synthesis of β-Keto Thioesters by Direct Crossed-Claisen Coupling of Thioesters and N-Acylbenzotriazoles

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Issue 18/2009

Nguyen, Thanh Binh; Martel, Arnaud; Dhal, Robert; Dujardin, Gilles: A Large-Scale Low-Cost Preparation of N-Benzylhydroxylamine Hydrochloride

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Issue 16/2009

Cvengroš, Ján; Stolz, Daniel; Togni, Antonio: A Concise Synthesis of ortho-Iodobenzyl Alcohols via Addition of ortho-Iodophenyl Grignard Reagent to Aldehydes and Ketones

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Issue 15/2009

Godineau, Edouard; Landais, Yannick: Synthesis of Piperidinones through a Radical Cascade

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Issue 14/2009

Maji, Modhu Sudan; Studer, Armido: Transition-Metal-Free Oxidative Homocoupling of Aryl, Alkenyl, and Alkynyl Grignard Reagents with TEMPO

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Issue 13/2009

Gooßen, Lukas J.; Blanchot, Mathieu; Salih, Kifah S. M.; Gooßen, Käthe: Ruthenium-Catalyzed Addition of Primary Amides to Alkynes: A Stereoselective Synthesis of Secondary Enamides

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He, Rongjun; Maruoka, Keiji: Binaphthyl-Modified Quaternary Phosphonium Salts as Chiral Phase Transfer Catalysts: Application to Asymmetric Amination of β-Keto Esters

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Issue 12/2009

Berkessel, A.; Seelig, B.: A Simplified Synthesis of Takemoto’s Catalyst

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Issue 11/2009

Csuk, René; Stark, Sebastian; Barthel, Alexander; Kluge, Ralph; Ströhl, Dieter: A Robust Synthesis of N^ε-(Carboxymethyl)-l-lysine (CML)

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Leogane, Olivier; Lebel, Hélène: One-Pot Curtius Rearrangement Processes from Carboxylic Acids

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Issue 10/2009

Besset, Tatiana; Morin, Christophe: Synthesis of 3,6-Dimethoxybenzene-1,2-diamine and of 4,7-Dimethoxy-2-methyl-1H-benzimidazole

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Ortmann, Regina; Schlitzer, Martin: An Inexpensive Procedure for Reductive Aminations Using Dimethylamineborane on Millimolar and Molar Scale

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Issue 09/2009

Owston, Nathan A.; Nixon, Tracy D.; Parker, Alexandra J.; Whittlesey, Michael K.; Williams, Jonathan M. J.: Conversion of Primary Alcohols and Aldehydes into Methyl Esters by Ruthenium-Catalysed Hydrogen Transfer Reactions

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Issue 08/2009

Parthasarathy, Kanniyappan; Cheng, Chien-Hong: Rhodium-Catalyzed Gram-Scale Synthesis of Highly Substituted Pyridine Derivatives

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Whitaker, John M.; Ronald, Robert C.: Enantioselective Synthesis of (R)-Propylene Carbonate from Ethyl (S)-Lactate

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Issue 07/2009

Yamaguchi, Ryohei; Mingwen, Zhu; Kawagoe, Shoko; Asai, Chiho; Fujita, Ken-ichi: A New Atom-Economical and Selective Synthesis of Secondary and Tertiary Alkylamines by Means of Cp*Iridium Complex Catalyzed Multiple N-Alkylation of Ammonium Salts with Alcohols without Solvent

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Castro, Juan C.; Malakhov, Andrey; Burgess, Kevin: Synthesis of Regioisomerically Pure 5-Functionalized 2′,7′-Dichloro­fluoresceins

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Issue 06/2009

Yang, Jie; Teng, Yun; Ara, Shamim; Rallapalli, Sundari; Cook, James M.: An Improved Process for the Synthesis of 4H-Imidazo[1,5-a][1,4]benzo­diazepines

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Melzig, Laurin; Rauhut, Christian B.; Knochel, Paul: Meta- and Para-Difunctionalization of Arenes via an Ortho-Magnesiation and a Subsequent Sulfoxide-Magnesium Exchange

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Issue 05/2009

Navarro, Cristina; Csákÿ, Aurelio G.: Diastereoselective Synthesis of 1,2,3-Trisubstituted Indanes via Rhodium(I)-Catalyzed Tandem Conjugate Additions

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Wallentin, Carl Johan; Orentas, Edvinas; Butkus, Eugenijus; Wärnmark, Kenneth: Baker’s Yeast for Sweet Dough Enables Large-Scale Synthesis of Enantiomerically Pure Bicyclo[3.3.1]nonane-2,6-dione

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Issue 04/2009

Dong, Zhibing; Manolikakes, Georg; Li, Jinshan; Knochel, Paul: Palladium-Catalyzed Cross-Couplings of Unsaturated Halides Bearing Relatively Acidic Hydrogen Atoms with Organozinc Reagents

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Phillips, Eric M.; Wadamoto, Manabu; Scheidt, Karl A.: Synthesis of Enantioenriched α,α-Disubstituted Cyclopentenes Catalyzed by N-Heterocyclic Carbenes

