Synlett 1996; 1996(9): 820-822
DOI: 10.1055/s-1996-5606
letter
© Georg Thieme Verlag, Rüdigerstr. 14, 70469 Stuttgart, Germany. All rights reserved. This journal, including all individual contributions and illustrations published therein, is legally protected by copyright for the duration of the copyright period. Any use, exploitation or commercialization outside the narrow limits set by copyright legislation, without the publisher's consent, is illegal and liable to criminal prosecution. This applies in particular to photostat reproduction, copying, cyclostyling, mimeographing or duplication of any kind, translating, preparation of microfilms, and electronic data processing and storage.

A Concise Route to Tetrahydrophenanthridinones and Functionalised Isoquinolones

Harry Heaney* , Mutasem O. Taha
  • *Department of Chemistry, Loughborough University, Loughborough, Leicestershire, LE11 3TU, Fax +44 (1509) 223925, E-mail h.heaney@lboro.ac.uk
Further Information

Publication History

Publication Date:
31 December 2000 (online)

Reaction of homophthalic anhydride with benzylamine and β-arylethylamine derivatives followed by alkylation, regioselective reduction, and treatment with Lewis acids generate acyliminium ions which, after rearrangement and loss of a proton, give tetrahydrophenanthridinones or isoquinolones.