Synthesis 2022; 54(10): 2487-2493
DOI: 10.1055/a-1730-8186
paper

Room Temperature, Metal-Free, Regioselective Arylselenation of Anilines Using Diselenides as Selenium Source

Rekha Bai
,
Kamlesh Kumar Dabaria
,
The Council of Scientific and Industrial Research [No. 02(0341)/18/EMR-II] and SERB-DST, New Delhi (CRG/2020/003634).


This work is dedicated to Professor Deevi Basavaiah (University of Hyderabad) on his 71st birthday.

Abstract

A metal-free direct C–H selenation of aniline derivatives via an iodine-catalyzed C–Se bond formation using diselenides as a selenium source at ambient temperature is described. A variety of aniline derivatives underwent regioselective C–H selenation with different diselenides to afford the corresponding aryl selenoethers in good to excellent yields.

Supporting Information



Publikationsverlauf

Eingereicht: 03. August 2021

Angenommen nach Revision: 04. Januar 2022

Accepted Manuscript online:
04. Januar 2022

Artikel online veröffentlicht:
08. März 2022

© 2022. Thieme. All rights reserved

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