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Issue 03/2009

Merkul, Eugen; Grotkopp, Oliver; Müller, Thomas J. J.: 2-Oxazol-5-ylethanones by Consecutive Three-Component Amidation-Coupling-Cycloisomerization (ACCI) Sequence

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Fairlamb, Ian J. S.; Sehnal, Petr; Taylor, Richard J. K.: Suzuki-Miyaura Cross-Couplings Mediated by trans-PdBr(N-Succ)(PPh₃)₂: A Convenient Synthetic Method for Diarylmethanes and Aryl(heteroaryl)methanes

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Issue 02/2009

Taft, Benjamin R.; Swift, Elizabeth C.; Lipshutz, Bruce H.: A Convenient Preparation of Di-p-chlorobenzyl Azodicarboxylate (DCAD) for Mitsunobu Couplings

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Cook, Matthew J.; Rovis, Tomislav: Enantioselective Rhodium-Catalyzed Alkylative Desymmetrization of 3,5-Dimethylglutaric Anhydride

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Issue 24/2008

L’Helgoual’ch, Jean-Martial; Bentabed-Ababsa, Ghenia; Chevallier, Floris; Derdour, Aïcha; Mongin, Florence: Synthesis of 2,5-Diiodopyrazine by Deprotonative Dimetalation of Pyrazine

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Yin, Yan; Chai, Zhuo; Ma, Wen-Ying; Zhao, Gang: Synthesis of Indoles via Diethylzinc-Mediated Intramolecular Hydroamination Reactions of Alkynyl Sulfonamides

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Issue 23/2008

Kanao, Keiichiro; Matsuzawa, Hiroshi; Miyake, Yoshihiro; Nishibayashi, Yoshiaki: Ruthenium-Catalyzed Enantioselective Propargylation of Indoles with Propargylic Alcohols

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Eagon, Scott; Kim, Jinsoo; Singaram, Bakthan: Mild and Practical Reductions of Prochiral Ketones to Chiral Alcohols Using the Chiral Boronic Ester TarB-H

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Issue 22/2008

Mosrin, Marc; Petrera, Marilena; Knochel, Paul: Multiple Regio- and Chemoselective Functionalizations of Pyrimidine Derivatives Using TMPMgCl×LiCl and TMP₂Mg×2 LiCl

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Hashimoto, Takuya; Maruoka, Keiji: Design of an Axially Chiral Dicarboxylic Acid and Its Application in Syntheses of Optically Active β-Amino Acids and β-Amino Phosphonic Acid Derivatives

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Issue 21/2008

Clarke, Paul A.; Zaytsev, Andrey V.; Whitwood, Adrian C.: Pot, Atom, and Step Economic (PASE) Synthesis of Highly Substituted Piperidines: A Five-Component Condensation

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Sakai, Norio; Moriya, Toshimitsu; Fujii, Kohji; Konakahara, Takeo: Direct Reduction of Esters to Ethers with an Indium(III) Bromide/Triethylsilane Catalytic System

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Issue 20/2008

Schareina, Thomas; Zapf, Alexander; Cotté, Alain; Müller, Nikolaus; Beller, Matthias: A Bio-inspired Copper Catalyst System for Practical Catalytic Cyanation of Aryl Bromides

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Aponick, Aaron; Biannic, Berenger: Gold-Catalyzed Dehydrative Cyclization of Allylic Diols

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Issue 19/2008

Ishikawa, Shunpei; Manabe, Kei: Synthesis of Substituted Monohalobenzenes via Ortho-Selective Cross-Coupling of Dihalobenzenes with Electron-Donating Ortho-Directing Groups

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Issue 18/2008

Matsubara, Ryosuke; Kobayashi, Shu: DBU-Catalyzed Addition Reactions of Sulfonylimidates

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Issue 17/2008

Alcaide, Benito; Almendros, Pedro; Cabrero, Gema; Ruiz, M. Pilar: Direct Synthesis of Protected Enantiopure 5-Cyano-3,4-dihydroxypyrrolidin-2-ones from β-Lactam Aldehydes Catalyzed by Iodine

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Issue 16/2008

Donohoe, Timothy J.; Fishlock, Lisa P.; Procopiou, Panayiotis A.: Ring-Closing Metathesis as a Key Step in the Synthesis of 2-Pyridones and Pyridine Triflates

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Issue 15/2008

Bischop, Martina; Cmrecki, Vesna; Ophoven, Vera; Pietruszka, Jörg: Synthesis of (2R,3R)-1,4-Dimethoxy-1,1,4,4-tetraphenylbutane-2,3-diol

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Issue 14/2008

Hintermann, Lukas; Suzuki, Keisuke: 2,5-Dihydroxyterephthalates, 2,5-Dichloro-1,4-benzoquinone-3,6-dicarbox­ylates, and Polymorphic 2,5-Dichloro-3,6-dihydroxyterephthalates

