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Synlett 1999; 1999(12): 1957-1959
DOI: 10.1055/s-1999-2987
DOI: 10.1055/s-1999-2987
letter
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Two Efficient N-Acylation Methods Mediated by Solid-Supported Reagents for Weakly Nucleophilic Heterocyclic Amines
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Publication History
Publication Date:
31 December 1999 (online)
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Two efficient acylation methods utilizing solid-supported reagents have been developed for weakly nucleophilic heterocyclic amines. The novel approaches by chemoselective purification and polymeric-supported reagents facilitate library synthesis of diverse heterocyclic amides that are found in several pharmacophores.
acylation - amide - chemoselective purification - combinatorial chemistry - solid-supported reagents