Synthesis 1991; 1991(3): 244
DOI: 10.1055/s-1991-26437
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Synthesis of (±)-3-Amino-2-(4-chlorophenyl)propanesulfonic acid (Saclofen)

Chun-Sing Li* , W. Howson, Roland E. Dolle
  • *Department of Medicinal Chemistry, Smith Kline & French Research Ltd. The Frythe, Welwyn, Hertfordshire, AL6 9AR, England
Further Information

Publication History

Publication Date:
17 September 2002 (online)

An efficient synthesis of saclofen, a putative GABAB antagonist, is reported.