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Issue 13/2008

Lim, Daniel; Zhou, Guoqiang; Livanos, Alexandra E.; Fang, Fang; Coltart, Don M.: MgBr₂·OEt₂-Promoted Coupling of Ketones and Activated Acyl Donors via Soft Enolization: A Practical Synthesis of 1,3-Diketones

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Issue 11/2008

Eloy, Nathalie; Pasquinet, Eric; Grech, Eric; David-Quillot, Frank; Besnard, Olivier; Poullain, Didier: A One-Step, Safe Synthesis of 2,4-Dinitrostyrene and Related (Di)nitrodivinylbenzenes via Stille Coupling

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Issue 10/2008

Igawa, Kazunobu; Sakita, Kyohei; Murakami, Masanori; Tomooka, Katsuhiko: Partial Oxidation of Alkenylsilanes with Ozone: A Novel Stereoselective Approach to the Diol and Triol Derivatives

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Issue 09/2008

Parenty, Alexis D. C.; Cronin, Leroy: One-Pot Synthesis of Imidazopyridine Derivatives

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Issue 08/2008

de Figueiredo, Renata Marcia; Oczipka, Philipp; Fröhlich, Roland; Christmann, Mathias: Synthesis of 4-Maleimidobutyric Acid and Related Maleimides

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Itoh, Junji; Fuchibe, Kohei; Akiyama, Takahiko: Preparation of β-Amino Esters by a Chiral Brønsted Acid Catalyzed Mannich-Type Reaction

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Issue 07/2008

Ibrahem, Ismail; Rios, Ramon; Vesely, Jan; Zhao, Gui-Ling; Córdova, Armando: Catalytic Enantioselective 5-Hydroxyisoxazolidine Synthesis: An Asymmetric Entry to β-Amino Acids

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Luu, Thanh; Morisaki, Yasuhiro; Tykwinski, Rik R.: One-Pot Synthesis and Functionalization of Polyynes via Alkylidene Carbenoids

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Issue 06/2008

Gwiazda, Maciej; Reissig, Hans-Ulrich: Highly Substituted Imidazole Derivatives from a New Four-Component Synthesis Employing Methoxyallene

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Motti, Elena; Della Ca’, Nicola; Ferraccioli, Raffaella; Catellani, Marta: Unsymmetrical Aryl-Aryl Cross-Coupling Leading to 6H-Dibenzopyrans

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Issue 05/2008

Iso, Kentaro; Yudha, S. Salprima; Asao, Naoki: Preparation of 1,2-Dihydroisoquinolines by a Three-Component Reaction under Catalyst-Free Conditions

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Hill, Matthew D.; Movassaghi, Mohammad: Direct Synthesis of Substituted Pyrimidines and Quinazolines

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Issue 04/2008

Jin, Liqun; Zhao, Yingsheng; Wang, Haibo; Lei, Aiwen: Palladium-Catalyzed R(sp³)-Zn/R(sp)-SnBu₃ Oxidative Cross-Coupling

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Kessabi, Jilali; Beaudegnies, Renaud; Jung, Pierre M. J.; Martin, Benjamin; Montel, Florian; Wendeborn, Sebastian: A Convenient, High-Yielding Copper-Free Synthesis of Skipped 1,4-Diynes

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Issue 03/2008

Aznar, Fernando; García, Ana-Belén; Quiñones, Noelia; Cabal, María-Paz: Stereoselective Synthesis of meso- and cis-2,6-Diarylpiperidin-4-ones Catalyzed by l-Proline

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Carson, Cheryl A.; Young, Ian S.; Kerr, Michael A.: The Reaction of Nitrones with Cyclopropanes: A Convenient Preparation of Tetrahydro-1,2-oxazines

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Issue 02/2008

Bartoli, Giuseppe; Di Antonio, Giustino; Giuli, Sandra; Marcantoni, Enrico; Marcolini, Mauro; Paoletti, Melissa: The CeCl₃·7H₂O/NaI/SiO₂ System as an Efficient Promoter for the Friedel-Crafts Reaction of Indoles to Nitroalkenes under Solvent-Free Conditions

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Kabalka, George; Borella, Scott; Yao, Min-Liang: Boron Trihalide Mediated Substitution of Hydroxyl Groups with Alkenyl, Alkynyl, and Allyl Moieties

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Issue 01/2008

Naik, Anil D.; Marchand-Brynaert, Jacqueline; Garcia, Yann: A Simplified Approach to N- and N,N′-Linked 1,2,4-Triazoles by Transamination

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Parenty, Alexis D. C.; Cronin, Leroy: One-Pot Synthesis of Dihydroimidazo- and Imidazophenanthridinium Salts

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Issue 24/2007

Soorukram, Darunee; Boudet, Nadège; Malakhov, Vladimir; Knochel, Paul: Preparation of Polyfunctionalized 2,6-Dimethoxypyrimidine Derivatives via Chemo- and Regioselective Direct Zinc Insertion

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Palacios, Francisco; Vicario, Javier: Enantioselective Synthesis of γ-Functionalized α-Dehydroamino Esters

