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Synthesis 2001(12): 1775-1777
DOI: 10.1055/s-2001-17517
DOI: 10.1055/s-2001-17517
SHORTPAPER
© Georg Thieme Verlag Stuttgart · New York
An Expedient Synthesis of 1-[3-(Dimethylamino)propyl]-5-methyl-3-phenyl-1H-indazole (FS-32) - An Antidepressant
Weitere Informationen
Received
16 May 2001
Publikationsdatum:
11. August 2004 (online)
Publikationsverlauf
Publikationsdatum:
11. August 2004 (online)
Abstract
Intramolecular 1,3-dipolar cycloaddition of functionalized sydnone leading to the synthesis of 1-[3-(dimethylamino)propyl]-5-methyl-3-phenyl-lH-indazole (FS-32), an antidepressant drug candidate, is described.
Keywords
intramolecular 1,3-dipolar cycloaddition - sydnones - antidepressant - FS-32
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