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Issue 23/2007

Roseblade, Stephen J.; Pfaltz, Andreas: Kinetic Resolution of Pyridyl Alcohols by Cu(II)(Borabox)-Catalyzed Acylation

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Blay, Gonzalo; Fernández, Isabel; Marco-Aleixandre, Alícia; Pedro, José R.: Enantioselective Addition of Dimethylzinc to α-Keto Esters

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Issue 22/2007

Riveiros, Ricardo; Sestelo, José Pérez; Sarandeses, Luis A.: Synthesis of Allenes by Palladium-Catalyzed S_N2′ Reaction of Indium Organometallics with Propargylic Esters

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Issue 21/2007

Rauniyar, Vivek; Hall, Dennis G.: Preparation of a C₂-Symmetric Binol-Derived Diol and Its Application in the Catalytic Enantioselective and Catalyst-Controlled Diastereoselective Allylboration of Aldehydes

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Rhee, Jong Uk; Jones, Regan A.; Krische, Michael J.: Catalytic Enantioselective Reductive Cyclization of Acetylenic Aldehydes via Hydrogenation

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Issue 20/2007

Sanz, Roberto; Martínez, Alberto; Miguel, Delia; Álvarez-Gutiérrez, Julia M.; Rodríguez, Félix: Synthesis of 1,5-Enynes by Brønsted Acid Catalyzed Substitution of Propargylic Alcohols and One-Pot Synthesis of Bicyclo[3.1.0]hexenes

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Lipshutz, Bruce H.; Lee, Ching-Tien; Taft, Benjamin R.: A Conjugate Reduction Pathway to Chiral Silanes Using CuH

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Issue 19/2007

Plastina, Pierluigi; Gabriele, Bartolo; Salerno, Giuseppe: Palladium-Catalyzed Oxidative Aminocarbonylation of Alkynols

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Babudri, Francesco; Farinola, Gianluca M.; Naso, Francesco; Ragni, Roberta; Spina, Giulia: A Novel Stereoselective Synthesis of Symmetrical (1E,3E)-1,4-Diarylbuta-1,3-dienes

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Issue 18/2007

Dohi, Toshifumi; Morimoto, Koji; Ito, Motoki; Kita, Yasuyuki: Regioselective Bipyrrole Coupling of Pyrroles and 3-Substituted Pyrroles Using Phenyliodine(III) Bis(trifluoroacetate)

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Tanaka, Ken; Takeishi, Kenzo: Preparation of Enantioenriched Axially Chiral Anilides via [2+2+2] Cycloaddition of 1,6-Diynes with Trimethylsilylynamides

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Issue 17/2007

Cozzi, Pier Giorgio; Mignogna, Alessandro; Zoli, Luca: Practical Chloromanganese-Salen-Catalyzed Enantioselective Reformatsky Reaction with Ketones

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Göhler, Sabrina; Roth, Stefanie; Cheng, Huan; Göksel, Hülya; Rupp, Alexander; Haustedt, Lars O.; Stark, Christian B. W.: Multigram Synthesis of Diastereomerically Pure Tetrahydrofuran-diols

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Issue 16/2007

Rábai, József; Szíjjártó, Csongor; Ivanko, Peter; Szabó, Dénes: 3-(Perfluoroalkyl)propanols: Valuable Building Blocks for Fluorous Chemistry

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Issue 14/2007

Lee, Daehyung; Yang, Youngmin; Yun, Jaesook: Copper Hydride Catalyzed Enantioselective Conjugate Reduction of Unsaturated Nitriles

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Issue 13/2007

Panunzio, Mauro; Bandini, Elisa; D’Aurizio, Antonio; Millemaggi, Alessia; Xia, Zhining: EuFOD-Catalyzed Hetero-Diels-Alder (HDA) Reaction under Microwave Heating

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Issue 12/2007

Bellina, Fabio; Rossi, Renzo: An Efficient and Inexpensive Multigram Synthesis of 3,4-Dibromo- and 3,4-Dichlorofuran-2(5H)-one

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Mendonça, Francisco J. B.; dos Anjos, Janaína V.; Sinou, Denis; de Melo, Sebastiao J.; Srivastava, Rajendra M.: Palladium-Catalyzed Alkynylation (Sonogashira Coupling) at C-5 of the Uracil Moiety in Modified Unsaturated Pyranosyl Nucleosides

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Issue 11/2007

Sulzer-Mossé, Sarah; Laars, Marju; Kriis, Kadri; Kanger, Tõnis; Alexakis, Alexandre: Synthesis and Use of 3,3′-Bimorpholine Derivatives in Asymmetric Michael Addition and Intramolecular Aldol Reaction

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Bartali, Laura; Larini, Paolo; Guarna, Antonio; Occhiato, Ernesto G.: Preparation of Cyclopenta-Fused N-, O-, and S-Heterocycles by Lewis Acid Catalyzed Nazarov Reaction

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Issue 10/2007

Ward, Dale E.; Rasheed, M. Abdul; Gillis, H. Martin; Beye, Garrison E.; Jheengut, Vishal; Achonduh, George T.: Simple and Efficient Preparation of Reagents for Thiopyran Introduction:
Methyl Tetrahydro-4-oxo-2H-thiopyran-3-carboxylate, Tetrahydro-4H-thiopyran-4-one, and 3,6-Dihydro-4-trimethylsilyloxy-2H-thiopyran

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Bandini, Marco; Eichholzer, Astrid; Tommasi, Simona; Umani-Ronchi, Achille: Practical Aspects in the Gram-Scale Synthesis of Chiral Diamino-Bithiophene ‘DAT2’ Ligand

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Issue 09/2007

Couture, Axel; Deniau, Eric; Lamblin, Marc; Lorion, Magali; Grandclaudon, Pierre: Preparation of Poly and Diversely Substituted N-Alkylated and Free-NH Isoindolin-1-ones

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Issue 08/2007

Kienle, Marcel; Reddy Dubbaka, Srinivas; del Amo, Vicente; Knochel, Paul: Preparation of Tertiary Amines via the Oxidative Coupling of Polyfunctional Aryl and Heteroaryl Amidocuprates

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Issue 07/2007

Hill, Matthew D.; Movassaghi, Mohammad: Synthesis of Substituted Pyridines and Quinolines

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Issue 06/2007

Llamas, Tomás; Gómez Arrayás, Ramón; Carretero, Juan Carlos: Copper(I)-Catalyzed Enantioselective 1,3-Dipolar Cycloaddition of Azomethine Ylides with Vinyl Sulfones

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Issue 05/2007

Thibault, Michelle E.; Luska, Kylie L.; Schlaf, Marcel: An Improved Synthesis of 6,6′-Diamino-2,2′-bipyridine

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Issue 04/2007

Soorukram, Darunee; Knochel, Paul: A Practical Synthesis of Optically Active α-Substituted Ketones in High Enantiomeric­ Excess

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Issue 03/2007

Zhou, Guoqiang; Yost, Julianne M.; Coltart, Don M.: A Direct Aldol Addition of Simple Thioesters Employing Soft Enolization

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Issue 02/2007

Kazmaier, Uli; Dörrenbächer, Sandra; Wesquet, Alexander; Lucas, Simon; Kummeter, Manuela: Molybdenum-Catalyzed Synthesis of Stannylated Allylic Alcohol Derivatives and Their Synthetic Applications

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Issue 01/2007

Albrecht, Markus; Dehn, Sabrina; Schmid, Sören; DeGroot, Marita: Enantiomerically Pure Bis-β-diketones: Valuable Building Blocks for Metallosupramolecular Chemistry

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Issue 24/2006

Pietruszka, Jörg; Witt, Andreas: Synthesis of the Bestmann-Ohira Reagent

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Issue 22/2006

Nagase, Ryohei; Oguni, Yumiko; Misaki, Tomonori; Tanabe, Yoo: Practical and Robust Method for the Preparation of Seebach and Fráter’s Chiral Template, cis-2-Substituted 5-Methyl(or Phenyl)-1,3-dioxolan-4-ones

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Issue 20/2006

Widegren, Magnus; Dietz, Melanie; Friberg, Annika; Frejd, Torbjörn; Hahn-Hägerdal, Bärbel; Gorwa-Grauslund, Marie F.; Katz, Mikael: The Synthesis of Bicyclo[2.2.2]octan-2,6-dione Revisited

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Issue 18/2006

Page, T. Keri; Wirth, Thomas: Simple Direct Synthesis of [Bis(trifluoroacetoxy)iodo]arenes

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Issue 17/2006

Gaefke, Gerald; Enkelmann, Volker; Höger, Sigurd: A Practical Synthesis of 1,4-Diiodo-2,5-bis(chloromethyl)benzene and 1,4-Diiodo-2,5-bis(bromomethyl)benzene

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Issue 15/2006

Yang, Xiaoyin; Knochel, Paul: Preparation and Reactions of Functionalized Organocopper Reagents

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Issue 14/2006

Casabona, Diego; Cativiela, Carlos: Simple and Efficient Multigram Scale Synthesis of 1-Aminocyclopent-3-ene-1-carboxylic Acid

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Issue 11/2006

Rodríguez-Domínguez, Juan C.; Kirsch, Gilbert: Zirconyl Chloride: A Useful Catalyst in the Pechmann Coumarin Synthesis

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Issue 08/2006

Breuning, Matthias; Steiner, Melanie: Convenient Multigram Synthesis of (R)-Homopipecolic Acid Methyl Ester

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Issue 05/2006

Krasovskiy, Arkady; Knochel, Paul: Convenient Titration Method for Organometallic Zinc, Magnesium, and Lanthanide­ Reagents

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Issue 03/2006

Danielec, Holger; Klügge, Jan; Schlummer, Björn; Bach, Thorsten: FeCl₂-Catalyzed Intramolecular Chloroamination Reactions

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Issue 02/2006

Navarro, Oscar; Nolan, Steven P.: Large-Scale One-Pot Synthesis of N-Heterocyclic Carbene-Pd(allyl)Cl Complexes

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Issue 01/2006

Gingras, Marc; Chabre, Yoann M.; Raimundo, J.-M.: Tetrabutylammonium Difluorotriphenylstannate [Bu₄N][Ph₃SnF₂]: Delivering­ Carbon or Fluorine Ligands via Hypercoordination

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Issue 20/2005

Jeulin, Séverine; Champion, Nicolas; Dellis, Philippe; Ratovelomanana-Vidal, Virginie; Genêt, Jean-Pierre: Multigram-Scale Asymmetric Hydrogenation Reactions Using Ru-SYNPHOS^® and Ru-DIFLUORPHOS^® Catalysts

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Issue 18/2005

Fleming, Fraser F.; Zhang, Zhiyu; Wei, Guoqing: Preparation of 3-Oxocyclohex-1-ene-1-carbonitrile

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Issue 17/2005

Frieman, Bryan A.; Taft, Benjamin R.; Lee, Ching-Tien; Butler, Tom; Lipshutz, Bruce H.: Nickel-in-Charcoal (Ni/C): An Efficient Heterogeneous Catalyst for the Construction of C-C, C-N, and C-H Bonds

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Issue 16/2005

Takimiya, Kazuo; Jeon, Hyung Joon; Otsubo, Tetsuo: A Practical Two-Step Synthesis of Tetraselenafulvalene (TSF)

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Issue 15/2005

Kneisel, Florian F.; Leuser, Helena; Knochel, Paul: Preparation and Reactions of Highly Functionalized Bis-Arylzinc Reagents Using a Li(acac)-Catalyzed Iodine-Zinc Exchange

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Issue 14/2005

Barbaro, Pierluigi; Bianchini, Claudio; Giambastiani, Giuliano: Large-Scale Synthesis of Chiral Ferrocenyl Imino-Phosphines

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Brebion, Franck; Goddard, Jean Philippe; Fensterbank, Louis; Malacria, Max: Highly Diastereoselective Michael Additions onto Dienyl Bis-Sulfoxides

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Issue 13/2005

Hodgson, David M.; Chung, Ying Kit; Paris, Jean-Marc: Intramolecular Cyclopropanation of Epichlorohydrin-Derived Unsaturated Chlorohydrins

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Vijayasaradhi, Sivalenka; Beedimane, Manjunath Narayana; Aidhen, Indrapal Singh: Convenient Enantiopure Synthesis of (2S,3R)-2-O-Benzyl-3,4-O-isopropylidene-d-erythritol from d-(+)-Glucono-δ-lactone: A Potential C₄ Chiral Building Block

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Issue 12/2005

Wallace, Karl J.; Hanes, Robert; Anslyn, Eric; Morey, Jeroni; Kilway, Kathleen V.; Siegel, Jay: Preparation of 1,3,5-Tris(aminomethyl)-2,4,6-triethylbenzene from Two Versatile 1,3,5-Tri(halosubstituted) 2,4,6-Triethylbenzene Derivatives

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Hübner, Sandra; Neumann, Helfried; Wangelin, Axel Jacobi; Klaus, Stefan; Strübing, Dirk; Klein, Holger; Beller, Matthias: Efficient One-Pot Synthesis of Substituted 1-Acylaminocyclohex-2-enes

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Issue 11/2005

Paquet, Valérie; Lebel, Hélène: Rhodium-Catalyzed Synthesis of Terminal Alkenes

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Issue 10/2005

Kulinkovich, Oleg G.; Kozyrkov, Yurii Y.; Bekish, Andrei V.; Matiushenkov, Evgenii A.; Lysenko, Ivan L.: A Convenient Way for the Conversion of Carboxylic Esters into 2-Substituted Allyl Halides

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Issue 08/2005

Aggarwal, Varinder K.; Aragoncillo, Cristina; Winn, Caroline L.: Simple Preparation of Trans-Epoxides via Ylide Intermediates

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Issue 07/2005

Heutling, Andreas; Severin, René; Doye, Sven: Regioselective Preparation of 2-Phenylethylamines from 1-Phenyl-2-alkyl­alkynes by Hydroamination/Reduction Sequences

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Issue 06/2005

Kampmann, Detlef; Stuhlmüller, Georg; Simon, Roger; Cottet, Fabrice; Leroux, Frédéric; Schlosser, Manfred: A Large-Scale Low-Cost Access to the Lithium 2,2,6,6-Tetramethylpiperidide Precursor

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Issue 05/2005

Rudolph, Jens; Schmidt, Frank; Bolm, Carsten: Boronic Acids as Versatile Aryl Sources for the Highly Enantioselective Synthesis of Chiral Diarylmethanols on Multigram Scale

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Issue 04/2005

Dömling, Alexander; Illgen, Katrin: 1-Isocyano-2-dimethylamino-alkenes: Versatile Reagents in Diversity-Oriented Organic Synthesis

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Alcaide, Benito; Almendros, Pedro; Alonso, José M.; Luna, Amparo: Chemoselective Deprotection of Allylic Amines Catalyzed by Grubbs’ Carbene

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Issue 03/2005

Rodriquez, Manuela; Taddei, Maurizio: A Simple Procedure for the Transformation of l-Glutamic Acid into the Corresponding γ-Aldehyde

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Cai, Qian; Zhu, Wei; Zhang, Hui; Zhang, Yongda; Ma, Dawei: Preparation of N-Aryl Compounds by Amino Acid-Promoted Ullmann-Type Coupling Reactions

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Issue 02/2005

Srinivasan, Jayasree M.; Burks, Heather E.; Smith, Colin R.; Viswanathan, Rajesh; Johnston, Jeffrey N.: Free Radical-Mediated Aryl Amination: A Practical Synthesis of (R)- and (S)-7-Azaindoline α-Amino Acid

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Pineschi, Mauro; Del Moro, Federica; Crotti, Paolo; Di Bussolo, Valeria; Macchia, Franco: Copper-Catalyzed Highly Enantioselective Synthesis of Cyclic Allylic and Homoallylic Alcohols with Dialkylzinc Reagents

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Issue 01/2005

Larionov, Oleg V.; Kozhushkov, Sergei I.; de Meijere, Armin: Facile Preparation of tert-Butyl 1-tert-Butoxycarbonylaminocyclopent-3-enecarboxylate from Inexpensive Starting Materials

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Fayol, Aude; Housseman, Christopher; Sun, Xiaowen; Janvier, Pierre; Bienaymé, Hugues; Zhu, Jieping: Synthesis of α-Isocyano-α-alkyl(aryl)acetamides and their Use in the Multicomponent Synthesis of 5-Aminooxazole, Pyrrolo[3,4-b]pyridin-5-one and 4,5,6,7-Tetrahydrofuro[2,3-c]pyridine

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Issue 18/2004

Bartoli, Giuseppe; Bosco, Marcella; Marcantoni, Enrico; Massaccesi, Massimo; Rinaldi, Samuele; Sambri, Letizia: Highly Diastereoselective Synthesis of β-Hydroxy Amides from β-Keto Amides

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Issue 17/2004

Kabalka, George W.; Wu, Zhongzhi; Ju, Yuhong: A New Convenient, Efficient, and Regioselective Synthesis of 1,3-Diaryl- 1,3-dihalopropanes

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de Filippis, Arnault; Gomez Pardo, Domingo; Cossy, Janine: Simple Preparation of 3-Aryl 2-Piperidinones

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Issue 16/2004

Slätt, Johnny; Romero, Ivan; Bergman, Jan: Cyanoacetylation of Indoles, Pyrroles and Aromatic Amines with the Combination Cyanoacetic Acid and Acetic Anhydride

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Issue 15/2004

Tissot-Croset, Karine; Polet, Damien; Gille, Ségolène; Hawner, Christine; Alexakis, Alexandre: Synthesis and Use of a Phosphoramidite Ligand for the Copper-Catalyzed Enantioselective­ Allylic Substitution. Tandem Allylic Substitution/Ring-Closing­ Metathesis

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Ueno, Yuichiro; Jiao, Guan-Sheng; Burgess, Kevin: Preparation of 5- and 6-Carboxyfluorescein

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Issue 14/2004

Lomberget, Thierry; Bossharth, Emmanuel; Bouyssi, Didier; Monteiro, Nuno; Balme, Geneviève: A Straightforward Entry to Functionalized Carbo- and Heterocycles Based on Pd-Mediated Cyclizations

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Chinkov, Nicka; Majumdar, Swapan; Marek, Ilan: Stereoselective Synthesis and Reactivity of Dienyl Zirconocene Derivatives

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Issue 13/2004

Tietze, Lutz F.; Hölsken, Sören; Adrio, Jens; Kinzel, Tom; Wegner, Christoph: Facial-Selective Allylation of Methyl Ketones for the Asymmetric Synthesis of Tertiary Homoallylic Ethers

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Issue 12/2004

Chao, Wenchun; Meketa, Matthew L.; Weinreb, Steven M.: Ring-Closing Metathesis of Vinyl Chlorides for Formation of 5-, 6- and 7-Membered Carbocyclic and Heterocyclic Systems

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von Hirschheydt, Thomas; Voss, Edgar: Simple, Short and Efficient Procedure for the Preparation of Hydroxyl- and Hydroxymethyl-Substituted 2,6-Dichlorobenzaldehydes

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Issue 11/2004

Cacchi, Sandro; Fabrizi, Giancarlo; Parisi, Luca M.: Preparation of Indoles from o-Alkynyltrifluoroacetanilides Through the Aminopalladation­-Reductive Elimination Process

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Park, Taesik; Torres, Eduardo; Fuchs, Philip L.: Improved and Environmentally Friendly Large-Scale Preparation of Cyclohexadienyl-, Cycloheptadienyl Sulfone and Enantiopure Epoxy Cycloheptyl Sulfones

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Issue 10/2004

Alonso, Diego A.; Botella, Luis; Nájera, C.; Pacheco, Mª Carmen: Synthetic Applications of Oxime-Derived Palladacycles as Versatile Catalysts in Cross-Coupling Reactions

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Issue 08/2004

Wolff, Oliver; Waldvogel, Siegfried R.: Reliable Protocol for the Large Scale Synthesis of Diphenylphosphoryl Azide (DPPA)

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Issue 07/2004

Yus, Miguel; Moreno, Benjamín; Foubelo, Francisco: Reductive Ring Opening of Oxygen-Containing Benzo-Fused Heterocycles by an Arene-Catalysed Lithiation

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Issue 06/2004

Schleusner, Marcel; Koep, Stefan; Günter, Markus; Tiwari, Shashi K.; Gais, Hans-Joachim: Preparation of (2-Methyl-propane-2-sulfonylimino) Acetic Acid Ethyl Ester

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Issue 05/2004

Rubin, Michael; Gevorgyan, Vladimir: Simple Large-Scale Preparation of 3,3-Disubstituted Cyclopropenes: Easy Access to Stereodefined Cyclopropylmetals via Transition Metal-Catalyzed Hydrometalation

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Issue 04/2004

Hilt, Gerhard; Lüers, Steffen; Schmidt, Frank: Cobalt(I)-Catalyzed Diels-Alder, 1,4-Hydrovinylation and 1,4-Hydrosilyl­ation Reactions of Non-Activated Starting Materials on a Large Scale

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Issue 03/2004

Diver, Steven T.; Giessert, Anthony J.: Enyne Metathesis: A Catalytic, Cross-Selective Diene Synthesis

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Issue 02/2004

Bajracharya, Gan B.; Nogami, Tsutomu; Jin, Tienan; Matsuda, Kumiko; Gevorgyan, Vladimir; Yamamoto, Yoshinori: Reduction of Carbonyl Function to a Methyl Group

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Issue 01/2004

Ley, Steven V.; Michel, Patrick: Preparation of Butane-1,2-diacetal-protected l-Glyceraldehyde from d-Mannitol

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Issue 18/2003

Muñoz, Mª Paz; Méndez, María; Nevado, Cristina; Cárdenas, Diego J.; Echavarren, Antonio M.: Hydroxy- and Alkoxycyclizations of Enynes Catalyzed by Platinum(II) Chloride

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Issue 17/2003

Schaffner, Arnaud-Pierre; Becattini, Barbara; Ollivier, Cyril; Weber, Valéry; Renaud, Philippe: B-Alkylcatecholboranes as a Source of Radicals for Efficient Conjugate Additions­ and Allylations

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Issue 16/2003

Marion, Nicolas; Navarro, Oscar; Kelly III, Roy A.; Nolan, Steven P.: Synthesis of Biaryl, Arylamine and Aryl Ketone Compounds Using a Commercially Available Air- and Moisture-Stable Palladium Catalyst

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Issue 15/2003

Zwikker, Jan W.; Brandsma, Lambert; Verkruijsse, Hermann D.: Simplified Procedures for 1-Amino-2-propyne and Some Homologues

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Issue 14/2003

Gaulon, Catherine; Dhal, Robert; Dujardin, Gilles: Preparation of Chiral N-Vinyl Oxazolidinones by a Simple General Procedure

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Issue 13/2003

Kulesza, Anna; Jurczak, Janusz: The Diastereoselective Barbier-Type Addition to Chiral N-Tosylimines

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Issue 12/2003

Larionov, Oleg V.; Kozhushkov, Sergei I.; de Meijere, Armin: New Protocol for Efficient N-Chlorinations of Amides and Carbamates

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Issue 08/2003

Enders, Dieter; Breuer, Klaus; Kallfass, Ulrike; Balensiefer, Tim: Preparation and Application of 1,3,4-Triphenyl-4,5-dihydro-1H-1,2,4-triazol-5-ylidene, A Stable Carbene

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Issue 06/2003

Kozhushkov, Sergei I.; Leonov, Andrei; de Meijere, Armin: Simple Large-Scale Preparation of 1,2,3-Tris-Acceptor Substituted Cyclopropanes

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Issue 12/2002

Enders, Dieter; Voith, Matthias; Ince, Stuart J.: Preparation and Reactions of 2,2-Dimethyl-1,3-dioxan-5-one-SAMP-Hydrazone: A Versatile Chiral Dihydroxyacetone Equivalent

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Issue 10/2002

Peña, Diego; Cobas, Agustín; Pérez, Dolores; Guitián, Enrique: An Efficient Procedure for the Synthesis of ortho-Trialkylsilylaryl Triflates: Easy Access to Precursors of Functionalized Arynes

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Issue 08/2002

Tokuyama, Hidetoshi; Yokoshima, Satoshi; Lin, Shao-Cheng; Li, Leping; Fukuyama, Tohru: Reduction of Ethanethiol Esters to Aldehydes

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Issue 04/2002

Jensen, Anne Eeg; Dohle, Wolfgang; Sapountzis, Ioannis; Lindsay, David M.; Vu, Viet Anh; Knochel, Paul: Preparation and Reactions of Functionalized Arylmagnesium Reagents

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